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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 985 products of "5-HT Receptor"

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  • Clozapine-d8

    CAS:
    Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.
    Formula:C18H19ClN4
    Color and Shape:Solid
    Molecular weight:334.87
  • WAY-100635

    CAS:
    <p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>
    Formula:C25H34N4O2
    Purity:98.972%
    Color and Shape:Solid
    Molecular weight:422.56
  • Alosetron D3 Hydrochloride

    CAS:
    <p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>
    Formula:C17H19ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.83
  • Nefazodone

    CAS:
    Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.
    Formula:C25H32ClN5O2
    Purity:99.85%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:470.01
  • Cariprazine D6

    CAS:
    <p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>
    Formula:C21H26D6Cl2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.45
  • Dehydroaripiprazole

    CAS:
    <p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>
    Formula:C23H25Cl2N3O2
    Purity:98.7%
    Color and Shape:Solid
    Molecular weight:446.37
  • Vilazodone-d8

    CAS:
    Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.
    Formula:C26H27N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.57
  • Asenapine

    CAS:
    <p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>
    Formula:C17H16ClNO
    Purity:99.64%
    Color and Shape:Coa
    Molecular weight:285.77
  • Levomepromazine

    CAS:
    Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.
    Formula:C19H24N2OS
    Purity:99.15%
    Color and Shape:Solid
    Molecular weight:328.47
  • 3-Hydroxy agomelatine D3

    CAS:
    <p>3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).</p>
    Formula:C15H17NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:262.32
  • 5-HT2B antagonist-1

    CAS:
    Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.
    Formula:C11H14BrN5
    Purity:99.965%
    Color and Shape:Solid
    Molecular weight:296.17
  • 5-HT3 antagonist 5

    CAS:
    <p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>
    Formula:C16H13N3O2
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:279.29
  • Thioridazine

    CAS:
    Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.
    Formula:C21H26N2S2
    Color and Shape:Solid
    Molecular weight:370.57
  • Quetiapine-d8 Fumarate

    CAS:
    Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
    Formula:C25H21D8N3O6S
    Color and Shape:Solid
    Molecular weight:507.63
  • LY310762

    CAS:
    LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.
    Formula:C24H27FN2O2·HCl
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:430.94
  • Methiothepin mesylate

    CAS:
    <p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>
    Formula:C21H28N2O3S3
    Purity:98% - 99.92%
    Color and Shape:Solid
    Molecular weight:452.65
  • Quipazine

    CAS:
    <p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>
    Formula:C13H15N3
    Color and Shape:Solid
    Molecular weight:213.28
  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Formula:C21H25NO4
    Purity:99.8% - 99.91%
    Color and Shape:Off-White Solid
    Molecular weight:355.43
  • Cyclopiazonic acid

    CAS:
    <p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>
    Formula:C20H20N2O3
    Purity:99.27% - 99.80%
    Color and Shape:Solid
    Molecular weight:336.38
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Formula:C17H25N3O2S
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:335.47