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Casein Kinase

Casein Kinase

Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.

Found 130 products of "Casein Kinase"

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  • CymitQuimica logo
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    CK1-IN-4

    <p>CK1-IN-4 (Compound 59) is an inhibitor of casein kinase CK1δ with an IC50 of 2.74 μM. It exhibits neuroprotective activity in SH-SY5Y cells treated with Ethacrynic acid.</p>
    Color and Shape:Odour Solid

    Ref: TM-T89036

  • Casein kinase 1δ-IN-9
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    Casein kinase 1δ-IN-9

    CAS:
    <p>Casein kinase 1δ-IN-9 is a Quinone reductase 2 inhibitor with IC50 of 0.6μM.</p>
    Formula:C15H12ClN3
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:269.73

    Ref: TM-T64376

  • Casein kinase 1δ-IN-7
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    Casein kinase 1δ-IN-7

    CAS:
    <p>Casein kinase 1δ-IN-7 is a Casein kinase 1δ inhibitor for neurodegenerative diseases such as Alzheimer's disease.</p>
    Formula:C17H14N4O2S
    Purity:98.6%
    Color and Shape:Solid
    Molecular weight:338.38

    Ref: TM-T77708

  • WAY-297174
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    WAY-297174

    CAS:
    <p>WAY-297174 is a human protein kinase CK2 inhibitor with IC50 of &gt; 33 μM.</p>
    Formula:C11H12N2O2S2
    Purity:99.53%
    Color and Shape:Soild
    Molecular weight:268.36

    Ref: TM-T60067

  • Casein Kinase 2 Substrate Peptide
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    Casein Kinase 2 Substrate Peptide

    CAS:
    <p>CK2 Substrate Peptide, C-terminus linked to EDANS, used for CK2 activity assays.</p>
    Formula:C45H73N19O24
    Color and Shape:Solid
    Molecular weight:1264.17

    Ref: TM-T76411

  • Casein Kinase Substrates 3
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    Casein Kinase Substrates 3

    CAS:
    <p>Casein Kinase Substrates 3 is a substrate of casein kinase.</p>
    Formula:C85H139N27O35S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2131.24

    Ref: TM-TP1509

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    QXG-6442

    <p>QXG-6442 is a molecular glue degrader targeting CK1α, demonstrating a degradation potency with a DC50 of 5.7 nM and a Dmax of 90%. In the MOLM-14 cell line, QXG-6442 induces antiproliferative effects.</p>
    Formula:C21H17N5O4
    Color and Shape:Solid
    Molecular weight:403.39

    Ref: TM-T205020

  • CymitQuimica logo
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    CZP-IN-1

    <p>CZP-IN-1 (compound SH-1) is an inhibitor targeting the pathogen Trypanosoma cruzi protease (CZP) without affecting cathepsin L (IC50=28 nM). This compound is applicable in Chagas disease research.</p>
    Formula:C20H26N4O4S
    Color and Shape:Solid
    Molecular weight:418.51

    Ref: TM-T205551

  • Casein kinase 1δ-IN-14
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    Casein kinase 1δ-IN-14

    CAS:
    <p>Casein kinase 1δ-IN-14 (WAY-637081) can be used to study atherosclerosis-related cardiovascular disease.</p>
    Formula:C17H11ClN4O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:338.75

    Ref: TM-T77648

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    AH078

    <p>AH078 (compound 37) is a selective PROTAC degrader targeting CK1δ and CK1ε with low selectivity for CK1α. AH078 consists of a PROTAC linker (black part) Monomethyl octanoate, a target protein ligand (red part) CK1δ/CK1ε ligand-1, and an E3 ligase ligand (blue part) E3 Ligase Ligand 58. The E3 ligase ligand combined with the linker forms the conjugate E3 Ligase Ligand-linker Conjugate 163.</p>
    Formula:C51H60F2N10O5S
    Color and Shape:Solid
    Molecular weight:963.15

    Ref: TM-T205491

  • SGC-CK2-1
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    SGC-CK2-1

    CAS:
    <p>SGC-CK2-1, a CK2 inhibitor, is a inducer of insulin production and secretion in pancreatic β-cells.</p>
    Formula:C20H21N7O
    Purity:99.41%
    Color and Shape:Solid
    Molecular weight:375.43

    Ref: TM-T40131

  • FPFT-2216
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    FPFT-2216

    CAS:
    <p>FPFT-2216 is a "molecular glue" compound with potential anti-tumor activity that degrades IKZF6, IKZF1, DE1D and can be used to study immune system diseases.</p>
    Formula:C12H12N4O3S
    Purity:99.35% - 99.62%
    Color and Shape:Solid
    Molecular weight:292.31

    Ref: TM-T60608

  • MRT00033659
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    MRT00033659

    CAS:
    <p>MRT00033659 inhibits CK1 (IC50=0.9 μM), CHK1 (IC50=0.23 μM), activates p53, and destabilizes E2F-1; it's a pyrazolo-pyridine.</p>
    Formula:C15H14N4O
    Color and Shape:Solid
    Molecular weight:266.3

    Ref: TM-T16141

  • PF-5006739
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    PF-5006739

    CAS:
    <p>PF-5006739: potent, selective CK1δ/ε inhibitor (IC50: 3.9/17.0 nM); may treat psychiatric disorders, improves glucose tolerance, reduces opioid seeking.</p>
    Formula:C22H22FN7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:419.45

    Ref: TM-T16507

  • TA-01
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    TA-01

    CAS:
    <p>TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respectively.</p>
    Formula:C20H12F3N3
    Purity:99.55% - 99.94%
    Color and Shape:Solid
    Molecular weight:351.32

    Ref: TM-T4645

  • PF-670462
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    PF-670462

    CAS:
    <p>PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (&gt;30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.</p>
    Formula:C19H22Cl2FN5
    Purity:99.42% - 99.72%
    Color and Shape:Solid
    Molecular weight:410.32

    Ref: TM-T3073

  • CK1-IN-1
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    CK1-IN-1

    CAS:
    <p>CK1-IN-1, a CK1 inhibitor with IC50: 15nM CK1δ, 16nM CK1ε, 73nM p38σ; patent WO2015119579A1.</p>
    Formula:C24H15F2N3
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:383.39

    Ref: TM-T5393

  • Longdaysin
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    Longdaysin

    CAS:
    <p>Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 μM). It also can inhibit ERK2 (IC50: 52 μM).</p>
    Formula:C16H16F3N5
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:335.33

    Ref: TM-T5358

  • TBB
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    TBB

    CAS:
    <p>TBB (NSC-231634)(NSC-231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).</p>
    Formula:C6HBr4N3
    Purity:98.51% - 99.45%
    Color and Shape:Off-White Solid
    Molecular weight:434.71

    Ref: TM-T2695

  • LY294002
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    LY294002

    CAS:
    <p>LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).</p>
    Formula:C19H17NO3
    Purity:98% - 99.96%
    Color and Shape:Pale Yellow Solid
    Molecular weight:307.34

    Ref: TM-T2008