Fibroblast Growth Factor Receptor (FGFR)
FGFR inhibitors are targeted therapies that block the activity of fibroblast growth factor receptors (FGFRs), which are involved in cell proliferation, differentiation, and angiogenesis. FGFR signaling contributes to the formation of new blood vessels in tumors, promoting their growth and survival. Inhibiting FGFR can therefore reduce angiogenesis and tumor progression. At CymitQuimica, we provide a range of high-quality FGFR inhibitors to support your research in cancer, developmental biology, and angiogenesis.
Read more
FIIN-3
CAS:1637735-84-2
FIIN-3 is an irreversible inhibitor of FGFR.
Formula:
C34H36Cl2N8O4
Purity:
97.63% - 98.92%
Color and Shape:
Solid
Molecular weight:
691.61
Ref: TM-T3466
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 513.00 € | ||
| 200mg | 699.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Ponatinib
CAS:943319-70-8
Ponatinib (AP24534) is an orally available, multitargeted kinase inhibitor (IC50s: 0.37/1.1/1.5/2.2/5.4 nM for Abl, PDGFRα, …
Formula:
C29H27F3N6O
Purity:
98% - 99.74%
Color and Shape:
Solid
Molecular weight:
532.56
Ref: TM-T2372
| 10mg | 54.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 136.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
S49076
CAS:1265965-22-7
S49076 is a novel, potent inhibitor of MET, AXL/MER, and FGFR1/2/3, blocking cellular phosphorylation of …
Formula:
C22H22N4O4S
Purity:
95.35% - 97.4%
Color and Shape:
Solid
Molecular weight:
438.5
Ref: TM-T3274
| 1mg | 46.00 € | ||
| 2mg | 62.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 549.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Regorafenib
CAS:755037-03-7
Regorafenib (BAY 73-4506) is a multi-targeted receptor tyrosine kinase inhibitor that inhibits RET, C-RAF, VEGFR2, …
Formula:
C21H15ClF4N4O3
Purity:
98% - 99.95%
Color and Shape:
Solid
Molecular weight:
482.82
Ref: TM-T1792
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 142.00 € | ||
| 200mg | 181.00 € | ||
| 500mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
PD168393
CAS:194423-15-9
PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, …
Formula:
C17H13BrN4O
Purity:
99.13% - 99.7%
Color and Shape:
Solid
Molecular weight:
369.22
Ref: TM-T6932
| 1mg | 39.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Lenvatinib mesylate
CAS:857890-39-2
Lenvatinib mesylate (E7080 (mesylate)) is an oral and multi-targeted inhibitor of VEGFR1-3, FGFR1-4, PDGFR, KIT, …
Formula:
C22H23ClN4O7S
Purity:
99.03% - 99.79%
Color and Shape:
Solid
Molecular weight:
522.96
Ref: TM-T8541
| 10mg | 40.00 € | ||
| 25mg | 59.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 162.00 € | ||
| 500mg | 263.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
SSR128129E
CAS:848318-25-2
SSR128129E (SSR) is an allosteric and orally-active FGFR1 inhibitor (IC50: 1.9 μM), but not affecting …
Formula:
C18H15N2O4·Na
Purity:
98.79% - ≥95%
Color and Shape:
Solid
Molecular weight:
346.31
Ref: TM-T6082
| 2mg | 40.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 275.00 € | ||
| 100mg | 432.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
H3B-6527
CAS:1702259-66-2
H3B-6527 Is a Potent and Selective Inhibitor of FGFR4 in FGF19-Driven Hepatocellular Carcinoma, with antineoplastic …
Formula:
C29H34Cl2N8O4
Purity:
97.45%
Color and Shape:
Solid
Molecular weight:
629.54
Ref: TM-T7738
| 1mg | 69.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 268.00 € | ||
| 25mg | 518.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,040.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Futibatinib
CAS:1448169-71-8
Futibatinib (TAS-120) is an orally active, potent,and irreversible FGFR inhibitor of FGFR1, FGFR2, FGFR3, and …
Formula:
C22H22N6O3
Purity:
97.66% - 99.14%
Color and Shape:
Solid
Molecular weight:
418.45
Ref: TM-T5044
| 1mg | 52.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 168.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 503.00 € | ||
| 100mg | 650.00 € | ||
| 200mg | 927.00 € | ||
| 1mL*10mM (DMSO) | 133.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Dovitinib lactate hydrate
CAS:915769-50-5
Dovitinib lactate hydrate (TKI258) is the Lactate of Dovitinib, which is a multitargeted RTK inhibitor, …
Formula:
C24H27FN6O4
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
482.51
Ref: TM-T6479
| 5mg | 54.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 378.00 € | ||
| 200mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Fisogatinib
CAS:1707289-21-1
Fisogatinib (BLU-554) is a highly potent, selective, and orally active FGFR4 inhibitor.Cost-effective and quality-assured.
Formula:
C24H24Cl2N4O4
Purity:
99.27% - ≥95%
Color and Shape:
Solid
Molecular weight:
503.38
Ref: TM-T3456
| 1mg | 52.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 175.00 € | ||
| 25mg | 307.00 € | ||
| 50mg | 463.00 € | ||
| 100mg | 699.00 € | ||
| 500mg | 1,397.00 € | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Masitinib mesylate
CAS:1048007-93-7
Masitinib mesylate (AB-1010 mesylate) is a selective and orally bioavailable c-Kit inhibitor (IC50 of 200 …
Formula:
C29H34N6O4S2
Purity:
100% - 99.92%
Color and Shape:
Solid
Molecular weight:
594.75
Ref: TM-T8544
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 75.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 220.00 € | ||
| 500mg | 364.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Ferulic acid sodium
CAS:24276-84-4
Ferulic acid sodium (Sodium ferulic) is an agent used in the treatment of cardiovascular and …
Formula:
C10H9NaO4
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
216.16
Ref: TM-T2S0007
| 1g | 60.00 € | ||
| 100mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
S49076 HCl
CAS:1265966-31-1
S49076 HCl (S-49076 Hydrochloride) is an effective inhibitor of MET, AXL/MER, and FGFR1/2/3.
Formula:
C22H18ClN3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
439.85
Ref: TM-T3512
| 5mg | 115.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 288.00 € | ||
| 50mg | 456.00 € | ||
| 100mg | 826.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
ON123300
CAS:1357470-29-1
ON123300 is a potent and multi-targeted kinase inhibitor for CDK4/Ark5/PDGFRβ/FGFR1/RET/Fyn (IC50: 3.9/5/26/26/9.2/11 nM).
Formula:
C24H27N7O
Purity:
99.22% - 99.53%
Color and Shape:
Solid
Molecular weight:
429.52
Ref: TM-T6920
| 1mg | 46.00 € | ||
| 2mg | 61.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 146.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 437.00 € | ||
| 100mg | 635.00 € | ||
| 500mg | 1,291.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
R1530
CAS:882531-87-5
R1530 is a multikinase inhibitor with antineoplastic and antiangiogenesis activities.
Formula:
C18H14ClFN4O
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
356.78
Ref: TM-TQ0317
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 552.00 € | ||
| 100mg | 796.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Alofanib
CAS:1612888-66-0
Alofanib (RPT835) selectively inhibits FGFR2 in KATO III cells with IC50 <10 nM; doesn’t affect …
Formula:
C19H15N3O6S
Purity:
98.82% - 99.06%
Color and Shape:
Solid
Molecular weight:
413.4
Ref: TM-T5122
| 1mg | 37.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 463.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
XL 999
CAS:705946-27-6
Tyrosine kinase-IN-1 is a multi-targeted tyrosine kinase inhibitor(KDR, Flt-1, FGFR1 and PDGFRα with IC50s of …
Formula:
C26H28FN5O
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
445.53
Ref: TM-T5466
| 1mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 398.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
PD-166866
CAS:192705-79-6
PD-166866 is a selective FGFR tyrosine kinase inhibitor.
Formula:
C20H24N6O3
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
396.44
Ref: TM-T3492
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 448.00 € | ||
| 1mL*10mM (DMSO) | 61.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Derazantinib
CAS:1234356-69-4
Derazantinib (ARQ-087) is a potent, ATP-competitive, orally active tyrosine kinase inhibitor.Cost-effective and quality-assured.
Formula:
C29H29FN4O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
468.57
Ref: TM-TQ0228
| 1mg | 52.00 € | ||
| 5mg | 115.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 397.00 € | ||
| 100mg | 590.00 € | ||
| 200mg | 840.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
