GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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Bemegride
CAS:64-65-3
Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.
Formula:
C8H13NO2
Purity:
99.97%
Color and Shape:
Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)
Molecular weight:
155.19
Ref: TM-T1396
| 1g | 90.00 € | ||
| 100mg | 37.00 € | ||
| 200mg | 49.00 € | ||
| 500mg | 69.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Topiramate
CAS:97240-79-4
Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of …
Formula:
C12H21NO8S
Purity:
100% - ≥95%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
339.36
Ref: TM-T0675
| 25mg | 45.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 71.00 € | ||
| 200mg | 108.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Broflanilide
CAS:1207727-04-5
Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 …
Formula:
C25H14BrF11N2O2
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
663.29
Ref: TM-T10618
| 1mg | 51.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 345.00 € | ||
| 50mg | 567.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Flumazenil
CAS:78755-81-4
Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex …
Formula:
C15H14FN3O3
Purity:
100% - 99.62%
Color and Shape:
Less Crystals Colourless Crystals
Molecular weight:
303.29
Ref: TM-T1240
| 25mg | 50.00 € | ||
| 50mg | 70.00 € | ||
| 100mg | 94.00 € | ||
| 500mg | 202.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
LAU159
CAS:2055050-87-6
LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).
Formula:
C17H12ClN3O2
Purity:
98.70% - 99.38%
Color and Shape:
Solid
Molecular weight:
325.75
Ref: TM-T11822
| 1mg | 115.00 € | ||
| 2mg | 166.00 € | ||
| 5mg | 228.00 € | ||
| 10mg | 412.00 € | ||
| 25mg | 681.00 € | ||
| 50mg | 926.00 € | ||
| 100mg | 1,295.00 € | ||
| 500mg | 2,572.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Penicillin G sodium salt
CAS:69-57-8
Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of …
Formula:
C16H17N2NaO4S
Purity:
98.11%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
356.37
Ref: TM-T0958
| 25mg | 30.00 € | ||
| 100mg | 56.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 108.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
GABAA receptor agent 1
CAS:1571-87-5
GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of …
Formula:
C13H8ClN3O2
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
273.67
Ref: TM-T11349
| 1mg | 37.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 477.00 € | ||
| 200mg | 657.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Isoguvacine hydrochloride
CAS:68547-97-7
Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.
Formula:
C6H10ClNO2
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
163.6
Ref: TM-T11684
| 25mg | 39.00 € | ||
| 50mg | 62.00 € | ||
| 100mg | 93.00 € | ||
| 500mg | 203.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
FG 7142
CAS:78538-74-6
FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 …
Formula:
C13H11N3O
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
225.25
Ref: TM-T11277
| 2mg | 33.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | 322.00 € | ||
| 200mg | 446.00 € | ||
| 1mL*10mM (DMSO) | 40.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Nefiracetam
CAS:77191-36-7
Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 …
Formula:
C14H18N2O2
Purity:
100%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
246.3
Ref: TM-T0169
| 100mg | 41.00 € | ||
| 200mg | 50.00 € | ||
| 500mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
3-Methylglutaconic acid
CAS:5746-90-7
3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, …
Formula:
C6H8O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
144.13
Ref: TM-T78071
| 1mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
MIDD0301
CAS:2187489-08-1
MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of …
Formula:
C19H13BrFN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
414.23
Ref: TM-T9946
| 1mg | 184.00 € | ||
| 5mg | 411.00 € | ||
| 10mg | 615.00 € | ||
| 25mg | 1,107.00 € | ||
| 50mg | 1,661.00 € | ||
| 100mg | 2,491.00 € | ||
| 200mg | 3,736.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Furosemide sodium
CAS:41733-55-5
Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.
Formula:
C12H10ClN2NaO5S
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
352.73
Ref: TM-T35336
| 25mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
3-Aminopropylphosphonic Acid
CAS:13138-33-5
3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist …
Formula:
C3H10NO3P
Purity:
98.9%
Color and Shape:
Light Yellow Liquid
Molecular weight:
139.09
Ref: TM-T38205
| 10mg | 39.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | 82.00 € | ||
| 100mg | 112.00 € | ||
| 200mg | 166.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
6,7-dimethylisatin
CAS:20205-43-0
6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.
Formula:
C10H9NO2
Purity:
99.09%
Color and Shape:
Liquid
Molecular weight:
175.18
Ref: TM-T77568
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,699.00 € | ||
| 500mg | 3,428.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
DAA-1106
CAS:220551-92-8
DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective …
Formula:
C23H22FNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
395.42
Ref: TM-T3173
| 5mg | 47.00 € | ||
| 10mg | 79.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
GABA receptor Antagonist 1
GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 …
Purity:
98%
Ref: TM-T82357
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
Guvacine hydrobromide
CAS:6027-92-5
Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor …
Formula:
C6H10BrNO2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
208.05
Ref: TM-T80014
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
CGP 35348
CAS:123690-79-9
CGP 35348: GABAB receptor antagonist, EC50 = 34 μM, used in neonatal brain damage research …
Formula:
C8H20NO4P
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
225.22
Ref: TM-T21793
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 304.00 € | ||
| 50mg | 489.00 € | ||
| 100mg | 733.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Arecaidine hydrobromide
CAS:6013-57-6
Arecaidine hydrobromide, a pyridine alkaloid, functions as a potent GABA uptake inhibitor and acts as …
Formula:
C7H12BrNO2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
222.08
Ref: TM-T80013
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
