PPAR
Peroxisome Proliferator-Activated Receptors (PPARs) are a group of nuclear receptor proteins that function as transcription factors regulating the expression of genes involved in metabolism, particularly fatty acid storage and glucose metabolism. PPAR inhibitors are important tools for studying metabolic disorders such as diabetes, obesity, and cardiovascular diseases. These inhibitors can modulate lipid metabolism, insulin sensitivity, and inflammation, making them valuable in therapeutic research. At CymitQuimica, we offer a range of PPAR inhibitors to support your research in metabolic diseases, endocrinology, and drug development.
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GW590735
CAS:343321-96-0
GW590735: PPARα agonist, EC50=4 nM, >500x selective over PPARδ/γ, for dyslipidemia research.
Formula:
C23H21F3N2O4S
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
478.48
Ref: TM-T9766
| 1mg | 95.00 € | ||
| 5mg | 202.00 € | ||
| 10mg | 298.00 € | ||
| 25mg | 507.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 1,026.00 € | ||
| 1mL*10mM (DMSO) | 213.00 € |
Estimated delivery in United States, on Monday 12 May 2025
Mavodelpar free acid hydrochloride
Mavodelpar free acid hydrochloride (Pparδ agonist HCl) is a potent PPARδ agonist.
Formula:
C31H31ClFNO5
Purity:
99.39%
Color and Shape:
Soild
Molecular weight:
552.03
Ref: TM-T12527L
| 1mg | 313.00 € | ||
| 5mg | 758.00 € | ||
| 10mg | 1,035.00 € | ||
| 25mg | 1,568.00 € | ||
| 50mg | 2,118.00 € | ||
| 100mg | 2,783.00 € |
Estimated delivery in United States, on Monday 12 May 2025
PPARγ agonist 16
CAS:2218046-01-4
PPARγ agonist16 (Compound 4G) is a PPARγ agonist that competitively binds to the ligand-binding domain …
Formula:
C19H14BrNO4S
Color and Shape:
Solid
Molecular weight:
432.29
Ref: TM-T203519
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
PPARγ agonist 15
PPARγ agonist15 (Compound 7c) functions as an agonist of PPARγ, inhibiting the expression of α-amylase …
Formula:
C21H16N4O3S2
Color and Shape:
Solid
Molecular weight:
436.51
Ref: TM-T203583
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
E0924G
CAS:2909474-29-7
E0924G is an orally active PPARδ agonist with an EC50 of 2.82 μM. It enhances …
Formula:
C12H12N2O3
Color and Shape:
Solid
Molecular weight:
232.24
Ref: TM-T203555
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
(±)-CBCQ
CAS:2415352-36-0
(±)-CBCQ, an oxidation product of cannabidiol, exhibits an EC50 value of 14.7 μM for the …
Formula:
C21H28O3
Color and Shape:
Solid
Molecular weight:
328.45
Ref: TM-T203263
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
SP4e
SP4e, a PPAR-γ activator, exhibits an EC50 of 739 nM in HK-2 cells.
Purity:
98%
Color and Shape:
Odour Solid
Ref: TM-T81121
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
SP4f
SP4f, an activator of PPAR-γ, exhibits an EC50 value of 826 nM in HK-2 cells.
Purity:
98%
Color and Shape:
Odour Solid
Ref: TM-T81120
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
Foenumoside B
CAS:877661-00-2
Foenumoside B, a triterpene saponin extracted from Lysimachia foenum-graecum, stimulates AMPK signaling, suppresses PPARγ-induced adipogenesis, …
Formula:
C60H96O25
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1217.39
Ref: TM-T79949
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
PPAR α/PPARA Protein, Mouse, Recombinant (His)
PPAR alpha/PPARA Protein, Mouse, Recombinant (His) is expressed in E.
Color and Shape:
Liquid
Molecular weight:
31.49 kDa (predicted)
Ref: TM-TMPY-06837
| 50µg | 608.00 € | ||
| 500µg | 3,832.00 € |
Estimated delivery in United States, on Monday 12 May 2025
CP-868388 free base
CAS:702681-67-2
CP-868388 free base (CP-868388) is a PPARα agonist with hypolipidemic and anti-inflammatory activity and is …
Formula:
C26H33NO5
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
439.54
Ref: TM-T31083
| 1mg | 57.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Monday 12 May 2025
Balaglitazone
CAS:199113-98-9
Balaglitazone is a PPARγ agonist that regulates blood glucose and is used in studies of …
Formula:
C20H17N3O4S
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
395.43
Ref: TM-TQ0272
| 1mg | 90.00 € |
Estimated delivery in United States, on Monday 12 May 2025
PPAR α/PPARA Protein, Human, Recombinant (His)
PPAR alpha/PPARA Protein, Human, Recombinant (His) is expressed in E.
Color and Shape:
Lyophilized Powder
Molecular weight:
31.36 kDa (predicted)
Ref: TM-TMPY-06830
| 50µg | 608.00 € | ||
| 500µg | 3,832.00 € |
Estimated delivery in United States, on Monday 12 May 2025
L-165041
CAS:79558-09-1
L-165041 is a potent and selective agonist of the nuclear receptor PPARβ and PPARδ(Ki = …
Formula:
C22H26O7
Purity:
97.97%
Color and Shape:
Solid
Molecular weight:
402.44
Ref: TM-T7159
| 5mg | 48.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 338.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 16 May 2025
LJ570
CAS:2252488-69-8
LJ570 is the first PPARα/γ dual agonist (PPARα,PPARγ with EC50s of 1.05 and 0.12 μM, …
Formula:
C27H22O3
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
394.46
Ref: TM-T8374
| 1mg | 145.00 € | ||
| 2mg | 213.00 € | ||
| 5mg | 329.00 € | ||
| 10mg | 470.00 € | ||
| 25mg | 718.00 € | ||
| 50mg | 938.00 € | ||
| 100mg | 1,301.00 € | ||
| 500mg | 2,612.00 € | ||
| 1mL*10mM (DMSO) | 354.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Glabrone
CAS:60008-02-8
Glabrone shows antiviral activity against influenza virus.
Formula:
C20H16O5
Purity:
99.08% - 99.55%
Color and Shape:
Solid
Molecular weight:
336.34
Ref: TM-TN1693
| 1mg | 115.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 411.00 € | ||
| 25mg | 682.00 € | ||
| 50mg | 938.00 € | ||
| 100mg | 1,301.00 € |
Estimated delivery in United States, on Friday 16 May 2025
GSK3787
CAS:188591-46-0
GSK3787 is a specific and irreversible PPARδ inhibitor(pIC50= 6.6).
Formula:
C15H12ClF3N2O3S
Purity:
98% - 98.53%
Color and Shape:
Solid
Molecular weight:
392.78
Ref: TM-T1941
| 5mg | 55.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 173.00 € | ||
| 50mg | 309.00 € | ||
| 100mg | 520.00 € | ||
| 500mg | 1,111.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 16 May 2025
MK-886
CAS:118414-82-7
MK-886 (L 663536) is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP).
Formula:
C27H34ClNO2S
Purity:
98.9% - 99.78%
Color and Shape:
Solid
Molecular weight:
472.08
Ref: TM-T6893
| 1mg | 35.00 € | ||
| 2mg | 48.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 567.00 € | ||
| 500mg | 1,198.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Methyl oleanonate
CAS:1721-58-0
3-Oxoolean-12-en-28-oic acid methyl ester is a triterpenoid PPARγ agonist isolated from Pistacia with anticancer properties.
Formula:
C31H48O3
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
468.71
Ref: TM-TN7060
| 1mg | 88.00 € | ||
| 5mg | 202.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 512.00 € | ||
| 50mg | 730.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Oroxin A
CAS:57396-78-8
Oroxin A (Baicalein 7-O-glucoside) has antitussive and expectorant effects.
Formula:
C21H20O10
Purity:
98.05% - 99.74%
Color and Shape:
Solid
Molecular weight:
432.38
Ref: TM-T5S0788
| 1mg | 43.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 224.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 509.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Friday 16 May 2025
