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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • JTP-117968

    CAS:
    <p>JTP-117968: Non-steroidal SGRM, glucocorticoid receptor modulator, IC50 = 6.8 nM, offers better inhibitory/activatory balance.</p>
    Formula:C31H31F3N2O2
    Color and Shape:Solid
    Molecular weight:520.59
  • MB-07344 sodium


    <p>"MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."</p>
    Formula:C19H25NaO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:387.36
  • Mepixetil


    <p>Mepixetil is a potent angiotensin II receptor antagonist[1].</p>
    Formula:C12H18N2O3
    Color and Shape:Solid
    Molecular weight:238.28
  • Mopivabil


    <p>Mopivabil is the angiotensin II receptor antagonist[1].</p>
    Formula:C14H20O3
    Color and Shape:Solid
    Molecular weight:236.31
  • GPR84 antagonist 1


    <p>GPR84 antagonist 1 is a highly selective, high-affinity competitive antagonist of human GPR84.</p>
    Formula:C26H22N4O2
    Color and Shape:Solid
    Molecular weight:422.48
  • Mu opioid receptor antagonist 5


    <p>Compound NAP: MOR antagonist, crosses blood-brain barrier, EC50: 1.14 nM, Ki: 0.37 nM, useful for OUD research.</p>
    Formula:C26H29N3O4
    Color and Shape:Solid
    Molecular weight:447.53
  • ZD 7155 hydrochloride

    CAS:
    <p>ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.</p>
    Formula:C26H27ClN6O
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:474.98
  • GLPG0974

    CAS:
    <p>GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.</p>
    Formula:C25H25ClN2O4S
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:484.99
  • Cort108297

    CAS:
    <p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>
    Formula:C26H25F4N3O3S
    Purity:98.36% - 99.94%
    Color and Shape:Solid
    Molecular weight:535.55
  • Nalmefene

    CAS:
    <p>Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study of opioid overdose and alcohol dependence.</p>
    Formula:C21H25NO3
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:339.43
  • L-371,257

    CAS:
    <p>L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.</p>
    Formula:C28H33N3O6
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:507.58
  • (E/Z)-GSK5182

    CAS:
    <p>GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.</p>
    Formula:C27H31NO3
    Purity:97.58%
    Color and Shape:Solid
    Molecular weight:417.54
  • LSZ-102

    CAS:
    <p>LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.</p>
    Formula:C25H17F3O4S
    Purity:98.56%
    Color and Shape:Solid
    Molecular weight:470.46
  • (S)-Mapracorat

    CAS:
    <p>(S)-Mapracorat is a selective and less active agonist of the glucocorticoid receptor.</p>
    Formula:C25H26F4N2O2
    Color and Shape:Solid
    Molecular weight:462.48

    Ref: TM-T13451

    1mg
    Discontinued
    Discontinued product
  • ZK 216348

    CAS:
    <p>ZK 216348 also binds to Progesterone and mineralocorticoid receptors (IC50s: 20.4 nM and 79.9 nM, respectively). ZK 216348 is a nonsteroidal selective glucocorticoid receptor agonist (IC50: 20.3 nM). ZK 216348 has an anti-inflammatory activity similar to</p>
    Formula:C24H23F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:476.45

    Ref: TM-T17291

    1mg
    Discontinued
    Discontinued product
  • Mapracorat

    CAS:
    <p>Mapracorat (ZK-245186, BOL-303242X) is a selective glucocorticoid receptor agonist,anti-inflammatory agent for atopic dermatitis and allergic conjunctivitis.</p>
    Formula:C25H26F4N2O2
    Color and Shape:Solid
    Molecular weight:462.48

    Ref: TM-T13451L

    1mg
    Discontinued
    Discontinued product
  • PSN632408

    CAS:
    <p>PSN632408 is an optimized agonist of GPR119 receptors that display similar potency to OEA at both recombinant mouse and human GPR119 receptors (EC50: 5.6 and 7.9 uM, respectively).</p>
    Formula:C18H24N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:360.41

    Ref: TM-T16678

    1mg
    Discontinued
    Discontinued product
  • ML314

    CAS:
    <p>ML314 is a brain-permeable nonpeptide β-inhibin-biased neurotensin NTR1 receptor agonist (EC50: 1.9 μM), a biased neurotensin receptor ligand for methamphetamine abuse that inhibits NTR2 and GPR35.</p>
    Formula:C24H28N4O3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:420.504

    Ref: TM-TQ0075

    1mg
    Discontinued
    Discontinued product
  • Exemestane

    CAS:
    <p>Exemestane (EXE) is an Aromatase Inhibitor. The mechanism of action of exemestane is as an Aromatase Inhibitor.</p>
    Formula:C20H24O2
    Purity:99.35% - 99.35%
    Color and Shape:White To Light Yellow Crystal Powder
    Molecular weight:296.4

    Ref: TM-T1587

    1ml
    Discontinued
    Discontinued product
  • Relacorilant

    CAS:
    <p>Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.</p>
    Formula:C27H22F4N6O3S
    Purity:98.53% - 99%
    Color and Shape:Solid
    Molecular weight:586.56

    Ref: TM-T16727

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    500mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    1mL*10mM (DMSO)_old
    Discontinued
    Discontinued product