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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 942 products of "5-HT Receptor"

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  • S1RA hydrochloride

    CAS:
    <p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki &gt;</p>
    Formula:C20H24ClN3O2
    Purity:98% - 99.84%
    Color and Shape:Solid
    Molecular weight:373.87
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Formula:C19H21ClF2N4O
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:394.85
  • Eltoprazine

    CAS:
    <p>Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.</p>
    Formula:C12H16N2O2
    Color and Shape:Solid
    Molecular weight:220.27
  • Sarpogrelate

    CAS:
    <p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>
    Formula:C24H31NO6
    Color and Shape:Solid
    Molecular weight:429.51
  • SKF-83566

    CAS:
    <p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>
    Formula:C17H18BrNO
    Purity:95.00% - 99.82%
    Color and Shape:Solid
    Molecular weight:332.23
  • BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Formula:C22H33Cl2N3O3
    Purity:97.32% - 99.08%
    Color and Shape:Solid
    Molecular weight:458.42
  • Cinanserin

    CAS:
    <p>Cinanserin is a serotonin 5-HT2 antagonist.</p>
    Formula:C20H24N2OS
    Color and Shape:Solid
    Molecular weight:340.48
  • Methiothepin mesylate

    CAS:
    <p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>
    Formula:C21H28N2O3S3
    Purity:98% - 99.92%
    Color and Shape:Solid
    Molecular weight:452.65
  • ML 10302

    CAS:
    <p>ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.</p>
    Formula:C15H21ClN2O3
    Color and Shape:Solid
    Molecular weight:312.79
  • SAX-187

    CAS:
    <p>SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.</p>
    Formula:C15H13ClN4O2S2
    Purity:97.82% - 98%
    Color and Shape:Solid
    Molecular weight:380.87
  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Formula:C21H25NO4
    Purity:99.8% - 99.91%
    Color and Shape:Off-White Solid
    Molecular weight:355.43
  • Isocorynoxeine

    CAS:
    Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.
    Formula:C22H26N2O4
    Purity:98% - 99.9%
    Color and Shape:Solid
    Molecular weight:382.45
  • Nuciferine

    CAS:
    <p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>
    Formula:C19H21NO2
    Purity:98.76% - 99.79%
    Color and Shape:Solid
    Molecular weight:295.38
  • Naratriptan

    CAS:
    <p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>
    Formula:C17H25N3O2S
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:335.47
  • Zotepine

    CAS:
    <p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>
    Formula:C18H18ClNOS
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:331.86
  • Metoclopramide

    CAS:
    <p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>
    Formula:C14H22ClN3O2
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:299.80
  • Harmine

    CAS:
    <p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>
    Formula:C13H12N2O
    Purity:98.29% - 99.92%
    Color and Shape:Off-White Solid
    Molecular weight:212.25
  • Ramosetron hydrochloride

    CAS:
    <p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>
    Formula:C17H18ClN3O
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:315.8
  • Trazodone

    CAS:
    <p>Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.</p>
    Formula:C19H22ClN5O
    Purity:99.79% - 99.92%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:371.86
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Formula:C14H17ClN2
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:248.75