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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • Androstatrione
    Targetmol
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    Androstatrione

    CAS:
    <p>Androstatrione is an androgenic compound.</p>
    Formula:C19H26O3
    Color and Shape:Solid
    Molecular weight:302.41

    Ref: TM-T207371

  • BNTX
    Targetmol
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    BNTX

    CAS:
    <p>BNTX (7-Benzylidenenaltrexone) is a selective δ1-opioid receptor antagonist. It competitively counteracts the antisecretory effects of DPDPE, Deltorphin 2, and DAMGO. BNTX is applicable in research focused on antinociceptive effects.</p>
    Formula:C27H27NO4
    Color and Shape:Solid
    Molecular weight:429.508

    Ref: TM-T206469

  • Estrogen receptor antagonist 4
    Targetmol
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    Estrogen receptor antagonist 4

    CAS:
    <p>Estrogen receptor antagonist 4 blocks ER, impacting cell growth and cancer research potential.</p>
    Formula:C23H29BF4N4O2
    Color and Shape:Solid
    Molecular weight:480.31

    Ref: TM-T63106

  • ORIC-101
    Targetmol
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    ORIC-101

    CAS:
    <p>ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.</p>
    Formula:C34H47NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:501.74

    Ref: TM-T16404

  • Estrone acetate
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    Estrone acetate

    CAS:
    <p>Estrone acetate (Hogival) is an estrogen derivative and an activator of estrogen receptors (ER). This compound can enhance breast development, stimulate the secretion of pituitary prolactin, and induce both the proliferation and activation of lactotrophs, evidenced by the reduction in prolactin storage granule size and the increase in the volume density of the rough endoplasmic reticulum and Golgi apparatus. Estrone acetate holds potential for endocrinological research and for investigating the mechanisms by which estrogen influences pituitary function, prolactin regulation, and breast tumor models.</p>
    Formula:C20H24O3
    Color and Shape:Solid
    Molecular weight:312.403

    Ref: TM-T206611

  • AP5 sodium
    Targetmol
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    AP5 sodium

    CAS:
    <p>AP5 sodium: potent oral GPR40 agonist, enhances ligands, may aid type II diabetes research.</p>
    Formula:C28H27FNNaO4
    Color and Shape:Solid
    Molecular weight:483.515

    Ref: TM-T63202

  • AVE 0991
    Targetmol
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    AVE 0991

    CAS:
    <p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>
    Formula:C29H32N4O5S2
    Purity:98.69%
    Color and Shape:Solid
    Molecular weight:580.72

    Ref: TM-TQ0057

  • BMS-986118
    Targetmol
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    BMS-986118

    CAS:
    <p>BMS-986118 is a GPR40 full agonist targeting type II diabetes, prompting insulin release without hypoglycemia risk.</p>
    Formula:C25H28ClF3N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.96

    Ref: TM-T26868

  • (±)-J 113397
    Targetmol
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    (±)-J 113397

    CAS:
    <p>(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).</p>
    Formula:C24H37N3O2
    Color and Shape:Solid
    Molecular weight:399.57

    Ref: TM-T21999

  • LX1
    Targetmol
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    LX1

    CAS:
    <p>LX1, an anti-prostate cancer compound, specifically targets the androgen receptor (AR), AR variants, and the steroidogenic enzyme AKR1C3. It inhibits AKR1C3's enzymatic function, decreases the conversion of androstenedione to testosterone, and reduces the expression of both AR and AR-V7, subsequently downregulating their target genes. Additionally, LX1 is effective in overcoming tumor cell resistance to Enzalutamide, and when combined with Enzalutamide, it further suppresses tumor growth.</p>
    Formula:C22H15F6NO2
    Color and Shape:Solid
    Molecular weight:439.35

    Ref: TM-T200147

  • GLPG0492 (R enantiomer)
    Targetmol
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    GLPG0492 (R enantiomer)

    CAS:
    <p>GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, a novel selective androgen receptor modulator.</p>
    Formula:C19H14F3N3O3
    Color and Shape:Solid
    Molecular weight:389.33

    Ref: TM-T11410

  • GPR81 agonist 2
    Targetmol
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    GPR81 agonist 2

    CAS:
    <p>GPR81 agonist 2 is a potent agonist targeting the GPR81 receptor, demonstrating EC50 values of 0.023 µM for hGPR81 and 0.123 µM for hGPR109A, respectively.</p>
    Formula:C26H27ClN6O5S2
    Color and Shape:Solid
    Molecular weight:603.11

    Ref: TM-T72772

  • Dazucorilant
    Targetmol
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    Dazucorilant

    CAS:
    <p>Dazucorilant (CORT113176), a selective non-steroidal GR modulator, has high affinity with a K i &lt;1 nM, useful for neurological research.</p>
    Formula:C29H22F4N4O3S
    Color and Shape:Solid
    Molecular weight:582.57

    Ref: TM-T38983

  • TD-0212
    Targetmol
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    TD-0212

    CAS:
    <p>TD-0212: Oral dual antagonist for AT1 (pKi 8.9) &amp; NEP inhibitor (pIC50 9.2).</p>
    Formula:C28H34FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.65

    Ref: TM-T13125

  • LNS8801
    Targetmol
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    LNS8801

    CAS:
    <p>LNS8801 is an orally active agonist of the G protein-coupled estrogen receptor (GPER). By activating GPER, LNS8801 mediates downstream signaling pathways, such as promoting cAMP production and activating CREB signaling, which results in antitumor activities like inhibiting tumor cell proliferation, inducing cell differentiation, and enhancing tumor immunogenicity. It is applicable in research across various cancers, such as melanoma, pancreatic cancer, colorectal cancer, and lung cancer, as well as studies exploring the role of GPER in normal physiological and pathological processes.</p>
    Formula:C21H18BrNO3
    Color and Shape:Solid
    Molecular weight:412.277

    Ref: TM-T206565

  • C108297
    Targetmol
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    C108297

    CAS:
    <p>C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.</p>
    Formula:C30H36FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.69

    Ref: TM-T26935

  • FSH receptor antagonist 1
    Targetmol
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    FSH receptor antagonist 1

    CAS:
    <p>FSH receptor antagonist 1 (compound 10) is a potent antagonist of the G(s) protein-coupled human follicle-stimulating hormone (FSH) receptor. It exhibits an IC50 value of 28 nM in cell lines expressing the human FSH receptor. This compound significantly inhibits follicle growth and ovulation in in vitro mouse models.</p>
    Formula:C33H32N2O2
    Color and Shape:Solid
    Molecular weight:488.619

    Ref: TM-T204299

  • SDM25N hydrochloride
    Targetmol
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    SDM25N hydrochloride

    CAS:
    <p>δ receptor antagonist</p>
    Formula:C26H27ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:450.96

    Ref: TM-T23341

  • Estrogen receptor-agonist-1
    Targetmol
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    Estrogen receptor-agonist-1

    CAS:
    <p>Estrogen receptor-agonist-1 (compound 4e) is an estrogen receptor (ER) agonist that binds to ERα with high affinity.</p>
    Formula:C24H22N2O2
    Color and Shape:Solid
    Molecular weight:370.444

    Ref: TM-T204741

  • CymitQuimica logo
    Targetmol
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    ERRγ agonist-1

    <p>ERRγ agonist-1 can be used in neuropsychological disorders research.</p>
    Formula:C17H21N5O
    Color and Shape:Solid
    Molecular weight:311.38

    Ref: TM-T60772