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Glutaminase

Glutaminase

Glutaminase inhibitors are compounds that inhibit glutaminase, an enzyme that catalyzes the conversion of glutamine to glutamate, a critical step in cellular metabolism, especially in cancer cells. Glutaminase plays a key role in providing energy and biosynthetic precursors for rapidly proliferating cells. Inhibitors of glutaminase are important for exploring metabolic dependencies in cancer cells and developing potential therapeutic strategies. At CymitQuimica, we provide glutaminase inhibitors to support your research in cancer metabolism, cellular bioenergetics, and therapeutic discovery.

Found 48 products for "Glutaminase".

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  • ZM39923
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    ZM39923

    CAS:
    ZM39923 is an effective JAK3 inhibitor (IC50=79 nM), simultaneously inhibiting TGM2 and Factor XIIIa (IC50=10/25 nM).
    Formula:C23H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.45

    Ref: TM-T17295

  • NC9 TG2 inhibitor
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    NC9 TG2 inhibitor

    CAS:
    NC9 is an irreversible inhibitor of transglutaminase 2 (TG2) and also inhibits Factor XIIIA (FXIIIA).
    Formula:C35H47N5O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:697.84

    Ref: TM-T28137

  • Duazomycin
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    Duazomycin

    CAS:
    Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.
    Formula:C8H11N3O4
    Color and Shape:Solid
    Molecular weight:213.19

    Ref: TM-T27217

  • VA4 TG2 inhibitor
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    VA4 TG2 inhibitor

    CAS:
    VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.
    Formula:C33H41N5O6S
    Color and Shape:Solid
    Molecular weight:635.77

    Ref: TM-T69933

  • α-Glucosidase-IN-5
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    α-Glucosidase-IN-5

    CAS:
    α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.
    Formula:C15H13NO3
    Color and Shape:Solid
    Molecular weight:255.27

    Ref: TM-T60389

  • Glutaminase-IN-4
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    Glutaminase-IN-4

    CAS:
    Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).
    Formula:C23H22N6O2S2
    Color and Shape:Solid
    Molecular weight:478.59

    Ref: TM-T63137

  • CP4d inhibitor
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    CP4d inhibitor

    CAS:
    CP4d is a novel reversible tg2 transamidase site-specific inhibitor
    Formula:C18H13N5O5
    Color and Shape:Solid
    Molecular weight:379.33

    Ref: TM-T71477

  • THDP-17
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    THDP-17

    CAS:
    THDP-17 is a inhibitor of glutaminase. THDP-17 shows a partial uncompetitive inhibition in vitro.
    Formula:C12H16N2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:220.33

    Ref: TM-T28961

  • GLS1 Inhibitor
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    GLS1 Inhibitor

    CAS:
    GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.
    Formula:C19H21N7O2S
    Color and Shape:Solid
    Molecular weight:411.48

    Ref: TM-T37222

  • JHU-083
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    JHU-083

    CAS:
    JHU-083 is a glutaminase antagonist that improves cognition and normalizes aberrant hippocampal glutaminase activity in APOE4 mice.
    Formula:C14H24N4O4
    Purity:97.89% - 99.53%
    Color and Shape:Solid
    Molecular weight:312.3648

    Ref: TM-T15613

  • AA9 TG2 inhibitor
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    AA9 TG2 inhibitor

    CAS:
    AA9 is a novel transglutaminase (TG2) inhibitor.
    Formula:C32H36N4O5
    Color and Shape:Solid
    Molecular weight:556.65

    Ref: TM-T69878

  • AA10 TG2 inhibitor
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    AA10 TG2 inhibitor

    CAS:
    AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).
    Formula:C32H36N4O5
    Color and Shape:Solid
    Molecular weight:556.65

    Ref: TM-T26494

  • GLS1 Inhibitor-3
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    GLS1 Inhibitor-3

    CAS:
    GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.
    Formula:C30H32N10O2S
    Color and Shape:Solid
    Molecular weight:596.71

    Ref: TM-T64211

  • UPGL00004
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    UPGL00004

    CAS:
    UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.
    Formula:C25H26N8O2S2
    Purity:97.93%
    Color and Shape:Red Solid
    Molecular weight:534.656

    Ref: TM-T17206

  • TG-2-IN-1
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    TG-2-IN-1

    CAS:
    TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].
    Formula:C8H13ClN2OS
    Purity:99.88%
    Color and Shape:White Solid
    Molecular weight:220.72

    Ref: TM-T60274

  • IPN60090
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    IPN60090

    CAS:
    IPN60090: potent oral GLS1 inhibitor, IC50 of 31 nM, potential for anticancer and immunomodulation.
    Formula:C24H27F3N8O3
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:532.5182

    Ref: TM-T11412

  • TG2-IN-3h
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    TG2-IN-3h

    CAS:
    TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitor
    Formula:C21H26N4O4S
    Purity:98.51% - 99.76%
    Color and Shape:Yellow Solid
    Molecular weight:430.52

    Ref: TM-T70413

  • Sirpiglenastat
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    Sirpiglenastat

    CAS:
    Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.
    Formula:C22H27N5O5
    Purity:98.01% - 99.25%
    Color and Shape:Solid
    Molecular weight:441.48

    Ref: TM-T62560

  • KCC009
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    KCC009

    CAS:
    KCC009 is a TG2 inhibitor; IC50=20 μM; blocks survival signaling; cancer chemotherapy sensitization; glioblastoma research.
    Formula:C21H22BrN3O5
    Purity:98.68%
    Color and Shape:White Solid
    Molecular weight:476.32

    Ref: TM-T27717

  • ZED-1227
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    ZED-1227

    CAS:
    ZED-1227 (TAK-227) is a TG2 inhibitor with anticancer activity that blocks inflammation-induced TG2 expression and activation for the treatment of Celiac Diseas
    Formula:C26H36N6O6
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:528.6006

    Ref: TM-T17289