Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3180 products of "Endocrinology/Hormones"
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(Glu2)-TRH
CAS:(Glu2)-TRH: Stable TRH analog; reduces TRH's cholinergic action; no thyroliberinase metabolism; neuroprotective with antidepressant, anticonvulsant effects.Formula:C15H22N4O6Color and Shape:SolidMolecular weight:354.36[Arg8]-Vasotocin
CAS:<p>[Arg8]-Vasotocin is a hormone present in the neurohypophysis of nonmammalian vertebrates that is related to vasopressin and oxytocin.</p>Formula:C43H67N15O12S2Purity:98%Color and Shape:SolidMolecular weight:1050.22N-Acetyl-α-Endorphin
CAS:N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Formula:C79H122N18O27SPurity:98%Color and Shape:SolidMolecular weight:1787.98Dynorphin A (1-8)
CAS:<p>Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin.</p>Formula:C46H72N14O10Purity:98%Color and Shape:SolidMolecular weight:981.15[Ala17]-MCH TFA
<p>'[Ala17]-MCH TFA is an MCH analogue, a selective MCHR1 ligand (Ki=0.16 nM) with high affinity (Kd=0.37 nM), and low MCHR2 affinity (Ki=34 nM).</p>Formula:C99H156F3N29O28S4Color and Shape:SolidMolecular weight:2385.73MCH(human, mouse, rat) TFA
<p>MCH TFA, a peptide, selectively binds MCH1R and MCH2R with IC50 of 0.3nM, 1.5nM; EC50s are 3.9nM (MCH1R) and 0.1nM (MCH2R) in CHO cells.</p>Formula:C107H161F3N30O28S4Color and Shape:SolidMolecular weight:2500.861-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone
CAS:<p>1-Methyl-quinolone alkaloid inhibits DAG acyltransferase, blocks angiotensin II receptor (IC50s: 20.1 & 34.1 μM), and fights H. pylori (MIC: 10 μg/mL).</p>Formula:C23H31NOColor and Shape:SolidMolecular weight:337.5SL910102
CAS:<p>SL910102 is a nonpeptide angiotensin antagonist of the AT1 receptor.</p>Formula:C30H30N6OPurity:98%Color and Shape:SolidMolecular weight:490.60OT antagonist 1 demethyl derivative
<p>OT antagonist 1 demethyl derivative is the demethyl derivative of OT antagonist 1. OT antagonist 1 is a selective Oxytocin antagonist (Ki of 50 nM. )</p>Formula:C21H20N4O3Purity:98%Color and Shape:SolidMolecular weight:376.41PROTAC ER Degrader-15
<p>PROTAC ER Degrader-15 (Compound 40) is an orally active estrogen receptor (ER) degrader with anticancer properties, suitable for breast cancer research.</p>Formula:C47H47F4N5O5Color and Shape:SolidMolecular weight:837.9Floramanoside C
CAS:<p>Floramanoside C exhibits 2,2-diphenyl-1-picrylhydrazyl scavenging and aldose reductase inhibitory activities [1].</p>Formula:C21H18O15Color and Shape:SolidMolecular weight:510.36SR 43845
CAS:<p>SR 43845 is an inhibitor of renin.</p>Formula:C44H64N8O8Purity:98%Color and Shape:SolidMolecular weight:833.044Abaloparatide
CAS:<p>Abaloparatide (BA 058) is a selective PTHR1 analog that promotes bone growth and may be researched for osteoporosis.</p>Formula:C174H300N56O49Color and Shape:SolidMolecular weight:3960.59CTOP
CAS:<p>Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (>10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.</p>Formula:C50H67N11O11S2Purity:98%Color and Shape:SolidMolecular weight:1062.28Aclerastide
CAS:<p>Aclerastide, an angiotensin receptor agonist, decreases fibrosis in wounds; effect increases with use duration, blocked by AT antagonist.</p>Formula:C42H64N12O11Color and Shape:SolidMolecular weight:913.03Locicortolone
CAS:<p>Locicortolone is a synthetic glucocorticoid corticosteroid which was never marketed.</p>Formula:C22H28Cl2O3Color and Shape:SolidMolecular weight:411.36Handle region peptide, rat
CAS:<p>Rat handle region peptide acts as prorenin receptor blocker, curbs diabetic kidney disease, and reduces eye inflammation.</p>Formula:C54H101N15O12SPurity:98%Color and Shape:SolidMolecular weight:1184.54Linuron
CAS:<p>Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.</p>Formula:C9H10Cl2N2O2Purity:99.08%Color and Shape:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An HerbicideMolecular weight:249.09Prednicarbate
CAS:<p>Prednicarbate (Hoe 777), a corticosteroid, has antipruritic, anti-inflammatory effects, reduces lymphocytes, and inhibits vasodilators.</p>Formula:C27H36O8Purity:99.88%Color and Shape:SolidMolecular weight:488.57Ditekiren
CAS:<p>Ditekiren is a renin inhibitor with orally active.</p>Formula:C50H75N9O8Purity:98%Color and Shape:SolidMolecular weight:930.19OP-3633
CAS:<p>OP-3633: potent GR antagonist (IC50: 29 nM), low PR agonism, AR antagonism, inhibits GR transcription.</p>Formula:C30H39NO2Purity:98%Color and Shape:SolidMolecular weight:445.64RTI-13951-33 hydrochloride
<p>RTI-13951-33 HCl: potent, selective GPR88 agonist; brain-penetrant; EC50 = 25nM; curbs rat alcohol behaviors.</p>Formula:C28H35Cl2N3O3Purity:98%Color and Shape:SolidMolecular weight:532.5GLL 398
CAS:<p>GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.</p>Formula:C25H23BO4Purity:98%Color and Shape:SolidMolecular weight:398.26Hemorphin-7
CAS:<p>Hemorphin-7, an atypical opioid peptide from hemoglobin, may enhance memory, promote cell growth, and is a potential breast cancer biomarker.</p>Formula:C49H64N12O11Purity:98%Color and Shape:SolidMolecular weight:997.11TAN67
CAS:<p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>Formula:C23H26Br2N2OColor and Shape:SolidMolecular weight:506.282PROTAC ERα Degrader-8
CAS:<p>PROTAC ERα Degrader-8 (compound ii-56), a highly potent degrader of Erα, achieves a DC50 of just 0.000006 μM in MCF7 cells [1].</p>Formula:C47H51N5O4Color and Shape:SolidMolecular weight:749.947β-Hydroxy-epi-androsterone
CAS:<p>7β-Hydroxy-epi-androsterone (7β-Hydroxy-EpiA) is an endogenous androgenic derivative of dehydroepiandrosterone that possesses the ability to bind to ERβ,</p>Formula:C19H30O3Color and Shape:SolidMolecular weight:306.44Lactandrate
CAS:<p>Lactandrate is a homo-aza-steroidal ester of p-bis(2-chloroethyl) amino phenyl acetic acid.</p>Formula:C31H44Cl2N2O3Color and Shape:SolidMolecular weight:563.6BAM-22P
CAS:<p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>Formula:C130H184N38O31S2Purity:98%Color and Shape:SolidMolecular weight:2839.2211-Ketodihydrotestosterone
CAS:<p>11-Ketodihydrotestosterone is a metabolite of 11β-Hydroxyandrostenedione. It is an active androgen and is also a potent androgen receptor (AR) agonist (Ki: 20.4 nM, EC50: 1.35 nM for human AR).</p>Formula:C19H28O3Color and Shape:SolidMolecular weight:304.42Zankiren
CAS:<p>Zankiren is a renin inhibitor. Zankiren can reduce blood pressure, plasma renin activity, and angiotension II.</p>Formula:C35H55N5O6S2Color and Shape:SolidMolecular weight:705.97D3R/MOR antagonist 1
<p>Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nM</p>Formula:C22H27Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:420.38ICI 174,864
CAS:<p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>Formula:C38H53N5O7Purity:98%Color and Shape:White SolidMolecular weight:691.87Nociceptin(1-7)
CAS:<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Formula:C31H41N7O9Purity:98%Color and Shape:SolidMolecular weight:655.709KOR agonist 4
<p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>Formula:C21H25N3Color and Shape:SolidMolecular weight:319.44Vasopressin Dimer (anti-parallel) (TFA)
<p>Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate four G protein-coupled receptors: V1aR, V1bR,</p>Formula:C94H131F3N30O26S4Purity:98%Color and Shape:SolidMolecular weight:2282.49Raloxifene 4'-glucuronide
CAS:<p>Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene.</p>Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71MT-7716 free base
CAS:<p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>Formula:C27H28N4O2Purity:98%Color and Shape:SolidMolecular weight:440.54[Nphe1]Nociceptin(1-13)NH2 TFA
<p>[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.</p>Formula:C63H101F3N22O17Color and Shape:SolidMolecular weight:1495.614A7C-301
<p>4A7C-301, a Nurr1 agonist, exhibits potent neuroprotective effects in vitro and markedly mitigates neuropathological abnormalities while enhancing motor and</p>Color and Shape:Odour SolidCJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formula:C34H35N5O4Color and Shape:SolidMolecular weight:577.67Orphanin FQ(1-11)
CAS:<p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>Formula:C49H75N15O14Purity:98%Color and Shape:SolidMolecular weight:1098.2RS 21314
CAS:<p>RS 21314 is a thiol ester corticosteroid that is topical.</p>Formula:C24H30F2O5SColor and Shape:SolidMolecular weight:468.55SNIPER(ER)-87
CAS:<p>SNIPER(ER)-87 is a chemical compound composed of a derivative of the inhibitor of apoptosis protein (IAP) ligand LCL161 conjugated to the estrogen receptor α (</p>Formula:C59H73N5O10SPurity:98%Color and Shape:SolidMolecular weight:1044.32Triphenylethylene
CAS:<p>Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formula:C20H16Color and Shape:White PowderMolecular weight:256.34Angiotensin II (1-4), human TFA
<p>Angiotensin II is a potent direct vasoconstrictor, causing arteries and veins to constrict, so leading to an increase in blood pressure.</p>Formula:C26H38F3N7O10Purity:98%Color and Shape:SolidMolecular weight:665.62KOR agonist 5
<p>KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD).</p>Formula:C38H38N2O5Color and Shape:SolidMolecular weight:602.72Inocoterone acetate
CAS:<p>Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.</p>Formula:C18H26O3Color and Shape:SolidMolecular weight:290.4018-Oxocortisol
CAS:<p>18-Oxocortisol, a naturally occurring mineralocorticoid and adrenal biomarker, is produced by CYP11B2.</p>Formula:C21H28O6Color and Shape:SolidMolecular weight:376.449Imlunestrant tosylate
CAS:<p>Imlunestrant (LY-3484356) tosylate, an oral SERD, targets ER+ aBC/EEC by blocking estrogen receptors and gene transcription.</p>Formula:C36H32F4N2O6SColor and Shape:SolidMolecular weight:696.71
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