Sodium Channel
Sodium channels are essential membrane proteins that allow the passage of sodium ions (Na+) across the cell membrane, generating and propagating electrical signals in neurons, muscle cells, and other excitable tissues. These channels are vital for the initiation and conduction of action potentials, making them crucial in processes such as nerve impulse transmission, muscle contraction, and cardiac function. Dysregulation of sodium channels can lead to neurological disorders, arrhythmias, and chronic pain conditions. At CymitQuimica, we provide a variety of sodium channel modulators to support your research in neurobiology, cardiology, and pain management.
Found 259 products of "Sodium Channel"
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µ-Conotoxin SIIIA
CAS:μ-Conotoxin SIIIA, a tetrodotoxin (TTX)-resistant sodium channel blocker, is a toxic peptide derived from Conus snail venom.Formula:C83H123N33O27S6Purity:98%Color and Shape:SolidMolecular weight:2207.461-(1-Methyl-1h-pyrazol-4-yl)-ethanone
CAS:1-(1-Methyl-1h-pyrazol-4-yl)-ethanone is a high purity biochemical reagent that can be used in research related to life sciences.Formula:C6H8N2OPurity:99.92%Color and Shape:SolidMolecular weight:124.14Myomodulin
CAS:Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A theFormula:C36H67N11O8S2Purity:98%Color and Shape:SolidMolecular weight:846.12SLC26A3-IN-2
CAS:Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.Formula:C19H13ClN2O2SPurity:99.86%Color and Shape:SolidMolecular weight:368.84PF-06456384 trihydrochloride
CAS:PF-06456384 trihydrochloride is a selective NaV1.7 inhibitor acting through protein-ligand binding. intravenous infusion and pain research.Formula:C35H35Cl3F3N7O3S2Purity:99.16%Color and Shape:SolidMolecular weight:829.18Mepivacaine hydrochloride
CAS:Mepivacaine hydrochloride (Mepivacaine HCl) is the hydrochloride salt form of mepivacaine, an amide derivative with local anesthetic properties.Formula:C15H22N2O·HClPurity:98.76% - 99.94%Color and Shape:White Or Off White Crystalline PowderMolecular weight:282.81Benzonatate (PEGn)
CAS:Benzonatate (PEGn) is a unique non-narcotic cough suppressant featuring sodium channel blocking properties and anesthetic effects on respiratory tract stretch receptors.Formula:(C2H4O)nC12H17NO2Color and Shape:SolidAnthopleurin-C
Anthopleurin-C (APE 2-1) is a cardiotonic polypeptide exhibiting a potent positive inotropic effect [1].Formula:C210H316N62O61S6Purity:98%Color and Shape:SolidMolecular weight:4877.52Pterinotoxin-1
Pterinotoxin-1 is a peptide toxin that functions as an inhibitor of sodium channels [1].Formula:C163H251N49O53S7Purity:98%Color and Shape:SolidMolecular weight:3969.49BmK-M1
BmK-M1, a scorpion-derived toxin, consists of a 64-amino acid polypeptide stabilized by four disulfide bridges.Formula:C313H467N91O91S8Purity:98%Color and Shape:SolidMolecular weight:7217.13Dc1a
Dc1a, a toxin isolated from the desert bush spider Diguetia canities [1], potently facilitates the opening of the German cockroach Na v channel (BgNa v 1).Formula:C276H414N76O84S8Purity:98%Color and Shape:SolidMolecular weight:6397.22ProTx II
CAS:Selective NaV1.7 inhibitor, alters activation, reduces current, 100x more selective for 1.7 over other Na+ channels.
Formula:C168H250N46O41S8Purity:98%Color and Shape:SolidMolecular weight:3826.59Hm1a
Hm1a, a disulfide-rich spider-venom peptide and NaV1.1 activator, reestablishes the function of inhibitory interneurons in a Dravet syndrome (DS) mouse model [1Formula:C170H239N47O54S6Purity:98%Color and Shape:SolidMolecular weight:3997.39Zandatrigine
CAS:Zandatrigine (NBI-921352) is a blocker of sodium channel protein type 8 subunit alpha and can be used in studies about nervous system pathologies of epilepsyFormula:C22H25FN4O2S2Purity:99.98%Color and Shape:SolidMolecular weight:460.59Ref: TM-T39630
1mg111.00€2mg164.00€5mg268.00€10mg439.00€25mg707.00€50mg1,009.00€100mg1,333.00€1mL*10mM (DMSO)294.00€Amlenetug
Amlenetug is a humanized IgG1κ antibody targeting SNCA, with its corresponding isotype control being HumanIgG1kappa, Isotype Control.Purity:95%Color and Shape:Odour Liquidμ-Conotoxin PIIIA
CAS:μ-Conotoxin PIIIA, isolated from Conus purpurascens [1] [2], is a blocker of the sodium channel NaV 1.4.Formula:C103H166N40O28S6Purity:98%Color and Shape:SolidMolecular weight:2605.06ETD001
CAS:ETD001 is a long-acting ENaC inhibitor with an IC50 value of 57.5 nM in HBE cells. It is applicable for research in cystic fibrosis.Formula:C41H57F6N9O16Color and Shape:SolidMolecular weight:1045.93Ion Channel Targeted Library
A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;
Color and Shape:Odour SolidSolpecainol
CAS:solpecainol is a sodium channel blocker used in the study of neurological and cardiovascular diseases.Formula:C18H23NO3Purity:99.71%Color and Shape:SoildMolecular weight:301.38Batrachotoxin
CAS:Batrachotoxin (BTX), a potent neurotoxin and cardiotoxin, is found in the skin of the Colombian dart frog (Phyllobates aurotaenia). As an activator of sodium channels (sodium channel), it interferes with normal sodium channel closure by binding to voltage-gated sodium channels (sodium channel) on the cell membrane. This interaction causes a continuous influx of sodium ions into the cells, leading to persistent depolarization.Formula:C31H42N2O6Color and Shape:SolidMolecular weight:538.67Anthopleurin-A
CAS:Anthopleurin-A, a sodium channel toxin, is selective for cardiac channels and has a cardiotonic effect. It can be isolated from the sea anemone [1] [2].Formula:C220H326N64O67S6Color and Shape:SolidMolecular weight:5131.72PF-04856264
CAS:PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.Formula:C20H15N5O3S2Purity:97.43%Color and Shape:SolidMolecular weight:437.5Ref: TM-T33943
1mg50.00€5mg105.00€10mg170.00€25mg340.00€50mg532.00€100mg893.00€1mL*10mM (DMSO)117.00€Ethacizine hydrochloride
CAS:Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.Formula:C22H28ClN3O3SPurity:98.08% - 98.08%Color and Shape:SolidMolecular weight:449.9910,11-Dihydro-10-hydroxycarbamazepine-d4
CAS:10,11-Dihydro-10-hydroxycarbamazepine-d4 is a deuterated compound of 10,11-Dihydro-10-hydroxycarbamazepine.Formula:C15H10D4N2O2Molecular weight:258.31AM-2099
CAS:AM-2099 is a selective voltage-gated sodium channel Nav1.7 inhibitor used in pain research.Formula:C19H13F3N4O3S2Color and Shape:SolidMolecular weight:466.46Bulleyaconitine A
CAS:Bulleyaconitine A, an analgesic and antiinflammatory drug isolated from Aconitum plants, has several potential targets, such as voltage-gated Na+ channels.Formula:C35H49NO9Purity:99.56% - 99.76%Color and Shape:SolidMolecular weight:627.76Dibucaine hydrochloride
CAS:Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.Formula:C20H30ClN3O2Purity:99.66%Color and Shape:White PowderMolecular weight:379.92Mexiletine-d6 hydrochloride
CAS:Mexiletine D6 hydrochloride is a non-selective voltage-gated sodium channel blocker,is a Class IB antianhythmic.Formula:C11H18ClNOPurity:98%Color and Shape:SolidMolecular weight:221.763,3-Diethylthiacarbocyanine iodide
CAS:3, 3-diethylthiacarbocyanine iodide is a cyanine dye. Can be used for photochemical methods.Formula:C21H21IN2S2Purity:99.79%Color and Shape:SolidMolecular weight:492.44Mepivacaine
CAS:Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.Formula:C15H22N2OPurity:99.86%Color and Shape:SolidMolecular weight:246.35Triamterene D5
CAS:Triamterene D5 is a deuterium-labeled Triamterene and can block epithelial Na+ channel (ENaC) in a voltage-dependent manner, used as a mild diuretic.Formula:C12H11N7Purity:98%Color and Shape:SolidMolecular weight:258.29BI-9627
CAS:BI-9627 is an inhibitor of sodium-hydrogen exchanger isoform 1 (NHE1) (EC50: 31 nM).Formula:C16H19F3N4O2Purity:99.77%Color and Shape:SolidMolecular weight:356.34Poneratoxin acetate
Poneratoxin acetate is a neurotoxic peptide and modulator of NaV1.6/NaV1.7, lowering the activation threshold of voltage-gated sodium channels and causing pain.Formula:C129H215N33O31S·xC2H4O2Color and Shape:SolidMolecular weight:2756.35 (free base)Nicainoprol
CAS:Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.Formula:C21H27N3O3Purity:99.54%Color and Shape:SolidMolecular weight:369.46Ref: TM-T4539
1mg133.00€5mg326.00€10mg485.00€25mg770.00€50mg1,035.00€100mg1,395.00€1mL*10mM (DMSO)333.00€Ropivacaine hydrochloride monohydrate
CAS:Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.Formula:C17H29ClN2O2Purity:99.94% - 99.95%Color and Shape:White SolidMolecular weight:328.88GNE-131
CAS:GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).Formula:C23H30N4O3SPurity:98.54% - 99.59%Color and Shape:SolidMolecular weight:442.57Ref: TM-TQ0014
1mg105.00€5mg250.00€10mg356.00€25mg597.00€50mg835.00€100mg1,108.00€1mL*10mM (DMSO)268.00€Flecainide acetate
CAS:Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).Formula:C19H24F6N2O5Purity:99.42%Color and Shape:SolidMolecular weight:474.39Fosphenytoin disodium
CAS:Fosphenytoin disodium (ACC-9653) is a prodrug of phenytoin that is rapidly converted to phenytoin, a voltage-gated sodium channel blockerFormula:C16H13N2Na2O6PPurity:99.97%Color and Shape:White Crystalline PowderMolecular weight:406.24DS-1971a
CAS:DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.Formula:C20H21ClFN5O3SPurity:99.66%Color and Shape:SolidMolecular weight:465.93Cariporide
CAS:Cariporide (HOE-642), an NHE1 inhibitor, reduces human platelet degranulation, platelet-leukocyte aggregates, and GPIIb/IIIa activation.Formula:C12H17N3O3SPurity:95.4% - 99.88%Color and Shape:SolidMolecular weight:283.35Rimeporide hydrochloride
CAS:Rimeporide hydrochloride (EMD-87580 hydrochloride) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.Formula:C11H16ClN3O5S2Purity:99.82%Color and Shape:SolidMolecular weight:369.84Licarbazepine
CAS:Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partialFormula:C15H14N2O2Purity:99.11%Color and Shape:SolidMolecular weight:254.28Nav1.8-IN-1
CAS:Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8
Formula:C20H15ClF3N3O2Purity:97.59%Color and Shape:SolidMolecular weight:421.8QX-222 chloride
CAS:QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.Formula:C13H21ClN2OPurity:97.37%Color and Shape:SolidMolecular weight:256.77Carbamazepine
CAS:Carbamazepine: a tricyclic with anticonvulsant and analgesic effects, treats trigeminal neuralgia.Formula:C15H12N2OPurity:99.78% - 99.79%Color and Shape:SolidMolecular weight:236.27λ-Cyhalothrin
CAS:λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.Formula:C23H19ClF3NO3Purity:99.76%Color and Shape:SolidMolecular weight:449.85Rimeporide
CAS:Rimeporide (EMD-87580) (EMD-87580) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.Formula:C11H15N3O5S2Purity:97.66%Color and Shape:SolidMolecular weight:333.38Ref: TM-T5319
1mg46.00€2mg62.00€5mg90.00€10mg166.00€25mg358.00€50mg523.00€100mg747.00€1mL*10mM (DMSO)108.00€Flecainide hydrochloride
CAS:Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.Formula:C17H21ClF6N2O3Purity:97.79%Color and Shape:SolidMolecular weight:450.81Raxatrigine
CAS:Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.Formula:C18H19FN2O2Purity:98% - 99.43%Color and Shape:SolidMolecular weight:314.35N-Me-aminopyrimidinone9
CAS:N-Me-aminopyrimidinone9 is a sodium channel antagonistFormula:C16H21N3OSPurity:99.21%Color and Shape:SolidMolecular weight:303.42Ref: TM-T8444
1mg58.00€5mg116.00€10mg172.00€25mg281.00€50mg396.00€100mg537.00€200mg712.00€1mL*10mM (DMSO)116.00€Levobupivacaine
CAS:Levobupivacaine is an amino-amide local anaesthetic drug belonging to the family of n-alkylsubstituted pipecoloxylidide.Formula:C18H28N2OPurity:99.72%Color and Shape:SolidMolecular weight:288.43Ref: TM-T1787
5mg46.00€10mg59.00€25mg87.00€50mg129.00€100mg178.00€200mg268.00€500mg460.00€1mL*10mM (DMSO)47.00€Propafenone hydrochloride
CAS:Propafenone hydrochloride (Arythmol8) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial.Formula:C21H27NO3·HClPurity:99.67%Color and Shape:White SolidMolecular weight:377.9Benzocaine xHCl(94-09-7(free base))
Benzocaine shares a common receptor with all othe rLAs in the voltage-gated Na+ channel(IC50 of 0.8 mM tested with a potential of +30 mV).Formula:C9H11NO2·xHClPurity:99.37%Color and Shape:SolidMolecular weight:N/AVX-150
CAS:VX-150 is a highly selective NaV1.8 inhibitor relative to the other sodium channel subtypes (>400-fold).Formula:C21H17F4N2O7PPurity:97.58%Color and Shape:SolidMolecular weight:516.34Ref: TM-T9683
1mg63.00€5mg137.00€10mg222.00€25mg447.00€50mg715.00€100mg1,144.00€1mL*10mM (DMSO)156.00€PF-01247324
CAS:PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).Formula:C13H10Cl3N3OPurity:99.22%Color and Shape:SolidMolecular weight:330.6PF 05089771
CAS:PF 05089771 is a Selective inhibitor of Nav1.7 (IC50 = 11 nM) that interacts with the voltage-sensor domain of domain IV.Formula:C18H12Cl2FN5O3S2Purity:99.03% - 99.42%Color and Shape:SolidMolecular weight:500.35PF-05186462
CAS:PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.Formula:C19H10ClF4N5O3S2Purity:99.10% - 99.37%Color and Shape:SolidMolecular weight:531.89Ralfinamide mesylate
CAS:Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.Formula:C18H23FN2O5SPurity:99.83%Color and Shape:SolidMolecular weight:398.45Ref: TM-T7547
1mg52.00€5mg112.00€10mg170.00€25mg280.00€50mg371.00€100mg525.00€200mg705.00€1mL*10mM (DMSO)172.00€Ajmaline
CAS:Ajmaline, a class Ia anti-arrhythmic, diagnoses Brugada syndrome and treats tachycardia; inhibits cardiac Kv1.5/Kv4.3 channels.Formula:C20H26N2O2Purity:99.67% - 99.87%Color and Shape:SolidMolecular weight:326.43ICA-121431
CAS:ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.Formula:C23H19N3O3S2Purity:98.06%Color and Shape:SolidMolecular weight:449.55(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purity:97% - ≥95%Color and Shape:White Fine PowderMolecular weight:230.26Benzamil
CAS:Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.Formula:C13H14ClN7OPurity:99.79%Color and Shape:SolidMolecular weight:319.7520(S)-Ginsenoside Rg3
CAS:20(S)-Ginsenoside Rg3 (Rg3) possess an ability to inhibit the lung metastasis of tumor cells via inhibition of the adhesion and invasion of tumor cells.Formula:C42H72O13Purity:98.11% - 99.93%Color and Shape:SolidMolecular weight:785.01Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5SPurity:98.85% - 99.99%Color and Shape:SolidMolecular weight:556.76Evenamide
CAS:Evenamide (NW-3509) is a sodium channel blocker. Which shows efficacy in a broad spectrum of rodent models of psychosis, mania, depression, and aggressiveness.Formula:C16H26N2O2Purity:96.74% - 99.15%Color and Shape:SolidMolecular weight:278.39Ref: TM-T15260
1mg39.00€5mg84.00€10mg120.00€25mg236.00€50mg378.00€100mg612.00€200mg850.00€1mL*10mM (DMSO)93.00€Metaflumizone
CAS:Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.Formula:C24H16F6N4O2Purity:98.73%Color and Shape:SolidMolecular weight:506.40Cyfluthrin
CAS:Cyfluthrin binds to voltage-sensitive sodium channel such as Nav 1.8 sodium channel and modify their gating kinetics, thereby disrupting nerve function of pestsFormula:C22H18Cl2FNO3Purity:99.76%Color and Shape:SolidMolecular weight:434.29A-803467
CAS:A-803467 is a selective NaV1.8 channel blocker.Formula:C19H16ClNO4Purity:96.94% - 98%Color and Shape:SolidMolecular weight:357.79Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Formula:C25H29N3O2Purity:99.83% - 99.97%Color and Shape:SolidMolecular weight:403.52Tenapanor
CAS:Tenapanor (RDX 5791), an NHE3 inhibitor, regulates sodium in the gut and kidney with a strong preclinical safety record and minimal side effects.Formula:C50H66Cl4N8O10S2Purity:99.49% - 99.85%Color and Shape:SolidMolecular weight:1145.05Dimethyl lithospermate B
CAS:Dimethyl lithospermate B (dmLSB) is a selective Na+ channel agonist.Formula:C38H34O16Purity:97.18% - 99.62%Color and Shape:SolidMolecular weight:746.67Ref: TM-T8299
1mg137.00€2mg202.00€5mg356.00€10mg522.00€25mg820.00€50mg1,099.00€100mg1,485.00€200mg2,008.00€1mL*10mM (DMSO)502.00€Eslicarbazepine Acetate
CAS:Eslicarbazepine Acetate (Zebinix) is an anticonvulsant medication approved for use as an adjunctive therapy for partial-onset seizures.Formula:C17H16N2O3Purity:99.58% - >99.99%Color and Shape:White To Off-White SolidMolecular weight:296.32Ref: TM-T3285
5mg35.00€10mg52.00€25mg87.00€50mg117.00€100mg161.00€200mg254.00€500mg371.00€1mL*10mM (DMSO)52.00€β-Pompilidotoxin Acetate
β-Pompilidotoxin Acetate is a wasp venom peptide.Formula:C73H128N22O19Purity:98.64%Color and Shape:SolidMolecular weight:1617.93Ref: TM-T21769L
2mg44.00€5mg63.00€10mg94.00€25mg145.00€50mg210.00€100mg298.00€200mg419.00€1mL*10mM (DMSO)129.00€Ranolazine
CAS:Ranolazine (RS 43285-003) inhibits calcium uptake, treats chronic angina by targeting sodium/calcium channels to modulate intracellular sodium.Formula:C24H33N3O4Purity:98.13%Color and Shape:White SolidMolecular weight:427.54Sodium ionophore III
CAS:Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.Formula:C34H52N2O4Purity:99.51% - 99.78%Color and Shape:SolidMolecular weight:552.79BI 01383298
CAS:BI 01383298 is a selective inhibitor of the sodium-citrate co-transporter (SLC13A5).Formula:C19H19Cl2FN2O3SPurity:99.71%Color and Shape:SolidMolecular weight:445.34GS967
CAS:GS967 is a potent, and selective inhibitor of cardiac late sodium current (late INa ).
Formula:C14H7F6N3OPurity:98% - >99.99%Color and Shape:SolidMolecular weight:347.22Ref: TM-T2049
2mg35.00€5mg52.00€10mg79.00€25mg159.00€50mg284.00€100mg495.00€200mg718.00€500mg1,111.00€Pilsicainide HCl
CAS:Pilsicainide HCl (SUN 1165) is a pure sodium channel blockerFormula:C17H25ClN2OPurity:99.01% - 99.80%Color and Shape:SolidMolecular weight:308.85AZ194
CAS:CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.Formula:C34H31F2N3O3Purity:99.61%Color and Shape:SolidMolecular weight:567.62Ref: TM-T9461
1mg77.00€5mg166.00€10mg260.00€25mg485.00€50mg700.00€100mg982.00€500mg1,963.00€1mL*10mM (DMSO)178.00€RY785
CAS:RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.Formula:C21H20N4O2SPurity:99.78%Color and Shape:SolidMolecular weight:392.47Ref: TM-T12786
1mg49.00€5mg137.00€10mg222.00€25mg378.00€50mg530.00€100mg745.00€200mg1,035.00€1mL*10mM (DMSO)118.00€6-Benzoylheteratisine
CAS:6-Benzoylheteratisine (Heteratisan-14-one, 6-(benzoyloxy)-20-ethyl-8-hydroxy-1-methoxy-4-meth) is a Aconitum alkaloid.Formula:C29H37NO6Purity:99.87%Color and Shape:SolidMolecular weight:495.61Benzonatate
CAS:Benzonatate is an antagonist of sodium channel protein.Formula:C30H53NO11Purity:99.92%Color and Shape:Colorless To Faintly Yellow Oil LiquidMolecular weight:603.74PF-06869206
CAS:PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).Formula:C15H14ClF3N4O2Purity:99.79% - 99.88%Color and Shape:SolidMolecular weight:374.75Levobupivacaine hydrochloride
CAS:Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.Formula:C18H28N2O·HClPurity:99.74%Color and Shape:White Crystalline PowderMolecular weight:324.893-Deoxyaconitine
CAS:3- Deoxyaconitine is a derivative of Aconitine (A189875), which activates tetrodotoxin-sensitive Na+ channels, inducing presynaptic depolarization, thusFormula:C34H47NO10Purity:98.31%Color and Shape:SolidMolecular weight:629.74Ralfinamide
CAS:Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.Formula:C17H19FN2O2Purity:99.41%Color and Shape:SolidMolecular weight:302.34Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.Formula:C8H5F3N2OSPurity:99.71% - 99.88%Color and Shape:PowderMolecular weight:234.24’-Hydroxybupivacaine
CAS:Controlled ProductApplications 4’-Hydroxybupivacaine is a metabolite of Bupivacaine. Bupivacaine is an amide-type, long-acting local anesthetic.
References Lindberg, R., et al.: J. Chromatogr. Biomed. Appl., 383, 357 (1986)Formula:C18H28N2O2Color and Shape:NeatMolecular weight:304.4276-(Propylamino)-N-(2,6-dimethylphenyl)hexanamide
Controlled ProductApplications 6-(Propylamino)-N-(2,6-dimethylphenyl)-hexanamide is a derivative of Bupivacaine (B689560), a sodium channel blocker, local anesthetic.
References Wilson, T.D., et al.: Anal. Profiles Drug Subs., 19, 59 (1990), McClellan, K.J., et al.: Drugs, 56, 355 (1998),Formula:C17H28N2OColor and Shape:NeatMolecular weight:276.417Propoxycaine hydrochloride
CAS:Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.Formula:C16H27ClN2O3Purity:97.25%Color and Shape:SolidMolecular weight:330.85Benzocaine N-Glucoside (a/b mixture)
CAS:Controlled ProductStability Hygroscopic
Applications The N-Glucoside of Benzocaine (B202970) with anesthetic activity. A potential sun-screening agent.
References Rybczynska, B. et al.: Parfum. Kosm., 48, 125 (1967); Nikolin, A. et al.: Glas. Hemi. Tehnol. Bosne Herceg., 16, 93 (1968);Formula:C15H21NO7Color and Shape:NeatMolecular weight:327.33Oxethazaine
CAS:Controlled ProductApplications A potent local anesthetic that is active even in acidic conditions. It is used (usually in combination with an antacid) for the relief of pain associated with peptic ulcer disease or esophagitis.
References Detrain, M. et al.: Acta. Gastro-Enterol. Belg., 28, 360 (1965); Barbezat, G.O. et al.: Scand. J. Gastroenterol., 13, 321 (1978); Masuda, Y. et al.: Biochem. Pharmacol., 64, 677 (2002);Formula:C28H41N3O3Color and Shape:NeatMolecular weight:467.6410,11-Dihydro-10-hydroxy Carbamazepine-d4
CAS:10,11-Dihydro-10-hydroxy Carbamazepine-d4 is a deuterated compound of 10,11-Dihydro-10-hydroxy Carbamazepine. 10,11-Dihydro-10-hydroxy Carbamazepine has a CAS number of 29331-92-8. Licarbazepine is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial seizures and bipolar disorders.Formula:C15H10D4N2O2Color and Shape:SolidMolecular weight:258.31Propafenone-d5 HCl
CAS:Propafenone-d5 HCl is a deuterated compound of Propafenone HCl. Propafenone HCl has a CAS number of 34183-22-7. Propafenone HCl is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial and ventricular arrhythmias.Formula:C21H23D5ClNO3Molecular weight:382.943-(2-Chloropropionyl)amino-4-methyl-2-methoxycarbonylthiophene
CAS:Controlled ProductApplications 3-(2-Chloropropionyl)amino-4-methyl-2-methoxycarbonylthiophene is an intermediate in the synthesis of Articaine-d7 Hydrochloride which is the labelled form of Articaine Hydrochloride (A777905). Articaine Hydrochloride is the Hydrochloride Salt of Articaine (A777900). Articaine is an amide based short-acting local anesthetic use for regional anaesthesia in day-case settings such arthroscopy, hand, food surgery and in dentistry.
References Malamed, S.F., et al.: J. Am. Dent. Assoc., 132, 177 (2001); Luan, F., et al.: Bioorg. Med. Chem., 21, 1870 (2013)Formula:C10H12ClNO3SColor and Shape:NeatMolecular weight:261.73Deacetamide Acetonitrile-pentisomide
CAS:Controlled ProductApplications Deacetamide Acetonitrile-pentisomide is an intermediate in the synthesis of Pentisomide (P275600). Pentisomide is a sodium channel blocker; derivative of disopyramide. Antiarrhythmic (class I).
References Kuhlkamp, V., et al.: Int. J. Cardiol., 36, 69 (1992); Yuan, S., et al.: Cardiovasc. Drug Rev., 11, 74 (1993)Formula:C19H31N3Color and Shape:NeatMolecular weight:301.472-(3-Bromopropyl)-1,2,4-triazolo-pyridin-3-one
CAS:Controlled ProductApplications Used in the preparation of bicycloamine derivatives as sodium channel inhibitors for treatment of pain, epilepsy and insomnia.
Formula:C9H10BrN3OColor and Shape:NeatMolecular weight:256.1N-(Chloroacetyl)-2,5-dimethylaniline
CAS:Controlled ProductApplications N-(Chloroacetyl)-2,5-dimethylaniline is an intermediate in the synthesis of impurities of Lidocaine (L397800), an anesthetic local agent and antiarrythmic class IB agent.
References Groningsson, K., et al.: Anal. Profiles Drug Subs., 14, 207 (1985), Davies, P.S., et al.: Drugs, 64, 937 (2004),Formula:C10H12ClNOColor and Shape:NeatMolecular weight:197.66Propafenone D7 hydrochloride
CAS:Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.Formula:C21H28ClNO3Purity:98%Color and Shape:SolidMolecular weight:384.95Methocarbamol D5
CAS:Methocarbamol is a central muscle relaxant. Methocarbamol D5 is deuterium labeled Methocarbamol.Formula:C11H15NO5Purity:98%Color and Shape:SolidMolecular weight:246.27
