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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3359 products of "Endocrinology/Hormones"

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  • GLPG0492 (R enantiomer)
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    GLPG0492 (R enantiomer)

    CAS:
    GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, a novel selective androgen receptor modulator.
    Formula:C19H14F3N3O3
    Color and Shape:Solid
    Molecular weight:389.33

    Ref: TM-T11410

  • EN171
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    EN171

    CAS:
    EN171, a covalent ligand, selectively binds to C38 and C96 on 14-3-3, intensifying 14-3-3's interactions with ERα, YAP, and TAZ. This action impairs both estrogen receptor and Hippo pathway transcriptional activities. Beyond serving as a molecular glue to augment native protein interactions, EN171 also functions as a covalent recruiter for 14-3-3 in heterobifunctional molecules. This facilitates the sequestration of nuclear neo-substrates, such as BRD4 and BLC6, into the cytosol.
    Formula:C17H22N2O
    Color and Shape:Solid
    Molecular weight:270.37

    Ref: TM-T200403

  • MB-07344 sodium
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    MB-07344 sodium

    "MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."
    Formula:C19H25NaO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:387.36

    Ref: TM-T11954L

  • AVE 0991
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    AVE 0991

    CAS:
    AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.
    Formula:C29H32N4O5S2
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:580.72

    Ref: TM-TQ0057

  • AP5 sodium
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    AP5 sodium

    CAS:
    AP5 sodium: potent oral GPR40 agonist, enhances ligands, may aid type II diabetes research.
    Formula:C28H27FNNaO4
    Color and Shape:Solid
    Molecular weight:483.515

    Ref: TM-T63202

  • GNTI dihydrochloride
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    GNTI dihydrochloride

    CAS:
    κ opioid receptor antagonist
    Formula:C27H30ClN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.01

    Ref: TM-T22802

  • J-113397
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    J-113397

    CAS:
    J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).
    Formula:C24H37N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.57

    Ref: TM-T27649

  • Estrone acetate
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    Estrone acetate

    CAS:
    Estrone acetate (Hogival) is an estrogen derivative and an activator of estrogen receptors (ER). This compound can enhance breast development, stimulate the secretion of pituitary prolactin, and induce both the proliferation and activation of lactotrophs, evidenced by the reduction in prolactin storage granule size and the increase in the volume density of the rough endoplasmic reticulum and Golgi apparatus. Estrone acetate holds potential for endocrinological research and for investigating the mechanisms by which estrogen influences pituitary function, prolactin regulation, and breast tumor models.
    Formula:C20H24O3
    Color and Shape:Solid
    Molecular weight:312.403

    Ref: TM-T206611

  • Fonsartan free acid
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    Fonsartan free acid

    CAS:
    Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.
    Formula:C26H32N4O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:544.69

    Ref: TM-T27347

  • ORIC-101
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    ORIC-101

    CAS:
    ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.
    Formula:C34H47NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:501.74

    Ref: TM-T16404

  • PD 134922
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    PD 134922

    CAS:
    PD 134922 is a HIV-1 protease inhibitors. Inactivation of the protease prevents infectious virion formation.
    Formula:C37H61N5O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:719.97

    Ref: TM-T28329

  • Estrogen receptor antagonist 4
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    Estrogen receptor antagonist 4

    CAS:
    Estrogen receptor antagonist 4 blocks ER, impacting cell growth and cancer research potential.
    Formula:C23H29BF4N4O2
    Color and Shape:Solid
    Molecular weight:480.31

    Ref: TM-T63106

  • BNTX maleate
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    BNTX maleate

    CAS:
    δ1 opioid receptor antagonist
    Formula:C31H31NO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:545.58

    Ref: TM-T22613

  • Androstatrione
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    Androstatrione

    CAS:
    <p>Androstatrione is an androgenic compound.</p>
    Formula:C19H26O3
    Color and Shape:Solid
    Molecular weight:302.41

    Ref: TM-T207371

  • SC13
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    SC13

    CAS:
    SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.
    Formula:C26H30N2O5
    Color and Shape:Solid
    Molecular weight:450.53

    Ref: TM-T62722

  • Metahexestrol
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    Metahexestrol

    CAS:
    Metahexestrol is an inhibitor of the estrogen receptor (E2R) with antitumor activity. It significantly inhibits the proliferation of estrogen receptor-positive MCF-7 human breast cancer cell line with an ED50 of 1.0 μM. Additionally, Metahexestrol shows inhibitory activity in estrogen receptor-negative MDA-MB-231 cell lines, and its antiproliferative effect is not reversed by estrogen, suggesting that its mechanism may be partially independent of the E2R pathway. Metahexestrol is applicable in research on estrogen-dependent breast cancer.
    Formula:C18H22O2
    Color and Shape:Solid
    Molecular weight:270.366

    Ref: TM-T206528

  • Daeatal
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    Daeatal

    CAS:
    Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.
    Formula:C56H93N19O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1192.46

    Ref: TM-T23963

  • GC 14
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    GC 14

    CAS:
    GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 200 nM and 35 nM for hTRα and hTRβ, respectively.
    Formula:C26H27NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.5

    Ref: TM-T11376

  • CymitQuimica logo
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    σ1 Receptor/μ Opioid receptor modulator 2

    CAS:
    Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM). It demonstrates significant analgesic effects in various pain models.
    Formula:C23H31N3O
    Molecular weight:365.51

    Ref: TM-T208835

  • LIT-001 free base
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    LIT-001 free base

    CAS:
    LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.
    Formula:C28H33N7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.67

    Ref: TM-T11856