AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Vecuronium bromide
CAS:50700-72-6
Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking …
Formula:
C34H57BrN2O4
Purity:
99.63% - 99.92%
Color and Shape:
White Powder
Molecular weight:
637.73
Ref: TM-T1594
| 10mg | 35.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 95.00 € | ||
| 500mg | 203.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
VU 0365114
CAS:1208222-39-2
VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: …
Formula:
C22H14F3NO3
Purity:
97.29%
Color and Shape:
Solid
Molecular weight:
397.35
Ref: TM-T13325
| 2mg | 37.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | 324.00 € | ||
| 200mg | 452.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
(±)-Acetylcarnitine chloride
CAS:2504-11-2
(±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can …
Formula:
C9H18ClNO4
Purity:
99.98%
Color and Shape:
White Crystalline Powder
Molecular weight:
239.7
Ref: TM-T21655
| 5mg | 39.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 124.00 € | ||
| 500mg | 292.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Hydroxybupropion
CAS:92264-81-8
Hydroxybupropion (6-Hydroxybupropion) is the major active metabolite of Bupropion and an antagonist of nACh receptor. …
Formula:
C13H18ClNO2
Purity:
98.61%
Color and Shape:
Off-White Solid
Molecular weight:
255.74
Ref: TM-T11588
| 1mg | 115.00 € | ||
| 2mg | 170.00 € | ||
| 5mg | 276.00 € | ||
| 10mg | 430.00 € | ||
| 25mg | 690.00 € | ||
| 50mg | 917.00 € | ||
| 100mg | 1,272.00 € | ||
| 1ml*10 (DMSO) | 276.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
8-Aminoadenine
CAS:28128-33-8
8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.
Formula:
C5H6N6
Purity:
90%
Color and Shape:
Solid
Molecular weight:
150.14
Ref: TM-T22013
| 1mg | 44.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 303.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 2 Dec 2024
bPiDDB
CAS:525596-66-1
bPiDDB (N,N'-Dodecylbis-Picolinium Bromide) is a nicotinic receptor (nAChR) antagonist.
Formula:
C24H38Br2N2
Purity:
98.72%
Color and Shape:
Liquid
Molecular weight:
514.38
Ref: TM-T37818
| 5mg | 59.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 403.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Simpinicline
CAS:753015-44-0
Simpinicline (OC-02) (OC-02) is an nAChR agonist that activates the trigeminal parasympathetic pathway and can …
Formula:
C10H13N3
Purity:
98.54% - 99.63%
Color and Shape:
Solid
Molecular weight:
175.23
Ref: TM-T40867
| 1mg | 375.00 € | ||
| 5mg | 915.00 € | ||
| 10mg | 1,217.00 € | ||
| 25mg | 1,839.00 € | ||
| 50mg | 2,471.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Emraclidine
CAS:2170722-84-4
Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive …
Formula:
C20H21F3N4O
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
390.4
Ref: TM-T9694
| 1mg | 125.00 € | ||
| 5mg | 301.00 € | ||
| 10mg | 539.00 € | ||
| 25mg | 867.00 € | ||
| 50mg | 1,183.00 € | ||
| 100mg | 1,576.00 € | ||
| 1mL*10mM (DMSO) | 335.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
TMPH
CAS:849461-90-1
TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. …
Formula:
C16H31NO2
Purity:
99.78%
Color and Shape:
Soild
Molecular weight:
269.42
Ref: TM-T60080
| 2mg | 37.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 136.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 307.00 € | ||
| 200mg | 433.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
M4 mAChR agonist-1
CAS:785705-53-5
M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).
Formula:
C14H18N4OS
Purity:
98.25%
Color and Shape:
Solid
Molecular weight:
290.38
Ref: TM-T9889
| 2mg | 46.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 402.00 € | ||
| 500mg | 904.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
(Rac)-Sabcomeline HCl
CAS:133642-67-8
Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.
Formula:
C10H16ClN3O
Purity:
99.03%
Color and Shape:
Soild
Molecular weight:
229.71
Ref: TM-T68135L
| 1mg | 183.00 € | ||
| 5mg | 402.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,262.00 € | ||
| 100mg | 1,699.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
9-Cyclopentyladenine
CAS:715-91-3
9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of …
Formula:
C10H13N5
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
203.24
Ref: TM-T29652
| 1mg | 182.00 € | ||
| 5mg | 402.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,698.00 € | ||
| 500mg | 3,438.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Rivanicline 2HCl
Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the …
Formula:
C10H16Cl2N2
Purity:
99.76%
Color and Shape:
Soild
Molecular weight:
235.15
Ref: TM-T12738L1
| 1mg | 35.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 242.00 € | ||
| 50mg | 434.00 € | ||
| 100mg | 637.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
(-)-OPC-51803
CAS:192514-57-1
(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and …
Formula:
C26H32ClN3O2
Purity:
100% - 100.00%
Color and Shape:
Soild
Molecular weight:
454
Ref: TM-T28257L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,271.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,416.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
(S)-Coclaurine
CAS:486-39-5
(S)-Coclaurine (Coclaurine) is an antagonist of nAChR isolated from Sarcopetalum harveyanum.
Formula:
C17H19NO3
Purity:
97.72%
Color and Shape:
Solid
Molecular weight:
285.34
Ref: TM-TN1519
| 1mg | 172.00 € | ||
| 5mg | 426.00 € | ||
| 10mg | 714.00 € | ||
| 25mg | 1,076.00 € | ||
| 50mg | 1,477.00 € | ||
| 100mg | 1,997.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
CDD0102 HCl
CAS:1196130-86-5
CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of …
Formula:
C8H13ClN4O
Purity:
99.7%
Color and Shape:
Soild
Molecular weight:
216.67
Ref: TM-T80662
| 1mg | 651.00 € | ||
| 5mg | 1,673.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Pozanicline hydrochloride
Pozanicline hydrochloride is an oral α4β2 nAChR agonist with a 16.7 nM Ki, insignificantly binding …
Formula:
C11H17ClN2O
Purity:
99.6%
Color and Shape:
Liquid
Molecular weight:
228.72
Ref: TM-T16563L
| 1mg | 113.00 € | ||
| 5mg | 244.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,031.00 € | ||
| 500mg | 2,070.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Cyclodrine
CAS:52109-93-0
Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.
Formula:
C19H29NO3
Purity:
98.3%
Color and Shape:
Soild
Molecular weight:
319.44
Ref: TM-T10914L
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,052.00 € | ||
| 500mg | 2,103.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Cevimeline hydrochloride hemihydrate
CAS:153504-70-2
Cevimeline hydrochloride hemihydrate is a novel muscarinic receptor agonist, used as a candidate therapeutic drug …
Formula:
C20H38Cl2N2O3S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
489.55
Ref: TM-T2390
| 2mg | 42.00 € | ||
| 5mg | 63.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
(-)-Coclaurine hydrochloride
CAS:3422-42-2
(-)-Coclaurine hydrochloride is an antagonist of nAChRs isolated from Sarcopetalum harveyanum.
Formula:
C17H20ClNO3
Purity:
97.75%
Color and Shape:
Soild
Molecular weight:
321.8
Ref: TM-TN1519L
| 1mg | 112.00 € | ||
| 5mg | 242.00 € | ||
| 10mg | 359.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,367.00 € | ||
| 1mL*10mM (DMSO) | 242.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
