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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • TRβ agonist 1
    Targetmol
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    TRβ agonist 1

    CAS:
    <p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>
    Formula:C29H25FN2O8
    Color and Shape:Solid
    Molecular weight:548.52

    Ref: TM-T63876

  • PD 134922
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    PD 134922

    CAS:
    <p>PD 134922 is a HIV-1 protease inhibitors. Inactivation of the protease prevents infectious virion formation.</p>
    Formula:C37H61N5O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:719.97

    Ref: TM-T28329

  • rel-SB-612111 hydrochloride
    Targetmol
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    rel-SB-612111 hydrochloride

    CAS:
    <p>NOP receptor antagonist</p>
    Formula:C24H30Cl3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.86

    Ref: TM-T23324

  • JNJ-1250132
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    JNJ-1250132

    CAS:
    <p>JNJ-1250132 is a steroidal progesterone receptor modulator that inhibits binding of the receptor to DNA in vitro.</p>
    Formula:C33H41NO4
    Color and Shape:Solid
    Molecular weight:515.68

    Ref: TM-T27662

  • GPR84 antagonist 3
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    GPR84 antagonist 3

    CAS:
    <p>Potent GPR84 antagonist 3 (compound 42), pIC50 8.28, inhibits GTPγS, with good pharmacokinetics.</p>
    Formula:C29H27N5O
    Color and Shape:Solid
    Molecular weight:461.56

    Ref: TM-T62918

  • Androgen receptor degrader-5
    Targetmol
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    Androgen receptor degrader-5

    CAS:
    <p>Androgen receptor degrader-5 (compound 14k) demonstrates superior capabilities, specifically in androgen receptor degradation and antiproliferative activity, showcasing its promising properties.</p>
    Formula:C29H25F4N5O2
    Color and Shape:Solid
    Molecular weight:551.53

    Ref: TM-T200197

  • Sunobinop
    Targetmol
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    Sunobinop

    CAS:
    <p>Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.</p>
    Formula:C26H33N3O3
    Color and Shape:Solid
    Molecular weight:435.56

    Ref: TM-T62482

  • Norbinaltorphimine dihydrochloride
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    Norbinaltorphimine dihydrochloride

    CAS:
    <p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>
    Formula:C40H45Cl2N3O6
    Purity:98.17% - 99.88%
    Color and Shape:Solid
    Molecular weight:734.71

    Ref: TM-T12241

  • SC13
    Targetmol
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    SC13

    CAS:
    <p>SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.</p>
    Formula:C26H30N2O5
    Color and Shape:Solid
    Molecular weight:450.53

    Ref: TM-T62722

  • FL442
    Targetmol
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    FL442

    CAS:
    <p>FL442 is an Androgen Receptor (AR) modulator. This compound exhibits potent inhibitory effects in AR-dependent prostate cancer cells, showing similar suppression efficiency to the traditional antiandrogen drugs Bicalutamide and Enzalutamide. It also maintains antiandrogen activity against the Enzalutamide-resistant AR mutant F876L. The pharmacokinetic properties of FL442 in mice reveal a longer half-life (8 hours), excellent targeting (prostate tissue), and metabolic stability. Additionally, it is effective at inhibiting LNCaP tumor growth at low plasma concentrations (30 ng/mL).</p>
    Formula:C15H13F3N2O
    Color and Shape:Solid
    Molecular weight:294.27

    Ref: TM-T200138

  • LY2066948
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    LY2066948

    CAS:
    <p>LY2066948 is a selective oral estrogen receptor modulator (SERM) with high affinity for estrogen receptors ERα and ERβ (Ki of 0.51 and 1.36 nM, respectively) and displays potent anti-estrogenic activity. It effectively blocks the increase in uterine weight induced by ethinylestradiol in immature rats. LY2066948 is utilized in the research of uterine fibroids and myomas.</p>
    Formula:C30H31NO5S
    Color and Shape:Solid
    Molecular weight:517.64

    Ref: TM-T200177

  • CCG258747
    Targetmol
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    CCG258747

    CAS:
    <p>CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.</p>
    Formula:C28H27FN4O4
    Color and Shape:Solid
    Molecular weight:502.54

    Ref: TM-T63411

  • MK-6913
    Targetmol
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    MK-6913

    CAS:
    <p>MK-6913 is a potent and selective agonist of estrogen receptor β.</p>
    Formula:C25H27N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.5

    Ref: TM-T13136

  • Elacestrant S enantiomer dihydrochloride
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    Elacestrant S enantiomer dihydrochloride

    <p>Elacestrant (RAD1901) dihydrochloride, an oral ERR degrader, has IC50 of 48 nM (ERα) and 870 nM (ERβ). Its S enantiomer has low activity.</p>
    Formula:C30H40Cl2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.56

    Ref: TM-T11173L

  • A 74273
    Targetmol
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    A 74273

    CAS:
    <p>A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.</p>
    Formula:C44H74N4O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:787.08

    Ref: TM-T26439

  • Estrogen receptor antagonist 6
    Targetmol
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    Estrogen receptor antagonist 6

    CAS:
    <p>Estrogen receptor antagonist 6 is a potent blocker of estrogen signaling, regulating various biological effects. (Compound 166)</p>
    Formula:C25H31F3N2O3
    Color and Shape:Solid
    Molecular weight:464.52

    Ref: TM-T62953

  • (+)-JJ-74-138
    Targetmol
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    (+)-JJ-74-138

    CAS:
    <p>(+)-JJ-74-138 is a novel non-competitive androgen receptor (AR) antagonist capable of inhibiting enzalutamide-resistant castration-resistant prostate cancer (CRPC).</p>
    Formula:C22H22F8N2OS
    Color and Shape:Solid
    Molecular weight:514.48

    Ref: TM-T200319

  • CymitQuimica logo
    Targetmol
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    Mu opioid receptor antagonist 4

    <p>Compound 31: Potent, selective MOR antagonist; crosses blood-brain barrier; Ki &amp; EC50: 0.38 nM; useful for OUD research.</p>
    Formula:C25H28N2O4S
    Color and Shape:Solid
    Molecular weight:452.57

    Ref: TM-T62768

  • CymitQuimica logo
    Targetmol
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    σ1 Receptor/μ Opioid receptor modulator 2

    CAS:
    <p>Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM). It demonstrates significant analgesic effects in various pain models.</p>
    Formula:C23H31N3O
    Molecular weight:365.51

    Ref: TM-T208835

  • RJG-2051
    Targetmol
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    RJG-2051

    CAS:
    <p>RJG-2051 is a selective covalent inhibitor of aldo-keto reductase family 1 member C3 (AKR1C3), with an IC50 value of 13 nM. It interferes with the metabolism of substrates such as androgens, estrogens, and prostaglandins through AKR1C3. RJG-2051 holds potential for cancer research.</p>
    Formula:C26H31N5O4S
    Color and Shape:Solid
    Molecular weight:509.62

    Ref: TM-T206799