Casein Kinase
Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
Found 150 products for "Casein Kinase".
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LY-294002 hydrochloride
CAS:LY-294002 HCl (NSC 697286) is a stable PI3K inhibitor (IC50: 0.5-0.97 µM) and prevents autophagosome formation.Formula:C19H17NO3·HClPurity:99.95% - 99.98%Color and Shape:Purple LiquidMolecular weight:343.81TTP 22
CAS:TTP 22: ATP-competitive CK2 inhibitor; IC50/Ki: 0.1 μM/40 nM; >250x selective over JNK3, ROCK1, MET.Formula:C16H14N2O2S2Purity:97.08% - 97.78%Color and Shape:SolidMolecular weight:330.42Umbralisib hydrochloride
CAS:Umbralisib hydrochloride: PI3Kδ inhibitor; IC50=22.2 nM, EC50=24.3 nM; active vs CK1ε, EC50=6.0 μM.Formula:C31H25ClF3N5O3Purity:98%Color and Shape:SolidMolecular weight:608.01DMAT
CAS:DMAT (Casein kinase II Inhibitor) is a potent and specific inhibitor of CK2(IC50 value of 130 nM).Formula:C9H7Br4N3Purity:99.48%Color and Shape:White SolidMolecular weight:476.79SR-3029
CAS:SR-3029 is a potent and highly specific CK1δ/CK1ε inhibitor.Formula:C23H19F3N8OPurity:99.64%Color and Shape:SolidMolecular weight:480.45D4476
CAS:D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).Formula:C23H18N4O3Purity:99.7% - 99.96%Color and Shape:SolidMolecular weight:398.41IWP-2
CAS:IWP-2 is a Wnt pathway inhibitor and an ATP-competitive CK1δ inhibitor. IWP-2 inhibits self-renewal of embryonic stem cells. Cost effective and quality assured.Formula:C22H18N4O2S3Purity:96.1% - 99.86%Color and Shape:White SolidMolecular weight:466.599Umbralisib
CAS:Umbralisib (TGR 1202) is a PI3Kδ inhibitor.Formula:C31H24F3N5O3Purity:99.56% - 99.56%Color and Shape:White SolidMolecular weight:571.55Ref: TM-T4976
1mg46.00€2mg62.00€5mg90.00€1mL*10mM (DMSO)114.00€10mg166.00€25mg324.00€50mg425.00€100mg623.00€Epiblastin A
CAS:Epiblastin A inhibits CK1, targets its isoenzymes, and converts EpiSCs to cESCs.Formula:C12H10ClN7Purity:99.45%Color and Shape:SolidMolecular weight:287.71Orobol
CAS:Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) is an inhibitor of tyrosine-specific protein kinase and phosphatidylinositol turnover.Formula:C15H10O6Purity:98% - 98%Color and Shape:SolidMolecular weight:286.24(E/Z)-GO289
CAS:(E/Z)-GO289, which strongly lengthened circadian period, is a potent and selective inhibitor of CK2.Formula:C17H15BrN4O2SPurity:98.1%Color and Shape:SolidMolecular weight:419.3Ref: TM-T9356
2mg34.00€5mg52.00€1mL*10mM (DMSO)54.00€10mg86.00€25mg170.00€50mg250.00€100mg354.00€200mg482.00€TA-01
CAS:TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respectively.Formula:C20H12F3N3Purity:99.55% - 99.94%Color and Shape:SolidMolecular weight:351.32Ref: TM-T4645
2mg34.00€5mg50.00€1mL*10mM (DMSO)67.00€10mg80.00€25mg147.00€50mg224.00€100mg313.00€200mg439.00€NCC007
CAS:NCC007 is a novel CKIα and CKIδ dual inhibitors by structural modification of N9 and C2 position of longdaysin.Formula:C22H28F3N7Purity:98.88%Color and Shape:SolidMolecular weight:447.5CK2-IN-1
CAS:CK2 inhibitorFormula:C14H9NO3Purity:97.28%Color and Shape:SolidMolecular weight:239.2262Silmitasertib
CAS:Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 nM).Formula:C19H12ClN3O2Purity:98% - 99.94%Color and Shape:SolidMolecular weight:349.77Ref: TM-T2259
1mg38.00€2mg49.00€5mg80.00€1mL*10mM (DMSO)88.00€10mg118.00€25mg197.00€50mg313.00€100mg492.00€500mg1,054.00€AS-252424
CAS:AS-252424 is a potent and selective inhibitor of PI3Kγ with IC50 of 33 nM; >10 fold selectivity for PI3Kγ versus PI3Kα.Formula:C14H8FNO4SPurity:99.06% - 99.09%Color and Shape:Orange SolidMolecular weight:305.28Ref: TM-T6208
1mg37.00€2mg52.00€5mg77.00€1mL*10mM (DMSO)84.00€10mg128.00€25mg205.00€50mg309.00€100mg447.00€500mg973.00€PF-4800567
CAS:PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.Formula:C17H18ClN5O2Purity:99.74% - 99.76%Color and Shape:White SolidMolecular weight:359.81LY294002
CAS:LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).Formula:C19H17NO3Purity:98% - 99.96%Color and Shape:White SolidMolecular weight:307.34PF-670462
CAS:PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.Formula:C19H22Cl2FN5Purity:99.42% - 99.72%Color and Shape:SolidMolecular weight:410.32TAK-715
CAS:TAK-715 is a p38 MAPK inhibitor for p38α.Formula:C24H21N3OSPurity:99.83%Color and Shape:White SolidMolecular weight:399.51Ref: TM-T6150
1mg38.00€2mg50.00€5mg82.00€1mL*10mM (DMSO)92.00€10mg94.00€25mg166.00€50mg306.00€100mg480.00€
