AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Pipecuronium bromide
CAS:52212-02-9
Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular …
Formula:
C35H62Br2N4O4
Purity:
100%
Color and Shape:
Powder
Molecular weight:
762.7
Ref: TM-T12481
| 1mg | 35.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 198.00 € | ||
| 50mg | 322.00 € | ||
| 100mg | 513.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
GSK-1034702
CAS:932373-87-0
GSK-1034702 is an M1 mAChR agonist that improves cognitive deficits and may be useful in …
Formula:
C18H24FN3O2
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
333.4
Ref: TM-T27446
| 1mg | 80.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 267.00 € | ||
| 25mg | 526.00 € | ||
| 50mg | 847.00 € | ||
| 100mg | 1,271.00 € | ||
| 500mg | 2,480.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
RPR121056
CAS:181467-56-1
RPR121056 is a Irinotecan metabolite, which is generated by CYP3A4. Irinotecan is an antineoplastic agent …
Formula:
C33H38N4O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
618.68
Ref: TM-T12766
| 2mg | 350.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
(±)-Darifenacin
CAS:133033-93-9
(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.
Formula:
C28H30N2O2
Color and Shape:
Solid
Molecular weight:
426.55
Ref: TM-T12680
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 86.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
(S)-(+)-Dimethindene maleate
CAS:136152-65-3
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist …
Formula:
C24H28N2O4
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
408.49
Ref: TM-T23297
| 1mg | 49.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
ML380
CAS:1627138-52-6
ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).
Formula:
C23H25F3N4O3S
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
494.53
Ref: TM-T28069
| 2mg | 50.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 516.00 € | ||
| 500mg | 1,133.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Blarcamesine
CAS:195615-83-9
Blarcamesine (AVex-73) is a muscarinic M1 agonist potentially for the treatment of Alzheimer's disease.
Formula:
C19H23NO
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
281.39
Ref: TM-T7780
| 5mg | 47.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 276.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PNU-120596
CAS:501925-31-1
PNU-120596 (NSC-216666) is a positive allosteric modulator of α7 nAChR with EC50 of 216 nM.
Formula:
C13H14ClN3O4
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
311.72
Ref: TM-T6950
| 5mg | 40.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 361.00 € | ||
| 200mg | 528.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Nitrocaramiphen hydrochloride
CAS:98636-73-8
Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in …
Formula:
C18H27ClN2O4
Purity:
98.94%
Color and Shape:
Solid
Molecular weight:
370.87
Ref: TM-T23071
| 5mg | 50.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 301.00 € | ||
| 200mg | 430.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BQCA
CAS:338747-41-4
BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.
Formula:
C18H15NO4
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
309.32
Ref: TM-T3993
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 421.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
VU 0238429
CAS:1160247-92-6
VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or …
Formula:
C17H12F3NO4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
351.28
Ref: TM-T8007
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 223.00 € | ||
| 100mg | 352.00 € | ||
| 500mg | 821.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mecamylamine hydrochloride
CAS:826-39-1
Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.
Formula:
C11H22ClN
Purity:
100% - 99.76%
Color and Shape:
White Solid
Molecular weight:
203.75
Ref: TM-T2141
| 5mg | 40.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 188.00 € | ||
| 100mg | 276.00 € | ||
| 200mg | 423.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ipratropium Bromide
CAS:22254-24-6
Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD …
Formula:
C20H30BrNO3
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
412.37
Ref: TM-T6547
| 50mg | 45.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 89.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SQ22536
CAS:17318-31-9
SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.
Formula:
C9H11N5O
Purity:
98.8%
Color and Shape:
Off-White Solid
Molecular weight:
205.22
Ref: TM-T2172
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 270.00 € | ||
| 100mg | 462.00 € | ||
| 200mg | 672.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Isopropamide Iodide
CAS:71-81-8
Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.
Formula:
C23H33IN2O
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
480.43
Ref: TM-T5051
| 10mg | 41.00 € | ||
| 25mg | 61.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 115.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Methylbenactyzium Bromide
CAS:3166-62-9
Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.
Formula:
C21H28BrNO3
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
422.36
Ref: TM-T6744
| 1g | 182.00 € | ||
| 25mg | 46.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 89.00 € | ||
| 200mg | 132.00 € | ||
| 500mg | 217.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Oxotremorine sesquifumarate
CAS:17360-35-9
Oxotremorine sesquifumarate is a muscarinic agonist.
Formula:
C12H18N2OC4H4O4
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
380.39
Ref: TM-T23116
| 5mg | 63.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 264.00 € | ||
| 100mg | 397.00 € | ||
| 200mg | 345.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
OXOMEMAZINE
CAS:3689-50-7
Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in …
Formula:
C18H22N2O2S
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
330.44
Ref: TM-T9353
| 10mg | 35.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
JHU37160
CAS:2369979-68-8
JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for …
Formula:
C19H20ClFN4
Purity:
99.25%
Color and Shape:
Solid
Molecular weight:
358.84
Ref: TM-T9018
| 10mg | 49.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 121.00 € | ||
| 100mg | 183.00 € | ||
| 1mL*10mM (DMSO) | 38.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Isoxazole
CAS:288-14-2
Isoxazole (1,2-oxazole) is the inhibitor of acetylcholinesterase (AChE). The ligands of Isoxazole bind to and …
Formula:
C3H3NO
Purity:
100%
Color and Shape:
Colorless Liquid
Molecular weight:
69.06
Ref: TM-T7500
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
