Tyrosine Kinase/Adaptors
Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.
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Subcategories of "Tyrosine Kinase/Adaptors"
ALK
CSF-1R
EGFR
Ephrin Receptor
FLT
Fibroblast Growth Factor Receptor (FGFR)
HER
Hck
IGF-1R
PDGFR
PYK2
Src
TAM Receptor
Tie-2
Trk receptor
Tyrosine Kinases
VEGFR
c-Fms
c-Kit
c-Met/HGFR
c-RET
Show 13 more subcategories
Products of "Tyrosine Kinase/Adaptors"
EGFR-IN-85
CAS:1956378-29-2
EGFR-IN-85 (Compound 1), an EGFR inhibitor, exhibits potent activity with an IC50 of 0.19 μM …
Formula:
C26H30N8O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
486.57
Ref: TM-T78574
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
EGFR-IN-61
CAS:2890261-81-9
EGFR-IN-61 inhibits EGFR kinase (IC50: 42 nM L858R/T790M, 137 nM L858R/T790M/C797S, 743 nM WT) and …
Formula:
C33H37ClN8O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
629.15
Ref: TM-T73128
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
FGFR4-IN-8
CAS:2765240-52-4
FGFR4-IN-8 is a selective, ATP-competitive FGFR4 inhibitor with IC50s as low as 0.25 nM, halting …
Formula:
C32H34Cl2FN7O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
654.56
Ref: TM-T73121
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
JGK-068S
CAS:2490431-16-6
Compound I (JGK-068S) is a potent inhibitor of the epidermal growth factor receptor (EGFR) [1].
Formula:
C22H23BrFN5O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
488.35
Ref: TM-T79124
| 5mg | 1,290.00 € | ||
| 50mg | 2,618.00 € | ||
| 100mg | 3,484.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
TG 100572 Hydrochloride
CAS:867331-64-4
TG 100572 Hydrochloride is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and …
Formula:
C26H27Cl2N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
512.43
Ref: TM-T13156L
| 1mg | 370.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
FGFR3-IN-6
CAS:2833703-72-1
FGFR3-IN-6 is a potent, selective inhibitor of FGFR 3, exhibiting an IC50 value of less …
Formula:
C25H23FN8O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
486.5
Ref: TM-T82405
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Feb 2025
Methyl 12-methyltridecanoate
CAS:5129-58-8
Methyl 12-methyltridecanoate ((R)-betaxolol hydrochloride), a biosurfactant derived from Brevibacterium casei LS14, enhances the biocompatibility of
Formula:
C15H30O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
242.4
Ref: TM-T79159
| 1mg | 141.00 € | ||
| 5mg | 394.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
Labuxtinib
CAS:1426449-01-5
Labutinib is a selective inhibitor of the c-kit tyrosine kinase [1].
Formula:
C20H16FN5O2
Purity:
99.77%
Color and Shape:
Liquid
Molecular weight:
377.37
Ref: TM-T79851
| 1mg | 138.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 533.00 € | ||
| 25mg | 1,059.00 € | ||
| 50mg | 1,523.00 € | ||
| 100mg | 2,046.00 € | ||
| 200mg | 2,763.00 € | ||
| 1mL*10mM (DMSO) | 369.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
c-Fms-IN-14
CAS:1898210-99-5
c-Fms-IN-14 (Example 76) is a potent inhibitor of the c-Fms kinase with an IC50 of …
Formula:
C26H24N6O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
436.51
Ref: TM-T79815
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Feb 2025
AXL-IN-15
CAS:1954722-22-5
AXL-IN-15 (cpd391) is a potent inhibitor of Axl, exhibiting both a dissociation constant (K i) …
Formula:
C26H32F3N9O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
575.59
Ref: TM-T79045
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Feb 2025
Vepafestinib
CAS:2129515-96-2
Vepafestinib is a RET inhibitor with potential antineoplastic activity[1].
Formula:
C26H30N6O3
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
474.55
Ref: TM-T9445
| 1mg | 127.00 € | ||
| 5mg | 305.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
UniPR1447
CAS:1809170-68-0
UniPR1447 is a dual antagonist for both EphA2 and EphB2 receptors, exhibiting an IC50 value …
Formula:
C36H50N2O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
574.79
Ref: TM-T80897
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Feb 2025
Zongertinib
CAS:2728667-27-2
Zongertinib is a human HER2-selective tyrosine kinase inhibitor, a novel TK that is highly selective …
Formula:
C29H29N9O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
535.6
Ref: TM-T69534
| 1mg | 143.00 € | ||
| 5mg | 347.00 € | ||
| 10mg | 464.00 € | ||
| 25mg | 696.00 € | ||
| 50mg | 906.00 € | ||
| 100mg | 1,149.00 € | ||
| 200mg | 1,560.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
TAK-020
CAS:1627603-21-7
TAK-020 is a potent covalent inhibitor of Btk with potential antitumor activity for the study …
Formula:
C18H17N5O3
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
351.36
Ref: TM-T9529
| 1mg | 143.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 616.00 € | ||
| 25mg | 1,277.00 € | ||
| 50mg | 1,977.00 € | ||
| 100mg | 3,044.00 € | ||
| 1mL*10mM (DMSO) | 375.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
UniPR505
CAS:2938227-14-4
UniPR505 is a potent EphA2 antagonist (IC50: 0.95 µM), a novel 3α-carbamoyloxy derivative with antiangiogenic …
Formula:
C39H57N3O5
Purity:
99.23%
Color and Shape:
Liquid
Molecular weight:
647.89
Ref: TM-T73368
| 1mg | 493.00 € | ||
| 5mg | 1,087.00 € | ||
| 25mg | 1,825.00 € | ||
| 50mg | 2,209.00 € | ||
| 100mg | 2,890.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
BEBT-109
CAS:2050906-40-4
BEBT-109 is a potent selective inhibitor of pan-mutant EGFR with enhanced pharmacokinetic properties, suitable for …
Formula:
C27H32N8O3
Purity:
99.01%
Color and Shape:
Liquid
Molecular weight:
516.59
Ref: TM-T80643
| 1mg | 187.00 € | ||
| 5mg | 462.00 € | ||
| 10mg | 662.00 € | ||
| 25mg | 1,033.00 € | ||
| 50mg | 1,425.00 € | ||
| 100mg | 1,885.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
EGFR-IN-1 hydrochloride
CAS:2227455-78-7
EGFR-IN-1 HCl targets L858R/T790M EGFR mutants over wild-type; IC50: 4 nM in H1975, 28 nM …
Formula:
C28H31ClN6O4
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
551.04
Ref: TM-T11157L
| 1mg | 95.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 737.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,033.00 € | ||
| 1mL*10mM (DMSO) | 335.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
MK-2461
CAS:917879-39-1
MK-2461 is a novel inhibitor that targets multiple proteins and competitively binds to ATP sites, …
Formula:
C24H25N5O5S
Purity:
95.41% - 99.53%
Color and Shape:
Solid
Molecular weight:
495.55
Ref: TM-T6094
| 1mg | 52.00 € | ||
| 5mg | 117.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 350.00 € | ||
| 50mg | 533.00 € | ||
| 100mg | 811.00 € | ||
| 200mg | 1,115.00 € | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
BTK-IN-25
CAS:2562351-92-0
BTK-IN-25 (compound 71) is a potent BTK inhibitor, demonstrating an IC50 of 0.77 nM against …
Formula:
C28H27F2N3O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
523.53
Ref: TM-T79113
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Feb 2025
EGFR/ErbB-2 inhibitor-1
CAS:1135150-79-6
EGFR/ErbB-2 inhibitor-1 is a selective ErbB2/HER2 inhibitor that effectively blocks ErbB2 and HER2 signaling.
Formula:
C23H15ClFN3OS2
Purity:
97.55%
Color and Shape:
Liquid
Molecular weight:
467.97
Ref: TM-T79861
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,004.00 € | ||
| 50mg | 1,385.00 € | ||
| 100mg | 1,831.00 € | ||
| 500mg | 3,652.00 € |
Estimated delivery in United States, on Wednesday 12 Feb 2025
