GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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Pentetrazol
CAS:54-95-5
Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and …
Formula:
C6H10N4
Purity:
100% - 99.95%
Color and Shape:
Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)
Molecular weight:
138.17
Ref: TM-T1413
| 25mg | 53.00 € | ||
| 50mg | 76.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Pivagabine
CAS:69542-93-4
Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.
Formula:
C9H17NO3
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
187.24
Ref: TM-T12492
| 1mg | 36.00 € | ||
| 2mg | 48.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 367.00 € | ||
| 500mg | 832.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Chlormezanone
CAS:80-77-3
Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has …
Formula:
C11H12ClNO3S
Purity:
99.89% - 99.97%
Color and Shape:
Crystals Solid
Molecular weight:
273.74
Ref: TM-T0715
| 100mg | 54.00 € | ||
| 200mg | 68.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
L-Cycloserine
CAS:339-72-0
L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.
Formula:
C3H6N2O2
Purity:
99.45% - ≥95%
Color and Shape:
Crystals White Powder
Molecular weight:
102.09
Ref: TM-T0710
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 50mg | 72.00 € | ||
| 100mg | 94.00 € | ||
| 200mg | 138.00 € | ||
| 500mg | 221.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Fluxametamide
CAS:928783-29-3
Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and …
Formula:
C20H16Cl2F3N3O3
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
474.26
Ref: TM-T11307
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 616.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
γ-Aminobutyric acid
CAS:56-12-2
γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.
Formula:
C4H9NO2
Purity:
≥95%
Color and Shape:
White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid Powder
Molecular weight:
103.12
Ref: TM-T0508
| 50mg | 36.00 € | ||
| 100mg | 50.00 € | ||
| 200mg | 63.00 € | ||
| 500mg | 90.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Etifoxine hydrochloride
CAS:56776-32-0
Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.
Formula:
C17H18Cl2N2O
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
337.24
Ref: TM-T13690
| 5mg | 38.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 182.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Nikethamide
CAS:59-26-7
Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former …
Formula:
C10H14N2O
Purity:
98.75%
Color and Shape:
Followed By A Faint Sensation Of The Warmth (Ntp 1992)
Molecular weight:
178.23
Ref: TM-T0048
| 1g | 77.00 € | ||
| 5g | 168.00 € | ||
| 200mg | 37.00 € | ||
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Broflanilide
CAS:1207727-04-5
Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 …
Formula:
C25H14BrF11N2O2
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
663.29
Ref: TM-T10618
| 1mg | 51.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 345.00 € | ||
| 50mg | 567.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Phenibut
CAS:1078-21-3
Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter …
Formula:
C10H13NO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
179.22
Ref: TM-T2990
| 10mg | 34.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 84.00 € | ||
| 200mg | 107.00 € | ||
| 500mg | 168.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
Clomethiazole
CAS:533-45-9
Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It …
Formula:
C6H8ClNS
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
161.65
Ref: TM-T14983
| 100mg | 48.00 € | ||
| 200mg | 63.00 € | ||
| 500mg | 93.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 5 Nov 2024
6,7-dimethylisatin
CAS:20205-43-0
6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.
Formula:
C10H9NO2
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
175.18
Ref: TM-T77568
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,699.00 € | ||
| 500mg | 3,428.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
3-Methylglutaconic acid
CAS:5746-90-7
3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, …
Formula:
C6H8O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
144.13
Ref: TM-T78071
| 1mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
MIDD0301
CAS:2187489-08-1
MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of …
Formula:
C19H13BrFN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
414.23
Ref: TM-T9946
| 1mg | 184.00 € | ||
| 5mg | 411.00 € | ||
| 10mg | 615.00 € | ||
| 25mg | 1,107.00 € | ||
| 50mg | 1,661.00 € | ||
| 100mg | 2,491.00 € | ||
| 200mg | 3,736.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
Arecaidine hydrobromide
CAS:6013-57-6
Arecaidine hydrobromide, a pyridine alkaloid, functions as a potent GABA uptake inhibitor and acts as …
Formula:
C7H12BrNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
222.08
Ref: TM-T80013
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
DAA-1106
CAS:220551-92-8
DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective …
Formula:
C23H22FNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
395.42
Ref: TM-T3173
| 5mg | 47.00 € | ||
| 10mg | 79.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
3-Aminopropylphosphonic Acid
CAS:13138-33-5
3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist …
Formula:
C3H10NO3P
Purity:
98.9%
Color and Shape:
Light Yellow Liquid
Molecular weight:
139.09
Ref: TM-T38205
| 10mg | 39.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | 82.00 € | ||
| 100mg | 112.00 € | ||
| 200mg | 166.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
CGP 35348
CAS:123690-79-9
CGP 35348: GABAB receptor antagonist, EC50 = 34 μM, used in neonatal brain damage research …
Formula:
C8H20NO4P
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
225.22
Ref: TM-T21793
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 304.00 € | ||
| 50mg | 489.00 € | ||
| 100mg | 733.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
GABA receptor Antagonist 1
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 …
Purity:
98%
Ref: TM-T82357
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
Guvacine hydrobromide
CAS:6027-92-5
Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor …
Formula:
C6H10BrNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
208.05
Ref: TM-T80014
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
