PAI-1
Plasminogen Activator Inhibitor-1 (PAI-1) is a serine protease inhibitor that regulates fibrinolysis by inhibiting tissue plasminogen activator (tPA) and urokinase (uPA). Elevated levels of PAI-1 are associated with an increased risk of thrombosis, cardiovascular diseases, and metabolic syndrome. PAI-1 inhibitors are being investigated for their potential to treat these conditions. At CymitQuimica, we offer PAI-1 inhibitors to support your research in hematology, cardiovascular health, and metabolic diseases.
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Upamostat
CAS:590368-25-5
Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) …
Formula:
C32H47N5O6S
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
629.81
Ref: TM-T13257
| 1mg | 96.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 378.00 € | ||
| 25mg | 630.00 € | ||
| 50mg | 898.00 € | ||
| 100mg | 1,216.00 € | ||
| 1mL*10mM (DMSO) | 325.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Angstrom6
CAS:220334-14-5
Angstrom6 (A-6 peptide) is an 8 amino acid peptide derived from single chain urokinase fibrinogen …
Formula:
C39H62N10O15
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
910.97
Ref: TM-T26629
| 1mg | 54.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 490.00 € | ||
| 100mg | 700.00 € | ||
| 500mg | 1,406.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
TM5275 sodium
CAS:1103926-82-4
TM5275 sodium (TM5275 sodium salt) is an inhibitor of plasminogen activator inhibitor 1 (PAI-1).
Formula:
C28H27ClN3NaO5
Purity:
99.02% - 99.55%
Color and Shape:
Solid
Molecular weight:
543.98
Ref: TM-T4255
| 2mg | 42.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 245.00 € | ||
| 100mg | 353.00 € | ||
| 200mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Tiplaxtinin
CAS:393105-53-8
Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with …
Formula:
C24H16F3NO4
Purity:
99.16% - 99.75%
Color and Shape:
Solid
Molecular weight:
439.38
Ref: TM-T2030
| 2mg | 44.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 512.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
TM5441
CAS:1190221-43-2
TM5441 is an orally bioavailable fibrinogen activator inhibitor-1 inhibitor that inhibits several cancer cell lines …
Formula:
C21H17ClN2O6
Purity:
97.62% - 99.09%
Color and Shape:
Solid
Molecular weight:
428.82
Ref: TM-T4254
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 469.00 € | ||
| 100mg | 665.00 € | ||
| 500mg | 1,388.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
UK-371804
CAS:256477-09-5
UK-371804: potent uPA blocker; candidate for chronic skin ulcer preclinical studies.
Formula:
C14H16ClN5O4S
Purity:
95.81% - 99.26%
Color and Shape:
Solid
Molecular weight:
385.83
Ref: TM-T3442
| 1mg | 52.00 € | ||
| 2mg | 66.00 € | ||
| 5mg | 108.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 487.00 € | ||
| 100mg | 705.00 € | ||
| 500mg | 1,473.00 € | ||
| 1mL*10mM (DMSO) | 117.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Loureirin B
CAS:119425-90-0
Loureirin B suppresses fibrosis by modulating MMPs/TIMPs, hindering fibroblast growth, and targeting TGF-β1/Smad2/3 pathway.
Formula:
C18H20O5
Purity:
99.33% - 99.86%
Color and Shape:
Solid
Molecular weight:
316.35
Ref: TM-T3876
| 1mg | 52.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 620.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
TM5007
CAS:342595-05-5
TM5007 is a poent inhibitor of plasminogen activator inhibitor-1 (PAI-1; IC50 of 29 uM).
Formula:
C24H20N2O6S4
Purity:
96.91%
Color and Shape:
Solid
Molecular weight:
560.69
Ref: TM-T8962
| 1mg | 145.00 € | ||
| 5mg | 288.00 € | ||
| 10mg | 434.00 € | ||
| 25mg | 712.00 € | ||
| 50mg | 1,008.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Toddalolactone
CAS:483-90-9
Toddalolactone ((+)-Toddalolactone) is an anti-inflammatory and analgesic.
Formula:
C16H20O6
Purity:
99.06% - 99.85%
Color and Shape:
Solid
Molecular weight:
308.33
Ref: TM-T4S0592
| 20mg | 99.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
AZ3976
CAS:1418747-15-5
AZ3976 is an inhibitor of PAI-1 with an IC50 of 16 μM in a plasma …
Formula:
C15H19N5O3
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
317.34
Ref: TM-T23764
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 306.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Diaplasinin
CAS:481631-45-2
Diaplasinin (PAI-749) is a potent inhibitor of plasminogen activator inhibitor-1 (PAI-1) with antithrombotic activity, used …
Formula:
C32H31N5O
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
501.62
Ref: TM-T25915
| 1mg | 90.00 € | ||
| 5mg | 207.00 € | ||
| 10mg | 309.00 € | ||
| 25mg | 520.00 € | ||
| 50mg | 750.00 € | ||
| 100mg | 1,216.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Aleplasinin
CAS:481629-87-2
Aleplasinin (PAZ 417) is a selective and orally active inhibitor of Plasminogen activator inhibitor-1(PAI-1) and …
Formula:
C28H27NO3
Purity:
97.51%
Color and Shape:
Solid
Molecular weight:
425.52
Ref: TM-T29856
| 1mg | 57.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 188.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 655.00 € | ||
| 100mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 145.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
GW-6604
CAS:452342-37-9
GW-6604 is an ALK5 inhibitor and shows clear antifibrotic effects resulting in liver function improvement.
Formula:
C19H14N4
Purity:
99.26%
Color and Shape:
Liquid
Molecular weight:
298.34
Ref: TM-T9947
| 1mg | 35.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 279.00 € | ||
| 100mg | 405.00 € |
Estimated delivery in United States, on Tuesday 17 Jun 2025
ZK824190
CAS:2254001-81-3
ZK824190: oral uPA inhibitor, IC50 - uPA 237 nM, tPA 1600 nM, Plasmin 1850 nM.
Formula:
C22H20F2N2O4
Purity:
98.84%
Color and Shape:
Solid
Molecular weight:
414.4
Ref: TM-T13408
| 1mg | 259.00 € | ||
| 5mg | 540.00 € | ||
| 10mg | 775.00 € | ||
| 25mg | 1,188.00 € | ||
| 50mg | 1,596.00 € | ||
| 100mg | 2,157.00 € | ||
| 1mL*10mM (DMSO) | 560.00 € |
Estimated delivery in United States, on Tuesday 17 Jun 2025
