5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
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Itasetron
CAS:123258-84-4
Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer …
Formula:
C16H20N4O2
Purity:
100% - 99.63%
Color and Shape:
Solid
Molecular weight:
300.36
Ref: TM-T24184
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,547.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
LP44 hydrochloride
CAS:824958-12-5
LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice …
Formula:
C27H38ClN3OS
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
488.13
Ref: TM-T22931
| 1mg | 38.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
WAY208466 dihydrochloride
CAS:1207064-61-6
WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.
Formula:
C17H20Cl2FN3O2S
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
420.33
Ref: TM-T23527
| 1mg | 64.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Piclozotan
CAS:182415-09-4
Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral …
Formula:
C23H24ClN3O2
Purity:
99%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T28414
| 25mg | 1,410.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Lecozotan HCl
CAS:433282-68-9
Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) …
Formula:
C28H30ClN5O3
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
520.02
Ref: TM-T27806
| 1mg | 156.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 875.00 € | ||
| 50mg | 1,189.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,211.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
S 16924
CAS:734513-52-1
S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful …
Formula:
C22H24FNO4
Purity:
98.23% - 99.45%
Color and Shape:
Solid
Molecular weight:
385.43
Ref: TM-T28638
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
GR 113808
CAS:144625-51-4
GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates …
Formula:
C19H27N3O4S
Purity:
98.16%
Color and Shape:
Solid
Molecular weight:
393.5
Ref: TM-T15414
| 1mg | 38.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
PNU-142633
CAS:187665-65-2
PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.
Formula:
C24H30N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
422.52
Ref: TM-T16556
| 10mg | 771.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Lesopitron
CAS:132449-46-8
Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.
Formula:
C15H21ClN6
Purity:
98.60% - 98.92%
Color and Shape:
Solid
Molecular weight:
320.82
Ref: TM-T25672
| 1mg | 138.00 € | ||
| 5mg | 337.00 € | ||
| 10mg | 495.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,960.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Adatanserin
CAS:127266-56-2
Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C …
Formula:
C21H31N5O
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
369.5
Ref: TM-T23631
| 1mg | 279.00 € | ||
| 5mg | 686.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Clovoxamine
CAS:54739-19-4
Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant …
Formula:
C14H21ClN2O2
Purity:
98.88% - 99.16%
Color and Shape:
Solid
Molecular weight:
284.78
Ref: TM-T27047
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
TIK-301
CAS:118702-11-7
TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 …
Formula:
C14H17ClN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
280.75
Ref: TM-T17095
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
RS 56812 hydrochloride
CAS:143339-12-2
5-HT3 partial agonist
Formula:
C18H22ClN3O2
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
347.84
Ref: TM-T23264
| 1mg | 64.00 € | ||
| 2mg | 90.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 431.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Felcisetrag
CAS:916075-84-8
Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi …
Formula:
C25H37N5O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
455.59
Ref: TM-T28934
| 1mg | 151.00 € | ||
| 5mg | 371.00 € | ||
| 10mg | 547.00 € | ||
| 25mg | 878.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,226.00 € | ||
| 1mL*10mM (DMSO) | 411.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CP 96021
CAS:139401-43-7
"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating …
Formula:
C29H21FN4OS
Purity:
97.81% - 99.11%
Color and Shape:
Soild
Molecular weight:
492.57
Ref: TM-T10872L
| 1mg | 181.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 614.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,756.00 € | ||
| 500mg | 3,531.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
PRX933 hydrochloride
CAS:639029-42-8
PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in …
Formula:
C16H22ClN5O2
Purity:
97.99% - 99.72%
Color and Shape:
Solid
Molecular weight:
351.84
Ref: TM-T12565
| 1mg | 349.00 € | ||
| 5mg | 556.00 € | ||
| 10mg | 886.00 € | ||
| 25mg | 1,309.00 € | ||
| 50mg | 1,773.00 € | ||
| 100mg | 2,377.00 € | ||
| 1mL*10mM (DMSO) | 649.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Deramciclane
CAS:120444-71-5
Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.
Formula:
C20H31NO
Color and Shape:
Solid
Molecular weight:
301.47
Ref: TM-T10996
| 25mg | 1,002.00 € | ||
| 50mg | 1,320.00 € | ||
| 100mg | 1,863.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Iferanserin
CAS:58754-46-4
Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity …
Formula:
C23H28N2O
Color and Shape:
Solid
Molecular weight:
348.48
Ref: TM-T15552
| 25mg | 1,299.00 € | ||
| 50mg | 1,704.00 € | ||
| 100mg | 2,340.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Pancopride
CAS:121650-80-4
Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen …
Formula:
C18H24ClN3O2
Purity:
93.64%
Color and Shape:
Solid
Molecular weight:
349.86
Ref: TM-T16433
| 1mg | 650.00 € | ||
| 5mg | 1,682.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
PNU-282987 free base
CAS:711085-63-1
PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for …
Formula:
C14H17ClN2O
Purity:
99.64%
Color and Shape:
Liquid
Molecular weight:
264.75
Ref: TM-T60437
| 1mg | 55.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,020.00 € | ||
| 500mg | 2,039.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
