Tyrosine Kinase/Adaptors

Subcategories of "Tyrosine Kinase/Adaptors"

ALK

CSF-1R

EGFR

Ephrin Receptor

FLT

Fibroblast Growth Factor Receptor (FGFR)

HER

Hck

IGF-1R

PDGFR

PYK2

Src

TAM Receptor

Tie-2

Trk receptor

Tyrosine Kinases

VEGFR

c-Fms

c-Kit

c-Met/HGFR

c-RET

Show 13 more subcategories

Products of "Tyrosine Kinase/Adaptors"

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products per page. 1202 products on this category.

Product data	Purity	Price range	Estimated delivery
CGP52411 REF: TM-T10782CAS: 145915-58-8	99.56%	46.00 €~603.00 €	Tue 03 Sep 24
FLT3-IN-4 REF: TM-T11299CAS: 2304799-09-3	98.96%	91.00 €~1,838.00 €	Tue 03 Sep 24
FIIN-4 REF: TM-T27319CAS: 2093088-81-2	100%	306.00 €~2,721.00 €	Tue 03 Sep 24
(E)-FeCP-oxindole REF: TM-T22755CAS: 884338-18-5	99.62%	107.00 €~2,319.00 €	Tue 03 Sep 24
EML4-ALK kinase inhibitor 1 REF: TM-T11184CAS: 1373409-08-5	99.14%	95.00 €~1,833.00 €	Tue 03 Sep 24
SI-2 hydrochloride REF: TM-T12906CAS: 1992052-49-9	98.18%	To inquire	Tue 03 Sep 24
Cloperastine fendizoate REF: TM-T13619CAS: 85187-37-7	99.85%	49.00 €~51.00 €	Tue 03 Sep 24
DMH4 REF: TM-T22737CAS: 515880-75-8	98.68%	To inquire	Tue 03 Sep 24
INDY REF: TM-T15579CAS: 1169755-45-6	98.15%	60.00 €~155.00 €	Tue 03 Sep 24
(±)-Zanubrutinib REF: TM-TQ0039CAS: 1633350-06-7	98.19%	52.00 €~1,464.00 €	Tue 03 Sep 24
EGFR-IN-89 REF: TM-T79775CAS: 2413029-40-8	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
IACS-9439 REF: TM-T69759CAS: 2231259-57-5	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
Sotuletinib dihydrochloride REF: TM-T78603CAS: 2222138-40-9	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
Protein kinase inhibitor 5 REF: TM-T79125CAS: 2278204-94-5	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
TRK-IN-23 REF: TM-T78968CAS: 2924344-29-4	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
EGFR-IN-73 REF: TM-T73165CAS: 2857033-34-0	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
EGFR-IN-82 REF: TM-T78788CAS: 2568086-81-5	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
TRK II-IN-1 REF: TM-T73033CAS: 2904690-41-9	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
Antiproliferative agent-34 REF: TM-T79368CAS: 2910858-34-1	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
Infigratinib phosphate REF: TM-T16364CAS: 1310746-10-1	99.6%	To inquire	Tue 03 Sep 24
JNJ-64264681 REF: TM-T79019CAS: 2101524-34-7	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
ER-27319 REF: TM-T78641CAS: 201010-95-9	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
FGFR1 inhibitor-10 REF: TM-T79686CAS: 2426769-76-6	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
EGFR-IN-88 REF: TM-T79694CAS: 2944452-34-8	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
GZD856 REF: TM-T11523CAS: 1257628-64-0	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
Falnidamol REF: TM-TQ0271CAS: 196612-93-8	96.46%	48.00 €~756.00 €	Tue 03 Sep 24
EGFR-IN-16 REF: TM-T8525CAS: 133550-22-8	98%	118.00 €~346.00 €	Tue 03 Sep 24
Tarlox-TKI REF: TM-T11761CAS: 2135696-72-7	97.03%	To inquire	Tue 03 Sep 24
ProINDY REF: TM-T23186CAS: 719277-30-2	97.19%	89.00 €~1,013.00 €	Tue 03 Sep 24
PD 174265 REF: TM-T28339CAS: 216163-53-0	98.88%	54.00 €~181.00 €	Tue 03 Sep 24
Naluzotan REF: TM-T16265CAS: 740873-06-7	100%	650.00 €~1,671.00 €	Tue 03 Sep 24
SSR128129E free acid REF: TM-T13003CAS: 848463-13-8	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
ALK2-IN-2 REF: TM-T10287CAS: 2254409-25-9	99.55%	91.00 €~2,103.00 €	Tue 03 Sep 24
Lanraplenib monosuccinate REF: TM-T11824LCAS: 1800046-97-2	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
RU-302 REF: TM-T16806CAS: 1182129-77-6	99.45%	65.00 €~1,783.00 €	Tue 03 Sep 24
OD36 REF: TM-T35694CAS: 1638644-62-8	98%	73.00 €~867.00 €	Tue 03 Sep 24
EAI001 REF: TM-T61191CAS: 892772-75-7	100%	55.00 €~446.00 €	Tue 03 Sep 24
Mutated EGFR-IN-2 REF: TM-T12130CAS: 2050906-97-1	98%	1,000.00 €~2,617.00 €	Tue 03 Sep 24
(E/Z)-CP-724714 REF: TM-T6046CAS: 537705-08-1	98%	905.00 €~2,331.00 €	Tue 03 Sep 24
AC710 REF: TM-TQ0235CAS: 1351522-04-7	98%	35.00 €~417.00 €	Tue 03 Sep 24
Bezuclastinib REF: TM-T60976CAS: 1616385-51-3	99.81%	172.00 €~3,421.00 €	Tue 03 Sep 24
AMPK-IN-3 REF: TM-T62745CAS: 2417674-27-0	99.13%	108.00 €~1,473.00 €	Tue 03 Sep 24
Gilteritinib hemifumarate REF: TM-T71973CAS: 1254053-84-3	98.07%	40.00 €~425.00 €	Tue 03 Sep 24
TG 100572 REF: TM-T13156CAS: 867334-05-2	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
EGFR-IN-5 REF: TM-T11160CAS: 2225887-26-1	98.17%	106.00 €~2,349.00 €	Tue 03 Sep 24
Sitravatinib malate REF: TM-T12925CAS: 2244864-88-6	98%	904.00 €~2,329.00 €	Tue 03 Sep 24
c-Fms-IN-9 REF: TM-T10648CAS: 1628574-50-4	98%	1,000.00 €~2,617.00 €	Tue 03 Sep 24
Keap1-Nrf2-IN-1 REF: TM-T11752CAS: 2232112-72-8	98%	347.00 €~2,321.00 €	Tue 03 Sep 24
Glesatinib hydrochloride REF: TM-T15383CAS: 1123838-51-6	98%	885.00 €~1,861.00 €	Tue 03 Sep 24
c-Kit-IN-3 REF: TM-T10651CAS: 2363169-01-9	99.43%	85.00 €~1,545.00 €	Tue 03 Sep 24
(R)-Zanubrutinib REF: TM-T13447CAS: 1691249-44-1	98.04%	69.00 €~1,839.00 €	Tue 03 Sep 24
Spebrutinib besylate REF: TM-T14357CAS: 1360053-81-1	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
Sovleplenib REF: TM-T32088CAS: 1415792-84-5	98.51%	206.00 €~2,089.00 €	Tue 03 Sep 24
TG-46 REF: TM-T20743CAS: 936091-15-5	100%	181.00 €~2,357.00 €	Tue 03 Sep 24
ALK-IN-5 REF: TM-T10283CAS: 2351929-66-1	98%	908.00 €~2,338.00 €	Tue 03 Sep 24
c-Fms-IN-2 REF: TM-T10775CAS: 791587-67-2	97.34%	95.00 €~1,040.00 €	Tue 03 Sep 24
A-935142 REF: TM-T14077CAS: 1031335-85-9	100%	326.00 €~4,547.00 €	Tue 03 Sep 24
(Z)-FeCP-oxindole REF: TM-T23554CAS: 1137967-28-2	98.13%	46.00 €~1,331.00 €	Tue 03 Sep 24
A 419259 trihydrochloride REF: TM-TQ0132CAS: 1435934-25-0	100%	52.00 €~1,551.00 €	Tue 03 Sep 24
QL-X-138 REF: TM-T38960CAS: 1469988-63-3	98.41%	182.00 €~1,850.00 €	Tue 03 Sep 24
Tyrphostin AG 112 REF: TM-T8534CAS: 144978-82-5	97.01%	46.00 €~649.00 €	Tue 03 Sep 24
Larotinib REF: TM-T73334CAS: 1438072-11-7	98.45%	90.00 €~2,032.00 €	Tue 03 Sep 24
H-9 dihydrochloride REF: TM-T22833CAS: 116700-36-8	96.57%	69.00 €~1,203.00 €	Tue 03 Sep 24
Tyrphostin A25 REF: TM-T21622CAS: 118409-58-8	98.76%	54.00 €~392.00 €	Tue 03 Sep 24
Glesatinib REF: TM-T15384CAS: 936694-12-1	98%	1,000.00 €~2,617.00 €	Tue 03 Sep 24
Epertinib REF: TM-T11213LCAS: 908305-13-5	98%	423.00 €~2,336.00 €	Tue 03 Sep 24
c-Kit-IN-2 REF: TM-T10650CAS: 2121515-37-3	98%	1,000.00 €~2,617.00 €	Tue 03 Sep 24
S49076 HCl REF: TM-T3512CAS: 1265966-31-1	98%	115.00 €~826.00 €	Tue 03 Sep 24
CHMFL-ABL/KIT-155 REF: TM-T10801CAS: 2081093-21-0	98%	1,000.00 €~2,617.00 €	Tue 03 Sep 24
EGFR-IN-99 REF: TM-T35901CAS: 2068806-31-3	97.75%	125.00 €~2,639.00 €	Tue 03 Sep 24
JTV-519 free base REF: TM-T11731CAS: 145903-06-6	98%	904.00 €~2,329.00 €	Tue 03 Sep 24
R916562 REF: TM-T12650CAS: 1037798-41-6	98%	908.00 €~2,338.00 €	Tue 03 Sep 24
EGFR-IN-11 REF: TM-T11158CAS: 2463200-44-2	99.37%	To inquire	Tue 03 Sep 24
PP58 REF: TM-T13824CAS: 212391-58-7	99.21%	46.00 €~370.00 €	Tue 03 Sep 24
CGP60474 REF: TM-T14943CAS: 164658-13-3	98%	35.00 €~537.00 €	Tue 03 Sep 24
TG 100801 Hydrochloride REF: TM-T13157LCAS: 1018069-81-2	98%	904.00 €~2,329.00 €	Tue 03 Sep 24
OXSI-2 REF: TM-T28281CAS: 622387-85-3	98%	86.00 €~437.00 €	Tue 03 Sep 24
TL02-59 dihydrochloride REF: TM-T13186LCAS: 2415263-06-6	98%	734.00 €~3,073.00 €	Tue 03 Sep 24
RO9021 REF: TM-T16776CAS: 1446790-62-0	97.19%	85.00 €~1,813.00 €	Tue 03 Sep 24
Pz-1 REF: TM-T12598CAS: 1800505-64-9	99.95%	35.00 €~453.00 €	Tue 03 Sep 24
TGFBR1-IN-1 REF: TM-T13138CAS: 2170830-26-7	98%	904.00 €~2,329.00 €	Tue 03 Sep 24
YK-2-69 REF: TM-T69564CAS: 2619846-89-6	99.57%	274.00 €~2,330.00 €	Tue 03 Sep 24
SDZ281-977 REF: TM-T16866CAS: 150779-71-8	98%	97.00 €~1,884.00 €	Tue 03 Sep 24
FGFR2-IN-1 REF: TM-T61304CAS: 2677709-76-9	- - -	60.00 €~1,419.00 €	Tue 03 Sep 24
DDR Inhibitor REF: TM-T10985CAS: 1644069-80-6	97.75%	114.00 €~1,597.00 €	Tue 03 Sep 24
c-Fms-IN-6 REF: TM-T10645CAS: 1628574-81-1	98%	1,000.00 €~2,617.00 €	Tue 03 Sep 24
Cenisertib REF: TM-T14925CAS: 871357-89-0	- - -	113.00 €~1,741.00 €	Tue 03 Sep 24
Trk-IN-4 REF: TM-T17169CAS: 1799788-94-5	98%	To inquire	Tue 03 Sep 24
Tilfrinib REF: TM-T17098CAS: 1600515-49-8	99.73%	45.00 €~1,374.00 €	Tue 03 Sep 24
Epitinib succinate REF: TM-T35914CAS: 2252334-12-4	97.43%	74.00 €~1,653.00 €	Tue 03 Sep 24
EGFR-IN-9 REF: TM-T11163CAS: 1226549-39-8	99.46%	85.00 €~882.00 €	Tue 03 Sep 24
CHMFL-BTK-01 REF: TM-T14956CAS: 2095280-64-9	98%	998.00 €~2,611.00 €	Tue 03 Sep 24
PKI-166 REF: TM-T16549CAS: 187724-61-4	99.76%	55.00 €~1,967.00 €	Tue 03 Sep 24
TG-89 REF: TM-T20742CAS: 936091-56-4	98.8%	60.00 €~1,476.00 €	Tue 03 Sep 24
SU16f REF: TM-T16947CAS: 251356-45-3	98%	46.00 €~427.00 €	Tue 03 Sep 24
EGFR-IN-2 REF: TM-T11159CAS: 1643497-70-4	98%	907.00 €~2,337.00 €	Tue 03 Sep 24
Tafetinib REF: TM-T28911CAS: 1032265-57-8	96.66%	233.00 €~4,532.00 €	Tue 03 Sep 24
Syk-IN-3 REF: TM-T13045CAS: 1312534-69-2	97.99%	370.00 €~2,351.00 €	Tue 03 Sep 24
OD36 hydrochloride REF: TM-T61424CAS: 2387510-88-3	99.85%	182.00 €~2,320.00 €	Tue 03 Sep 24
MMPP REF: TM-T28077CAS: 1895957-18-2	100%	238.00 €~1,710.00 €	Tue 03 Sep 24

+ info

CGP52411

CAS:145915-58-8

CGP52411 is an orally active, and ATP-competitive inhibitor of EGFR (IC50: 0.3 μM).

Formula:

C₂₀H₁₅N₃O₂

Purity:

99.56%

Color and Shape:

Solid

Molecular weight:

329.35

Ref: TM-T10782

1mg		46.00 €
1ml		104.00 €
5mg		94.00 €
10mg		152.00 €
25mg		294.00 €
50mg		429.00 €
100mg		603.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

FLT3-IN-4

CAS:2304799-09-3

FLT3-IN-4 (FLT3 inhibitor 9u) is a potent and orally effective Fms-like tyrosine receptor kinase 3 …

Formula:

C₂₃H₂₅N₇O₂

Purity:

98.96%

Color and Shape:

Solid

Molecular weight:

431.49

Ref: TM-T11299

1mg		91.00 €
1ml		248.00 €
5mg		221.00 €
10mg		328.00 €
25mg		527.00 €
50mg		713.00 €
100mg		917.00 €
500mg		1,838.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

FIIN-4

CAS:2093088-81-2

FIIN-4 is a covalent inhibitor of FGFR and can be used in studies about metastatic …

Formula:

C₃₅H₃₈N₈O₄

Purity:

100%

Color and Shape:

Solid

Molecular weight:

634.73

Ref: TM-T27319

1mg		306.00 €
5mg		744.00 €
10mg		1,013.00 €
25mg		1,532.00 €
50mg		2,079.00 €
100mg		2,721.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

(E)-FeCP-oxindole

CAS:884338-18-5

(E)-FeCP-oxindole is an inhibitor of VEGFR2 with IC50 of 214 nM.

Formula:

C₁₉H₁₅FeNO

Purity:

99.62%

Color and Shape:

Solid

Molecular weight:

329.17

Ref: TM-T22755

1mg		107.00 €
5mg		239.00 €
10mg		358.00 €
25mg		602.00 €
50mg		859.00 €
100mg		1,161.00 €
500mg		2,319.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

EML4-ALK kinase inhibitor 1

CAS:1373409-08-5

Potent oral EML4-ALK inhibitor with a 1 nM IC50.

Formula:

C₃₁H₄₈N₈O₃

Purity:

99.14%

Color and Shape:

Solid

Molecular weight:

580.76

Ref: TM-T11184

1mg		95.00 €
1ml		269.00 €
5mg		208.00 €
10mg		310.00 €
25mg		500.00 €
50mg		682.00 €
100mg		922.00 €
500mg		1,833.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

SI-2 hydrochloride

CAS:1992052-49-9

SI-2 hydrochloride, an SRC-3 inhibitor, induces breast cancer cell death (IC50: 3-20 nM) with good …

Formula:

C₁₅H₁₆ClN₅

Purity:

98.18%

Color and Shape:

Solid

Molecular weight:

301.77

Ref: TM-T12906

5mg		35.00 €
10mg		46.00 €
25mg		63.00 €
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Sep 2024

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+ info

Cloperastine fendizoate

CAS:85187-37-7

Cloperastine fendizoate (Hustazol) inhibits the hERG K+ currents in a concentration-dependent manner (IC50: 27 nM).

Formula:

C₄₀H₃₈ClNO₅

Purity:

99.85%

Color and Shape:

Solid

Molecular weight:

648.19

Ref: TM-T13619

1ml		51.00 €
500mg		49.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

DMH4

CAS:515880-75-8

DMH4 is a potent and selective inhibitor of VEGFR2 with an IC50 of 0.16 µM.

Formula:

C₂₄H₂₄N₄O₂

Purity:

98.68%

Color and Shape:

Solid

Molecular weight:

400.47

Ref: TM-T22737

1mg		41.00 €
5mg		81.00 €
10mg		103.00 €
25mg		171.00 €
50mg		244.00 €
100mg		361.00 €
500mg		To inquire

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

INDY

CAS:1169755-45-6

INDY is an ATP-competitive inhibitor of Dyrk1A and Dyrk1B with IC50s of 0.24 μM and …

Formula:

C₁₂H₁₃NO₂S

Purity:

98.15%

Color and Shape:

Solid

Molecular weight:

235.3

Ref: TM-T15579

1ml		65.00 €
5mg		60.00 €
10mg		79.00 €
25mg		109.00 €
50mg		155.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

(±)-Zanubrutinib

CAS:1633350-06-7

(±)-Zanubrutinib ((±)-BGB-3111) is a potent and orally available Bruton's tyrosine kinase (Btk) inhibitor that demonstrates …

Formula:

C₂₇H₂₉N₅O₃

Purity:

98.19%

Color and Shape:

Solid

Molecular weight:

471.55

Ref: TM-TQ0039

1mg		52.00 €
1ml		116.00 €
5mg		109.00 €
10mg		172.00 €
25mg		307.00 €
50mg		508.00 €
100mg		728.00 €
500mg		1,464.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-89

CAS:2413029-40-8

EGFR-IN-89 (compound 13k) is a fourth-generation inhibitor selectively targeting EGFR mutations, exhibiting potent activity with …

Formula:

C₂₆H₃₁FN₈O₂S

Purity:

98%

Molecular weight:

538.64

Ref: TM-T79775

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

IACS-9439

CAS:2231259-57-5

IACS-9439 is a potent, selective, and orally active inhibitor of CSF1R, exhibiting a K(i) of …

Formula:

C₂₃H₂₆ClN₇O₃S

Purity:

98%

Molecular weight:

516.02

Ref: TM-T69759

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Sotuletinib dihydrochloride

CAS:2222138-40-9

Sotuletinib (BLZ945) dihydrochloride is an orally administered, blood-brain barrier-permeable inhibitor specifically targeting CSF1-R with an …

Formula:

C₂₀H₂₄Cl₂N₄O₃S

Purity:

98%

Molecular weight:

471.4

Ref: TM-T78603

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Protein kinase inhibitor 5

CAS:2278204-94-5

Protein kinase inhibitor 5 is a potent inhibitor of TRK-A, demonstrating an IC50 of 1.8 …

Formula:

C₂₉H₃₁F₂N₇O

Purity:

98%

Molecular weight:

531.6

Ref: TM-T79125

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

TRK-IN-23

CAS:2924344-29-4

TRK-IN-23 (compound 24b) is a potent, orally active inhibitor of TRK with IC50s of 0.5 …

Formula:

C₂₀H₁₇FN₄O₂

Purity:

98%

Molecular weight:

364.37

Ref: TM-T78968

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-73

CAS:2857033-34-0

EGFR-IN-73 (Compound 3f) effectively inhibits the prevalent EGFR mutation, EGFR Del19, exhibiting an IC50 value …

Formula:

C₁₉H₁₇ClFN₃O₄

Purity:

98%

Molecular weight:

405.81

Ref: TM-T73165

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-82

CAS:2568086-81-5

EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of …

Formula:

C₃₂H₄₁BrN₉O₂P

Purity:

98%

Molecular weight:

694.6

Ref: TM-T78788

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

TRK II-IN-1

CAS:2904690-41-9

TRK II-IN-1 is a potent type II inhibitor of tropomyosin receptor kinases (TRK), demonstrating inhibitory …

Formula:

C₂₉H₃₁F₃N₈O

Purity:

98%

Molecular weight:

564.6

Ref: TM-T73033

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Antiproliferative agent-34

CAS:2910858-34-1

Antiproliferative Agent-34 (Compound A14), a multitarget kinase inhibitor, demonstrates IC50 values of 177 nM for …

Formula:

C₂₇H₂₇N₇O₅

Purity:

98%

Molecular weight:

529.55

Ref: TM-T79368

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Infigratinib phosphate

CAS:1310746-10-1

Infigratinib phosphate (BGJ-398 phosphate) is an effective inhibitor of the FGFR family (IC50: 0.9 nM, …

Formula:

C₂₆H₃₄Cl₂N₇O₇P

Purity:

99.6%

Color and Shape:

Solid

Molecular weight:

658.47

Ref: TM-T16364

1ml		46.00 €
5mg		47.00 €
10mg		61.00 €
25mg		83.00 €
50mg		95.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

JNJ-64264681

CAS:2101524-34-7

JNJ-64264681 is a potent, orally active, selective, and irreversible covalent inhibitor of Bruton's tyrosine kinase …

Formula:

C₂₇H₃₀N₆O₃S

Purity:

98%

Molecular weight:

518.63

Ref: TM-T79019

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

ER-27319

CAS:201010-95-9

ER-27319, an acridone derivative, serves as a potent and selective inhibitor of spleen tyrosine kinase …

Formula:

C₂₀H₂₂N₂O₅

Purity:

98%

Molecular weight:

370.4

Ref: TM-T78641

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

FGFR1 inhibitor-10

CAS:2426769-76-6

FGFR1 inhibitor-10 (Compound 4i), with an IC50 of 28 nM, effectively inhibits FGFR1 phosphorylation. This …

Formula:

C₂₆H₃₀F₃N₇O₂S

Purity:

98%

Molecular weight:

561.62

Ref: TM-T79686

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-88

CAS:2944452-34-8

EGFR-IN-88 (Compound 4i), an EGFR inhibitor with an IC50 of 87 nM, exhibits cytotoxic effects …

Formula:

C₂₂H₁₈Cl₂N₄O₂S

Purity:

98%

Molecular weight:

473.37

Ref: TM-T79694

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

GZD856

CAS:1257628-64-0

GZD856 is an orally bioavailable PDGFRα/β inhibitor (IC50s: 68.6 and 136.6 nM) with anti-lung cancer …

Formula:

C₂₉H₂₇F₃N₆O

Purity:

98%

Color and Shape:

Solid

Molecular weight:

532.56

Ref: TM-T11523

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Falnidamol

CAS:196612-93-8

Falnidamol (BIBX 1382), an oral selective EGFR inhibitor, IC50 3 nM, weak on ErbB2 and …

Formula:

C₁₈H₁₉ClFN₇

Purity:

96.46%

Color and Shape:

Solid

Molecular weight:

387.84

Ref: TM-TQ0271

1mg		48.00 €
1ml		95.00 €
5mg		93.00 €
10mg		167.00 €
25mg		313.00 €
50mg		547.00 €
100mg		756.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-16

CAS:133550-22-8

EGFR-IN-16 (AG473) is an inhibitor of EGFR in human A431 cells.

Formula:

C₁₆H₁₁NO₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

265.26

Ref: TM-T8525

5mg		118.00 €
10mg		183.00 €
25mg		346.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Tarlox-TKI

CAS:2135696-72-7

Tarlox-TKI (Kinase inhibitor-1) is a pan-ErbB inhibitor, the active ingredient of Tarloxotinib, which has antitumor …

Formula:

C₁₉H₁₈BrClN₆O

Purity:

97.03%

Color and Shape:

Solid

Molecular weight:

461.74

Ref: TM-T11761

1mg		142.00 €
1ml		253.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

ProINDY

CAS:719277-30-2

ProINDY (Pro-indy) is a potent DYRK inhibitor that activates NFAT for the study of Down …

Formula:

C₁₄H₁₅NO₃S

Purity:

97.19%

Color and Shape:

Solid

Molecular weight:

277.34

Ref: TM-T23186

1mg		89.00 €
5mg		210.00 €
10mg		312.00 €
25mg		523.00 €
50mg		728.00 €
100mg		1,013.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

PD 174265

CAS:216163-53-0

PD 174265 is an effective, selective and reversible inhibitor of epidermal growth factor receptor (EGFR) …

Formula:

C₁₇H₁₅BrN₄O

Purity:

98.88%

Color and Shape:

Solid

Molecular weight:

371.23

Ref: TM-T28339

1ml		69.00 €
5mg		54.00 €
10mg		69.00 €
25mg		92.00 €
50mg		130.00 €
100mg		181.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Naluzotan

CAS:740873-06-7

Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of …

Formula:

C₂₃H₃₈N₄O₃S

Purity:

100%

Color and Shape:

Solid

Molecular weight:

450.64

Ref: TM-T16265

1mg		650.00 €
5mg		1,671.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

SSR128129E free acid

CAS:848463-13-8

SSR128129E free acid is an orally available and allosteric inhibitor of FGFR(IC50 of 1.9 μM …

Formula:

C₁₈H₁₆N₂O₄

Purity:

98%

Color and Shape:

Solid

Molecular weight:

324.33

Ref: TM-T13003

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

ALK2-IN-2

CAS:2254409-25-9

ALK2-IN-2 is a potent and selective inhibitor of activin receptor-like kinase 2 (ALK2) (IC50: 9 …

Formula:

C₂₈H₂₇N₅O₂S

Purity:

99.55%

Color and Shape:

Solid

Molecular weight:

497.61

Ref: TM-T10287

1mg		91.00 €
1ml		238.00 €
2mg		134.00 €
5mg		215.00 €
10mg		343.00 €
25mg		541.00 €
50mg		742.00 €
100mg		1,028.00 €
500mg		2,103.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Lanraplenib monosuccinate

CAS:1800046-97-2

Lanraplenib monosuccinate inhibits SYK activity in platelets via the glycoprotein VI (GPVI) receptor without prolonging …

Formula:

C₂₇H₃₁N₉O₅

Purity:

98%

Color and Shape:

Solid

Molecular weight:

561.59

Ref: TM-T11824L

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

RU-302

CAS:1182129-77-6

RU-302 is a pan inhibitor of TAM Receptor blocking the interface between the TAM Ig1 …

Formula:

C₂₄H₂₄F₃N₃O₂S

Purity:

99.45%

Color and Shape:

Solid

Molecular weight:

475.53

Ref: TM-T16806

1mg		65.00 €
1ml		159.00 €
2mg		95.00 €
5mg		142.00 €
10mg		237.00 €
25mg		423.00 €
50mg		624.00 €
100mg		888.00 €
500mg		1,783.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

OD36

CAS:1638644-62-8

OD36: Potent RIPK2 inhibitor, IC50=5.3 nM; hinders ALK2 signaling and osteogenesis, KD=37 nM; targets ALK2 …

Formula:

C₁₆H₁₅ClN₄O₂

Purity:

98%

Color and Shape:

Solid

Molecular weight:

330.77

Ref: TM-T35694

1mg		73.00 €
5mg		157.00 €
10mg		230.00 €
25mg		384.00 €
50mg		576.00 €
100mg		867.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EAI001

CAS:892772-75-7

EAI001 is a potent and selective mutant epidermal growth factor receptor (EGFR) variant inhibitor that …

Formula:

C₁₉H₁₅N₃O₂S

Purity:

100%

Color and Shape:

Solid

Molecular weight:

349.41

Ref: TM-T61191

5mg		55.00 €
10mg		96.00 €
25mg		172.00 €
50mg		276.00 €
100mg		446.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Mutated EGFR-IN-2

CAS:2050906-97-1

Mutated EGFR-IN-2 is an inhibitor of mutant-selective EGFR.

Formula:

C₂₉H₃₅FN₈O₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

562.64

Ref: TM-T12130

25mg		1,549.00 €
50mg		2,038.00 €
100mg		2,617.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

(E/Z)-CP-724714

CAS:537705-08-1

(E/Z)-CP-724714, comprising racemic mixtures of (E)-CP-724714 and (Z)-CP-724714 isomers, is a potent, selective, and orally …

Formula:

C₂₇H₂₇N₅O₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

469.54

Ref: TM-T6046

25mg		1,410.00 €
50mg		1,847.00 €
100mg		2,331.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

AC710

CAS:1351522-04-7

AC710 is a potent PDGFR inhibitor (Kds: 0.6, 1, 1.57, 1.3, 1 nM for FLT3, …

Formula:

C₃₁H₄₂N₆O₄

Purity:

98%

Color and Shape:

Solid

Molecular weight:

562.7

Ref: TM-TQ0235

1mg		35.00 €
1ml		87.00 €
2mg		45.00 €
5mg		68.00 €
10mg		95.00 €
25mg		185.00 €
50mg		277.00 €
100mg		417.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Bezuclastinib

CAS:1616385-51-3

Bezuclastinib (CGT9486) is a novel, potent and highly selective tyrosine kinase and c-kit D816V inhibitor …

Formula:

C₁₉H₁₇N₅O

Purity:

99.81%

Color and Shape:

Solid

Molecular weight:

331.37

Ref: TM-T60976

1mg		172.00 €
5mg		422.00 €
10mg		675.00 €
25mg		1,344.00 €
50mg		2,151.00 €
100mg		3,421.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

AMPK-IN-3

CAS:2417674-27-0

AMPK-IN-3: potent, selective AMPK (α2/α1) & KDR inhibitor; IC50: 60.7/107/3820 nM; anticancer in K562 cells.

Formula:

C₂₅H₃₃N₅O₃

Purity:

99.13%

Color and Shape:

Solid

Molecular weight:

451.56

Ref: TM-T62745

1mg		108.00 €
5mg		246.00 €
10mg		395.00 €
25mg		810.00 €
50mg		1,086.00 €
100mg		1,473.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Gilteritinib hemifumarate

CAS:1254053-84-3

Gilteritinib hemifumarate (ASP2215 hemifumarate) is a potent ATP-competitive dual FLT3 (IC50: 0.29 nM) and AXL …

Formula:

C₂₉H₄₄N₈O₃C₄H₄O₄

Purity:

98.07%

Color and Shape:

Solid

Molecular weight:

610.35

Ref: TM-T71973

1mg		40.00 €
5mg		87.00 €
10mg		118.00 €
25mg		185.00 €
50mg		269.00 €
100mg		425.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

TG 100572

CAS:867334-05-2

TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src …

Formula:

C₂₆H₂₆ClN₅O₂

Purity:

98%

Color and Shape:

Solid

Molecular weight:

475.97

Ref: TM-T13156

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-5

CAS:2225887-26-1

EGFR-IN-5 inhibits EGFR & mutants; IC50: EGFR 10.4nM, L858R 1.1nM, L858R/T790M 34nM, L858R/T790M/C797S 7.2nM.

Formula:

C₃₁H₃₈FN₉O

Purity:

98.17%

Color and Shape:

Solid

Molecular weight:

571.69

Ref: TM-T11160

1mg		106.00 €
5mg		249.00 €
10mg		442.00 €
25mg		887.00 €
50mg		1,346.00 €
100mg		2,349.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Sitravatinib malate

CAS:2244864-88-6

Sitravatinib malate is an orally bioavailable receptor inhibitor of tyrosine kinase (RTK) (IC50s of 1.5 …

Formula:

C₃₇H₃₅F₂N₅O₉S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

763.76

Ref: TM-T12925

25mg		1,410.00 €
50mg		1,845.00 €
100mg		2,329.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

c-Fms-IN-9

CAS:1628574-50-4

c-Fms-IN-9 inhibits c-FMS/uFMS and uKIT with IC50 <0.01μM and 0.1-1μM, from patent WO2014145023A1.

Formula:

C₂₁H₂₃N₇O₂

Purity:

98%

Color and Shape:

Solid

Molecular weight:

405.45

Ref: TM-T10648

25mg		1,549.00 €
50mg		2,038.00 €
100mg		2,617.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Keap1-Nrf2-IN-1

CAS:2232112-72-8

Keap1-Nrf2 IN-1, a protein interaction inhibitor with 43 nM IC50, boosts Nrf2 cytoprotection and counters …

Formula:

C₂₄H₂₄N₂O₇S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

484.52

Ref: TM-T11752

25mg		1,327.00 €
50mg		1,734.00 €
100mg		2,321.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Glesatinib hydrochloride

CAS:1123838-51-6

Glesatinib hydrochloride is an orally active and potent dual inhibitor of MET/SMO.

Formula:

C₃₁H₂₈ClF₂N₅O₃S₂

Purity:

98%

Color and Shape:

Solid

Molecular weight:

656.16

Ref: TM-T15383

25mg		885.00 €
50mg		1,160.00 €
100mg		1,861.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

c-Kit-IN-3

CAS:2363169-01-9

c-Kit-IN-3 is a selective inhibitor of c-KIT kinase with IC50s of 4 nM and 8 …

Formula:

C₂₆H₂₀ClF₃N₂O₄

Purity:

99.43%

Color and Shape:

Solid

Molecular weight:

516.9

Ref: TM-T10651

1mg		85.00 €
1ml		333.00 €
5mg		159.00 €
10mg		249.00 €
25mg		411.00 €
50mg		551.00 €
100mg		771.00 €
500mg		1,545.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

(R)-Zanubrutinib

CAS:1691249-44-1

(R)-Zanubrutinib ((R)-BGB-3111) is a selective inhibitor of Bruton tyrosine kinase (BTK).

Formula:

C₂₇H₂₉N₅O₃

Purity:

98.04%

Color and Shape:

Solid

Molecular weight:

471.55

Ref: TM-T13447

1mg		69.00 €
1ml		165.00 €
5mg		149.00 €
10mg		270.00 €
25mg		453.00 €
50mg		664.00 €
100mg		917.00 €
500mg		1,839.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Spebrutinib besylate

CAS:1360053-81-1

Spebrutinib besylate (AVL-292 benzenesulfonate; CC-292 besylate) is a Btk kinase activity inhibitor (IC50<0.5 nM, …

Formula:

C₂₈H₂₈FN₅O₆S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

581.62

Ref: TM-T14357

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Sovleplenib

CAS:1415792-84-5

Sovleplenib (HMPL-523), oral SYK inhibitor, IC50 25 nM, targets tumors & ITP studies.

Formula:

C₂₄H₃₀N₆O₃S

Purity:

98.51%

Color and Shape:

Solid

Molecular weight:

482.6

Ref: TM-T32088

1mg		206.00 €
1ml		584.00 €
5mg		523.00 €
10mg		738.00 €
25mg		1,142.00 €
50mg		1,557.00 €
100mg		2,089.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

TG-46

CAS:936091-15-5

TG-46 (TG46) inhibits JAK2, FLT3, RET, JAK3 and can be used to study glaucoma.

Formula:

C₂₆H₃₄N₆O₃S

Purity:

100%

Color and Shape:

Solid

Molecular weight:

510.65

Ref: TM-T20743

1mg		181.00 €
5mg		402.00 €
10mg		604.00 €
25mg		1,031.00 €
50mg		1,570.00 €
100mg		2,357.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

ALK-IN-5

CAS:2351929-66-1

ALK-IN-5 is a potent, selective, and brain-penetrant inhibitor of anaplastic lymphoma kinase (ALK, IC50: 2.9 …

Formula:

C₂₄H₂₅FN₆O₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

464.49

Ref: TM-T10283

25mg		1,410.00 €
50mg		1,852.00 €
100mg		2,338.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

c-Fms-IN-2

CAS:791587-67-2

c-Fms-IN-2 is an inhibitor of c-FMS kinase (IC50 = 24 nM).

Formula:

C₁₉H₂₁N₃O₃

Purity:

97.34%

Color and Shape:

Solid

Molecular weight:

339.39

Ref: TM-T10775

1mg		95.00 €
1ml		188.00 €
5mg		249.00 €
10mg		367.00 €
25mg		550.00 €
50mg		775.00 €
100mg		1,040.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

A-935142

CAS:1031335-85-9

A-935142 enhances hERG (Kv 11.1) channels, slows inactivation, promotes activation, and shortens repolarization.

Formula:

C₁₈H₁₉F₃N₂O₂

Purity:

100%

Color and Shape:

Solid

Molecular weight:

352.35

Ref: TM-T14077

1mg		326.00 €
5mg		769.00 €
10mg		1,050.00 €
25mg		1,486.00 €
50mg		1,850.00 €
100mg		2,322.00 €
500mg		4,547.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

(Z)-FeCP-oxindole

CAS:1137967-28-2

(Z)-FeCP-oxindole is a selective inhibitor of VEGFR2 with an IC50 of 200 nM for human. …

Formula:

C₁₉H₁₅FeNO

Purity:

98.13%

Color and Shape:

Solid

Molecular weight:

329.17

Ref: TM-T23554

1mg		46.00 €
1ml		96.00 €
5mg		92.00 €
10mg		131.00 €
25mg		261.00 €
50mg		418.00 €
100mg		645.00 €
500mg		1,331.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

A 419259 trihydrochloride

CAS:1435934-25-0

A 419259 trihydrochloride (RK 20449 trihydrochloride) is an Src family kinases inhibitor (IC50s: 9 nM, …

Formula:

C₂₉H₃₇Cl₃N₆O

Purity:

100%

Color and Shape:

Solid

Molecular weight:

592

Ref: TM-TQ0132

1mg		52.00 €
2mg		73.00 €
5mg		105.00 €
10mg		167.00 €
25mg		312.00 €
50mg		546.00 €
100mg		779.00 €
500mg		1,551.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

QL-X-138

CAS:1469988-63-3

QL-X-138 is a potent and selective BTK and MNK dual kinase inhibitor that binds covalently …

Formula:

C₂₅H₁₉N₅O₂

Purity:

98.41%

Color and Shape:

Solid

Molecular weight:

421.45

Ref: TM-T38960

1mg		182.00 €
2mg		295.00 €
5mg		546.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Tyrphostin AG 112

CAS:144978-82-5

Tyrphostin AG 112 is an inhibitor of EGFR phosphorylation.

Formula:

C₁₃H₈N₄O

Purity:

97.01%

Color and Shape:

Solid

Molecular weight:

236.23

Ref: TM-T8534

5mg		46.00 €
10mg		69.00 €
25mg		123.00 €
50mg		180.00 €
100mg		267.00 €
500mg		649.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Larotinib

CAS:1438072-11-7

Larotinib is an orally active, potent, and broad-spectrum tyrosine kinase inhibitor (TKI) with an IC50 …

Formula:

C₂₄H₂₆ClFN₄O₄

Purity:

98.45%

Color and Shape:

Solid

Molecular weight:

488.94

Ref: TM-T73334

1mg		90.00 €
5mg		202.00 €
10mg		298.00 €
25mg		504.00 €
50mg		727.00 €
100mg		1,012.00 €
500mg		2,032.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

H-9 dihydrochloride

CAS:116700-36-8

H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.

Formula:

C₁₁H₁₅Cl₂N₃O₂S

Purity:

96.57%

Color and Shape:

Solid

Molecular weight:

324.23

Ref: TM-T22833

1mg		69.00 €
5mg		143.00 €
10mg		208.00 €
25mg		465.00 €
50mg		894.00 €
100mg		1,203.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Tyrphostin A25

CAS:118409-58-8

Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist …

Formula:

C₁₀H₆N₂O₃

Purity:

98.76%

Color and Shape:

Yellow Green Powder /Off-White Solid

Molecular weight:

202.17

Ref: TM-T21622

1mg		54.00 €
5mg		73.00 €
10mg		93.00 €
25mg		150.00 €
50mg		258.00 €
100mg		392.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Glesatinib

CAS:936694-12-1

Glesatinib is an orally active and potent dual inhibitor of MET/SMO.

Formula:

C₃₁H₂₇F₂N₅O₃S₂

Purity:

98%

Color and Shape:

Solid

Molecular weight:

619.7

Ref: TM-T15384

25mg		1,549.00 €
50mg		2,038.00 €
100mg		2,617.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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Epertinib

CAS:908305-13-5

Epertinib is a reversible and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 (IC50s: …

Formula:

C₃₀H₂₇ClFN₅O₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

560.02

Ref: TM-T11213L

25mg		1,262.00 €
50mg		1,644.00 €
100mg		2,336.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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c-Kit-IN-2

CAS:2121515-37-3

c-Kit-IN-2 is a c-KIT inhibitor (IC50: 82 nM), shows superior antiproliferative activities against all the …

Formula:

C₂₅H₂₉N₉O₂S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

519.62

Ref: TM-T10650

25mg		1,549.00 €
50mg		2,038.00 €
100mg		2,617.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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S49076 HCl

CAS:1265966-31-1

S49076 HCl (S-49076 Hydrochloride) is an effective inhibitor of MET, AXL/MER, and FGFR1/2/3.

Formula:

C₂₂H₁₈ClN₃O₅

Purity:

98%

Color and Shape:

Solid

Molecular weight:

439.85

Ref: TM-T3512

5mg		115.00 €
10mg		176.00 €
25mg		288.00 €
50mg		456.00 €
100mg		826.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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+ info

CHMFL-ABL/KIT-155

CAS:2081093-21-0

CHMFL-ABL/KIT-155 is a highly potent and orally active type II ABL/c-KIT dual kinase inhibitor (IC50s: …

Formula:

C₃₃H₃₈F₃N₅O₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

609.68

Ref: TM-T10801

25mg		1,545.00 €
50mg		2,038.00 €
100mg		2,617.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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EGFR-IN-99

CAS:2068806-31-3

EGFR-IN-99 (JBJ-03-142-02) is an EGFR and HER2 Exon 20 insertion mutation inhibitor for the study …

Formula:

C₂₅H₂₂FN₇O₃

Purity:

97.75%

Color and Shape:

Solid

Molecular weight:

487.49

Ref: TM-T35901

1mg		125.00 €
5mg		297.00 €
10mg		441.00 €
25mg		714.00 €
50mg		979.00 €
100mg		1,324.00 €
500mg		2,639.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

JTV-519 free base

CAS:145903-06-6

JTV-519 free base (K201 free base), recognized for its antiarrhythmic and cardioprotective properties, functions as …

Formula:

C₂₅H₃₂N₂O₂S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

424.6

Ref: TM-T11731

25mg		1,410.00 €
50mg		1,845.00 €
100mg		2,329.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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R916562

CAS:1037798-41-6

R916562 is an orally active and selective Axl/VEGF-R2 inhibitor with IC50s of 136 nM and …

Formula:

C₂₆H₃₀ClN₉S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

536.09

Ref: TM-T12650

25mg		1,410.00 €
50mg		1,852.00 €
100mg		2,338.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

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EGFR-IN-11

CAS:2463200-44-2

EGFR-IN-11 selectively blocks EGFR-tyrosine kinase and promotes apoptosis; targets EGFRL858R/T790M/C797S, IC50=18 nM; halts cell cycle …

Formula:

C₂₉H₃₅N₉O₂S

Purity:

99.37%

Color and Shape:

Solid

Molecular weight:

573.71

Ref: TM-T11158

1mg		85.00 €
1ml		236.00 €
5mg		182.00 €
10mg		313.00 €
25mg		496.00 €
50mg		686.00 €
100mg		911.00 €
500mg		To inquire

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

PP58

CAS:212391-58-7

PP58 is an inhibitor of PDGFR, FGFR and Src family.

Formula:

C₂₂H₁₉Cl₂N₅O₂

Purity:

99.21%

Color and Shape:

Solid

Molecular weight:

456.32

Ref: TM-T13824

1mg		46.00 €
1ml		96.00 €
5mg		90.00 €
10mg		142.00 €
25mg		239.00 €
50mg		370.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

CGP60474

CAS:164658-13-3

CGP60474 is an inhibitor of VEGFR-2 (IC50 = 84 nM) and an inhibitor of ATP-competitive …

Formula:

C₁₈H₁₈ClN₅O

Purity:

98%

Color and Shape:

Solid

Molecular weight:

355.82

Ref: TM-T14943

1mg		35.00 €
1ml		82.00 €
2mg		47.00 €
5mg		73.00 €
10mg		95.00 €
25mg		183.00 €
50mg		324.00 €
100mg		537.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

TG 100801 Hydrochloride

CAS:1018069-81-2

TG 100801: prodrug for macular degeneration. TG 100572: inhibits kinases (VEGFRs, FGFRs, PDGFRβ, Src family), …

Formula:

C₃₃H₃₁Cl₂N₅O₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

616.54

Ref: TM-T13157L

25mg		1,410.00 €
50mg		1,845.00 €
100mg		2,329.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

OXSI-2

CAS:622387-85-3

OXSI-2 (Syk Inhibitor) is an inhibitor of Syk with an EC50 of 313 nM and …

Formula:

C₁₈H₁₅N₃O₃S

Purity:

98%

Color and Shape:

Dark Orange Solid

Molecular weight:

353.39

Ref: TM-T28281

1mg		136.00 €
10mg		437.00 €
500µg		86.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

TL02-59 dihydrochloride

CAS:2415263-06-6

TL02-59 dihydrochloride is an orally active inhibitor of Src-family kinase Fgr (IC50: 0.03 nM).

Formula:

C₃₂H₃₆Cl₂F₃N₅O₄

Purity:

98%

Color and Shape:

Solid

Molecular weight:

682.56

Ref: TM-T13186L

10mg		734.00 €
50mg		3,073.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

RO9021

CAS:1446790-62-0

RO9021 is an orally bioavailable, novel ATP-competitive SYK inhibitor (average IC50: 5.6 nM).

Formula:

C₁₈H₂₅N₇O

Purity:

97.19%

Color and Shape:

Solid

Molecular weight:

355.44

Ref: TM-T16776

1mg		85.00 €
5mg		184.00 €
10mg		277.00 €
25mg		459.00 €
50mg		668.00 €
100mg		909.00 €
500mg		1,813.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Pz-1

CAS:1800505-64-9

Pz-1 is an inhibitor of VEGFR2 and RET (rearranged during transfection) tyrosine kinase that blocks …

Formula:

C₂₆H₂₆N₆O₂

Purity:

99.95%

Color and Shape:

Solid

Molecular weight:

454.52

Ref: TM-T12598

1ml		58.00 €
2mg		35.00 €
5mg		52.00 €
10mg		90.00 €
25mg		184.00 €
50mg		313.00 €
100mg		453.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

TGFBR1-IN-1

CAS:2170830-26-7

TGFBR1-IN-1 is an inhibitor of ALK5 (IC50 of 10-100 nM).

Formula:

C₂₃H₁₇N₅O₂S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

427.48

Ref: TM-T13138

25mg		1,410.00 €
50mg		1,845.00 €
100mg		2,329.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

YK-2-69

CAS:2619846-89-6

YK-2-69 selectively blocks DYRK2 at Lys-231 and Lys-234, outperforming enzalutamide in prostate cancer treatment.

Formula:

C₂₅H₂₇FN₈OS

Purity:

99.57%

Color and Shape:

Solid

Molecular weight:

506.6

Ref: TM-T69564

1mg		274.00 €
5mg		673.00 €
10mg		920.00 €
25mg		1,417.00 €
50mg		1,846.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

SDZ281-977

CAS:150779-71-8

SDZ 281-977 is a derivative of Lavendustin A which is the EGF receptor tyrosine kinase …

Formula:

C₁₈H₂₀O₅

Purity:

98%

Color and Shape:

Solid

Molecular weight:

316.35

Ref: TM-T16866

1mg		97.00 €
1ml		257.00 €
5mg		231.00 €
10mg		369.00 €
25mg		739.00 €
50mg		1,146.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

FGFR2-IN-1

CAS:2677709-76-9

FGFR2-IN-1 is an FGFR inhibitor that inhibits FGFR1, FGFR2, and FGFR3, and can be used …

Formula:

C₂₂H₁₉N₃O₂

Color and Shape:

Solid

Molecular weight:

357.41

Ref: TM-T61304

1mg		60.00 €
5mg		130.00 €
10mg		198.00 €
25mg		333.00 €
50mg		495.00 €
100mg		704.00 €
500mg		1,419.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

DDR Inhibitor

CAS:1644069-80-6

DDR inhibitor is a potent discidin domain receptor (DDR) inhibitor. The IC50 of DDR2 is …

Formula:

C₂₃H₂₀FN₅O₂

Purity:

97.75%

Color and Shape:

Solid

Molecular weight:

417.44

Ref: TM-T10985

1mg		114.00 €
1ml		258.00 €
5mg		230.00 €
10mg		369.00 €
25mg		741.00 €
50mg		1,179.00 €
100mg		1,597.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

c-Fms-IN-6

CAS:1628574-81-1

c-Fms-IN-6 is a potent inhibitor of c-FMS (IC50 ≤10 nM for unphosphorylated c-FMS) and also …

Formula:

C₂₂H₂₅N₇O₂

Purity:

98%

Color and Shape:

Solid

Molecular weight:

419.48

Ref: TM-T10645

25mg		1,549.00 €
50mg		2,038.00 €
100mg		2,617.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Cenisertib

CAS:871357-89-0

Cenisertib is A potent ATP-competitive multi-kinase inhibitor, showing inhibitory effects on the activity of Aurora-kinase-A/B, …

Formula:

C₂₄H₃₀FN₇O

Molecular weight:

451.54

Ref: TM-T14925

25mg		916.00 €
50mg		1,273.00 €
100mg		1,741.00 €
1ml*10 (DMSO)		342.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Trk-IN-4

CAS:1799788-94-5

Trk-IN-4 is an effective pan-Trk inhibitor in cell-based assays (IC50s: 1.9 nM, 2.6 nM, and …

Formula:

C₂₄H₂₃F₄N₅O₄

Purity:

98%

Color and Shape:

Solid

Molecular weight:

521.46

Ref: TM-T17169

1mg		40.00 €
2mg		To inquire

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Tilfrinib

CAS:1600515-49-8

Tilfrinib is an effective and selective inhibitor of breast tumor kinase(Brk, IC50 = 3.15 nM) …

Formula:

C₁₇H₁₃N₃O

Purity:

99.73%

Color and Shape:

Solid

Molecular weight:

275.3

Ref: TM-T17098

1mg		45.00 €
1ml		87.00 €
2mg		59.00 €
5mg		96.00 €
10mg		134.00 €
25mg		250.00 €
50mg		455.00 €
100mg		665.00 €
500mg		1,374.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

Epitinib succinate

CAS:2252334-12-4

Epitinib succinate (HMPL-813 succinate) is an orally active and brain penetration EGFR tyrosine kinase inhibitor …

Formula:

C₂₈H₃₂N₆O₆

Purity:

97.43%

Color and Shape:

Solid

Molecular weight:

548.59

Ref: TM-T35914

1mg		74.00 €
2mg		95.00 €
5mg		167.00 €
10mg		266.00 €
25mg		440.00 €
50mg		602.00 €
100mg		825.00 €
500mg		1,653.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-9

CAS:1226549-39-8

EGFR-IN-9 is a potent EGFR kinase inhibitor with IC50s of 7 nM, 28 nM for …

Formula:

C₂₉H₂₄N₄O₃

Purity:

99.46%

Color and Shape:

Solid

Molecular weight:

476.53

Ref: TM-T11163

1mg		85.00 €
1ml		205.00 €
5mg		183.00 €
10mg		294.00 €
25mg		480.00 €
50mg		665.00 €
100mg		882.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

CHMFL-BTK-01

CAS:2095280-64-9

CHMFL-BTK-01 is an irreversible inhibitor of BTK (IC50: 7 nM) and also potently inhibits BTK …

Formula:

C₃₈H₄₁N₅O₅

Purity:

98%

Color and Shape:

Solid

Molecular weight:

647.76

Ref: TM-T14956

25mg		1,549.00 €
50mg		2,033.00 €
100mg		2,611.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

PKI-166

CAS:187724-61-4

PKI-166: oral EGF-R tyrosine kinase inhibitor (IC50: 0.7 nM), halts growth & spread of many …

Formula:

C₂₀H₁₈N₄O

Purity:

99.76%

Color and Shape:

Solid

Molecular weight:

330.38

Ref: TM-T16549

1mg		55.00 €
1ml		130.00 €
5mg		118.00 €
10mg		189.00 €
25mg		370.00 €
50mg		620.00 €
100mg		985.00 €
500mg		1,967.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

TG-89

CAS:936091-56-4

TG-89 is an inhibitor of JAK2, JAK3, RET and FLT3, and has an IC50 value …

Formula:

C₂₆H₃₄N₆O₃S

Purity:

98.8%

Color and Shape:

Solid

Molecular weight:

510.65

Ref: TM-T20742

1mg		60.00 €
5mg		151.00 €
10mg		232.00 €
25mg		386.00 €
50mg		549.00 €
100mg		741.00 €
500mg		1,476.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

SU16f

CAS:251356-45-3

SU16f, a 3-substituted indolin-2-one, is a selective PDGFRβ inhibitor; IC50: 10 nM (PDGFRβ), 140 nM …

Formula:

C₂₄H₂₂N₂O₃

Purity:

98%

Color and Shape:

Solid

Molecular weight:

386.44

Ref: TM-T16947

1mg		46.00 €
1ml		97.00 €
5mg		95.00 €
10mg		124.00 €
25mg		199.00 €
50mg		296.00 €
100mg		427.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

EGFR-IN-2

CAS:1643497-70-4

EGFR-IN-2 is a non-covalent, mutation-selective and irreversible second-generation EGFR inhibitor.

Formula:

C₂₆H₃₃N₉O₃S

Purity:

98%

Color and Shape:

Solid

Molecular weight:

551.66

Ref: TM-T11159

25mg		1,410.00 €
50mg		1,851.00 €
100mg		2,337.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Tafetinib

CAS:1032265-57-8

Tafetinib (SIM-010603) is a novel potent and orally available tyrosine kinase inhibitor with anti-angiogenic and …

Formula:

C₂₄H₂₉FN₄O₂

Purity:

96.66%

Color and Shape:

Solid

Molecular weight:

424.51

Ref: TM-T28911

1mg		233.00 €
5mg		581.00 €
10mg		824.00 €
25mg		1,234.00 €
50mg		1,654.00 €
100mg		2,265.00 €
500mg		4,532.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

Syk-IN-3

CAS:1312534-69-2

Syk-IN-3 is a Syk inhibitor with potential anti-inflammatory and anticancer activity and can be used …

Formula:

C₂₄H₂₈N₄O₃S

Purity:

97.99%

Color and Shape:

Solid

Molecular weight:

452.57

Ref: TM-T13045

1mg		370.00 €
5mg		913.00 €
25mg		1,410.00 €
50mg		1,862.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

+ info

OD36 hydrochloride

CAS:2387510-88-3

OD36 hydrochloride (OD-36 hydrochloride) is a potent RIPK2 inhibitor with an IC50 of 5.3 nM.OD36 …

Formula:

C₁₆H₁₆Cl₂N₄O₂

Purity:

99.85%

Color and Shape:

Solid

Molecular weight:

367.23

Ref: TM-T61424

25mg		1,197.00 €
50mg		1,561.00 €
100mg		2,320.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info

MMPP

CAS:1895957-18-2

MMPP is a VEGFR2 inhibitor with anti-inflammatory activity, inhibits STAT3 , inhibits angiogenesis, and can …

Formula:

C₁₇H₁₈O₃

Purity:

100%

Color and Shape:

Solid

Molecular weight:

270.32

Ref: TM-T28077

1mg		238.00 €
5mg		590.00 €
10mg		843.00 €
25mg		1,266.00 €
50mg		1,710.00 €

Estimated delivery in United States, on Tuesday 3 Sep 2024

+ info