5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 1025 products of "5-HT Receptor"
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SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purity:97.82% - 98%Color and Shape:SolidMolecular weight:380.87Ref: TM-T3183
1mg79.00€5mg152.00€10mg245.00€25mg398.00€50mg532.00€100mg735.00€200mg973.00€1mL*10mM (DMSO)166.00€Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.57Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Formula:C20H33NO7Purity:99.26%Color and Shape:White Crystalline PowdeMolecular weight:399.48SB399885
CAS:SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35Ref: TM-T19669
1mg67.00€5mg123.00€10mg177.00€25mg291.00€50mg393.00€100mg553.00€200mg743.00€1mL*10mM (DMSO)150.00€Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purity:99.75%Color and Shape:SolidMolecular weight:299.80Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg38.00€2mg50.00€5mg84.00€10mg118.00€25mg220.00€50mg403.00€100mg582.00€500mg1,198.00€1mL*10mM (DMSO)120.00€Eptapirone
CAS:Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formula:C16H23N7O2Purity:99.39% - 99.65%Color and Shape:SolidMolecular weight:345.4Harmine
CAS:Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.Formula:C13H12N2OPurity:98.29% - 99.92%Color and Shape:Off-White SolidMolecular weight:212.25Ramosetron hydrochloride
CAS:Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formula:C17H18ClN3OPurity:99.95%Color and Shape:SolidMolecular weight:315.8Alprenolol benzoate
CAS:Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formula:C22H29NO4Color and Shape:SolidMolecular weight:371.48Trazodone
CAS:Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formula:C19H22ClN5OPurity:99.79% - 99.92%Color and Shape:White To Off-White Crystalline PowderMolecular weight:371.861-(1-Naphthyl) piperazine hydrochloride
CAS:1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multipleFormula:C14H17ClN2Purity:98.27%Color and Shape:SolidMolecular weight:248.75A-582941 dihydrochloride
CAS:A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partialFormula:C17H22Cl2N4Purity:99.55%Color and Shape:SolidMolecular weight:353.29Ref: TM-T22016
1mg42.00€5mg88.00€10mg120.00€25mg235.00€50mg354.00€100mg533.00€200mg743.00€1mL*10mM (DMSO)87.00€Sertindole
CAS:Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).Formula:C24H26ClFN4OPurity:99.87% - 99.92%Color and Shape:Off-White To Pale Yellow SolidMolecular weight:440.94Flibanserin hydrochloride
CAS:Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.Formula:C20H22ClF3N4OColor and Shape:SolidMolecular weight:426.87Rizatriptan benzoate
CAS:Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormula:C22H25N5O2Purity:99% - 99.79%Color and Shape:White To Off-White Crystalline PowderMolecular weight:391.47Ref: TM-T1512
10mg44.00€25mg74.00€50mg119.00€100mg173.00€200mg259.00€500mg437.00€1mL*10mM (DMSO)48.00€PU02
CAS:PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Formula:C16H12N4SPurity:99.35%Color and Shape:SolidMolecular weight:292.36Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Formula:C19H26ClNOSPurity:99.53% - 99.56%Color and Shape:Almost White To White Crystalline PowderMolecular weight:351.93LY334370
CAS:LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormula:C21H22FN3OPurity:99.32%Color and Shape:SolidMolecular weight:351.42Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formula:C10H13ClN2SColor and Shape:SolidMolecular weight:228.74Almotriptan Malate
CAS:Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formula:C17H25N3O2S·C4H6O5Purity:99.95%Color and Shape:Pale Yellow SolidMolecular weight:469.55Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formula:C22H23FN2O5Purity:97.39% - 99.73%Color and Shape:White SolidMolecular weight:414.43Ref: TM-T6493
1g268.00€10mg37.00€25mg52.00€50mg63.00€100mg86.00€200mg118.00€500mg187.00€1mL*10mM (DMSO)42.00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32Serotonin hydrochloride
CAS:Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (Formula:C10H13ClN2OPurity:98.05% - 99.93%Color and Shape:White To Cream PowderMolecular weight:212.676Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formula:C19H25NOSPurity:98.08% - 99.59%Color and Shape:SolidMolecular weight:315.47Ref: TM-T6647
5mg50.00€10mg73.00€25mg138.00€50mg241.00€100mg358.00€200mg523.00€500mg822.00€1mL*10mM (DMSO)52.00€5-HT1A modulator 2 hydrochloride
CAS:5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.Formula:C11H16ClNOPurity:98.5%Color and Shape:SolidMolecular weight:213.7Metadoxine
CAS:Metadoxine (Metadoxil) is a neurotransmitter stimulant.Formula:C8H11NO3·C5H7NO3Purity:99.19%Color and Shape:Off-White PowderMolecular weight:298.29Azaphen
CAS:Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formula:C16H21Cl2N5OPurity:97.62%Color and Shape:SolidMolecular weight:370.28PRX-07034 hydrochloride
CAS:PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.Formula:C21H29Cl2N3O4SPurity:98.5%Color and Shape:SolidMolecular weight:490.44Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Formula:C20H30N2O3S2Purity:99.70%Color and Shape:White To Off-White SolidMolecular weight:410.59Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFormula:C21H32Cl2N4OPurity:99.68% - 99.87%Color and Shape:SolidMolecular weight:427.41Ref: TM-T4577
1mg49.00€5mg92.00€10mg145.00€25mg281.00€50mg394.00€100mg550.00€200mg780.00€1mL*10mM (DMSO)103.00€7-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Formula:C10H6F3NO2Purity:97.31% - 97.84%Color and Shape:Yellow PowderMolecular weight:229.16Sumatriptan hydrochloride
CAS:Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Formula:C14H22ClN3O2SColor and Shape:SolidMolecular weight:331.86Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formula:C8H11N5Purity:99.54%Color and Shape:SolidMolecular weight:177.21Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formula:C23H24FN3O2Purity:99.2%Color and Shape:SolidMolecular weight:393.45F-15599
CAS:F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).Formula:C19H21ClF2N4OPurity:98.72%Color and Shape:SolidMolecular weight:394.85Ref: TM-T7281
1mg49.00€5mg92.00€10mg152.00€25mg295.00€50mg477.00€100mg715.00€200mg982.00€1mL*10mM (DMSO)104.00€Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formula:C17H21ClN4SColor and Shape:SolidMolecular weight:348.89Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formula:C28H36N4O2SPurity:99.78% - 99.91%Color and Shape:SolidMolecular weight:492.68WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formula:C25H34N4O2·C4H4O4Purity:98.44% - 99.46%Color and Shape:SolidMolecular weight:538.64Ref: TM-T2631
2mg43.00€5mg63.00€10mg89.00€25mg170.00€50mg315.00€100mg470.00€200mg680.00€500mg1,054.00€1mL*10mM (DMSO)74.00€Eltoprazine
CAS:Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.Formula:C12H16N2O2Color and Shape:SolidMolecular weight:220.27Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Formula:C16H23Cl2N3O2Color and Shape:SolidMolecular weight:360.28Loxapine hydrochloride
CAS:Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.Formula:C18H19Cl2N3OColor and Shape:SolidMolecular weight:364.27Adoprazine hydrochloride
CAS:Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formula:C24H25ClFN3O2Color and Shape:SolidMolecular weight:441.93ARC-239
CAS:ARC-239 is an agonist of α2-adrenergic receptor.Formula:C24H29N3O3Color and Shape:SolidMolecular weight:407.51(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formula:C12H14O5Purity:99.83%Color and Shape:SolidMolecular weight:238.24VUF 10166
CAS:VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Formula:C13H15ClN4Purity:99.66%Color and Shape:SolidMolecular weight:262.74(S)-Amisulpride
CAS:(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.Formula:C17H27N3O4SPurity:98.38%Color and Shape:SolidMolecular weight:369.48Ref: TM-T26375
1mg34.00€5mg84.00€10mg123.00€25mg225.00€50mg358.00€100mg485.00€200mg622.00€1mL*10mM (DMSO)94.00€Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formula:C22H24ClN3O3SColor and Shape:SolidMolecular weight:445.96
