Glucocorticoid Receptor
The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.
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Amcinonide
CAS:51022-69-6
Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid …
Formula:
C28H35FO7
Purity:
98.33% - 99.62%
Color and Shape:
Solid
Molecular weight:
502.57
Ref: TM-T0261
| 25mg | 41.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 101.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Relacorilant
CAS:1496510-51-0
Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating …
Formula:
C27H22F4N6O3S
Purity:
98.91% - 99%
Color and Shape:
Solid
Molecular weight:
586.56
Ref: TM-T16727
| 1mg | 109.00 € | ||
| 5mg | 263.00 € | ||
| 10mg | 416.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 979.00 € | ||
| 100mg | 1,324.00 € | ||
| 1mL*10mM (DMSO) | 338.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Rofleponide
CAS:144459-70-1
Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.
Formula:
C25H34F2O6
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
468.53
Ref: TM-T34383
| 1mg | 246.00 € | ||
| 5mg | 606.00 € | ||
| 10mg | 863.00 € | ||
| 25mg | 1,296.00 € | ||
| 50mg | 1,746.00 € | ||
| 100mg | 2,364.00 € | ||
| 500mg | 4,612.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Miricorilant
CAS:1400902-13-7
Miricorilant (CORT 118335) is a glucocorticoid receptor modulator for the study of digestive and metabolic …
Formula:
C24H23F3N2O2
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
428.45
Ref: TM-T33393
| 1mg | 272.00 € | ||
| 5mg | 670.00 € | ||
| 10mg | 916.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,837.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
EX-A5386
CAS:2452396-89-1
EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50/EC50<100nM.
Formula:
C29H27FN4O2
Purity:
99.69%
Color and Shape:
Soild
Molecular weight:
482.55
Ref: TM-T67742
| 1mg | 87.00 € | ||
| 5mg | 200.00 € | ||
| 10mg | 302.00 € | ||
| 25mg | 504.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Hydrocortisone aceponate
CAS:74050-20-7
Hydrocortisone aceponate (Hydrocortisone 17-propionate 21-acetate) is an effective topical glucocorticoid used in the form of …
Formula:
C26H36O7
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
460.56
Ref: TM-T32114
| 10mg | 39.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 137.00 € | ||
| 200mg | 184.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
NR3C1 Protein, Human, Recombinant (His)
NR3C1 (Nuclear Receptor Subfamily 3 Group C Member 1) is a Protein Coding gene.
Color and Shape:
Solid
Molecular weight:
10.95 kDa (predicted)
Ref: TM-TMPY-06836
| 100µg | 687.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Canrenoate potassium
CAS:2181-04-6
Canrenoate potassium (Soldactone) is a synthetic pregnadiene derivative with anti-aldosterone activity.
Formula:
C22H29KO4
Purity:
97.39% - 98.28%
Color and Shape:
Light Yellow To Tan Powder
Molecular weight:
396.56
Ref: TM-T3096
| 100mg | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Cortodoxone
CAS:152-58-9
Cortodoxone (11-Desoxycortisol) is a glucocorticoid steroid hormone that is an intermediate in the biosynthesis of …
Formula:
C21H30O4
Purity:
99.26% - 99.87%
Color and Shape:
Solid
Molecular weight:
346.46
Ref: TM-T2748
| 20mg | 47.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Deoxycorticosterone acetate
CAS:56-47-3
Deoxycorticosterone acetate (Cortexone acetate) is the 21-acetate derivative of desoxycorticosterone, used for intramuscular injection.
Formula:
C23H32O4
Purity:
99% - 99.81%
Color and Shape:
White Solid
Molecular weight:
372.5
Ref: TM-T3033
| 50mg | 48.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 78.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Diflorasone
CAS:2557-49-5
Diflorasone is a synthetic glucocorticoid. It has anti-inflammatory and immunosuppressive effects by acting on gene …
Formula:
C22H28F2O5
Purity:
99.02% - 99.92%
Color and Shape:
Solid
Molecular weight:
410.45
Ref: TM-T2548
| 5mg | 42.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 75.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 128.00 € | ||
| 200mg | 174.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AL 082D06
CAS:256925-03-8
AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding …
Formula:
C23H24ClN3O2
Purity:
99.06% - ≥95%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T1749
| 5mg | 50.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 338.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LY404039
CAS:635318-11-5
LY404039 (pomaglumetad) is an effective agonist of recombinant human mGlu2(Ki =149 nM)/mGlu3(Ki =92 nM).
Formula:
C7H9NO6S
Purity:
99% - 99.16%
Color and Shape:
Solid
Molecular weight:
235.22
Ref: TM-T6022
| 10mg | 50.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 166.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Osilodrostat
CAS:928134-65-0
Osilodrostat (LCI699) is a potent inhibitor of human 11β-hydroxylase (CYP11B1) and aldosterone synthase (CYP11B2).Cost-effective and …
Formula:
C13H10FN3
Purity:
98% - 99.12%
Color and Shape:
Solid
Molecular weight:
227.24
Ref: TM-T4277
| 1mg | 51.00 € | ||
| 2mg | 66.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 193.00 € | ||
| 50mg | 374.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Apararenone
CAS:945966-46-1
Apararenone (MT-3995) is a receptor antagonist of mineralocorticoid receptor which can be used to treat …
Formula:
C17H17FN2O4S
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
364.39
Ref: TM-T14301
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 178.00 € | ||
| 100mg | 257.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Fluorometholone
CAS:426-13-1
Fluorometholone (Fluoromethalone) is a corticosteroid, most often used after laser-based refractive surgery.
Formula:
C22H29FO4
Purity:
98.21%
Color and Shape:
Solid
Molecular weight:
376.46
Ref: TM-T3316
| 25mg | 52.00 € | ||
| 50mg | 70.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Hydrocortisone hemisuccinate
CAS:2203-97-6
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) is a corticosteroid used as an analytical and chromatography reagent.
Formula:
C25H34O8
Purity:
98.01% - 98.8%
Color and Shape:
Solid
Molecular weight:
462.53
Ref: TM-T4602
| 10mg | 36.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 66.00 € | ||
| 100mg | 85.00 € | ||
| 500mg | 181.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Methylprednisolone succinate
CAS:2921-57-5
Methylprednisolone succinate (Methylprednisolone hemisuccinate) is a synthetic glucocorticoid and is widely used as an anti-inflammatory …
Formula:
C26H34O8
Purity:
98.41% - 99.60%
Color and Shape:
White Or Almost-White Solid Powder
Molecular weight:
474.54
Ref: TM-T22367
| 25mg | 45.00 € | ||
| 50mg | 69.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Actriol
CAS:547-81-9
Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist.
Formula:
C18H24O3
Purity:
95.35% - 95.35%
Color and Shape:
Solid
Molecular weight:
288.38
Ref: TM-T1683
| 1mg | 52.00 € | ||
| 5mg | 98.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
(20S)-Protopanaxatriol
CAS:34080-08-5
(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor …
Formula:
C30H52O4
Purity:
95% - 99%
Color and Shape:
Solid
Molecular weight:
476.73
Ref: TM-T2810
| 5mg | 57.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 243.00 € | ||
| 100mg | 389.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
