Casein Kinase
Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
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LH846
CAS:639052-78-1
LH846 is a selective inhibitor of CK1δ (IC50 values are 290 nM, 1.3 uM and …
Formula:
C16H13ClN2OS
Purity:
90% - 98.13%
Color and Shape:
Solid
Molecular weight:
316.81
Ref: TM-T1877
| 5mg | 63.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 231.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TBB
CAS:17374-26-4
TBB (NSC-231634)(NSC-231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).
Formula:
C6HBr4N3
Purity:
98.51% - 99.45%
Color and Shape:
Off-White Solid
Molecular weight:
434.71
Ref: TM-T2695
| 5mg | 45.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 119.00 € | ||
| 200mg | 173.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
CK1-IN-1
CAS:1784751-20-7
CK1-IN-1, a CK1 inhibitor with IC50: 15nM CK1δ, 16nM CK1ε, 73nM p38σ; patent WO2015119579A1.
Formula:
C24H15F2N3
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
383.39
Ref: TM-T5393
| 1mg | 50.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 304.00 € | ||
| 50mg | 468.00 € | ||
| 100mg | 703.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
DMAT
CAS:749234-11-5
DMAT (Casein kinase II Inhibitor) is a potent and specific inhibitor of CK2(IC50 value of …
Formula:
C9H7Br4N3
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
476.79
Ref: TM-T7390
| 5mg | 62.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 270.00 € | ||
| 100mg | 351.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Longdaysin
CAS:1353867-91-0
Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 μM). It also can inhibit …
Formula:
C16H16F3N5
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
335.33
Ref: TM-T5358
| 5mg | 50.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 315.00 € | ||
| 200mg | 451.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PF-670462
CAS:950912-80-8
PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with …
Formula:
C19H22Cl2FN5
Purity:
99.42% - 99.56%
Color and Shape:
Solid
Molecular weight:
410.32
Ref: TM-T3073
| 2mg | 49.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 371.00 € | ||
| 100mg | 548.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TA-01
CAS:1784751-18-3
TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 …
Formula:
C20H12F3N3
Purity:
98.77% - 99.94%
Color and Shape:
Solid
Molecular weight:
351.32
Ref: TM-T4645
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 150.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 318.00 € | ||
| 200mg | 447.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Epiblastin A
CAS:16470-02-3
Epiblastin A inhibits CK1, targets its isoenzymes, and converts EpiSCs to cESCs.
Formula:
C12H10ClN7
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
287.71
Ref: TM-T8987
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 159.00 € | ||
| 100mg | 261.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
IWP-2
CAS:686770-61-6
IWP-2 is a Wnt pathway inhibitor and an ATP-competitive CK1δ inhibitor. IWP-2 inhibits self-renewal of …
Formula:
C22H18N4O2S3
Purity:
96.1% - 99.76%
Color and Shape:
Solid
Molecular weight:
466.6
Ref: TM-T2702
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 196.00 € | ||
| 100mg | 293.00 € | ||
| 200mg | 440.00 € | ||
| 500mg | 720.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Umbralisib
CAS:1532533-67-7
Umbralisib (TGR 1202) is a PI3Kδ inhibitor.
Formula:
C31H24F3N5O3
Purity:
99.56% - 99.83%
Color and Shape:
White Solid
Molecular weight:
571.55
Ref: TM-T4976
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 335.00 € | ||
| 50mg | 440.00 € | ||
| 100mg | 644.00 € | ||
| 1mL*10mM (DMSO) | 121.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
MLN8054
CAS:869363-13-3
MLN8054 is a potent and selective Aurora A kinase inhibitor with an IC50 of 4 …
Formula:
C25H15ClF2N4O2
Purity:
98.07% - 98.26%
Color and Shape:
Solid
Molecular weight:
476.86
Ref: TM-T6315
| 1mg | 52.00 € | ||
| 2mg | 71.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 562.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
NCC007
CAS:2342583-66-6
NCC007 is a novel CKIα and CKIδ dual inhibitors by structural modification of N9 and …
Formula:
C22H28F3N7
Purity:
98.11%
Color and Shape:
Solid
Molecular weight:
447.5
Ref: TM-T7949
| 5mg | 44.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 169.00 € | ||
| 100mg | 241.00 € | ||
| 200mg | 347.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
SR-3029
CAS:1454585-06-8
SR-3029 is a potent and highly specific CK1δ/CK1ε inhibitor.
Formula:
C23H19F3N8O
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
480.45
Ref: TM-T3972
| 1mg | 35.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 388.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TTP 22
CAS:329907-28-0
TTP 22: ATP-competitive CK2 inhibitor; IC50/Ki: 0.1 μM/40 nM; >250x selective over JNK3, ROCK1, MET.
Formula:
C16H14N2O2S2
Purity:
97.08% - 97.78%
Color and Shape:
Solid
Molecular weight:
330.42
Ref: TM-T1828
| 1mg | 38.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 108.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 477.00 € | ||
| 1mL*10mM (DMSO) | 98.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
LY294002
CAS:154447-36-6
LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 …
Formula:
C19H17NO3
Purity:
98% - 99.96%
Color and Shape:
Pale Yellow Solid
Molecular weight:
307.34
Ref: TM-T2008
| 5mg | 39.00 € | ||
| 10mg | 50.00 € | ||
| 50mg | 71.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 121.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Silmitasertib
CAS:1009820-21-6
Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 …
Formula:
C19H12ClN3O2
Purity:
98% - ≥95%
Color and Shape:
Solid
Molecular weight:
349.77
Ref: TM-T2259
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 508.00 € | ||
| 500mg | 1,086.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
D4476
CAS:301836-43-1
D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) …
Formula:
C23H18N4O3
Purity:
99.02% - 99.96%
Color and Shape:
Solid
Molecular weight:
398.41
Ref: TM-T2449
| 1mg | 42.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 401.00 € | ||
| 200mg | 584.00 € | ||
| 500mg | 917.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Orobol
CAS:480-23-9
Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) is an inhibitor of tyrosine-specific protein kinase and phosphatidylinositol turnover.
Formula:
C15H10O6
Purity:
98% - 98%
Color and Shape:
Solid
Molecular weight:
286.24
Ref: TM-TN2019
| 1mg | 178.00 € | ||
| 2mg | 268.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PF-4800567
CAS:1188296-52-7
PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with …
Formula:
C17H18ClN5O2
Purity:
98.23%
Color and Shape:
Solid
Molecular weight:
359.81
Ref: TM-T5056
| 5mg | 44.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 191.00 € | ||
| 100mg | 276.00 € | ||
| 200mg | 400.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
LY-294002 hydrochloride
CAS:934389-88-5
LY-294002 HCl (NSC 697286) is a stable PI3K inhibitor (IC50: 0.5-0.97 µM) and prevents autophagosome …
Formula:
C19H17NO3·HCl
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
343.81
Ref: TM-T4079
| 1mg | 43.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 440.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
