GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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Fenobam
CAS:57653-26-6
Fenobam shows inverse agonist activity which blocks the mGlu5 receptor basal activity(IC50: 84 nM).
Formula:
C11H11ClN4O2
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
266.68
Ref: TM-T15275
| 1mg | 35.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 349.00 € | ||
| 200mg | 483.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Decoglurant
CAS:911115-16-7
Decoglurant (RO4995819) is a negative allosteric modulator of mGluR2 and mGluR3 and it also is …
Formula:
C21H11F6N5
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
447.34
Ref: TM-T15090
| 1mg | 54.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 302.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 588.00 € | ||
| 200mg | 792.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
DHPG
CAS:146255-66-5
DHPG is a potent Group I mGluR agonist; doesn't affect Group II/III; linked to phospholipase …
Formula:
C8H9NO4
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
183.16
Ref: TM-T11032
| 5mg | 50.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 216.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
(R)-ADX-47273
CAS:851881-59-9
(R)-ADX-47273 is a potent mGluR5 positive allosteric modulator(EC50 of 168 nM for potentiation ).
Formula:
C20H17F2N3O2
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
369.36
Ref: TM-T13441
| 2mg | 41.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 377.00 € | ||
| 200mg | 525.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Piracetam
CAS:7491-74-9
Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy …
Formula:
C6H10N2O2
Purity:
99.72%
Color and Shape:
Crystals From Isopropanol Solid
Molecular weight:
142.16
Ref: TM-T0426
| 1g | 62.00 € | ||
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 54.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
VU0650786
CAS:1809085-30-0
VU0650786: selective mGlu3 NAM, CNS-penetrant, IC50 392 nM, shows antidepressant/anxiolytic effects in rodents.
Formula:
C18H15ClFN5O2
Purity:
98.96%
Color and Shape:
Solid
Molecular weight:
387.8
Ref: TM-T13318
| 1mg | 95.00 € | ||
| 5mg | 232.00 € | ||
| 10mg | 326.00 € | ||
| 25mg | 553.00 € | ||
| 50mg | 790.00 € | ||
| 100mg | 1,088.00 € | ||
| 1mL*10mM (DMSO) | 256.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Org-26576
CAS:1026791-61-6
Org-26576 is a positive allosteric modulator of the AMPA receptor.
Formula:
C11H12N2O2
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
204.23
Ref: TM-T16402
| 5mg | 45.00 € | ||
| 10mg | 68.00 € | ||
| 25mg | 101.00 € | ||
| 50mg | 145.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 365.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
GET73
CAS:202402-01-5
GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.
Formula:
C13H16F3NO2
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
275.27
Ref: TM-T11393
| 1mg | 63.00 € | ||
| 5mg | 127.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 331.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 620.00 € | ||
| 200mg | 817.00 € | ||
| 1mL*10mM (DMSO) | 173.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Basimglurant
CAS:802906-73-6
Basimglurant (CTEP Derivative) is a potent, selective and orally available modulator of mGlu5 negative allosteric(Kd …
Formula:
C18H13ClFN3
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
325.77
Ref: TM-T12717
| 1mg | 81.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 246.00 € | ||
| 25mg | 406.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 682.00 € | ||
| 200mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 190.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
AZD-8529 mesylate
CAS:1314217-69-0
AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: …
Formula:
C25H28F3N5O6S
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
583.58
Ref: TM-T10432L
| 1mg | 91.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,079.00 € | ||
| 1mL*10mM (DMSO) | 218.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
(S)-3,4-DCPG
CAS:201730-11-2
(S)-3,4-DCPG ((S)-3,4-Dicarboxyphenylglycine) is a selective agonist of human metabotropic glutamate receptor 8a (mGluR8a).
Formula:
C10H9NO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
239.18
Ref: TM-T23288
| 1mg | 86.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 473.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
LY339434 HCl
LY339434 HCl is a low affinity GluR5 erythrocyte receptor agonist.LY339434 HCl causes rapid neuronal death …
Formula:
C18H20ClNO4
Purity:
99% - 99.32%
Color and Shape:
Soild
Molecular weight:
349.81
Ref: TM-T27947L
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,262.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,416.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Pomaglumetad methionil anhydrous
CAS:635318-55-7
LY2140023, potential schizophrenia treatment, is an oral prodrug of LY404039, a selective mGlu2/3 agonist.
Formula:
C12H18N2O7S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
366.41
Ref: TM-T11907
| 10mg | 1,386.00 € | ||
| 25mg | 2,957.00 € | ||
| 50mg | 4,649.00 € | ||
| 100mg | 7,067.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
KRP-199 sodium
KRP-199 sodium sodium is highly potent and selective for AMPA-R in vitro and exhibits good …
Formula:
C22H12F3N5Na2O7
Purity:
96.85%
Color and Shape:
Soild
Molecular weight:
561.33
Ref: TM-T27748L
| 1mg | 181.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,384.00 € | ||
| 100mg | 1,829.00 € | ||
| 500mg | 3,648.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
mGluR3 modulator-1
CAS:374548-18-2
1-ethyl-3-morpholin-4-yl tetrahydroisoquinoline: mGluR3 modulator, potential for Parkinson's.
Formula:
C16H21N3O
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
271.36
Ref: TM-T9970
| 5mg | 63.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 325.00 € | ||
| 1mL*10mM (DMSO) | 61.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
MMPIP hydrochloride
CAS:1215566-78-1
MMPIP hydrochloride is a selective antagonist of allosteric mGluR7.
Formula:
C19H16ClN3O3
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
369.8
Ref: TM-T23008L
| 1mg | 58.00 € | ||
| 2mg | 85.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 198.00 € | ||
| 25mg | 407.00 € | ||
| 50mg | 603.00 € | ||
| 100mg | 864.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
KM02894
CAS:116850-74-9
KM02894 inhibits glutamate release, potentially reducing cancer-induced bone pain in tumor studies.
Formula:
C7H9N3OS2
Purity:
98.72%
Color and Shape:
Liquid
Molecular weight:
215.3
Ref: TM-T77581
| 25mg | 49.00 € | ||
| 50mg | 71.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
![1H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)-](https://static.cymitquimica.com/products/TM/thumb/T60224.jpg)
1H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)-
CAS:175340-21-3
1H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)- is a low activity isomer of S 18986.
Formula:
C10H12N2O2S
Purity:
99.69%
Color and Shape:
Soild
Molecular weight:
224.28
Ref: TM-T60224
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 1mL*10mM (DMSO) | 218.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
(R)-3,4-DCPG HCl
(R)-3,4-DCPG HCl is a potent and selective mGlu8a receptor agonist that activates metabotropic glutamate receptors …
Formula:
C10H10ClNO6
Purity:
98.36% - 99.64%
Color and Shape:
Soild
Molecular weight:
275.64
Ref: TM-T23215L
| 1mg | 182.00 € | ||
| 5mg | 411.00 € | ||
| 10mg | 602.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,736.00 € | ||
| 500mg | 3,463.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
NBQX Disodium
CAS:479347-86-9
NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and …
Formula:
C12H6N4Na2O6S
Purity:
98.22%
Color and Shape:
Solid
Molecular weight:
380.24
Ref: TM-T25853
| 1mg | 67.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 308.00 € | ||
| 50mg | 456.00 € | ||
| 100mg | 666.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
