AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Desfesoterodine
CAS:207679-81-0
Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.
Formula:
C22H31NO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
341.49
Ref: TM-T6364
| 1mg | 65.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 539.00 € | ||
| 100mg | 774.00 € | ||
| 500mg | 1,576.00 € | ||
| 1mL*10mM (DMSO) | 159.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Tiquizium
CAS:149755-23-7
Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary …
Formula:
C19H24NS2
Purity:
99.02%
Color and Shape:
Liquid
Molecular weight:
330.53
Ref: TM-T9877
| 1mg | 113.00 € | ||
| 5mg | 244.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,031.00 € | ||
| 500mg | 2,070.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
α-Muricholic acid
CAS:2393-58-0
α-Muricholic acid is the most abundant primary bile acid in rodents.
Formula:
C24H40O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
408.57
Ref: TM-T19623
| 1mg | 278.00 € | ||
| 5mg | 936.00 € | ||
| 10mg | 1,774.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
5-AAM-2-CP
CAS:175424-74-5
5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a …
Formula:
C8H9ClN2O
Purity:
90%
Color and Shape:
Solid
Molecular weight:
184.62
Ref: TM-T37196
| 25mg | 37.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 84.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
V-11-0711 HCl
V-11-0711 HCl is a selective and highly effective choline kinase α (ChoKα) inhibitor that inhibits …
Formula:
C27H36ClNO3
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
458.03
Ref: TM-T29083L
| 1mg | 195.00 € | ||
| 5mg | 659.00 € | ||
| 10mg | 1,030.00 € | ||
| 25mg | 1,540.00 € | ||
| 50mg | 2,078.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Tazomeline
CAS:131987-54-7
Tazomeline is a muscarinic M1 receptor agonist with neuroprotective activity.
Formula:
C14H23N3S2
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
297.48
Ref: TM-T68153
| 1mg | 104.00 € | ||
| 5mg | 242.00 € | ||
| 10mg | 365.00 € | ||
| 25mg | 607.00 € | ||
| 50mg | 867.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,350.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
TC-2216
CAS:646055-67-6
TC-2216 is a partial agonist at the neural nicotinic acetylcholine receptor and is used to …
Formula:
C12H17N3
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
203.28
Ref: TM-T68154
| 1mg | 93.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 743.00 € | ||
| 100mg | 1,016.00 € | ||
| 500mg | 2,083.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SSR 180
CAS:298198-52-4
SSR 180 is a potent and subtype-selective α7 agonist with applications in the study of …
Formula:
C14H17BrN2O2
Purity:
98.95%
Color and Shape:
Soild
Molecular weight:
325.20
Ref: TM-T84293
| 1mg | 182.00 € | ||
| 5mg | 450.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,388.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Methyllycaconitine citrate
CAS:351344-10-0
Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the …
Formula:
C43H58N2O17
Purity:
98.03% - 98.69%
Color and Shape:
Solid
Molecular weight:
874.92
Ref: TM-T12017
| 5mg | 143.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
(Rac)-Sabcomeline
CAS:149156-36-5
(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such …
Formula:
C10H15N3O
Purity:
99.14%
Color and Shape:
Liquid
Molecular weight:
193.25
Ref: TM-T68135L1
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,389.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SIB 1553A
CAS:191611-76-4
SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to …
Formula:
C13H19NOS
Purity:
99.64%
Color and Shape:
Soild
Molecular weight:
237.36
Ref: TM-T16881L
| 1mg | 185.00 € | ||
| 5mg | 458.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € | ||
| 100mg | 1,868.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
(S)-UFR2709 hydrochloride
CAS:2934318-93-9
(S)-UFR2709 HCl: competitive nAChR blocker, prefers α4β2 over α7, lessens anxiety & alcohol intake in …
Formula:
C13H18ClNO2
Purity:
98.94%
Color and Shape:
Liquid
Molecular weight:
255.74
Ref: TM-T37094
| 1mg | 42.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 121.00 € | ||
| 25mg | 234.00 € | ||
| 50mg | 352.00 € | ||
| 100mg | 547.00 € | ||
| 500mg | 1,152.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Monepantel
CAS:887148-69-8
Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.
Formula:
C20H13F6N3O2S
Purity:
99.76%
Color and Shape:
White Powder
Molecular weight:
473.39
Ref: TM-T16126
| 1mg | 97.00 € | ||
| 5mg | 244.00 € | ||
| 10mg | 351.00 € | ||
| 25mg | 692.00 € | ||
| 50mg | 993.00 € | ||
| 100mg | 1,420.00 € | ||
| 1mL*10mM (DMSO) | 268.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Metixene hydrochloride hydrate
CAS:7081-40-5
Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and …
Formula:
C20H26ClNOS
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
363.95
Ref: TM-TQ0304
| 5mg | 41.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 171.00 € | ||
| 100mg | 269.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Velufenacin
CAS:1648737-78-3
Velufenacin is an antagonist of muscarinic receptor[1].
Formula:
C19H20ClFN2O2
Purity:
98.88%
Color and Shape:
Liquid
Molecular weight:
362.83
Ref: TM-T9771
| 1mg | 64.00 € | ||
| 5mg | 141.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 393.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 758.00 € | ||
| 200mg | 998.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
NBTGR
CAS:13153-27-0
NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).
Formula:
C17H18N6O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
434.43
Ref: TM-T12191
| 2mg | 84.00 € | ||
| 5mg | 141.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Ispronicline
CAS:252870-53-4
Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, …
Formula:
C14H22N2O
Purity:
96.49% - 96.54%
Color and Shape:
Solid
Molecular weight:
234.34
Ref: TM-T27636
| 2mg | 45.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 150.00 € | ||
| 50mg | 206.00 € | ||
| 100mg | 305.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Biperiden
CAS:514-65-8
Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.
Formula:
C21H29NO
Purity:
99.65%
Color and Shape:
Crystals Solid
Molecular weight:
311.46
Ref: TM-T0218
| 1mg | 49.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Tolterodine
CAS:124937-51-5
Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive …
Formula:
C22H31NO
Purity:
99.71%
Color and Shape:
White Like Or Light Brown Crystalline Powder
Molecular weight:
325.49
Ref: TM-T23229
| 5mg | 35.00 € | ||
| 10mg | 42.00 € | ||
| 25mg | 61.00 € | ||
| 50mg | 86.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
SSR180711 hydrochloride
CAS:446031-79-4
SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used …
Formula:
C14H18BrClN2O2
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
361.66
Ref: TM-T28856
| 1mg | 36.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 179.00 € | ||
| 50mg | 272.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
