PPAR
Peroxisome Proliferator-Activated Receptors (PPARs) are a group of nuclear receptor proteins that function as transcription factors regulating the expression of genes involved in metabolism, particularly fatty acid storage and glucose metabolism. PPAR inhibitors are important tools for studying metabolic disorders such as diabetes, obesity, and cardiovascular diseases. These inhibitors can modulate lipid metabolism, insulin sensitivity, and inflammation, making them valuable in therapeutic research. At CymitQuimica, we offer a range of PPAR inhibitors to support your research in metabolic diseases, endocrinology, and drug development.
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Gemfibrozil
CAS:25812-30-0
Gemfibrozil, a fibric acid derivative, stimulates PPARalpha, boosts fatty acid oxidation, LPL, lowers VLDL-C, apoC-III, …
Formula:
C15H22O3
Purity:
99.53% - 99.88%
Color and Shape:
Crystals From Hexane Solid
Molecular weight:
250.33
Ref: TM-T1415
| 25mg | 35.00 € | ||
| 50mg | 46.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 69.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
5-Aminosalicylic Acid
CAS:89-57-6
5-ASA, an anti-inflammatory salicylate, treats inflammatory bowel disease, active part of sulphalazine.
Formula:
C7H7NO3
Purity:
98.88% - 99.98%
Color and Shape:
Purplish-Tan Solid Powder
Molecular weight:
153.14
Ref: TM-T0646
| 500mg | 49.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Oleoylethanolamide
CAS:111-58-0
Oleoylethanolamide (N-Oleoylethanolamide) is a high affinity endogenous agonist of PPAR-α.
Formula:
C20H39NO2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
325.53
Ref: TM-T12296
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 376.00 € | ||
| 200mg | 550.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Fenofibrate
CAS:49562-28-9
Fenofibrate (Lipanthyl) is a PPARα agonist. Fenofibrate inhibits cytochrome P450 isoforms. Fenofibrate exhibits antihyperlipidemic activity. …
Formula:
C20H21ClO4
Purity:
99.13% - 99.95%
Color and Shape:
Crystals From Isopropanol Solid
Molecular weight:
360.83
Ref: TM-T1149
| 100mg | 38.00 € | ||
| 200mg | 49.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Rosiglitazone maleate
CAS:155141-29-0
Rosiglitazone maleate (BRL 49653) is an oral antidiabetic and potential anticancer agent.
Formula:
C22H23N3O7S
Purity:
99.33% - 99.51%
Color and Shape:
Off-White Solid
Molecular weight:
473.5
Ref: TM-T1622
| 50mg | 34.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 144.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Magnolol
CAS:528-43-8
Magnolol (5,5'-Diallyl-2,2'-biphenyldiol) is a dual agonist of RXRα( EC50=10.4 μM) and PPARγ(EC50=17.7 μM). It blocks …
Formula:
C18H18O2
Purity:
99.49%
Color and Shape:
A Bioactive Compound Found In The Bark Of The Houpu Magnolia
Molecular weight:
266.33
Ref: TM-T3000
| 1g | 543.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 72.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 153.00 € | ||
| 500mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Pioglitazone hydrochloride
CAS:112529-15-4
Pioglitazone hydrochloride (AD 4833) is the hydrochloride salt of an orally-active thiazolidinedione with antidiabetic properties …
Formula:
C19H20N2O3S·HCl
Purity:
100% - 99.66%
Color and Shape:
White Crystals Or Crystalline Powder
Molecular weight:
392.9
Ref: TM-T0214L
| 50mg | 42.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 80.00 € | ||
| 500mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Anandamide
CAS:94421-68-8
Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but …
Formula:
C22H37NO2
Purity:
98.76% - 99.22%
Color and Shape:
Light Yellow Oil
Molecular weight:
347.53
Ref: TM-T14046
| 2mg | 72.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 435.00 € | ||
| 100mg | 640.00 € | ||
| 500mg | 1,359.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Daidzein
CAS:486-66-8
Daidzein (Isoflavone) is an isoflavone extract from soy, which is an inactive analog of the …
Formula:
C15H10O4
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
254.24
Ref: TM-T1238
| 1g | 63.00 € | ||
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Retinoic acid
CAS:302-79-4
Retinoic acid (Tretinoin) binds to and activates RARs, thereby inducing changes in gene expression that …
Formula:
C20H28O2
Purity:
97.21% - 99.6%
Color and Shape:
Yellow-Orange Powder
Molecular weight:
300.44
Ref: TM-T1051
| 50mg | 39.00 € | ||
| 100mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Clofibric acid
CAS:882-09-7
Clofibric acid (Chlorofibrinic acid) is an antilipemic agent that is the biologically active metabolite of …
Formula:
C10H11ClO3
Purity:
99.47% - 99.8%
Color and Shape:
Pale Yellow Solid
Molecular weight:
214.65
Ref: TM-T0061
| 1g | 37.00 € | ||
| 5g | 77.00 € | ||
| 10g | 97.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Arhalofenate
CAS:24136-23-0
Arhalofenate (JNJ 39659100) is a selective partial agonist of peroxisome proliferator-activated receptor PPARγ. It is …
Formula:
C19H17ClF3NO4
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
415.79
Ref: TM-T16022
| 1mg | 131.00 € | ||
| 5mg | 286.00 € | ||
| 10mg | 430.00 € | ||
| 25mg | 710.00 € | ||
| 50mg | 998.00 € | ||
| 100mg | 1,349.00 € | ||
| 500mg | 2,688.00 € | ||
| 1mL*10mM (DMSO) | 330.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
NSC-87877
CAS:56990-57-9
NSC-87877 inhibits Shp2 (IC50=0.318μM), Shp1 (IC50=0.355μM), and DUSP26 phosphatases.
Formula:
C19H13N3O7S2
Purity:
97.35%
Color and Shape:
Solid
Molecular weight:
459.45
Ref: TM-T16350
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 465.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
GW7647
CAS:265129-71-3
GW 7647 is an effective and highly selective PPARα agonist. GW 7647 can reduce the …
Formula:
C29H46N2O3S
Purity:
99.30% - 99.34%
Color and Shape:
Solid
Molecular weight:
502.75
Ref: TM-T15453
| 1mg | 49.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 605.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
LY518674
CAS:425671-29-0
LY518674 (LY-674) decreases triglycerides and increases HDL-C and is used for the treatment of atherosclerosis.
Formula:
C23H27N3O4
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
409.48
Ref: TM-T15821
| 1mg | 170.00 € | ||
| 5mg | 359.00 € | ||
| 10mg | 533.00 € | ||
| 25mg | 847.00 € | ||
| 50mg | 1,159.00 € | ||
| 100mg | 1,568.00 € | ||
| 1mL*10mM (DMSO) | 398.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Mifobate
CAS:76541-72-5
Mifobate (SR-202) 是一种有效且特异性的 PPARγ拮抗剂,可选择性抑制噻唑烷二酮 (TZD) 诱导的 PPARγ 转录活性,IC50为140 μM,具有抗肥胖和抗糖尿病作用。
Formula:
C11H17ClO7P2
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
358.65
Ref: TM-T16074
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 303.00 € | ||
| 50mg | 449.00 € | ||
| 100mg | 645.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Pioglitazone
CAS:111025-46-8
Pioglitazone (U 72107) is an insulin sensitizing agent and thiazolidinedione that is indicated for the …
Formula:
C19H20N2O3S
Purity:
95% - 99.57%
Color and Shape:
White Powder
Molecular weight:
356.44
Ref: TM-T0214
| 5mg | 42.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 97.00 € | ||
| 100mg | 140.00 € | ||
| 500mg | 334.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
CUDA
CAS:479413-68-8
CUDA is an effective soluble cyclohydrolase inhibitor with IC50 of 11.1 nM and 112 nM …
Formula:
C19H36N2O3
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
340.5
Ref: TM-T10900
| 5mg | 48.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 334.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
MA-0204
CAS:2095128-17-7
MA-0204 is a highly selective and orally available peroxisome proliferator-activated receptor δ (PPARδ) modulator (EC50s: …
Formula:
C25H27F3N2O4
Purity:
97.80%
Color and Shape:
Solid
Molecular weight:
476.49
Ref: TM-T15945
| 1mg | 96.00 € | ||
| 5mg | 178.00 € | ||
| 10mg | 301.00 € | ||
| 25mg | 490.00 € | ||
| 50mg | 677.00 € | ||
| 100mg | 900.00 € | ||
| 200mg | 1,206.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Fenofibric acid
CAS:42017-89-0
Fenofibric acid (FNF acid) is the active form of fenofibrate, a synthetic phenoxy-isobutyric acid derivate …
Formula:
C17H15ClO4
Purity:
99.36%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
318.75
Ref: TM-T1402
| 1g | 37.00 € | ||
| 5g | 74.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
