5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 1025 products of "5-HT Receptor"
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LY 344864 S-enantiomer
CAS:LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.Formula:C21H22FN3OPurity:98%Color and Shape:SolidMolecular weight:351.42PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formula:C23H21ClFN5O4SPurity:97.59%Color and Shape:SolidMolecular weight:517.96Ref: TM-T6959
1mg79.00€5mg168.00€10mg220.00€25mg398.00€50mg587.00€100mg835.00€200mg1,134.00€1mL*10mM (DMSO)380.00€Bopindolol fumarate
CAS:Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.Formula:C27H32N2O7Color and Shape:SolidMolecular weight:496.56DR4485 hydrochloride
CAS:5-HT7 antagonistFormula:C26H29Cl3N2OPurity:98%Color and Shape:SolidMolecular weight:491.88OSU 6162 hydrochloride
CAS:Dopamine stabilizerFormula:C15H24ClNO2SPurity:98%Color and Shape:SolidMolecular weight:317.88S-15535
CAS:S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.Formula:C21H24N2O2Purity:98%Color and Shape:SolidMolecular weight:336.43Etoperidone hydrochloride
CAS:Etoperidone hydrochloride is an antidepressant agent.Formula:C19H29Cl2N5OColor and Shape:SolidMolecular weight:414.37SLV-310
CAS:SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.Formula:C25H24FN3O2Purity:99.39%Color and Shape:SolidMolecular weight:417.48Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purity:98%Color and Shape:SolidMolecular weight:393.74Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Formula:C27H41ClN4O5Color and Shape:SolidMolecular weight:537.09Fonazine
CAS:Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.Formula:C19H25N3O2S2Color and Shape:SolidMolecular weight:391.55Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Formula:C26H32N2O7Color and Shape:SolidMolecular weight:484.549(R)-Viloxazine Hydrochloride
CAS:(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.Formula:C13H20ClNO3Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:273.76Ref: TM-T22413
1mg52.00€5mg111.00€10mg162.00€25mg235.00€50mg330.00€100mg452.00€200mg607.00€1mL*10mM (DMSO)101.00€LEK 8841
CAS:LEK 8841 is an ergoline derivative that is a potential antipsychotic.Formula:C21H24BrN3O4SPurity:98%Color and Shape:SolidMolecular weight:494.4AP-521 (Free base)
CAS:AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.Formula:C20H18N2O3SColor and Shape:SolidMolecular weight:366.43Trimipramine
CAS:Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.Formula:C20H26N2Purity:98%Color and Shape:SolidMolecular weight:294.435-HT2A receptor agonist-2
CAS:Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.Formula:C20H21ClN2O3Color and Shape:SolidMolecular weight:372.85Alniditan
CAS:Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.Formula:C17H26N4OPurity:98%Color and Shape:SolidMolecular weight:302.41OPC-14523 hydrochloride
CAS:OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.Formula:C23H29Cl2N3O2Purity:99.60%Color and Shape:SolidMolecular weight:450.4Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Formula:C26H31FN2O4Purity:98%Color and Shape:SolidMolecular weight:454.53CGS-12066 maleate salt
CAS:CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.Formula:C21H21F3N4O4Color and Shape:SolidMolecular weight:450.41TMPPAA
CAS:TMPPAA is an allosteric agonist of 5-HT3 receptor.Formula:C15H21NO2Purity:98%Color and Shape:SolidMolecular weight:247.33Lofepramine hydrochloride
CAS:Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.Formula:C26H28Cl2N2OPurity:98%Color and Shape:Off-White SolidMolecular weight:455.42GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Formula:C19H20N2O2Purity:98%Color and Shape:SolidMolecular weight:308.37LY320135
CAS:CB1 receptor antagonist/inverse agonistFormula:C24H17NO4Purity:98%Color and Shape:SolidMolecular weight:383.4Pruvanserin hydrochloride
CAS:Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.Formula:C22H22ClFN4OPurity:99.6%Color and Shape:SolidMolecular weight:412.89Nexopamil racemate
CAS:Nexopamil racemate（(Rac)-Nexopamil） is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.Formula:C24H40N2O3Purity:98.61%Color and Shape:SolidMolecular weight:404.59Oxetorone fumarate
CAS:Oxetorone fumarate is a non-selective, orally active antagonist of serotonin and 5-HT receptors,used for migraine treatment.Formula:C25H25NO6Purity:99.809%Color and Shape:SolidMolecular weight:435.48Tertatolol
CAS:Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.Formula:C16H25NO2SPurity:98%Color and Shape:SolidMolecular weight:295.44YM 114
CAS:YM 114 is an anatagonist of 5-HT(3) receptor.Formula:C16H18ClN3OPurity:98%Color and Shape:SolidMolecular weight:303.79Bifeprunox Mesylate
CAS:Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.Formula:C25H27N3O5SPurity:98%Color and Shape:SolidMolecular weight:481.56SB-737050A
CAS:SB-737050A, a 5-HT antagonist, is used potentially for the treatment of schizophrenia.Formula:C22H23ClN2O3S2Color and Shape:SolidMolecular weight:463.01GR-55562 dihydrobromide
CAS:GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.Formula:C23H26ClN3O2Purity:98%Color and Shape:SolidMolecular weight:411.93SDZ 21009
CAS:β-adrenoceptor and 5-HT1A/1B receptor antagonistFormula:C19H28N2O4Purity:98%Color and Shape:SolidMolecular weight:348.44S 14063
CAS:S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.Formula:C22H29Cl2N3O2SColor and Shape:SolidMolecular weight:470.45SEP-363856
CAS:SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.Formula:C9H13NOSPurity:98%Color and Shape:SolidMolecular weight:183.27(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:5-HT1A serotonin receptor agonistFormula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Formula:C18H22BrNSPurity:99.65%Color and Shape:SolidMolecular weight:364.34ATC0065 HCl
CAS:ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.Formula:C25H31BrCl2F3N5OColor and Shape:SolidMolecular weight:625.35SB 272183
CAS:SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.Formula:C29H28ClN5OPurity:98%Color and Shape:SolidMolecular weight:498.02ATC0065
CAS:ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.Formula:C25H29BrF3N5OColor and Shape:SolidMolecular weight:552.43LY 393558
CAS:Dual 5-HT1B/1D receptor antagonistFormula:C26H31FN4O4S2Purity:98%Color and Shape:SolidMolecular weight:546.68UCSF686
CAS:UCSF686, a UCSF678 analog, lacks 5-HT5A potency but keeps affinity for 5-HT1A, 5-HT2B, 5-HT7, and serves as a control.Formula:C14H19N3O2SColor and Shape:SolidMolecular weight:293.38Amitifadine hydrochloride
CAS:Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).Formula:C11H12Cl3NPurity:98%Color and Shape:SolidMolecular weight:264.58LY 302148
CAS:LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.Formula:C19H23FN4Purity:98%Color and Shape:SolidMolecular weight:326.41RG-12915
CAS:RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).Formula:C20H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:360.88LY314228
CAS:LY314228 is an antagonist of 5-HT2A receptor.Formula:C20H24N4O3Color and Shape:SolidMolecular weight:368.43CP 135807
CAS:CP 135807 is a 5-HT1D receptor agonist.Formula:C19H21N5O2Purity:98%Color and Shape:SolidMolecular weight:351.4SGS518 oxalate
CAS:SGS518 oxalate is a 5-HT6 antagonist.Formula:C23H24F2N2O7SPurity:98%Color and Shape:SolidMolecular weight:510.51Altanserin hydrochloride
CAS:Altanserin hydrochloride is a 5-HT2A receptor antagonist.Formula:C22H23ClFN3O2SPurity:98%Color and Shape:SolidMolecular weight:447.95GW-876167
CAS:GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.Formula:C16H21N5O2Purity:98%Color and Shape:SolidMolecular weight:315.37Penbutolol
CAS:Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.Formula:C18H29NO2Purity:98%Color and Shape:SolidMolecular weight:291.43SDZ 205-557 hydrochloride
CAS:5-HT3/5-HT4 receptor antagonistFormula:C14H22Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:337.245-HT6/5-HT2A receptor ligand-2
CAS:Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.Formula:C20H18FN3O2Color and Shape:SolidMolecular weight:351.37CGS 12066B dimaleate
CAS:5-HT1B full agonistFormula:C25H25F3N4O8Purity:98%Color and Shape:SolidMolecular weight:566.485-Nonyloxytryptamine oxalate
CAS:5-HT1B agonistFormula:C21H32N2O5Purity:98%Color and Shape:SolidMolecular weight:392.49(Rac)-SEP-363856
CAS:(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a uniqueFormula:C9H13NOSPurity:98%Color and Shape:SolidMolecular weight:183.27Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Formula:C15H17Cl2NO2Purity:99.77%Color and Shape:SolidMolecular weight:314.21Deramciclane
CAS:Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Formula:C20H31NOColor and Shape:SolidMolecular weight:301.47Captodiame
CAS:Captodiame is an antihistamine agent.Formula:C21H29NS2Purity:98%Color and Shape:SolidMolecular weight:359.59CP 93129 dihydrochloride
CAS:5-HT1B agonist, potent and highly selectiveFormula:C12H14ClN3OPurity:98%Color and Shape:SolidMolecular weight:251.71S(-)-8-Hydroxy-DPAT hydrobromide
CAS:S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.Formula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29SB-221284
CAS:5-HT2C/2B receptor antagonistFormula:C16H14F3N3OSPurity:98%Color and Shape:SolidMolecular weight:353.36SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Formula:C19H27IN2O4Color and Shape:SolidMolecular weight:474.33Ampreloxetine
CAS:Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.Formula:C18H18F3NOPurity:98%Color and Shape:SolidMolecular weight:321.34SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purity:98%Color and Shape:SolidMolecular weight:403.86Alaproclate
CAS:Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.Formula:C13H18ClNO2Purity:98.29% - 98.64%Color and Shape:SolidMolecular weight:255.742-Methyl-5-HT maleate
CAS:2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.Formula:C15H18N2O5Purity:98%Color and Shape:SolidMolecular weight:306.31TC-2153
CAS:TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.Formula:C7H5ClF3NS5Color and Shape:SolidMolecular weight:355.89FR260010
CAS:FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.Formula:C22H19N5Color and Shape:SolidMolecular weight:353.42Opiranserin
CAS:Opiranserin is a development as an injectable agent for the treatment of postoperative pain.Formula:C21H34N2O5Purity:98%Color and Shape:SolidMolecular weight:394.51Palonosetron
CAS:Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).Formula:C19H24N2OPurity:98%Color and Shape:SolidMolecular weight:296.41Alniditan dihydrochloride
CAS:Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.Formula:C17H28Cl2N4OColor and Shape:SolidMolecular weight:375.34Iferanserin
CAS:Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.Formula:C23H28N2OColor and Shape:SolidMolecular weight:348.48LY 125180
CAS:LY 125180 is a serotonin antagonist.Formula:C18H24ClNOPurity:98%Color and Shape:SolidMolecular weight:305.84WAY 161503 hydrochloride
CAS:WAY 161503 hydrochloride is a 5-HT2C receptor agonist.Formula:C11H12Cl3N3OPurity:98%Color and Shape:SolidMolecular weight:308.59Zicronapine
CAS:Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.Formula:C22H27ClN2Color and Shape:SolidMolecular weight:354.92Pancopride
CAS:Pancopride（LAS 30451） is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-inducedFormula:C18H24ClN3O2Purity:93.64%Color and Shape:SolidMolecular weight:349.86Tacitin
CAS:Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.Formula:C18H20ClNPurity:98%Color and Shape:SolidMolecular weight:285.81PF-4479745
CAS:PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.Formula:C17H22N4Purity:98%Color and Shape:SolidMolecular weight:282.38Masupirdine mesylate
CAS:Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's diseaseFormula:C23H32BrN3O9S3Purity:99.57%Color and Shape:SolidMolecular weight:670.61Piclozotan
CAS:Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)Formula:C23H24ClN3O2Purity:98.59%Color and Shape:SolidMolecular weight:409.91Ipsapirone
CAS:Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
Formula:C19H23N5O3SPurity:99.51%Color and Shape:SolidMolecular weight:401.48SUN-C5174
CAS:"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."Formula:C22H29FN4O2Purity:98%Color and Shape:SolidMolecular weight:400.49SB357134
CAS:SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.Formula:C17H18Br2FN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.21Levemopamil HCl
CAS:Levemopamil HCl is used as a calcium channel blocker.Formula:C23H31ClN2Purity:98%Color and Shape:SolidMolecular weight:370.96DAT 582
CAS:DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agentFormula:C22H28ClN5OPurity:98%Color and Shape:SolidMolecular weight:413.95QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Formula:C23H28N2O2Purity:>99.99%Color and Shape:SolidMolecular weight:364.48SB 206553 hydrochloride
CAS:SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disordersFormula:C17H17ClN4OPurity:99.56%Color and Shape:SolidMolecular weight:328.8(4E)-SUN9221
CAS:(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormula:C25H31FN4O3Purity:97.79%Color and Shape:SolidMolecular weight:454.54ST1936
CAS:ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Formula:C13H17ClN2Purity:98%Color and Shape:SolidMolecular weight:236.74Ref: TM-T23396
1mg44.00€5mg111.00€10mg178.00€25mg316.00€50mg470.00€100mg682.00€200mg954.00€1mL*10mM (DMSO)123.00€UCSF678
CAS:UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.Formula:C15H18N2O2SColor and Shape:SolidMolecular weight:290.38CP-809101
CAS:CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H17ClN4OPurity:98%Color and Shape:SolidMolecular weight:304.775-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurity:99.75%Color and Shape:SolidMolecular weight:480.62Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Formula:C19H21NPurity:99.15% - 99.66%Color and Shape:SolidMolecular weight:263.38E-3620
CAS:E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formula:C20H27Cl2N3O2Purity:98.88% - 98.88%Color and Shape:SolidMolecular weight:412.35Ro 04-6790
CAS:Ro 04-6790 is a 5-HT6 receptor antagonist.Formula:C12H16N6O2SPurity:98%Color and Shape:SolidMolecular weight:308.36T 82
CAS:T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.Formula:C56H62N6O8Purity:98%Color and Shape:SolidMolecular weight:947.146SKF-83566 hydrobromide
CAS:D1-like dopamine receptor antagonistFormula:C17H19BrClNOPurity:98%Color and Shape:SolidMolecular weight:368.7GR 55562 dihydrochloride
CAS:5-HT1B (5-HT1Dβ) silent antagonistFormula:C23H27Cl2N3O2Purity:99.45%Color and Shape:SolidMolecular weight:448.39
