GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
Found 255 products of "GluR"
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(1S,3R)-ACPD
CAS:<p>(1S,3R)-ACPD is a group I and II mGlu receptor agonist.</p>Formula:C7H11NO4Purity:98%Color and Shape:SolidMolecular weight:173.17VU0404251
CAS:<p>VU0404251 is a positive allosteric modulator of mGlu5.</p>Formula:C19H23FN2O2Color and Shape:SolidMolecular weight:330.4Mavoglurant racemate
CAS:<p>Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant.</p>Formula:C19H23NO3Purity:98%Color and Shape:SolidMolecular weight:313.39ACPT-II
CAS:<p>metabotropic receptor antagonist</p>Formula:C8H11NO6Purity:98%Color and Shape:SolidMolecular weight:217.18DL-AP4 Sodium salt
CAS:<p>Broad spectrum EAA ligand</p>Formula:C4H10NNaO5PPurity:98%Color and Shape:SolidMolecular weight:206.09UPF-523
CAS:<p>group I metabotropic glutamate receptors (mGlu1a) antagonist</p>Formula:C11H11NO4Purity:98%Color and Shape:White SolidMolecular weight:221.21JNJ-46356479
CAS:<p>JNJ-46356479: Selective, oral mGlu2 receptor PAM, EC50=78 nM, Emax=256%.</p>Formula:C22H22F5N5Color and Shape:SolidMolecular weight:451.44ACPT-I
CAS:<p>Agonist for group III mGlu receptors</p>Formula:C8H11NO6Purity:98%Color and Shape:SolidMolecular weight:217.18VU0364289
CAS:<p>VU0364289 is a positive allosteric modulator of mGlu5.</p>Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.4(S)-4C3HPG
CAS:<p>group I mGlu1a/1a receptor antagonist and mGluR2 agonist</p>Formula:C9H9NO5Purity:98%Color and Shape:SolidMolecular weight:211.17LSN2814617
CAS:<p>LSN2814617: oral, brain-penetrant mGlu5 PAM, EC50 = 52 nM (human), 42 nM (rat). Promotes wakefulness, useful in schizophrenia study.</p>Formula:C18H20FN5OPurity:98%Color and Shape:SolidMolecular weight:341.38RO4988546
CAS:<p>RO4988546 is a potent negative allosteric modulator of mGlu₂/₃.</p>Formula:C21H10F6N4O3SPurity:98%Color and Shape:SolidMolecular weight:512.38mGluR2 modulator 1
CAS:<p>Potent mGluR2 modulator 1 crosses blood-brain barrier, EC50: 0.03 μM, useful for psychiatric research.</p>Formula:C21H20F3N3O3Color and Shape:SolidMolecular weight:419.4NPEC-caged-LY379268
CAS:<p>NPEC-caged-LY379268 is a type II mGluR agonist [1].</p>Formula:C16H16N2O9Color and Shape:SolidMolecular weight:380.31A 841720
CAS:<p>Potent, selective mGlu1 antagonist A-841720; IC50: 10 nM; 34x selectivity vs mGlu5; analgesic potential.</p>Formula:C17H21N5OSColor and Shape:SolidMolecular weight:343.45RO5488608
CAS:<p>RO5488608 is a new type of high-efficiency mGlu2/3 NAM.</p>Formula:C23H17F3N2O4SColor and Shape:SolidMolecular weight:474.45Talaglumetad hydrochloride
CAS:<p>Talaglumetad hydrochloride, a prodrug of Eglumegad, targets mGluR2/3 to treat psychiatric disorders.</p>Formula:C11H17ClN2O5Color and Shape:SolidMolecular weight:292.72mGluR2 modulator 2
CAS:<p>mGluR2 modulator 2: potent, selective, oral, EC50 = 0.13 μM, for antipsychotic research.</p>Formula:C20H22FN3Color and Shape:SolidMolecular weight:323.41VU0418506
CAS:<p>VU0418506 is a positive allosteric modulator (PAM) of the metabotropic glutamate receptor 4 (mGlu4).</p>Formula:C12H8ClFN4Purity:98%Color and Shape:SolidMolecular weight:262.67ACDPP hydrochloride
CAS:<p>mGlu5 receptor antagonist</p>Formula:C12H13ClN6OPurity:98%Color and Shape:SolidMolecular weight:292.72
