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Histamine Receptor

Histamine Receptor

Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.

Found 385 products of "Histamine Receptor"

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  • Hydroxyzine D8

    CAS:
    Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.
    Formula:C21H27ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.95
  • Tiotidine

    CAS:
    Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).
    Formula:C10H16N8S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.42
  • WZ4141

    CAS:
    WZ4141 is an intermediate in compound synthesis.
    Formula:C16H13N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.29
  • Diphenylpyraline

    CAS:
    Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.
    Formula:C19H23NO
    Color and Shape:Solid
    Molecular weight:281.39
  • Cetirizine D8

    CAS:
    Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
    Formula:C21H25ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.94
  • Hydroxyzine dihydrochloride-d4

    CAS:
    Hydroxyzine dihydrochloride-d4 is a deuterated compound of Hydroxyzine dihydrochloride.
    Formula:C21H25D4Cl3N2O2
    Color and Shape:Solid
    Molecular weight:451.85
  • Cetirizine D4

    CAS:
    Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
    Formula:C21H25ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.91
  • 1-Methyl-4-imidazoleacetic Acid (hydrochloride)

    CAS:
    MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.
    Formula:C6H9ClN2O2
    Color and Shape:Solid
    Molecular weight:176.601
  • Acrivastine D7

    CAS:
    Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.
    Formula:C22H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.48
  • Doxepin D3 Hydrochloride

    CAS:
    Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and
    Formula:C19H22ClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.86
  • Fexofenadine-d6

    CAS:
    Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.
    Formula:C32H39NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:507.69
  • Emedastine Difumarate

    CAS:
    Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.
    Formula:C25H34N4O9
    Color and Shape:Solid
    Molecular weight:534.56
  • Gizzerosine

    CAS:
    Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.
    Formula:C11H20N4O2
    Color and Shape:Solid
    Molecular weight:240.3
  • Emedastine

    CAS:
    <p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>
    Formula:C17H26N4O
    Purity:97.1% - 97.76%
    Color and Shape:Oil
    Molecular weight:302.41
  • Fexofenadine hydrochloride

    CAS:
    Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,
    Formula:C32H39NO4·HCl
    Purity:99.39% - ≥95%
    Color and Shape:Solid
    Molecular weight:538.13
  • Conessine

    CAS:
    <p>Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.</p>
    Formula:C24H40N2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:356.59
  • Chlorpheniramine

    CAS:
    Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.
    Formula:C16H19ClN2
    Color and Shape:Solid
    Molecular weight:274.79
  • VUF10460

    CAS:
    VUF10460 is a non-imidazole histamine H4 receptor agonist.
    Formula:C15H19N5
    Purity:99.44% - 99.57%
    Color and Shape:Solid
    Molecular weight:269.34
  • Hydroxyzine

    CAS:
    Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
    Formula:C21H27ClN2O2
    Purity:99.54% - ≥95%
    Color and Shape:Oil Solid
    Molecular weight:374.9
  • Dimaprit dihydrochloride

    CAS:
    Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.
    Formula:C6H15N3S·2HCl
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:234.19