MLK
GW806742X
CAS:579515-63-2
GW806742X is an inhibitor of Mixed Lineage Kinase Domain-Like protein (MLKL) which binds the MLKL …
Formula:
C25H22F3N7O4S
Purity:
99.07%
Color and Shape:
Solid
Molecular weight:
573.55
Ref: TM-T11520
2mg | 35.00 € | |
5mg | 51.00 € | |
10mg | 69.00 € | |
25mg | 118.00 € | |
50mg | 184.00 € | |
100mg | 343.00 € | |
1ml*10 (DMSO) | 65.00 € |
Estimated delivery in United States, on Friday 3 May 2024
MLKL-IN-2
CAS:899759-16-1
MLKL-IN-2 is an MLKL inhibitor with potential tumorigenic activity for the study of cellular necrosis-related …
Formula:
C26H25N5O
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
423.51
Ref: TM-T41027
1mg | 102.00 € | |
5mg | 245.00 € | |
10mg | 368.00 € | |
25mg | 755.00 € | |
50mg | 1,198.00 € | |
100mg | 1,839.00 € | |
500mg | 3,675.00 € | |
1ml*10 (DMSO) | 269.00 € |
Estimated delivery in United States, on Monday 6 May 2024
Cerdulatinib hydrochloride
CAS:1369761-01-2
Cerdulatinib hydrochloride (PRT2070 hydrochloride) is an oral active, multi-targeted tyrosine kinase inhibitor with IC50 of …
Formula:
C20H28ClN7O3S
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
482
Ref: TM-T6104
1mg | 44.00 € | |
5mg | 94.00 € | |
10mg | 114.00 € | |
25mg | 208.00 € | |
50mg | 365.00 € | |
100mg | 544.00 € | |
500mg | 1,179.00 € | |
1ml*10 (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 6 May 2024
AZ7550 trimesylate salt
CAS:2319837-99-3
AZ7550 trimesylate salt (AZ7550 Mesylate) is the active metabolite of ositinib, AZ7550 trimesylate salt inhibits …
Formula:
C30H43N7O11S3
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
773.9
Ref: TM-T13564L2
5mg | To inquire | |
10mg | To inquire | |
50mg | To inquire | |
100mg | To inquire |
Estimated delivery in United States, on Monday 6 May 2024
IM-54
CAS:861891-50-1
IM-54 is a cell-permeable, effective, and selective necrosis inhibitor.
Formula:
C19H23N3O2
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
325.4
Ref: TM-T24160
1mg | 56.00 € | |
5mg | 128.00 € | |
10mg | 184.00 € | |
25mg | 308.00 € | |
50mg | 452.00 € | |
100mg | 647.00 € | |
500mg | 1,328.00 € |
Estimated delivery in United States, on Monday 6 May 2024
URMC-099
CAS:1229582-33-5
URMC-099 is an orally bioavailable, brain penetrant MLK inhibitor (IC50: 19/42/14/150 nM, for MLK1/MLK2/MLK3/DLK), and …
Formula:
C27H27N5
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
421.54
Ref: TM-T6057
5mg | 56.00 € | |
10mg | 85.00 € | |
25mg | 138.00 € | |
50mg | 217.00 € | |
100mg | 371.00 € | |
1ml*10 (DMSO) | 58.00 € |
Estimated delivery in United States, on Friday 10 May 2024
(E/Z)-Necrosulfonamide
CAS:432531-71-0
(E/Z)-Necrosulfonamide is a novel inhibitor of MLKL.
Formula:
C18H15N5O6S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
461.47
Ref: TM-T7129
5mg | 54.00 € | |
10mg | 77.00 € | |
25mg | 116.00 € | |
50mg | 191.00 € | |
100mg | 286.00 € | |
1ml*10 (DMSO) | 73.00 € |
Estimated delivery in United States, on Friday 10 May 2024
AZ7550
CAS:1421373-99-0
AZ7550, an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).
Formula:
C27H31N7O2
Purity:
97.07%
Color and Shape:
Solid
Molecular weight:
485.58
Ref: TM-T13564
1mg | 129.00 € | |
5mg | 282.00 € | |
10mg | 417.00 € | |
25mg | 689.00 € | |
50mg | 920.00 € | |
100mg | 1,287.00 € |
Estimated delivery in United States, on Friday 10 May 2024
Necrosulfonamide
CAS:1360614-48-7
(E)-Necrosulfonamide ((E)-Necrosulfonamide) is an inhibitor of necroptosis. Blocks mixed lineage kinase domain-like protein (MLKL), a …
Formula:
C18H15N5O6S2
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
461.47
Ref: TM-T6904
5mg | 56.00 € | |
10mg | 73.00 € | |
25mg | 138.00 € | |
50mg | 211.00 € | |
100mg | 370.00 € | |
500mg | 875.00 € | |
1ml*10 (DMSO) | 56.00 € |
Estimated delivery in United States, on Friday 10 May 2024
PRT062607 hydrochloride
CAS:1370261-97-4
PRT062607 hydrochloride (P505-15 Hydrochloride) is a selective inhibitor of Syk (IC50: 1 nM). It displays …
Formula:
C19H23N9O·HCl
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
429.91
Ref: TM-T2696
1mg | 59.00 € | |
2mg | 84.00 € | |
5mg | 124.00 € | |
10mg | 183.00 € | |
25mg | 320.00 € | |
50mg | 489.00 € | |
200mg | 926.00 € | |
1ml*10 (DMSO) | 137.00 € |
Estimated delivery in United States, on Friday 10 May 2024
LY-364947
CAS:396129-53-6
LY-364947 (HTS466284) is a potent ATP-competitive inhibitor of TGFβR-I.
Formula:
C17H12N4
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
272.3
Ref: TM-T2048
5mg | 69.00 € | |
10mg | 86.00 € | |
25mg | 141.00 € | |
50mg | 254.00 € | |
100mg | 365.00 € | |
200mg | 547.00 € | |
500mg | 858.00 € | |
1ml*10 (DMSO) | 71.00 € |
Estimated delivery in United States, on Friday 10 May 2024