CaMK
Calcium/Calmodulin-Dependent Protein Kinase (CaMK) inhibitors are compounds that block the activity of CaMK, a kinase involved in regulating various cellular processes, including synaptic plasticity, memory formation, and gene expression in the nervous system. CaMK plays a critical role in translating calcium signals into cellular responses, and its dysregulation is associated with neurological disorders. Inhibitors of CaMK are valuable tools for studying synaptic signaling, learning, and memory. At CymitQuimica, we offer CaMK inhibitors to support your research in synaptic plasticity, cognitive function, and neuropharmacology.
Found 69 products for "CaMK".
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Calmodulin Binding Peptide 1
CAS:Calmodulin Binding Peptide 1, a high-affinity MLCK-derived inhibitor, blocks IP3-induced Ca2+ release.Formula:C231H373N69O70S2Purity:98%Color and Shape:SolidMolecular weight:5301.1Cloxacepride
CAS:cloxacepride is a CaM antagonist that is used to treat asthma disease.Formula:C22H27Cl2N3O4Purity:99.76%Color and Shape:SolidMolecular weight:468.37CaMKIIα-PHOTAC
CaMKIIα-PHOTAC is a photochemically targeted chimera (PHOTAC) that specifically targets Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα).Formula:C54H58Cl2N10O11Purity:98%Color and Shape:SolidMolecular weight:1094TAT-CN21 (scrambled)
TAT-CN21(scrambled) is a control peptide lacking specific targeting activity and serves as a negative control for TatCN21. TatCN21 is an effective and selective inhibitory peptide for calcium/calmodulin-dependent protein kinase II (CaMKII).Color and Shape:Odour SolidCAMKIV Protein, Human, Recombinant (GST)
CAMKIV Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag.Color and Shape:Lyophilized PowderMolecular weight:79 kDa (predicted); 100 kDa (reducing conditions)A-484954
CAS:A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.Formula:C13H15N5O3Purity:97.47% - 99.86%Color and Shape:SolidMolecular weight:289.29Ref: TM-TQ0137
1mg40.00€2mg52.00€5mg84.00€1mL*10mM (DMSO)98.00€10mg137.00€25mg289.00€50mg515.00€100mg733.00€KN-92 hydrochloride
CAS:KN-92 hydrochloride is an inactive derivative of KN-93.Formula:C24H26Cl2N2O3SPurity:99.68%Color and Shape:White SolidMolecular weight:493.45KN-93
CAS:KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase.Formula:C26H29ClN2O4SPurity:99.56% - 99.95%Color and Shape:White SolidMolecular weight:501.04Ref: TM-T2697
1mg54.00€2mg74.00€5mg107.00€1mL*10mM (DMSO)120.00€10mg146.00€25mg289.00€50mg358.00€100mg523.00€KN-62
CAS:KN-62 is a potent and specific Ca2+/calmodulin-dependent protein kinase II (CaMKII) inhibitor with Ki of 0.9 μM.Formula:C38H35N5O6S2Purity:99.80% - >99.99%Color and Shape:SolidMolecular weight:721.84Ref: TM-T2694
1mg34.00€2mg49.00€5mg71.00€10mg105.00€1mL*10mM (DMSO)105.00€25mg207.00€50mg404.00€100mg592.00€Trifluoperazine
CAS:Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.Formula:C21H24F3N3SPurity:98.3% - 99.46%Color and Shape:White To Yellowish Crystalline PowderMolecular weight:407.5NH125
CAS:NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.Formula:C27H45IN2Purity:98.60%Color and Shape:SolidMolecular weight:524.56Ref: TM-T6605
1mg38.00€2mg50.00€5mg84.00€1mL*10mM (DMSO)93.00€10mg113.00€25mg250.00€50mg430.00€100mg620.00€STO-609
CAS:STO-609 inhibits CaM-KKα/KKβ (Ki: 80/15 ng/mL), is specific, cell-permeable, and targets Ca2+/calmodulin-dependent protein kinase kinase.Formula:C19H10N2O3Purity:97.14% - 99.35%Color and Shape:SolidMolecular weight:314.29Ref: TM-T3546
1mg39.00€5mg84.00€1mL*10mM (DMSO)93.00€10mg120.00€25mg250.00€50mg400.00€100mg620.00€200mg873.00€Autocamtide 2 TFA(129198-88-5 free base)
Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.Formula:C67H119F3N22O22Purity:99.86%Color and Shape:SolidMolecular weight:1641.79CaMKII-IN-1
CAS:CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM).Formula:C29H30ClN5O2SPurity:99.69%Color and Shape:SolidMolecular weight:548.1Ref: TM-T14860
1mg50.00€2mg71.00€5mg113.00€1mL*10mM (DMSO)137.00€10mg166.00€25mg334.00€50mg520.00€100mg750.00€lavendustin C
CAS:lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.Formula:C14H13NO5Purity:98.06%Color and Shape:Yellow To Tan PowderMolecular weight:275.26Ref: TM-T4185
1mg42.00€2mg55.00€1mL*10mM (DMSO)90.00€5mg93.00€10mg152.00€25mg330.00€50mg492.00€100mg707.00€Autocamtide-2-related inhibitory peptide
CAS:Autocamtide-2-related inhibitory peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.Formula:C64H116N22O19Purity:>99.99%Color and Shape:SolidMolecular weight:1497.74CaMKP Inhibitor
CAS:CaMKP Inhibitor can inhibit CaMKP.Formula:C10H8NNaO7S2Purity:99.91% - 99.98%Color and Shape:SolidMolecular weight:341.28Ref: TM-T2159
1mg39.00€5mg82.00€1mL*10mM (DMSO)102.00€10mg120.00€25mg227.00€50mg334.00€100mg460.00€500mg1,035.00€Syntide 2 acetate(108334-68-5 free base)
Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM).Formula:C70H126N20O20Purity:99.87%Color and Shape:Purple LiquidMolecular weight:1567.85CALP2 acetate(261969-04-4 free base)
CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.Formula:C68H104N14O13SPurity:99.91%Color and Shape:SolidMolecular weight:1357.7KN-92
CAS:KN-92 is an inactive analog of the CaM kinase II inhibitor KN 93.Formula:C24H25ClN2O3SColor and Shape:SolidMolecular weight:456.98
