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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3348 products of "Endocrinology/Hormones"

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  • CymitQuimica logo
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    ST-CY14

    <p>ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.</p>
    Formula:C139H237N57O31S2
    Color and Shape:Solid
    Molecular weight:3266.86

    Ref: TM-TP3109

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    PTP1B/AKR1B1-IN-2

    <p>PTP1B/AKR1B1-IN-2 (Compound 7f) is a potent inhibitor targeting both PTP1B and AKR1B1 with IC50 values of 3.2 and 2.1 μM, respectively, and K i values of 4.0</p>
    Formula:C23H23NO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.56

    Ref: TM-T78703

  • AZ 1729
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    AZ 1729

    CAS:
    <p>FFA2 modulator; inhibits cAMP, enhances 35SGTPγS binding (pEC50: 6.9, 7.23); alters Gi/Gq signaling; affects lipolysis, neutrophil migration.</p>
    Formula:C18H16FN5OS
    Color and Shape:Solid
    Molecular weight:369.42

    Ref: TM-T37896

  • Estrogen receptor modulator 6
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    Estrogen receptor modulator 6

    CAS:
    <p>ER modulator 6 (3a) is a potent ERβ agonist with a K i of 0.44 nM; 19x more selective for ERβ than ERα.</p>
    Formula:C18H16F2O3
    Color and Shape:Solid
    Molecular weight:318.32

    Ref: TM-T40893

  • [DPro10] Dynorphin A (1-11)acetate,porcine
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    [DPro10] Dynorphin A (1-11)acetate,porcine

    [DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.
    Formula:C65H107N21O15
    Purity:99.59%
    Color and Shape:Soild
    Molecular weight:1422.7

    Ref: TM-T76341L

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    Nurr1 agonist 9

    <p>Nurr1 agonist 9 (Compound 36) acts as an agonist for Nurr1, with an EC50 of 0.090 µM and a Kd of 0.17 µM. It activates Nurr1 homodimers (NurRE, EC50 = 0.094 µM) and Nurr1-RXR heterodimers (DR5, EC50 = 0.165 µM). This compound induces the expression of Nurr1-regulated tyrosine hydroxylase (TH) in Parkinson's disease organoid models and can penetrate the human brain endothelial cell barrier.</p>
    Formula:C21H19ClN4O2
    Molecular weight:394.11965

    Ref: TM-T210048

  • Ro 64-6198
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    Ro 64-6198

    CAS:
    Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.
    Formula:C26H31N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.54

    Ref: TM-T16772

  • AKR1B10-IN-1
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    AKR1B10-IN-1

    CAS:
    AKR1B10-IN-1: potent AKR1B10 inhibitor, IC50 3.5 nM; hinders lung cancer cell growth, spread, and Cisplatin resistance.
    Formula:C19H16FNO4
    Color and Shape:Solid
    Molecular weight:341.338

    Ref: TM-T39594

  • [Orn8]-Urotensin II acetate
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    [Orn8]-Urotensin II acetate

    <p>[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.</p>
    Formula:C65H87N13O20S2
    Purity:98.63%
    Color and Shape:Solid
    Molecular weight:1434.59

    Ref: TM-T37527L

  • UFP-101
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    UFP-101

    CAS:
    <p>Strong, selective NOP receptor antagonist with pKi=10.24; &gt;3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>
    Formula:C82H138N32O21
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1908.19

    Ref: TM-TP2105

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    PF-06655075

    <p>PF-06655075 is a novel, non-brain-penetrant oxytocin receptor agonist that demonstrates enhanced selectivity for the oxytocin receptor and substantially</p>
    Formula:C75H130N14O22S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1644.05

    Ref: TM-T79172

  • T4-ATA (S-isomer)
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    T4-ATA (S-isomer)

    T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.
    Formula:C19H15I4NO6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:893.01

    Ref: TM-T19572

  • Estetrol
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    Estetrol

    CAS:
    <p>Estetrol (Donesta), a fetal liver-synthesized estrogen, selectively modulates estrogen receptors and may ease menopausal symptoms.</p>
    Formula:C18H24O4
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:304.38

    Ref: TM-T15248

  • U-54494A hydrochloride
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    U-54494A hydrochloride

    CAS:
    U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.
    Formula:C18H25Cl3N2O
    Color and Shape:Solid
    Molecular weight:391.76

    Ref: TM-T36372

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    [Sar1, Ile8]-Angiotensin II TFA

    [Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.
    Formula:C48H74F3N13O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1082.18

    Ref: TM-TP1224

  • Bazedoxifene hydrochloride
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    Bazedoxifene hydrochloride

    CAS:
    Bazedoxifene hydrochloride (TSE 424 hydrochloride) is an estrogen receptor modulator and an inhibitor of IL-6/GP130 protein interaction.
    Formula:C30H35ClN2O3
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:507.06

    Ref: TM-T6404

  • Awl 60
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    Awl 60

    CAS:
    Awl 60 is a substance P (6-11) non-competitive antagonist.
    Formula:C57H65N9O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1036.25

    Ref: TM-T25122

  • 7-FluorotryptaMine HCl
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    7-FluorotryptaMine HCl

    CAS:
    7-FluorotryptaMine HCl is a potent aromatic monoamine GPRC5A agonist that induces GPRC5A-mediated β-arrestin recruitment.7-FluorotryptaMine HCl can be used to
    Formula:C10H12ClFN2
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:214.67

    Ref: TM-T77673

  • Dimestrol
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    Dimestrol

    CAS:
    Dimestrol can induce DNA damage.
    Formula:C20H24O2
    Color and Shape:Solid
    Molecular weight:296.4

    Ref: TM-T31485

  • Herkinorin
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    Herkinorin

    CAS:
    Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.
    Formula:C28H30O8
    Color and Shape:Solid
    Molecular weight:494.53

    Ref: TM-T27534