GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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JNJ-40411813
CAS:1127498-03-6
JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor …
Formula:
C20H25ClN2O
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
344.88
Ref: TM-TQ0094
| 1mg | 54.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 179.00 € | ||
| 25mg | 299.00 € | ||
| 50mg | 426.00 € | ||
| 100mg | 547.00 € | ||
| 200mg | 724.00 € | ||
| 1mL*10mM (DMSO) | 128.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ro0711401
CAS:714971-87-6
Ro0711401 is an agonist of mGlu1 receptor.
Formula:
C18H11F3N2O3
Purity:
97.57%
Color and Shape:
Solid
Molecular weight:
360.29
Ref: TM-T9021
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 148.00 € | ||
| 50mg | 228.00 € | ||
| 100mg | 379.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
YM90K
CAS:154164-30-4
YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.
Formula:
C11H8ClN5O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
309.66
Ref: TM-T8435
| 1mg | 86.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 414.00 € | ||
| 50mg | 582.00 € | ||
| 100mg | 787.00 € | ||
| 200mg | 1,044.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
3-MATIDA
CAS:518357-51-2
3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).
Formula:
C8H9NO4S
Purity:
98.41% - 99.05%
Color and Shape:
Solid
Molecular weight:
215.23
Ref: TM-T3486
| 1mg | 43.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 586.00 € | ||
| 500mg | 1,254.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
trans-ACPD
CAS:67684-64-4
trans-ACPD ((±)-trans-ACPD) is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD.
Formula:
C7H11NO4
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
173.17
Ref: TM-T3484
| 1mg | 48.00 € | ||
| 2mg | 62.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 493.00 € | ||
| 100mg | 713.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
LY-404187
CAS:211311-95-4
LY404187 is a positive allosteric modulator of AMPA receptors
Formula:
C19H22N2O2S
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
342.46
Ref: TM-T7706
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 330.00 € | ||
| 200mg | 459.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
MTEP hydrochloride
CAS:1186195-60-7
MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 …
Formula:
C11H9ClN2S
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
236.72
Ref: TM-T7515
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 367.00 € | ||
| 100mg | 551.00 € | ||
| 200mg | 763.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
1-BCP
CAS:34023-62-6
1-BCP (Piperonylic acid piperidide) is a centrally active drug that modulates AMPA receptor gated currents.
Formula:
C13H15NO3
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
233.26
Ref: TM-T7579
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 159.00 € | ||
| 100mg | 236.00 € | ||
| 200mg | 339.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(S)-3-Hydroxyphenylglycine
CAS:71301-82-1
(S)-3-Hydroxyphenylglycine is an agonist of group I metabotropic glutamate receptors (mGluRs).
Formula:
C8H9NO3
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
167.16
Ref: TM-T23291
| 1mg | 82.00 € | ||
| 2mg | 93.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 206.00 € | ||
| 25mg | 345.00 € | ||
| 50mg | 494.00 € | ||
| 100mg | 676.00 € | ||
| 200mg | 909.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
ML 254
CAS:1428630-86-7
ML254 competitively interacts with the MPEP allosteric binding site.
Formula:
C18H15FN2O2
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
310.32
Ref: TM-T8862
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 427.00 € | ||
| 50mg | 631.00 € | ||
| 100mg | 897.00 € | ||
| 1mL*10mM (DMSO) | 153.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Transtorine
CAS:13593-94-7
Transtorine (1,4-DIHYDRO-4-OXOQUINOLINE-2-CARBOXYLIC ACID) is a GluR and NMDA inhibitor.
Formula:
C10H7NO3
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
189.17
Ref: TM-T8626
| 50mg | 46.00 € | ||
| 100mg | 61.00 € | ||
| 200mg | 86.00 € | ||
| 500mg | 131.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
MPEP hydrochloride
CAS:219911-35-0
MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype …
Formula:
C14H12ClN
Purity:
100% - 99.75%
Color and Shape:
Solid
Molecular weight:
229.7
Ref: TM-T2497
| 10mg | 47.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 134.00 € | ||
| 100mg | 206.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
TCN238
CAS:125404-04-8
TCN238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 (mGluR4with …
Formula:
C12H11N3
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
197.24
Ref: TM-T7494
| 5mg | 36.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 106.00 € | ||
| 50mg | 176.00 € | ||
| 100mg | 305.00 € | ||
| 200mg | 439.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CNQX
CAS:115066-14-3
CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM …
Formula:
C9H4N4O4
Purity:
≥95%
Color and Shape:
Pale Yellow Solid
Molecular weight:
232.15
Ref: TM-T7178
| 5mg | 48.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 120.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 296.00 € | ||
| 200mg | 442.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
NPS2390
CAS:226878-01-9
NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 …
Formula:
C19H21N3O
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
307.39
Ref: TM-T8457
| 5mg | 41.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 296.00 € | ||
| 200mg | 408.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(RS)-MCPG
CAS:146669-29-6
(RS)-MCPG ((±)-MCPG) is a non-selective group I/II metabotropic glutamate receptor antagonist.
Formula:
C10H11NO4
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
209.2
Ref: TM-T3479
| 1mg | 35.00 € | ||
| 2mg | 47.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 331.00 € | ||
| 100mg | 494.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ro 67-7476
CAS:298690-60-5
Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors.
Formula:
C17H18FNO2S
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
319.39
Ref: TM-T3478
| 1mg | 36.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 252.00 € | ||
| 50mg | 455.00 € | ||
| 100mg | 664.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CTEP
CAS:871362-31-1
CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor …
Formula:
C19H13ClF3N3O
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
391.77
Ref: TM-T6457
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 336.00 € | ||
| 200mg | 478.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
SIB-1757
CAS:31993-01-8
SIB-1757 (6-methyl-2-[(E)-phenyldiazenyl]pyridin-3) is a selective antagonist of mGlu5 metabotropic glutamate receptor subtype (hmGlu5, IC50 : …
Formula:
C12H11N3O
Purity:
97.37%
Color and Shape:
Solid
Molecular weight:
213.24
Ref: TM-T8434
| 2mg | 39.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 361.00 € | ||
| 200mg | 506.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PHCCC
CAS:179068-02-1
PHCCC is a Group I mGluR antagonist and enhances mGluR4 function; also blocks mGluR2/8.
Formula:
C17H14N2O3
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
294.3
Ref: TM-T3464
| 2mg | 46.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 519.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
