5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
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Methiothepin maleate
CAS:19728-88-2
Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.
Formula:
C24H28N2O4S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
472.62
Ref: TM-T4375
| 10mg | 86.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 437.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
AVN-322
CAS:1194574-68-9
AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive …
Formula:
C17H20ClN5O2S
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
393.89
Ref: TM-T26691
| 1mg | 276.00 € | ||
| 5mg | 679.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SB-215505
CAS:162100-15-4
SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, …
Formula:
C19H16ClN3O
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
337.8
Ref: TM-T28680
| 1mg | 209.00 € | ||
| 5mg | 521.00 € | ||
| 10mg | 726.00 € | ||
| 25mg | 1,081.00 € | ||
| 50mg | 1,493.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
GR 46611
CAS:185259-85-2
GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in …
Formula:
C23H27N3O2
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
377.48
Ref: TM-T22808
| 1mg | 52.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 136.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 620.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
5-HT3 antagonist 2
CAS:128199-93-9
5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.
Formula:
C18H21N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
295.38
Ref: TM-T12988
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
5-HT7 agonist 1
CAS:334974-31-1
5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).
Formula:
C19H20ClN3
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
325.84
Ref: TM-T10170
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,052.00 € | ||
| 1mL*10mM (DMSO) | 253.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SB228357
CAS:181629-93-6
SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, …
Formula:
C22H17F4N3O2
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
431.38
Ref: TM-T16856
| 1mg | 74.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 277.00 € | ||
| 25mg | 458.00 € | ||
| 50mg | 610.00 € | ||
| 100mg | 833.00 € | ||
| 1mL*10mM (DMSO) | 165.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
LY-2624803
CAS:879409-35-5
LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used …
Formula:
C22H25N3O3
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T24421
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 496.00 € | ||
| 25mg | 803.00 € | ||
| 50mg | 1,099.00 € | ||
| 100mg | 1,486.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
5HT6-ligand-1
CAS:1038988-11-2
5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).
Formula:
C20H22BrN3O2S
Purity:
98.48% - 98.95%
Color and Shape:
Solid
Molecular weight:
448.38
Ref: TM-T10053
| 1mg | 184.00 € | ||
| 5mg | 445.00 € | ||
| 10mg | 609.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,238.00 € | ||
| 100mg | 1,629.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
RS 67333 hydrochloride
CAS:168986-60-5
RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's …
Formula:
C19H30Cl2N2O2
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
389.36
Ref: TM-T23265
| 5mg | 50.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 252.00 € | ||
| 100mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
ST1936
CAS:1210-81-7
ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and …
Formula:
C13H17ClN2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
236.74
Ref: TM-T23396
| 1mg | 46.00 € | ||
| 5mg | 115.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 489.00 € | ||
| 100mg | 707.00 € | ||
| 200mg | 990.00 € | ||
| 1mL*10mM (DMSO) | 128.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
5-HT2 antagonist 1
CAS:191592-09-3
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.
Formula:
C22H29FN4O2
Purity:
99.25%
Color and Shape:
Solid
Molecular weight:
400.49
Ref: TM-T12597
| 1mg | 663.00 € | ||
| 5mg | 1,328.00 € | ||
| 10mg | 1,792.00 € | ||
| 25mg | 2,665.00 € | ||
| 50mg | 3,593.00 € | ||
| 100mg | 4,855.00 € | ||
| 1mL*10mM (DMSO) | 1,595.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Ampreloxetine
CAS:1227056-84-9
Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.
Formula:
C18H18F3NO
Purity:
98%
Color and Shape:
Solid
Molecular weight:
321.34
Ref: TM-T26622
| 25mg | 1,410.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
RG-12915
CAS:136174-04-4
RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).
Formula:
C20H25ClN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
360.88
Ref: TM-T12716
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Org-13011 fumarate
CAS:142494-13-1
Org-13011 fumarate1 is an agonist of the 5-HT1A receptor and can be used to study …
Formula:
C22H29F3N4O5
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
486.48
Ref: TM-T28258
| 1mg | 277.00 € | ||
| 5mg | 683.00 € | ||
| 10mg | 933.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 1,832.00 € | ||
| 100mg | 2,342.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Alniditan
CAS:152317-89-0
Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 …
Formula:
C17H26N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
302.41
Ref: TM-T14190
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Enciprazine
CAS:68576-86-3
Enciprazine (D-3112) shows anxiolytic activity, is used to treat anxiety disorders, and can be used …
Formula:
C23H32N2O6
Purity:
98.66%
Color and Shape:
Solid
Molecular weight:
432.51
Ref: TM-T27262
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,442.00 € | ||
| 50mg | 1,878.00 € | ||
| 100mg | 2,371.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
AP521
CAS:151227-08-6
AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).
Formula:
C20H19ClN2O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
402.89
Ref: TM-T10344
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
2-Methyl-5-HT maleate
CAS:78263-91-9
2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.
Formula:
C15H18N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
306.31
Ref: TM-T10075L
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
EMD 56551
CAS:133109-86-1
EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the …
Formula:
C24H31N3O2
Purity:
95.07% - 99.19%
Color and Shape:
Liquid
Molecular weight:
393.522
Ref: TM-T61816
| 1mg | 276.00 € | ||
| 5mg | 679.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,430.00 € | ||
| 50mg | 1,862.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
