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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • ACT 178882
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    ACT 178882

    CAS:
    <p>ACT 178882 is a new Renin inhibitor (IC50: 1.4 nM).</p>
    Formula:C33H38Cl3N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:647.03

    Ref: TM-T14123

  • Androgen receptor antagonist 11
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    Androgen receptor antagonist 11

    CAS:
    <p>Androgen receptor antagonist 11 (compound N29) is a selective, orally available antagonist.</p>
    Formula:C20H19F3N4O3S
    Color and Shape:Solid
    Molecular weight:452.45

    Ref: TM-T201269

  • J-113397
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    J-113397

    CAS:
    <p>J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).</p>
    Formula:C24H37N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.57

    Ref: TM-T27649

  • ER degrader 10
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    ER degrader 10

    CAS:
    <p>ER degrader 10 (Compound 51) is an orally active estrogen receptor (ER) selective degrader and antagonist, with a DC50 of 0.43 nM and an IC50 of 0.56 nM. It inhibits the proliferation of ER-positive cells, with an IC50 ranging from 0 to 15 nM. ER degrader 10 exhibits weak inhibitory activity on the hERG channel, with an IC50 greater than 40 μM. It has blood-brain barrier permeability, with a brain/plasma ratio (Kp) of 3.05. In mouse models, ER degrader 10 demonstrates antitumor activity.</p>
    Formula:C28H29F2NO3S
    Color and Shape:Solid
    Molecular weight:497.597

    Ref: TM-T204775

  • ADX61623
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    ADX61623

    CAS:
    <p>ADX61623 is an effective negative allosteric modulator (NAM) of the follicle-stimulating hormone receptor (FSHR). It also exhibits activity on the luteinizing hormone receptor (LH-R) but is inactive on the thyroid-stimulating hormone (TSH) receptor. ADX61623 can be utilized in research on estrogen-dependent diseases.</p>
    Formula:C19H20N2O3
    Color and Shape:Solid
    Molecular weight:324.37

    Ref: TM-T201265

  • ERα degrader 11
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    ERα degrader 11

    CAS:
    <p>ERα degrader11 (compound B16) is a selective estrogen receptor degrader designed for use as a probe in examining the ER status within ER-positive breast cancer cells.</p>
    Formula:C28H27F3N2O3
    Color and Shape:Solid
    Molecular weight:496.52

    Ref: TM-T200861

  • Fonsartan free acid
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    Fonsartan free acid

    CAS:
    <p>Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.</p>
    Formula:C26H32N4O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:544.69

    Ref: TM-T27347

  • Pentomone
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    Pentomone

    CAS:
    <p>Pentomone (LY-113935) is an anti-androgen compound that acts as a prostate growth inhibitor.</p>
    Formula:C24H26O5
    Color and Shape:Solid
    Molecular weight:394.46

    Ref: TM-T201000

  • Sob-AM2
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    Sob-AM2

    CAS:
    <p>Sob-AM2 is an effective substrate targeting the fatty acid amide hydrolase (FAAH) expressed in the brain, with a Km of 1.3 μM. It delivers higher concentrations of Sobetirome to the central nervous system at minimal peripheral systemic doses, thereby activating the central thyroid hormone receptor β (TRβ).</p>
    Formula:C21H27NO3
    Color and Shape:Solid
    Molecular weight:341.44

    Ref: TM-T200594

  • (S)-MCOPPB
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    (S)-MCOPPB

    CAS:
    <p>(S)-MCOPPB is the S-enantiomer of MCOPPB, an orally active selective agonist for the Nociceptin/Orphanin FQ-Receptor. It inhibits signal transduction in mouse brain NOP receptors and is utilized in anxiety disorder research.</p>
    Formula:C26H40N4
    Color and Shape:Solid
    Molecular weight:408.623

    Ref: TM-TYD-02076

  • L162389
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    L162389

    CAS:
    <p>L162389 is an angiotensin II receptor antagonist with a balanced affinity for AT1 and AT2 receptor and stimulates the conversion of phosphatidylinositol.</p>
    Formula:C31H38N4O4S
    Purity:99.11% - 99.57%
    Color and Shape:Solid
    Molecular weight:562.72

    Ref: TM-T11808

  • Androgen receptor ligand 1
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    Androgen receptor ligand 1

    CAS:
    <p>Androgen receptorligand 1 is a ligand for the androgen receptor (AR). It interacts with the CRBN E3 ligase via a linker to form an AR-PROTAC degrader. This compound is useful in prostate cancer research.</p>
    Formula:C19H16F4N2O
    Color and Shape:Solid
    Molecular weight:364.34

    Ref: TM-T207737

  • OT-R agonist 1 TFA
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    OT-R agonist 1 TFA

    CAS:
    <p>OT-R agonist 1 TFA (compound 5) is an oxytocin receptor (OT-R) agonist with an EC50 value of 0.39 nM. It exhibits V1A antagonist activity, with an EC50 value of 2432 nM, and can be utilized in studies related to central nervous system diseases.</p>
    Formula:C37H40F3N7O7S
    Color and Shape:Solid
    Molecular weight:783.82

    Ref: TM-T207687

  • Allyphenyline oxalate
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    Allyphenyline oxalate

    CAS:
    <p>The pKi values of Allyphenyline oxalate (compound 9) for the α2-adrenergic receptor subtypes α2A, α2B, and α2C are 7.24, 6.47, and 7.07, respectively.</p>
    Formula:C16H20N2O5
    Color and Shape:Solid
    Molecular weight:320.34

    Ref: TM-T204376

  • NSC 645827
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    NSC 645827

    CAS:
    <p>NSC 645827 is an inhibitor of NAD(P)H:quinone oxidoreductase 1 (NQO1), with an IC50 of 0.7 μM.</p>
    Formula:C17H17N5O2
    Color and Shape:Solid
    Molecular weight:323.349

    Ref: TM-T204942

  • CymitQuimica logo
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    AR antagonist 4

    <p>AR antagonist 4 (Compound 67-b) is an orally active androgen receptor (AR) antagonist that acts on wild-type AR (IC50: 246.6 nM).</p>
    Formula:C29H36N4O
    Color and Shape:Solid
    Molecular weight:456.62

    Ref: TM-T62838

  • CymitQuimica logo
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    ERα degrader 5

    <p>ERα degrader 5 is an orally active, selective estrogen receptor (ER) reducer that acts on ERα (EC50: 1.1 nM). ERα degrader 5 shows anti-tumour effects in vivo.</p>
    Formula:C29H25F4N3O2S
    Color and Shape:Solid
    Molecular weight:555.59

    Ref: TM-T63922

  • 5α-reductase-IN-1
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    5α-reductase-IN-1

    CAS:
    <p>5α-reductase-IN-1 is a potent inhibitor of the enzyme 5α-reductase.</p>
    Formula:C31H37NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:503.63

    Ref: TM-T10636

  • BU09059
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    BU09059

    CAS:
    <p>BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).</p>
    Formula:C28H37N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:495.61

    Ref: TM-T26919

  • Anticancer agent 257
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    Anticancer agent 257

    CAS:
    <p>Anticanceragent 257 (compound of formula (I)) is an anticancer agent that regulates Nur77 and Nurr1.</p>
    Formula:C15H9Cl2N3
    Color and Shape:Solid
    Molecular weight:302.158

    Ref: TM-T204917