Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 358 products of "Histamine Receptor"
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Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Formula:C21H28N2O2Purity:99.53%Color and Shape:White Or Similar To White PowderMolecular weight:340.46JNJ-5207852 dihydrochloride
CAS:<p>JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor</p>Formula:C20H34Cl2N2OPurity:99.51%Color and Shape:SolidMolecular weight:389.4Bepotastine Besilate
CAS:<p>Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).</p>Formula:C21H25ClN2O3·C6H6O3SPurity:99.83% - 99.9%Color and Shape:Brown Viscous LiquidMolecular weight:547.062-Pyridylethylamine dihydrochloride
CAS:<p>2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.</p>Formula:C7H12Cl2N2Purity:99.42%Color and Shape:SolidMolecular weight:195.09Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Formula:C16H14O2Purity:98.15%Color and Shape:SolidMolecular weight:238.2812Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Formula:C9H7N5O3Purity:98.25%Color and Shape:SolidMolecular weight:233.18BMY-25368
CAS:<p>BMY-25368 is a long-acting antagonist of the H2-receptor.</p>Formula:C19H25N3O3Color and Shape:SolidMolecular weight:343.42Alcaftadine
CAS:<p>Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.</p>Formula:C19H21N3OPurity:98% - 98.65%Color and Shape:SolidMolecular weight:307.39Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Formula:C15H19Cl2N3O3SPurity:98.48%Color and Shape:SolidMolecular weight:392.3Tribenoside
CAS:<p>Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.</p>Formula:C29H34O6Purity:≥98%Color and Shape:LiquidMolecular weight:478.58Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Formula:C19H20ClN3Purity:98% - 99.65%Color and Shape:SolidMolecular weight:325.84Mebhydrolin
CAS:<p>Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.</p>Formula:C19H20N2Purity:99.3% - ≥98%Color and Shape:SolidMolecular weight:276.38Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Formula:C18H24ClN3O2Color and Shape:SolidMolecular weight:349.86Pitolisant hydrochloride
CAS:<p>Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).</p>Formula:C17H27Cl2NOPurity:99.72% - 99.91%Color and Shape:SolidMolecular weight:332.31Bromodiphenhydramine hydrochloride
CAS:<p>Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.</p>Formula:C17H21BrClNOPurity:97.29%Color and Shape:SolidMolecular weight:370.71VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Formula:C15H19N5Purity:99.44% - 99.57%Color and Shape:SolidMolecular weight:269.34Chlorphenoxamine
CAS:<p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>Formula:C18H22ClNOPurity:99.44% - 99.85%Color and Shape:SolidMolecular weight:303.83Dimaprit dihydrochloride
CAS:<p>Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.</p>Formula:C6H15N3S·2HClPurity:99.79%Color and Shape:SolidMolecular weight:234.19Epinastine
CAS:<p>Epinastine (WAL801) is an antihistamine, mast cell stabilizer, and H1 antagonist with anti-allergic properties.</p>Formula:C16H15N3Purity:99.94%Color and Shape:SolidMolecular weight:249.31
