GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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E2730
CAS:1520073-91-9
E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying …
Formula:
C9H8F4N2O2S
Purity:
98.22% - 98.54%
Color and Shape:
Liquid
Molecular weight:
284.23
Ref: TM-T79399
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
U-89843A
CAS:157013-85-9
U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents …
Formula:
C16H24ClN5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
321.85
Ref: TM-T78560
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
DMCM hydrochloride
CAS:1215833-62-7
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.
Formula:
C17H19ClN2O4
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
350.8
Ref: TM-T11061
| 1mg | 37.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 464.00 € | ||
| 100mg | 655.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Phaclofen
CAS:114012-12-3
GABAB antagonist
Formula:
C9H13ClNO3P
Purity:
99.32%
Color and Shape:
White Solid
Molecular weight:
249.63
Ref: TM-T23147
| 1mg | 81.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 283.00 € | ||
| 25mg | 652.00 € | ||
| 50mg | 908.00 € | ||
| 100mg | 1,216.00 € | ||
| 200mg | 1,644.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Sarmazenil
CAS:78771-13-8
Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used …
Formula:
C15H14ClN3O3
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
319.74
Ref: TM-T16844
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
RWJ-51204
CAS:205701-85-5
RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:
C21H19F2N3O3
Purity:
100% - 99.57%
Color and Shape:
Solid
Molecular weight:
399.39
Ref: TM-T16811
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Riluzole hydrochloride
CAS:850608-87-6
Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).
Formula:
C8H6ClF3N2OS
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
270.66
Ref: TM-T41265
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
RO 4938581
CAS:883093-10-5
RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, …
Formula:
C13H8BrF2N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T16794
| 25mg | 1,169.00 € | ||
| 50mg | 1,529.00 € | ||
| 100mg | 2,517.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Progabide
CAS:62666-20-0
Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.
Formula:
C17H16ClFN2O2
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
334.77
Ref: TM-T16581
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 335.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Losigamone
CAS:112856-44-7
Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about …
Formula:
C12H11ClO4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
254.67
Ref: TM-T27845
| 1mg | 82.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 256.00 € | ||
| 25mg | 480.00 € | ||
| 50mg | 647.00 € | ||
| 100mg | 940.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Panadiplon
CAS:124423-84-3
Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, …
Formula:
C18H17N5O2
Purity:
100% - 99.75%
Color and Shape:
Solid
Molecular weight:
335.36
Ref: TM-T28294
| 1mg | 140.00 € | ||
| 5mg | 343.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Muscimol HBr
CAS:18174-72-6
Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.
Formula:
C4H7BrN2O2
Purity:
100%
Color and Shape:
Off-White Powder
Molecular weight:
195.01
Ref: TM-T20657
| 1mg | 119.00 € | ||
| 2mg | 172.00 € | ||
| 5mg | 253.00 € | ||
| 10mg | 406.00 € | ||
| 25mg | 657.00 € | ||
| 50mg | 948.00 € | ||
| 100mg | 1,264.00 € | ||
| 500mg | 2,555.00 € | ||
| 1mL*10mM (DMSO) | 215.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Anxiolytic/nonsedative agent-1
CAS:355022-97-8
TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy …
Formula:
C18H15N3O4
Purity:
97.05%
Color and Shape:
Solid
Molecular weight:
337.33
Ref: TM-T23445
| 1mg | 64.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 115.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 330.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 655.00 € | ||
| 500mg | 1,293.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Nerisopam
CAS:102771-12-0
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
Formula:
C18H19N3O2
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
309.36
Ref: TM-T28159
| 1mg | 93.00 € | ||
| 5mg | 200.00 € | ||
| 10mg | 303.00 € | ||
| 25mg | 490.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € | ||
| 500mg | 3,030.00 € | ||
| 1mL*10mM (DMSO) | 270.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Fengabine
CAS:80018-06-0
Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat …
Formula:
C17H17Cl2NO
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
322.23
Ref: TM-T27310
| 1mg | 50.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 154.00 € | ||
| 25mg | 288.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 933.00 € | ||
| 500mg | 1,872.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
SCH 50911
CAS:733717-87-8
SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow …
Formula:
C8H15NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
173.21
Ref: TM-T12867L
| 50mg | 2,480.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
GS 39783
CAS:39069-52-8
GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties …
Formula:
C15H23N5O2S
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
337.44
Ref: TM-T22813
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 592.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
SCH 50911 hydrochloride
CAS:160415-07-6
SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) …
Formula:
C8H16ClNO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
209.67
Ref: TM-T12867
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Pazinaclone
CAS:103255-66-9
Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.
Formula:
C25H23ClN4O4
Purity:
98.12% - 99%
Color and Shape:
Solid
Molecular weight:
478.93
Ref: TM-T28303
| 1mg | 138.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
3α,21-Dihydroxy-5α-pregnan-20-one
CAS:567-02-2
3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like …
Formula:
C21H34O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
334.49
Ref: TM-T26390
| 1mg | 146.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Monday 21 Apr 2025
