Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Read more
Trimebutine
CAS:39133-31-8
Trimebutine (Mebutin) is a spasmolytic agent that regulates intestinal and colonic motility and relieves abdominal …
Formula:
C22H29NO5
Purity:
98.13% - 99.49%
Color and Shape:
Solid
Molecular weight:
387.47
Ref: TM-T0918
| 1g | 36.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Trimebutine maleate
CAS:34140-59-5
Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.
Formula:
C26H33NO9
Purity:
99.76% - 99.88%
Color and Shape:
White Solid
Molecular weight:
503.55
Ref: TM-T1197
| 1g | 38.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Docusate sodium
CAS:577-11-7
Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to …
Formula:
C20H37NaO7S
Purity:
99.77%
Color and Shape:
White Wax-Like Solid With Water (Uscg 1999)
Molecular weight:
444.56
Ref: TM-T0929
| 50mg | 42.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 81.00 € | ||
| 500mg | 120.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
BTRX-335140
CAS:2244614-14-8
BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic …
Formula:
C25H32FN5O2
Purity:
98% - 98.45%
Color and Shape:
Solid
Molecular weight:
453.55
Ref: TM-T14835
| 1mg | 105.00 € | ||
| 2mg | 154.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 404.00 € | ||
| 25mg | 835.00 € | ||
| 50mg | 1,368.00 € | ||
| 100mg | 1,867.00 € | ||
| 200mg | 2,612.00 € | ||
| 1mL*10mM (DMSO) | 281.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Loperamide hydrochloride
CAS:34552-83-5
Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
Formula:
C29H34Cl2N2O2
Purity:
100% - 99.78%
Color and Shape:
Crystals Practically Insoluble In Water
Molecular weight:
513.498
Ref: TM-T0209
| 100mg | 59.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Naltrexone hydrochloride
CAS:16676-29-2
Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse …
Formula:
C20H24ClNO4
Purity:
100% - 99%
Color and Shape:
White Crystalline Powder
Molecular weight:
377.862
Ref: TM-T0963
| 100mg | 54.00 € | ||
| 200mg | 68.00 € | ||
| 500mg | 110.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Sinomenine hydrochloride
CAS:6080-33-7
Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.
Formula:
C19H24ClNO4
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
365.851
Ref: TM-T2921
| 50mg | 44.00 € | ||
| 100mg | 56.00 € | ||
| 200mg | 72.00 € | ||
| 500mg | 103.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
ZT 52656A hydrochloride
CAS:115730-24-0
ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or …
Formula:
C19H26ClF3N2O
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
390.87
Ref: TM-T13414
| 1mg | 528.00 € | ||
| 5mg | 1,169.00 € | ||
| 10mg | 1,744.00 € | ||
| 25mg | 2,959.00 € | ||
| 50mg | 3,831.00 € | ||
| 100mg | 5,000.00 € | ||
| 1mL*10mM (DMSO) | 1,253.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Alvimopan
CAS:156053-89-3
Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.
Formula:
C25H32N2O4
Purity:
99.78% - 99.97%
Color and Shape:
Solid
Molecular weight:
424.53
Ref: TM-T1242
| 1mg | 49.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 552.00 € | ||
| 500mg | 1,189.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
LY2940094
CAS:1307245-86-8
LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
Formula:
C22H23ClF2N4O2S
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
480.96
Ref: TM-T15799
| 1mg | 80.00 € | ||
| 2mg | 105.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 270.00 € | ||
| 25mg | 533.00 € | ||
| 50mg | 764.00 € | ||
| 100mg | 1,054.00 € | ||
| 1mL*10mM (DMSO) | 179.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Meptazinol hydrochloride
CAS:59263-76-2
Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic …
Formula:
C15H23NO·HCl
Purity:
99.83%
Color and Shape:
White Solid
Molecular weight:
269.81
Ref: TM-T0201
| 5mg | 48.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 166.00 € | ||
| 200mg | 222.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Matrine
CAS:519-02-8
Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor …
Formula:
C15H24N2O
Purity:
100% - 97.16%
Color and Shape:
Solid
Molecular weight:
248.36
Ref: TM-T2870
| 25mg | 42.00 € | ||
| 50mg | 57.00 € | ||
| 100mg | 80.00 € | ||
| 200mg | 115.00 € | ||
| 500mg | 245.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
6'-GNTI dihydrochloride
CAS:2410327-94-3
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over …
Formula:
C27H29N5O3·2ClH
Purity:
99.08%
Color and Shape:
Liquid
Molecular weight:
544.47
Ref: TM-T39988
| 1mg | 325.00 € | ||
| 5mg | 788.00 € | ||
| 10mg | 1,082.00 € | ||
| 25mg | 1,606.00 € | ||
| 50mg | 2,164.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Valorphin
CAS:144313-54-2
Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 …
Formula:
C44H61N9O11
Purity:
98%
Color and Shape:
Solid
Molecular weight:
892.01
Ref: TM-T7306
| 2mg | 79.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 438.00 € | ||
| 100mg | 656.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist …
Formula:
C37H47Cl2N5O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
680.71
Ref: TM-T79547
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
Adrenorphin
CAS:88377-68-8
Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C44H69N15O9S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
984.18
Ref: TM-T7567
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
Apitegromab
CAS:2278276-46-1
Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be …
Purity:
95%
Color and Shape:
Liquid
Ref: TM-T77445
| 1mg | 207.00 € | ||
| 5mg | 608.00 € | ||
| 10mg | 917.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Nociceptin (1-13), amide
CAS:178064-02-3
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 …
Formula:
C61H100N22O15
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1381.59
Ref: TM-TP1793
| 5mg | 98.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 323.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
SNC 80
CAS:156727-74-1
SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 …
Formula:
C28H39N3O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
449.63
Ref: TM-T8414
| 1mg | 41.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 389.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BPR1M97
CAS:2059904-66-2
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain …
Formula:
C18H18Cl2N2O
Purity:
98.13% - 99.15%
Color and Shape:
Solid
Molecular weight:
349.25
Ref: TM-T10593
| 1mg | 94.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 647.00 € | ||
| 50mg | 1,014.00 € | ||
| 100mg | 1,423.00 € | ||
| 500mg | 2,762.00 € | ||
| 1mL*10mM (DMSO) | 215.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
