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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

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  • LAS190792
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    LAS190792

    CAS:
    <p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>
    Formula:C39H43ClN4O9S2
    Color and Shape:Solid
    Molecular weight:811.36

    Ref: TM-T74709

  • Guanylyl Imidodiphosphate (lithium salt)
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    Guanylyl Imidodiphosphate (lithium salt)

    CAS:
    <p>Guanylyl Imidodiphosphate (lithium salt) is a non-hydrolyzable GTP analog that increases adenylate cyclase activity.</p>
    Formula:C10H13Li4N6O13P3
    Color and Shape:Solid
    Molecular weight:545.93

    Ref: TM-T36009

  • Lu AE51090
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    Lu AE51090

    CAS:
    <p>Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.</p>
    Formula:C24H29N3O3
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:407.51

    Ref: TM-T32913

  • Perindoprilat
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    Perindoprilat

    CAS:
    <p>Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.</p>
    Formula:C17H28N2O5
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:340.41

    Ref: TM-T1484

  • Soclenicant
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    Soclenicant

    CAS:
    <p>Soclenicant is a negative-altering modulator of α 7 -nAChR for anxiety, depression, and PTSD, due to its high selectivity, oral availability</p>
    Formula:C24H26N4O3
    Purity:99.57%
    Color and Shape:Soild
    Molecular weight:418.49

    Ref: TM-T203814

  • Br-PBTC
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    Br-PBTC

    CAS:
    <p>Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.</p>
    Formula:C14H15BrN2OS
    Color and Shape:Solid
    Molecular weight:339.25

    Ref: TM-T39286

  • α-Conotoxin EI
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    α-Conotoxin EI

    CAS:
    <p>Selective antagonist of neuromuscular nicotinic receptors α1β1γδ</p>
    Formula:C83H125N27O27S5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2093.37

    Ref: TM-TP2218

  • Perlapine
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    Perlapine

    CAS:
    <p>Perlapine is an effective and selective HM3DQ DREADD agonist (EC50 = 2.8 nM).</p>
    Formula:C19H21N3
    Color and Shape:Solid
    Molecular weight:291.39

    Ref: TM-T33937

  • Atracurium
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    Atracurium

    CAS:
    <p>Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.</p>
    Formula:C53H72N2O122
    Color and Shape:Solid
    Molecular weight:929.14

    Ref: TM-T75283

  • BTMPS
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    BTMPS

    CAS:
    <p>BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.</p>
    Formula:C28H52N2O4
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:480.72

    Ref: TM-T203537

  • Albanin A
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    Albanin A

    <p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>
    Formula:C20H18O6
    Color and Shape:Solid
    Molecular weight:354.358

    Ref: TM-T124310

  • Epiboxidine hydrochloride
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    Epiboxidine hydrochloride

    CAS:
    <p>Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.</p>
    Formula:C10H15ClN2O
    Color and Shape:Solid
    Molecular weight:214.69

    Ref: TM-T74131

  • (rel)-Asperparaline A
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    (rel)-Asperparaline A

    CAS:
    <p>Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.</p>
    Formula:C20H29N3O3
    Color and Shape:Solid
    Molecular weight:359.47

    Ref: TM-T37609

  • sabcomeline
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    sabcomeline

    CAS:
    <p>Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.</p>
    Formula:C10H15N3O
    Color and Shape:Solid
    Molecular weight:193.25

    Ref: TM-T68135

  • M 8218
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    M 8218

    CAS:
    <p>M 8218 is a bioactive chemical.</p>
    Formula:C20H29NO2
    Color and Shape:Solid
    Molecular weight:315.45

    Ref: TM-T33111

  • Anagyrine hydrochloride
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    Anagyrine hydrochloride

    CAS:
    <p>Anagyrine hydrochloride, a quinolizidine from Lupinus albus, targets muscarinic/nicotinic receptors; IC50: 132/2096 µM. It desensitizes nAChR directly.</p>
    Formula:C15H21ClN2O
    Color and Shape:Solid
    Molecular weight:280.79

    Ref: TM-T73856

  • Navafenterol saccharinate
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    Navafenterol saccharinate

    CAS:
    <p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>
    Formula:C45H47N7O9S3
    Color and Shape:Solid
    Molecular weight:926.09

    Ref: TM-T30265

  • NNC 11-1607
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    NNC 11-1607

    CAS:
    <p>NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.</p>
    Formula:C30H32N6O2S2
    Color and Shape:Solid
    Molecular weight:572.74

    Ref: TM-T28181

  • (-)-Coclaurine hydrochloride
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    (-)-Coclaurine hydrochloride

    CAS:
    <p>(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.</p>
    Formula:C17H20ClNO3
    Purity:99.07%
    Color and Shape:Soild
    Molecular weight:321.8

    Ref: TM-TN1519L

  • (Rac)-Sabcomeline
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    (Rac)-Sabcomeline

    CAS:
    <p>(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.</p>
    Formula:C10H15N3O
    Purity:99.14%
    Color and Shape:Solid
    Molecular weight:193.25

    Ref: TM-T68135L1