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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 940 products of "5-HT Receptor"

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  • Sumatriptan

    CAS:
    <p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>
    Formula:C14H21N3O2S
    Purity:99.93%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:295.4
  • Paliperidone Palmitate

    CAS:
    <p>Paliperidone: atypical antipsychotic, dopamine &amp; serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>
    Formula:C39H57FN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:664.89
  • Spiroxatrine

    CAS:
    <p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>
    Formula:C22H25N3O3
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:379.45
  • Clozapine-d8

    CAS:
    <p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>
    Formula:C18H19ClN4
    Color and Shape:Solid
    Molecular weight:334.87
  • Dehydroaripiprazole

    CAS:
    <p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>
    Formula:C23H25Cl2N3O2
    Purity:98.7%
    Color and Shape:Solid
    Molecular weight:446.37
  • Asenapine hydrochloride

    CAS:
    <p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>
    Formula:C17H17Cl2NO
    Color and Shape:Solid
    Molecular weight:322.23
  • Alosetron D3 Hydrochloride

    CAS:
    <p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>
    Formula:C17H19ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.83
  • Nefazodone

    CAS:
    <p>Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.</p>
    Formula:C25H32ClN5O2
    Purity:99.85%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:470.01
  • Cariprazine D6

    CAS:
    <p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>
    Formula:C21H26D6Cl2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.45
  • Ziprasidone amino acid

    CAS:
    <p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>
    Formula:C21H23ClN4O2S
    Color and Shape:Solid
    Molecular weight:430.95
  • Levomepromazine

    CAS:
    <p>Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.</p>
    Formula:C19H24N2OS
    Purity:99.15%
    Color and Shape:Solid
    Molecular weight:328.47
  • Vilazodone-d8

    CAS:
    <p>Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.</p>
    Formula:C26H27N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.57
  • 3-Hydroxy agomelatine D3

    CAS:
    <p>3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).</p>
    Formula:C15H17NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:262.32
  • 5-HT2B antagonist-1

    CAS:
    <p>Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.</p>
    Formula:C11H14BrN5
    Purity:99.965%
    Color and Shape:Solid
    Molecular weight:296.17
  • Asenapine

    CAS:
    <p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>
    Formula:C17H16ClNO
    Purity:99.64%
    Color and Shape:Coa
    Molecular weight:285.77
  • 5-HT3 antagonist 5

    CAS:
    <p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>
    Formula:C16H13N3O2
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:279.29
  • 4,4-Diphenylbutylamine hydrochloride

    CAS:
    <p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>
    Formula:C16H20ClN
    Color and Shape:Solid
    Molecular weight:261.79
  • WAY-100635

    CAS:
    <p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>
    Formula:C25H34N4O2
    Purity:98.972%
    Color and Shape:Solid
    Molecular weight:422.56
  • LY310762

    CAS:
    <p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>
    Formula:C24H27FN2O2·HCl
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:430.94
  • Melperone

    CAS:
    <p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>
    Formula:C16H22FNO
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:263.35