
Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 242 products of "Adenosine Receptor"
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CGS 15943
CAS:<p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>Formula:C13H8ClN5OPurity:97.4%Color and Shape:SolidMolecular weight:285.69Pentoxifylline
CAS:<p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>Formula:C13H18N4O3Purity:99.26% - 99.93%Color and Shape:SolidMolecular weight:278.31Acefylline
CAS:<p>Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.</p>Formula:C9H10N4O4Purity:99.57%Color and Shape:White Crystalline SolidMolecular weight:238.2AB928
CAS:<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Formula:C23H22N8OPurity:98.09% - >99.99%Color and Shape:SolidMolecular weight:426.47N6-Ethyladenosine
CAS:<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Formula:C12H17N5O4Purity:99.96%Color and Shape:SolidMolecular weight:295.29DPTN dihydrochloride
CAS:<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Formula:C22H20Cl2N4OSPurity:99.95%Color and Shape:SoildMolecular weight:459.39Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Formula:C24H29ClF3N5O5SPurity:96.56%Color and Shape:SoildMolecular weight:592.03Theophylline
CAS:<p>Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central</p>Formula:C7H8N4O2Purity:99.65% - 99.98%Color and Shape:White Solid PowderMolecular weight:180.16YT 146
CAS:<p>YT 146 is a biochemical.</p>Formula:C18H25N5O4Purity:98.81% - 99.25%Color and Shape:SolidMolecular weight:375.42Diphylline
CAS:<p>Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.</p>Formula:C10H14N4O4Purity:98.54%Color and Shape:Crystals From Alcohol SolidMolecular weight:254.24Adenosine A1 receptor activator T62
CAS:<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Formula:C15H14ClNOSPurity:97.83%Color and Shape:SolidMolecular weight:291.8Adenosine 5'-monophosphate monohydrate
CAS:<p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>Formula:C10H14N5O7P·H2OPurity:97.68% - 98.49%Color and Shape:White PowderMolecular weight:365.24Theophylline monohydrate
CAS:<p>Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium</p>Formula:C7H8N4O2·H2OPurity:99.78%Color and Shape:SolidMolecular weight:198.18Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formula:C14H15Cl2NSPurity:99.85% - >99.99%Color and Shape:White PowderMolecular weight:300.25Aminophylline
CAS:<p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>Formula:C7H8O2·C2H8N2Purity:99.31%Color and Shape:White Or Slightly Yellowish Granules Or Powder SolidMolecular weight:420.43Quercetin-3'-o-phosphate TEA
<p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>Formula:C21H26NO10PPurity:95.63%Color and Shape:SoildMolecular weight:483.41Pamabrom
CAS:<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Formula:C11H18BrN5O3Purity:99.84% - >99.99%Color and Shape:CoaMolecular weight:348.2Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formula:C11H14N4O4Purity:99.958% - >99.99%Color and Shape:SolidMolecular weight:266.25N6-Cyclohexyladenosine
CAS:<p>N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.</p>Formula:C16H23N5O4Purity:99.84% - 99.98%Color and Shape:SolidMolecular weight:349.38Adenosine receptor antagonist 1
CAS:<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Formula:C22H15ClFN7OColor and Shape:SolidMolecular weight:447.86Theophyllol
CAS:<p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>Formula:C9H10N4Na2O4Color and Shape:SolidMolecular weight:284.183F6-9G5
<p>3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.</p>Purity:>95%Color and Shape:Odour LiquidHeterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Formula:C86H115FN16O21Color and Shape:SolidMolecular weight:1727.93PSB 0777 ammonium salt
CAS:<p>adenosine A2A receptor full agonist</p>Formula:C18H24N6O7S2Purity:98%Color and Shape:SolidMolecular weight:500.55AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Formula:C21H25N5Color and Shape:SolidMolecular weight:347.211MRS-1706
CAS:<p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>Formula:C27H29N5O5Purity:99.00%Color and Shape:SolidMolecular weight:503.55A2A/A3 AR antagonist-1
<p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).</p>Formula:C56H71N15O12S2Color and Shape:SolidMolecular weight:1210.39Norisoboldine hydrochloride
CAS:<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Formula:C18H20ClNO4Color and Shape:SolidMolecular weight:349.81A3AR agonist 2
<p>Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.</p>Formula:C34H34N6O6Purity:98%Color and Shape:SolidMolecular weight:622.67LUF7690
CAS:<p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>Formula:C25H24FN5O6SColor and Shape:SolidMolecular weight:541.55Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Formula:C25H31F3N6O8Purity:98.08%Color and Shape:SoildMolecular weight:600.55Xanthine amine congener dihydrochloride
CAS:<p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>Formula:C21H30Cl2N6O4Color and Shape:SolidMolecular weight:501.41FSCPX
CAS:<p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>Formula:C23H27FN4O6SPurity:98%Color and Shape:SolidMolecular weight:506.55ABT-702
CAS:<p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>Formula:C22H19BrN6OPurity:99.57%Color and Shape:SoildMolecular weight:463.33PSB 0777 ammonium hydrate
<p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>Formula:C18H20N5O7S2·NH4·75H2OPurity:98%Color and Shape:SolidMolecular weight:532.09Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Formula:C12H14ClN5O2SeColor and Shape:SolidMolecular weight:374.68A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Formula:C23H25IN4Color and Shape:SolidMolecular weight:484.38hA3AR agonist 2
<p>hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.</p>Formula:C11H14ClN5O2SColor and Shape:SolidMolecular weight:315.78N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:<p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.428-Chloro caffeine
CAS:<p>8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.</p>Formula:C8H9ClN4O2Color and Shape:SolidMolecular weight:228.64GW-328267
CAS:<p>GW-328267 is an agonist of the adenosine A2 receptor.</p>Formula:C21H26N10O4Color and Shape:SolidMolecular weight:482.5Xanthine amine congener trihydrochloride
CAS:<p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>Formula:C21H29ClN6O4Purity:98.81%Color and Shape:SolidMolecular weight:464.95A3AR agonist 1
<p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>Formula:C28H34N6O6Purity:98%Color and Shape:SolidMolecular weight:550.61Danshenol B
<p>Danshenol B is a natural product that can be used as a reference standard.</p>Formula:C22H26O4Color and Shape:SolidMolecular weight:354.446A-286501
CAS:<p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>Formula:C11H14BrN5O2Purity:98%Color and Shape:SolidMolecular weight:328.17LUF6096
CAS:<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Formula:C22H21Cl2N3OPurity:99.5%Color and Shape:SolidMolecular weight:414.33LAS101057
CAS:<p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>Formula:C18H14FN5OPurity:99.03% - >99.99%Color and Shape:SolidMolecular weight:335.34GR79236
CAS:<p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>Formula:C15H21N5O5Color and Shape:SolidMolecular weight:351.36MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formula:C17H19N5OC2H2O4Purity:97.10%Color and Shape:SolidMolecular weight:354.39(Rac)-Mirabegron-d5
CAS:<p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>Formula:C21H24N4O2SPurity:98%Color and Shape:SolidMolecular weight:401.54CCPA
CAS:<p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>Formula:C15H20ClN5O4Purity:99.1%Color and Shape:Off-White To Light Yellow SolidMolecular weight:369.8A2B receptor antagonist 2
CAS:<p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>Formula:C12H15N5Purity:100%Color and Shape:SolidMolecular weight:229.28CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43Regadenoson hydrate
CAS:<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Formula:C15H20N8O6Purity:98%Color and Shape:SolidMolecular weight:408.37Tecadenoson
CAS:<p>Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.</p>Formula:C14H19N5O5Purity:98.83%Color and Shape:SolidMolecular weight:337.33Derenofylline
CAS:<p>Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)</p>Formula:C18H20N4OPurity:98.09%Color and Shape:SolidMolecular weight:308.385-Iodotubercidin
CAS:<p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>Formula:C11H13IN4O4Purity:99.98%Color and Shape:Tan SolidMolecular weight:392.15DPCPX
CAS:<p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>Formula:C16H24N4O2Purity:99.23% - 99.93%Color and Shape:White SolidMolecular weight:304.39Proxyphylline
CAS:<p>Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.</p>Formula:C10H14N4O3Purity:99.48%Color and Shape:SolidMolecular weight:238.24ABT-702 dihydrochloride
CAS:<p>ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.</p>Formula:C22H21BrCl2N6OPurity:98.42% - 98.98%Color and Shape:SolidMolecular weight:536.25ZM241385
CAS:<p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>Formula:C16H15N7O2Purity:97.02% - 99.69%Color and Shape:SolidMolecular weight:337.34N6,N6-Dimethyladenosine
CAS:<p>N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.</p>Formula:C12H17N5O4Purity:98.79%Color and Shape:White PowderMolecular weight:295.29CGS 21680 Hydrochloride
CAS:<p>CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.</p>Formula:C23H29N7O6·HClPurity:96.74% - 99.53%Color and Shape:SolidMolecular weight:535.98Piclidenoson
CAS:<p>Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.</p>Formula:C18H19IN6O4Purity:99.83% - ≥95%Color and Shape:SolidMolecular weight:510.29Swertisin
CAS:<p>Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.</p>Formula:C22H22O10Purity:99.74% - 99.89%Color and Shape:SolidMolecular weight:446.42-Chloroadenosine
CAS:<p>2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively</p>Formula:C10H12ClN5O4Purity:99.23%Color and Shape:White PowderMolecular weight:301.69VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Formula:C18H12F3NOSPurity:99.78%Color and Shape:SolidMolecular weight:347.35BAY-545
CAS:<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.451-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Formula:C6H9N3O2Purity:99.29%Color and Shape:SolidMolecular weight:155.15Regadenoson
CAS:<p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>Formula:C15H18N8O5Purity:99.57% - 99.81%Color and Shape:Off-White SolidMolecular weight:390.355'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Formula:C12H16N6O4Purity:98.95% - ≥95%Color and Shape:PowderMolecular weight:308.29Namodenoson
CAS:<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.73Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12CHEMBL241987
CAS:<p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>Formula:C16H11N3OPurity:99.81%Color and Shape:SolidMolecular weight:261.28Xanthine amine congener hydrochloride
CAS:<p>Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.</p>Formula:C21H29ClN6O4Color and Shape:SolidMolecular weight:464.95Vipadenant
CAS:<p>Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).</p>Formula:C16H15N7OPurity:97.25% - 97.36%Color and Shape:SolidMolecular weight:321.34Fostamatinib
CAS:<p>Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.</p>Formula:C23H26FN6O9PPurity:93.08% - 99.38%Color and Shape:SolidMolecular weight:580.46MIPS521
CAS:<p>MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.</p>Formula:C19H10ClF6NOSPurity:99.76%Color and Shape:SolidMolecular weight:449.88-Cyclopentyl-1,3-dimethylxanthine
CAS:<p>8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.</p>Formula:C12H16N4O2Purity:98.58% - >99.99%Color and Shape:SolidMolecular weight:248.28Adenosine receptor antagonist 4
CAS:<p>Adenosine receptor antagonist 4 is an adenosine receptor antagonist.</p>Formula:C10H13N3Purity:99.63% - 99.65%Color and Shape:Off-White PowderMolecular weight:175.23Inosine
CAS:<p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>Formula:C10H12N4O5Purity:99.51% - 99.89%Color and Shape:SolidMolecular weight:268.23Binodenoson
CAS:<p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>Formula:C17H25N7O4Purity:99.74%Color and Shape:SolidMolecular weight:391.42PD 117519
CAS:<p>PD 117519 (CI947) is an agonist of adenosine receptor</p>Formula:C19H21N5O4Purity:99.98%Color and Shape:SolidMolecular weight:383.4Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Formula:C25H29N9O3Purity:98.02% - 99.68%Color and Shape:SolidMolecular weight:503.56Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Adenosine amine congener
CAS:<p>Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.</p>Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6Alloxazine
CAS:<p>Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.</p>Formula:C10H6N4O2Purity:99.75%Color and Shape:SolidMolecular weight:214.18SDZ WAG 994
CAS:<p>SDZ WAG 994 is an A1 adenosine receptor agonist.</p>Formula:C17H25N5O4Purity:99.82%Color and Shape:SolidMolecular weight:363.41Istradefylline
CAS:<p>Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.</p>Formula:C20H24N4O4Purity:98.18% - 99.95%Color and Shape:SolidMolecular weight:384.43Norisoboldine
CAS:<p>Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.</p>Formula:C18H19NO4Purity:98.12% - 99.7%Color and Shape:SolidMolecular weight:313.35SCH442416
CAS:<p>SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).</p>Formula:C20H19N7O2Purity:99.58%Color and Shape:SolidMolecular weight:389.41Tozadenant
CAS:<p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>Formula:C19H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:406.5SCH 58261
CAS:<p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Enprofylline
CAS:<p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Capadenoson
CAS:<p>Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.</p>Formula:C25H18ClN5O2S2Purity:98.85% - 99.57%Color and Shape:SolidMolecular weight:520.03Reversine
CAS:<p>Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).</p>Formula:C21H27N7OPurity:98% - 98.42%Color and Shape:SolidMolecular weight:393.49AZD4635
CAS:<p>AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).</p>Formula:C15H11ClFN5Purity:99.15% - 99.90%Color and Shape:SolidMolecular weight:315.735'-Amino-5'-deoxyadenosine
CAS:<p>5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer</p>Formula:C10H14N6O3Purity:95.55%Color and Shape:SolidMolecular weight:266.26Rolofylline
CAS:<p>Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.</p>Formula:C20H28N4O2Purity:99.53%Color and Shape:SolidMolecular weight:356.46Theobromine
CAS:<p>Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.</p>Formula:C7H8N4O2Purity:99.69% - 99.91%Color and Shape:White To Yellow Crystalline PowderMolecular weight:180.16Trabodenoson
CAS:<p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>Formula:C15H20N6O6Purity:99.94%Color and Shape:SolidMolecular weight:380.36Blontuvetmab
CAS:<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Color and Shape:LiquidTC-G 1004
CAS:<p>adenosine A2A receptors antagonist</p>Formula:C22H27N7O2Purity:98%Color and Shape:SolidMolecular weight:421.5A2AR-agonist-1
CAS:<p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>Formula:C20H22N6O4Purity:99.9%Color and Shape:SolidMolecular weight:410.43hA2A/hCA XII modulator 1
CAS:<p>Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.</p>Formula:C24H19N7O4SColor and Shape:SolidMolecular weight:501.52IHCH-3064
CAS:<p>IHCH-3064: dual-action cancer immunotherapy, A2AR affinity (Ki 2.2 nM), selective HDAC1 inhibitor (IC50 80.2 nM).</p>Formula:C25H21N9O2Color and Shape:SolidMolecular weight:479.49MRS 1334
CAS:<p>antagonist for the human adenosine A3 receptor</p>Formula:C31H26N2O6Purity:98%Color and Shape:SolidMolecular weight:522.55LUF6000
CAS:<p>LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).</p>Formula:C22H20Cl2N4Color and Shape:SolidMolecular weight:411.33A2A/A1 AR antagonist-1
CAS:<p>A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).</p>Formula:C15H12N6O2Color and Shape:SolidMolecular weight:308.29LUF 5834
CAS:<p>A2A and A2B adenosine receptor partial agonist</p>Formula:C17H12N6OSPurity:98%Color and Shape:SolidMolecular weight:348.385'-(N-Cyclopropyl)carboxamidoadenosine
CAS:<p>adenosine A2 receptor agonist</p>Formula:C13H16N6O4Purity:98%Color and Shape:SolidMolecular weight:320.3A1AR antagonist 5
CAS:<p>A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].</p>Formula:C17H15ClN4OColor and Shape:SolidMolecular weight:326.78A1AR antagonist 3
CAS:<p>Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.</p>Formula:C25H20N2O3SColor and Shape:SolidMolecular weight:428.5XCC
CAS:<p>XCC is an Adenosine receptor antagonist.</p>Formula:C19H22N4O5Purity:98%Color and Shape:SolidMolecular weight:386.4A1AR antagonist 4
CAS:<p>Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.</p>Formula:C23H25N3O2Color and Shape:SolidMolecular weight:375.46MRS1097
CAS:<p>MRS1097 is a selective antagonist A3 adenosine receptor.</p>Formula:C26H27NO4Purity:98%Color and Shape:SolidMolecular weight:417.5MRS-1191
CAS:<p>MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).</p>Formula:C31H27NO4Color and Shape:SolidMolecular weight:477.55Apadenoson
CAS:<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Formula:C23H30N6O6Purity:98%Color and Shape:SolidMolecular weight:486.52Lu AA 47070
CAS:<p>adenosine A2A receptor antagonist</p>Formula:C17H20F2N3O6PSPurity:98%Color and Shape:SolidMolecular weight:463.39A1AR antagonist 2
CAS:<p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>Formula:C17H12N4OColor and Shape:SolidMolecular weight:288.3Adenosine receptor inhibitor 1
CAS:<p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>Formula:C17H19ClFN5O3Color and Shape:SolidMolecular weight:395.82A1/A3 AR antagonist 2
CAS:<p>The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.</p>Formula:C22H16N2O3SColor and Shape:SolidMolecular weight:388.44AB-MECA
CAS:<p>AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.</p>Formula:C18H21N7O4Purity:98%Color and Shape:SolidMolecular weight:399.4A2AAR/HDAC-IN-1
CAS:<p>A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.</p>Formula:C24H21N7O2Color and Shape:SolidMolecular weight:439.47LASSBio-1359
CAS:<p>LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.</p>Formula:C17H18N2O3Purity:98%Color and Shape:SolidMolecular weight:298.34PSB 11 hydrochloride
CAS:<p>PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.</p>Formula:C16H18ClN5OPurity:98%Color and Shape:SolidMolecular weight:331.8Adenosine receptor antagonist 3
CAS:<p>Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].</p>Formula:C16H14N6SColor and Shape:SolidMolecular weight:322.39Adentri
CAS:<p>Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.</p>Formula:C18H24N4O3Purity:98%Color and Shape:SolidMolecular weight:344.41A2A receptor antagonist 3
CAS:<p>A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).</p>Formula:C26H26N6O2Color and Shape:SolidMolecular weight:454.52MRS1186
CAS:<p>MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).</p>Formula:C16H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:341.75Adenosine receptor A1 antagonist 5
CAS:<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Formula:C17H20N4O2Purity:99.97%Color and Shape:SolidMolecular weight:312.37MRS1177
CAS:<p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>Formula:C20H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:389.79XU1
CAS:<p>XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or</p>Formula:C12H8N2OPurity:98.58% - 99.59%Color and Shape:SolidMolecular weight:196.2HEMADO
CAS:<p>HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).</p>Formula:C17H23N5O4Purity:98%Color and Shape:SolidMolecular weight:361.4A1AR antagonist 6
CAS:<p>A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].</p>Formula:C17H15N3O2Color and Shape:SolidMolecular weight:293.32Lu AA41063
CAS:<p>Lu AA41063 is a potent and selective antagonist of the hA2A receptor.</p>Formula:C16H17F2N3O2SColor and Shape:SolidMolecular weight:353.39Neladenoson dalanate HCl
CAS:<p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>Formula:C35H35Cl2N7O4S2Purity:98%Color and Shape:SolidMolecular weight:752.73A3AR antagonist 1
CAS:<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Formula:C32H24N4O4SColor and Shape:SolidMolecular weight:560.62Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Formula:C23H21FN8OColor and Shape:SolidMolecular weight:444.46CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Formula:C18H20N6Color and Shape:SolidMolecular weight:320.39VUF8507
CAS:<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Formula:C21H15N3OColor and Shape:SolidMolecular weight:325.36PD 81723
CAS:<p>Allosteric potentiator at the adenosine A1 receptor</p>Formula:C14H12F3NOSPurity:98%Color and Shape:SolidMolecular weight:299.31Sipagladenant
CAS:<p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>Formula:C20H19N3O4SColor and Shape:SolidMolecular weight:397.45SCH-202676 HBr
CAS:<p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>Formula:C15H13N3SPurity:98%Color and Shape:SolidMolecular weight:267.35A3AR antagonist 2
CAS:<p>A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.</p>Formula:C22H16N6O3Color and Shape:SolidMolecular weight:412.4TH-162
CAS:<p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>Formula:C19H23N5O4Color and Shape:SolidMolecular weight:385.42PQ-69
CAS:<p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>Formula:C20H19FN4OColor and Shape:SolidMolecular weight:350.39MRS 1523
CAS:<p>MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.</p>Formula:C23H29NO3SPurity:98%Color and Shape:SolidMolecular weight:399.55Inupadenant
CAS:<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Formula:C25H26F2N8O4S2Color and Shape:SolidMolecular weight:604.65CAY10680
CAS:<p>CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.</p>Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.4FR-194921
CAS:<p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>Formula:C23H23N5OColor and Shape:SolidMolecular weight:385.46CVT-2759
CAS:<p>CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.</p>Formula:C17H24N6O6Color and Shape:SolidMolecular weight:408.41Adenosine receptor inhibitor 2
CAS:<p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>Formula:C17H20BrN5O2Color and Shape:SolidMolecular weight:406.28Acefylline piperazine
CAS:<p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>Formula:C9H10N4O4·xC4H10N2Color and Shape:SolidMolecular weight:562.54JNJ-40255293
CAS:<p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>Formula:C23H22N4O3Purity:98%Color and Shape:SolidMolecular weight:402.45AK-IN-1
CAS:<p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42ATL-801
CAS:<p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>Formula:C24H25N7O3Color and Shape:SolidMolecular weight:459.5Kira8 Hydrochloride
CAS:<p>Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.</p>Formula:C31H30Cl2N6O3SPurity:98%Color and Shape:SolidMolecular weight:637.58A2AAR/HDAC-IN-2
CAS:<p>A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.</p>Formula:C23H26N6O4Color and Shape:SolidMolecular weight:450.49Theophylline sodium glycinate
CAS:<p>Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.</p>Formula:C9H12N5NaO4Color and Shape:SolidMolecular weight:277.216hA2AAR antagonist 1
CAS:<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Formula:C15H15N5OColor and Shape:SolidMolecular weight:281.31LUF5831
CAS:<p>LUF5831 is an agonist of adenosine A1 receptor.</p>Formula:C15H12N4O2SColor and Shape:SolidMolecular weight:312.35Draflazine
CAS:<p>Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.</p>Formula:C30H33Cl2F2N5O2Purity:98%Color and Shape:SolidMolecular weight:604.52LUF5981
CAS:<p>LUF5981 is a selective agonist of human adenosine A1 receptor.</p>Formula:C24H23N3Color and Shape:SolidMolecular weight:353.46Cirazoline hydrochloride
CAS:<p>Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.</p>Formula:C13H17ClN2OPurity:99.863%Color and Shape:SolidMolecular weight:252.74Bamifylline Hydrochloride
CAS:<p>Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.</p>Formula:C20H28ClN5O3Color and Shape:SolidMolecular weight:421.92MRS1067
CAS:<p>MRS1067 is an antagonist of A3 adenosine receptor.</p>Formula:C19H16Cl2O3Color and Shape:SolidMolecular weight:363.23MRE3008F20
CAS:<p>MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.</p>Formula:C21H20N8O3Purity:97.29%Color and Shape:SolidMolecular weight:432.44A2AR-antagonist-1
CAS:<p>Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.</p>Formula:C27H25N5O2Purity:98%Color and Shape:SolidMolecular weight:451.52VUF 5574
CAS:<p>VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.</p>Formula:C21H17N5O2Purity:99.53%Color and Shape:SolidMolecular weight:371.39ST3932
CAS:<p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>Formula:C12H16N8OPurity:98%Color and Shape:SolidMolecular weight:288.31APNEA
CAS:<p>APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.</p>Formula:C18H22N6O4Purity:99.88%Color and Shape:SolidMolecular weight:386.41N6-Cyclopentyladenosine
CAS:<p>N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of</p>Formula:C15H21N5O4Purity:99.84%Color and Shape:SolidMolecular weight:335.36Sonedenoson
CAS:<p>Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.</p>Formula:C18H20ClN5O5Purity:99.79%Color and Shape:SolidMolecular weight:421.84Evodenoson
CAS:<p>Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.</p>Formula:C23H29N7O6Purity:99.75% - 99.83%Color and Shape:SolidMolecular weight:499.52N-[(4-Aminophenyl)methyl]adenosine
CAS:<p>N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).</p>Formula:C17H20N6O4Purity:98.75%Color and Shape:SolidMolecular weight:372.38BAY 60-6583
CAS:<p>BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3</p>Formula:C19H17N5O2SPurity:98.46% - 99.8%Color and Shape:SolidMolecular weight:379.44ANR 94
CAS:<p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>Formula:C9H13N5OPurity:98.9%Color and Shape:SolidMolecular weight:207.23Adenosine antagonist-1
CAS:<p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>Formula:C18H13N7SPurity:99.28% - 99.95%Color and Shape:SolidMolecular weight:359.41ST-1535
CAS:<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Formula:C12H16N8Purity:99.64% - 99.69%Color and Shape:SolidMolecular weight:272.31MRS1220
CAS:<p>MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic</p>Formula:C21H14ClN5O2Purity:98.43%Color and Shape:SolidMolecular weight:403.82N 0861
CAS:<p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>Formula:C13H17N5Purity:98.78%Color and Shape:SolidMolecular weight:243.31Selodenoson
CAS:<p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>Formula:C17H24N6O4Purity:99.52%Color and Shape:SolidMolecular weight:376.41ISAM-140
CAS:<p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>Formula:C19H19N3O3Purity:99.51%Color and Shape:SolidMolecular weight:337.37GW-493838
CAS:<p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>Formula:C21H21ClFN7O4Purity:99.11% - 99.58%Color and Shape:SolidMolecular weight:489.89GS-9667
CAS:<p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>Formula:C21H24FN5O4SPurity:99.76% - 99.77%Color and Shape:SolidMolecular weight:461.51A2A receptor antagonist 1
CAS:<p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>Formula:C16H12FN5OPurity:99.52% - 99.93%Color and Shape:SolidMolecular weight:309.3LAS38096
CAS:<p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>Formula:C17H12N6OPurity:99.18% - 99.95%Color and Shape:SolidMolecular weight:316.32N6-(2-Phenylethyl)adenosine
CAS:<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Formula:C18H21N5O4Purity:99.83%Color and Shape:SolidMolecular weight:371.392'-MeCCPA
CAS:<p>2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.</p>Formula:C16H22ClN5O4Purity:99.93%Color and Shape:SolidMolecular weight:383.83KI-7
CAS:<p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>Formula:C23H18N2O2Purity:98.33%Color and Shape:SolidMolecular weight:354.4FK-453
CAS:<p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>Formula:C23H25N3O2Purity:99.44%Color and Shape:SolidMolecular weight:375.46GP3269
CAS:<p>GP3269 is a selective, potent, orally active human adenosine kinase (AK) inhibitor (IC50: 11 nM) with anticonvulsant effects in rats.</p>Formula:C23H21FN4O3Color and Shape:SolidMolecular weight:420.44PSB-1115 potassium salt
CAS:<p>PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1].</p>Formula:C14H13KN4O5SColor and Shape:SolidMolecular weight:388.44MRS3558
CAS:<p>MRS3558 is an agonist of A3 adenosine receptors.</p>Formula:C20H20Cl2N6O3Color and Shape:SolidMolecular weight:463.32ABT-702 hydrochloride
CAS:<p>ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].</p>Formula:C22H20BrClN6OColor and Shape:SolidMolecular weight:499.79KFM19
CAS:<p>KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.</p>Formula:C16H22N4O3Purity:98.62%Color and Shape:SolidMolecular weight:318.37Neladenoson dalanate
CAS:<p>Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.</p>Formula:C35H34ClN7O4S2Color and Shape:SolidMolecular weight:716.27Sulmazole
CAS:<p>Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.</p>Formula:C14H13N3O2SPurity:99.94%Color and Shape:SolidMolecular weight:287.34Xanthine amine congener
CAS:<p>Xanthine amine congener is an Adenosine receptor antagonist.</p>Formula:C21H28N6O4Purity:99.7%Color and Shape:SolidMolecular weight:428.48

