CymitQuimica logo
GABA Receptor

GABA Receptor

GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.

Found 336 products of "GABA Receptor"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Formula:C18H21ClF3N3O
    Purity:99.03% - 99.95%
    Color and Shape:Solid
    Molecular weight:387.83
  • Gabazine free base

    CAS:
    <p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>
    Formula:C15H17N3O3
    Color and Shape:Solid
    Molecular weight:287.31
  • Amentoflavone

    CAS:
    <p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>
    Formula:C30H18O10
    Purity:98.21% - 99.22%
    Color and Shape:Odourless Whitish Solid
    Molecular weight:538.46
  • U93631

    CAS:
    <p>GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.</p>
    Formula:C17H21N3O2
    Purity:99.65% - 99.76%
    Color and Shape:Solid
    Molecular weight:299.37
  • Ginsenoside Rc

    CAS:
    <p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>
    Formula:C53H90O22
    Purity:98.83% - 99.56%
    Color and Shape:White Powder
    Molecular weight:1079.27
  • NS11394

    CAS:
    <p>NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) &gt; α(3) &gt; α(2) &gt; α(</p>
    Formula:C23H19N3O
    Purity:99.44% - 99.86%
    Color and Shape:Solid
    Molecular weight:353.42
  • Loreclezole hydrochloride

    CAS:
    <p>Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.</p>
    Formula:C10H7Cl4N3
    Color and Shape:Solid
    Molecular weight:310.99
  • α-Thujone

    CAS:
    <p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>
    Formula:C10H16O
    Purity:97.02% - 98.41%
    Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)
    Molecular weight:152.23
  • Cholesterol myristate

    CAS:
    <p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>
    Formula:C41H72O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:597.01
  • Fipronil

    CAS:
    <p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>
    Formula:C12H4Cl2F6N4OS
    Purity:97.21%
    Color and Shape:Solid Powder
    Molecular weight:437.15
  • Acetoxyvalerensre

    CAS:
    <p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>
    Formula:C17H24O4
    Purity:98.22%
    Color and Shape:Solid
    Molecular weight:292.37
  • α-Asarone

    CAS:
    <p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>
    Formula:C12H16O3
    Purity:99.64% - 99.64%
    Color and Shape:Monoclinic Needles From Water Monoclinic Needles From Water
    Molecular weight:208.25
  • Tiagabine hydrochloride hydrate

    CAS:
    <p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>
    Formula:C20H28ClNO3S2
    Color and Shape:Solid
    Molecular weight:430.02
  • (+)-Kavain

    CAS:
    <p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>
    Formula:C14H14O3
    Purity:97% - ≥95%
    Color and Shape:White Fine Powder
    Molecular weight:230.26
  • Cyclothiazide

    CAS:
    <p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>
    Formula:C14H16ClN3O4S2
    Purity:98.23% - 99.49%
    Color and Shape:Crystals From Dilute Alcohol Solid
    Molecular weight:389.88
  • Pikamilone

    CAS:
    <p>Pikamilone (Picamilon) is an intelligent medicine.</p>
    Formula:C10H12N2O3
    Purity:99.38%
    Color and Shape:White Crystalline Powder
    Molecular weight:208.21
  • AZD-6280

    CAS:
    <p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>
    Formula:C20H22N4O3
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:366.41
  • Imidazenil

    CAS:
    <p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>
    Formula:C18H12BrFN4O
    Purity:98.4%
    Color and Shape:Solid
    Molecular weight:399.22
  • CL 218872

    CAS:
    <p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>
    Formula:C13H9F3N4
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:278.23
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Formula:C19H19FN4O2
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:354.38