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Adenosine Receptor

Adenosine Receptor

Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.

Found 242 products of "Adenosine Receptor"

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  • CGS 15943

    CAS:
    <p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>
    Formula:C13H8ClN5O
    Purity:97.4%
    Color and Shape:Solid
    Molecular weight:285.69
  • Pentoxifylline

    CAS:
    <p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>
    Formula:C13H18N4O3
    Purity:99.26% - 99.93%
    Color and Shape:Solid
    Molecular weight:278.31
  • Acefylline

    CAS:
    <p>Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.</p>
    Formula:C9H10N4O4
    Purity:99.57%
    Color and Shape:White Crystalline Solid
    Molecular weight:238.2
  • AB928

    CAS:
    <p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>
    Formula:C23H22N8O
    Purity:98.09% - >99.99%
    Color and Shape:Solid
    Molecular weight:426.47
  • N6-Ethyladenosine

    CAS:
    <p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>
    Formula:C12H17N5O4
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:295.29
  • DPTN dihydrochloride

    CAS:
    <p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>
    Formula:C22H20Cl2N4OS
    Purity:99.95%
    Color and Shape:Soild
    Molecular weight:459.39
  • Amp579 TFA


    <p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>
    Formula:C24H29ClF3N5O5S
    Purity:96.56%
    Color and Shape:Soild
    Molecular weight:592.03
  • Theophylline

    CAS:
    <p>Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central</p>
    Formula:C7H8N4O2
    Purity:99.65% - 99.98%
    Color and Shape:White Solid Powder
    Molecular weight:180.16
  • YT 146

    CAS:
    <p>YT 146 is a biochemical.</p>
    Formula:C18H25N5O4
    Purity:98.81% - 99.25%
    Color and Shape:Solid
    Molecular weight:375.42
  • Diphylline

    CAS:
    <p>Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.</p>
    Formula:C10H14N4O4
    Purity:98.54%
    Color and Shape:Crystals From Alcohol Solid
    Molecular weight:254.24
  • Adenosine A1 receptor activator T62

    CAS:
    <p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>
    Formula:C15H14ClNOS
    Purity:97.83%
    Color and Shape:Solid
    Molecular weight:291.8
  • Adenosine 5'-monophosphate monohydrate

    CAS:
    <p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>
    Formula:C10H14N5O7P·H2O
    Purity:97.68% - 98.49%
    Color and Shape:White Powder
    Molecular weight:365.24
  • Theophylline monohydrate

    CAS:
    <p>Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium</p>
    Formula:C7H8N4O2·H2O
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:198.18
  • Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Formula:C14H15Cl2NS
    Purity:99.85% - >99.99%
    Color and Shape:White Powder
    Molecular weight:300.25
  • Aminophylline

    CAS:
    <p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>
    Formula:C7H8O2·C2H8N2
    Purity:99.31%
    Color and Shape:White Or Slightly Yellowish Granules Or Powder Solid
    Molecular weight:420.43
  • Quercetin-3'-o-phosphate TEA


    <p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>
    Formula:C21H26NO10P
    Purity:95.63%
    Color and Shape:Soild
    Molecular weight:483.41
  • Pamabrom

    CAS:
    <p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>
    Formula:C11H18BrN5O3
    Purity:99.84% - >99.99%
    Color and Shape:Coa
    Molecular weight:348.2
  • Doxofylline

    CAS:
    <p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>
    Formula:C11H14N4O4
    Purity:99.958% - >99.99%
    Color and Shape:Solid
    Molecular weight:266.25
  • N6-Cyclohexyladenosine

    CAS:
    <p>N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.</p>
    Formula:C16H23N5O4
    Purity:99.84% - 99.98%
    Color and Shape:Solid
    Molecular weight:349.38
  • Adenosine receptor antagonist 1

    CAS:
    <p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>
    Formula:C22H15ClFN7O
    Color and Shape:Solid
    Molecular weight:447.86
  • Theophyllol

    CAS:
    <p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>
    Formula:C9H10N4Na2O4
    Color and Shape:Solid
    Molecular weight:284.18
  • 3F6-9G5


    <p>3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.</p>
    Purity:>95%
    Color and Shape:Odour Liquid
  • Heterobivalent ligand-1


    <p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>
    Formula:C86H115FN16O21
    Color and Shape:Solid
    Molecular weight:1727.93
  • PSB 0777 ammonium salt

    CAS:
    <p>adenosine A2A receptor full agonist</p>
    Formula:C18H24N6O7S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.55
  • AR ligand 40


    <p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>
    Formula:C21H25N5
    Color and Shape:Solid
    Molecular weight:347.211
  • MRS-1706

    CAS:
    <p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>
    Formula:C27H29N5O5
    Purity:99.00%
    Color and Shape:Solid
    Molecular weight:503.55
  • A2A/A3 AR antagonist-1


    <p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) &amp; 31.8 nM (hA3).</p>
    Formula:C56H71N15O12S2
    Color and Shape:Solid
    Molecular weight:1210.39
  • Norisoboldine hydrochloride

    CAS:
    <p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>
    Formula:C18H20ClNO4
    Color and Shape:Solid
    Molecular weight:349.81
  • A3AR agonist 2


    <p>Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.</p>
    Formula:C34H34N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:622.67
  • LUF7690

    CAS:
    <p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>
    Formula:C25H24FN5O6S
    Color and Shape:Solid
    Molecular weight:541.55
  • Apadenoson TFA


    <p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>
    Formula:C25H31F3N6O8
    Purity:98.08%
    Color and Shape:Soild
    Molecular weight:600.55
  • Xanthine amine congener dihydrochloride

    CAS:
    <p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>
    Formula:C21H30Cl2N6O4
    Color and Shape:Solid
    Molecular weight:501.41
  • FSCPX

    CAS:
    <p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>
    Formula:C23H27FN4O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.55
  • ABT-702

    CAS:
    <p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>
    Formula:C22H19BrN6O
    Purity:99.57%
    Color and Shape:Soild
    Molecular weight:463.33
  • PSB 0777 ammonium hydrate


    <p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>
    Formula:C18H20N5O7S2·NH4·75H2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:532.09
  • Adenosine receptor agonist 1


    <p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>
    Formula:C12H14ClN5O2Se
    Color and Shape:Solid
    Molecular weight:374.68
  • A3AR modulator 1


    <p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>
    Formula:C23H25IN4
    Color and Shape:Solid
    Molecular weight:484.38
  • hA3AR agonist 2


    <p>hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.</p>
    Formula:C11H14ClN5O2S
    Color and Shape:Solid
    Molecular weight:315.78
  • N6-Benzyl-5'-ethylcarboxamido adenosine

    CAS:
    <p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>
    Formula:C19H22N6O4
    Color and Shape:Solid
    Molecular weight:398.42
  • 8-Chloro caffeine

    CAS:
    <p>8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.</p>
    Formula:C8H9ClN4O2
    Color and Shape:Solid
    Molecular weight:228.64
  • GW-328267

    CAS:
    <p>GW-328267 is an agonist of the adenosine A2 receptor.</p>
    Formula:C21H26N10O4
    Color and Shape:Solid
    Molecular weight:482.5
  • Xanthine amine congener trihydrochloride

    CAS:
    <p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>
    Formula:C21H29ClN6O4
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:464.95
  • A3AR agonist 1


    <p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>
    Formula:C28H34N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:550.61
  • Danshenol B


    <p>Danshenol B is a natural product that can be used as a reference standard.</p>
    Formula:C22H26O4
    Color and Shape:Solid
    Molecular weight:354.446
  • A-286501

    CAS:
    <p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>
    Formula:C11H14BrN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.17
  • LUF6096

    CAS:
    <p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>
    Formula:C22H21Cl2N3O
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:414.33
  • LAS101057

    CAS:
    <p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>
    Formula:C18H14FN5O
    Purity:99.03% - >99.99%
    Color and Shape:Solid
    Molecular weight:335.34
  • GR79236

    CAS:
    <p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>
    Formula:C15H21N5O5
    Color and Shape:Solid
    Molecular weight:351.36
  • MRS-3777 hemioxalate

    CAS:
    <p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>
    Formula:C17H19N5OC2H2O4
    Purity:97.10%
    Color and Shape:Solid
    Molecular weight:354.39
  • (Rac)-Mirabegron-d5

    CAS:
    <p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>
    Formula:C21H24N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.54
  • CCPA

    CAS:
    <p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>
    Formula:C15H20ClN5O4
    Purity:99.1%
    Color and Shape:Off-White To Light Yellow Solid
    Molecular weight:369.8
  • A2B receptor antagonist 2

    CAS:
    <p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>
    Formula:C12H15N5
    Purity:100%
    Color and Shape:Solid
    Molecular weight:229.28
  • CPI-444

    CAS:
    <p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>
    Formula:C20H21N7O3
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:407.43
  • Regadenoson hydrate

    CAS:
    <p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>
    Formula:C15H20N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.37
  • Tecadenoson

    CAS:
    <p>Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.</p>
    Formula:C14H19N5O5
    Purity:98.83%
    Color and Shape:Solid
    Molecular weight:337.33
  • Derenofylline

    CAS:
    <p>Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)</p>
    Formula:C18H20N4O
    Purity:98.09%
    Color and Shape:Solid
    Molecular weight:308.38
  • 5-Iodotubercidin

    CAS:
    <p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>
    Formula:C11H13IN4O4
    Purity:99.98%
    Color and Shape:Tan Solid
    Molecular weight:392.15
  • DPCPX

    CAS:
    <p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>
    Formula:C16H24N4O2
    Purity:99.23% - 99.93%
    Color and Shape:White Solid
    Molecular weight:304.39
  • Proxyphylline

    CAS:
    <p>Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.</p>
    Formula:C10H14N4O3
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:238.24
  • ABT-702 dihydrochloride

    CAS:
    <p>ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.</p>
    Formula:C22H21BrCl2N6O
    Purity:98.42% - 98.98%
    Color and Shape:Solid
    Molecular weight:536.25
  • ZM241385

    CAS:
    <p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>
    Formula:C16H15N7O2
    Purity:97.02% - 99.69%
    Color and Shape:Solid
    Molecular weight:337.34
  • N6,N6-Dimethyladenosine

    CAS:
    <p>N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.</p>
    Formula:C12H17N5O4
    Purity:98.79%
    Color and Shape:White Powder
    Molecular weight:295.29
  • CGS 21680 Hydrochloride

    CAS:
    <p>CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.</p>
    Formula:C23H29N7O6·HCl
    Purity:96.74% - 99.53%
    Color and Shape:Solid
    Molecular weight:535.98
  • Piclidenoson

    CAS:
    <p>Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.</p>
    Formula:C18H19IN6O4
    Purity:99.83% - ≥95%
    Color and Shape:Solid
    Molecular weight:510.29
  • Swertisin

    CAS:
    <p>Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.</p>
    Formula:C22H22O10
    Purity:99.74% - 99.89%
    Color and Shape:Solid
    Molecular weight:446.4
  • 2-Chloroadenosine

    CAS:
    <p>2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively</p>
    Formula:C10H12ClN5O4
    Purity:99.23%
    Color and Shape:White Powder
    Molecular weight:301.69
  • VPC171

    CAS:
    <p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>
    Formula:C18H12F3NOS
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:347.35
  • BAY-545

    CAS:
    <p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>
    Formula:C18H22F3N3O4S
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:433.45
  • 1-Ethyl-6-aminouracil

    CAS:
    <p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>
    Formula:C6H9N3O2
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:155.15
  • Regadenoson

    CAS:
    <p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>
    Formula:C15H18N8O5
    Purity:99.57% - 99.81%
    Color and Shape:Off-White Solid
    Molecular weight:390.35
  • 5'-N-Ethylcarboxamidoadenosine

    CAS:
    <p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>
    Formula:C12H16N6O4
    Purity:98.95% - ≥95%
    Color and Shape:Powder
    Molecular weight:308.29
  • Namodenoson

    CAS:
    <p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>
    Formula:C18H18ClIN6O4
    Purity:98.97%
    Color and Shape:Solid
    Molecular weight:544.73
  • Taminadenant

    CAS:
    <p>Taminadenant is an adenosine receptor antagonist.</p>
    Formula:C10H8BrN7
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:306.12
  • CHEMBL241987

    CAS:
    <p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>
    Formula:C16H11N3O
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:261.28
  • Xanthine amine congener hydrochloride

    CAS:
    <p>Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.</p>
    Formula:C21H29ClN6O4
    Color and Shape:Solid
    Molecular weight:464.95
  • Vipadenant

    CAS:
    <p>Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).</p>
    Formula:C16H15N7O
    Purity:97.25% - 97.36%
    Color and Shape:Solid
    Molecular weight:321.34
  • Fostamatinib

    CAS:
    <p>Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.</p>
    Formula:C23H26FN6O9P
    Purity:93.08% - 99.38%
    Color and Shape:Solid
    Molecular weight:580.46
  • MIPS521

    CAS:
    <p>MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.</p>
    Formula:C19H10ClF6NOS
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:449.8
  • 8-Cyclopentyl-1,3-dimethylxanthine

    CAS:
    <p>8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.</p>
    Formula:C12H16N4O2
    Purity:98.58% - >99.99%
    Color and Shape:Solid
    Molecular weight:248.28
  • Adenosine receptor antagonist 4

    CAS:
    <p>Adenosine receptor antagonist 4 is an adenosine receptor antagonist.</p>
    Formula:C10H13N3
    Purity:99.63% - 99.65%
    Color and Shape:Off-White Powder
    Molecular weight:175.23
  • Inosine

    CAS:
    <p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>
    Formula:C10H12N4O5
    Purity:99.51% - 99.89%
    Color and Shape:Solid
    Molecular weight:268.23
  • Binodenoson

    CAS:
    <p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>
    Formula:C17H25N7O4
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:391.42
  • PD 117519

    CAS:
    <p>PD 117519 (CI947) is an agonist of adenosine receptor</p>
    Formula:C19H21N5O4
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:383.4
  • Preladenant

    CAS:
    <p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has &gt;1000-fold selectivity over all other adenosine</p>
    Formula:C25H29N9O3
    Purity:98.02% - 99.68%
    Color and Shape:Solid
    Molecular weight:503.56
  • Nitrobenzylthioinosine

    CAS:
    <p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>
    Formula:C17H17N5O6S
    Purity:99.69% - 99.74%
    Color and Shape:Off-White Solid
    Molecular weight:419.41
  • Adenosine amine congener

    CAS:
    <p>Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.</p>
    Formula:C28H32N8O6
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:576.6
  • Alloxazine

    CAS:
    <p>Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.</p>
    Formula:C10H6N4O2
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:214.18
  • SDZ WAG 994

    CAS:
    <p>SDZ WAG 994 is an A1 adenosine receptor agonist.</p>
    Formula:C17H25N5O4
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:363.41
  • Istradefylline

    CAS:
    <p>Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.</p>
    Formula:C20H24N4O4
    Purity:98.18% - 99.95%
    Color and Shape:Solid
    Molecular weight:384.43
  • Norisoboldine

    CAS:
    <p>Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.</p>
    Formula:C18H19NO4
    Purity:98.12% - 99.7%
    Color and Shape:Solid
    Molecular weight:313.35
  • SCH442416

    CAS:
    <p>SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).</p>
    Formula:C20H19N7O2
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:389.41
  • Tozadenant

    CAS:
    <p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>
    Formula:C19H26N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.5
  • SCH 58261

    CAS:
    <p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>
    Formula:C18H15N7O
    Purity:99.07% - 99.75%
    Color and Shape:Solid
    Molecular weight:345.36
  • Enprofylline

    CAS:
    <p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>
    Formula:C8H10N4O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:194.19
  • Capadenoson

    CAS:
    <p>Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.</p>
    Formula:C25H18ClN5O2S2
    Purity:98.85% - 99.57%
    Color and Shape:Solid
    Molecular weight:520.03
  • Reversine

    CAS:
    <p>Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).</p>
    Formula:C21H27N7O
    Purity:98% - 98.42%
    Color and Shape:Solid
    Molecular weight:393.49
  • AZD4635

    CAS:
    <p>AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).</p>
    Formula:C15H11ClFN5
    Purity:99.15% - 99.90%
    Color and Shape:Solid
    Molecular weight:315.73
  • 5'-Amino-5'-deoxyadenosine

    CAS:
    <p>5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer</p>
    Formula:C10H14N6O3
    Purity:95.55%
    Color and Shape:Solid
    Molecular weight:266.26
  • Rolofylline

    CAS:
    <p>Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.</p>
    Formula:C20H28N4O2
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:356.46
  • Theobromine

    CAS:
    <p>Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.</p>
    Formula:C7H8N4O2
    Purity:99.69% - 99.91%
    Color and Shape:White To Yellow Crystalline Powder
    Molecular weight:180.16
  • Trabodenoson

    CAS:
    <p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>
    Formula:C15H20N6O6
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:380.36
  • Blontuvetmab

    CAS:
    <p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>
    Color and Shape:Liquid
  • TC-G 1004

    CAS:
    <p>adenosine A2A receptors antagonist</p>
    Formula:C22H27N7O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.5
  • A2AR-agonist-1

    CAS:
    <p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>
    Formula:C20H22N6O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:410.43
  • hA2A/hCA XII modulator 1

    CAS:
    <p>Potent hA2AAR antagonist &amp; hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.</p>
    Formula:C24H19N7O4S
    Color and Shape:Solid
    Molecular weight:501.52
  • IHCH-3064

    CAS:
    <p>IHCH-3064: dual-action cancer immunotherapy, A2AR affinity (Ki 2.2 nM), selective HDAC1 inhibitor (IC50 80.2 nM).</p>
    Formula:C25H21N9O2
    Color and Shape:Solid
    Molecular weight:479.49
  • MRS 1334

    CAS:
    <p>antagonist for the human adenosine A3 receptor</p>
    Formula:C31H26N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:522.55
  • LUF6000

    CAS:
    <p>LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).</p>
    Formula:C22H20Cl2N4
    Color and Shape:Solid
    Molecular weight:411.33
  • A2A/A1 AR antagonist-1

    CAS:
    <p>A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).</p>
    Formula:C15H12N6O2
    Color and Shape:Solid
    Molecular weight:308.29
  • LUF 5834

    CAS:
    <p>A2A and A2B adenosine receptor partial agonist</p>
    Formula:C17H12N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.38
  • 5'-(N-Cyclopropyl)carboxamidoadenosine

    CAS:
    <p>adenosine A2 receptor agonist</p>
    Formula:C13H16N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.3
  • A1AR antagonist 5

    CAS:
    <p>A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].</p>
    Formula:C17H15ClN4O
    Color and Shape:Solid
    Molecular weight:326.78
  • A1AR antagonist 3

    CAS:
    <p>Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.</p>
    Formula:C25H20N2O3S
    Color and Shape:Solid
    Molecular weight:428.5
  • XCC

    CAS:
    <p>XCC is an Adenosine receptor antagonist.</p>
    Formula:C19H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.4
  • A1AR antagonist 4

    CAS:
    <p>Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.</p>
    Formula:C23H25N3O2
    Color and Shape:Solid
    Molecular weight:375.46
  • MRS1097

    CAS:
    <p>MRS1097 is a selective antagonist A3 adenosine receptor.</p>
    Formula:C26H27NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:417.5
  • MRS-1191

    CAS:
    <p>MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).</p>
    Formula:C31H27NO4
    Color and Shape:Solid
    Molecular weight:477.55
  • Apadenoson

    CAS:
    <p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>
    Formula:C23H30N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:486.52
  • Lu AA 47070

    CAS:
    <p>adenosine A2A receptor antagonist</p>
    Formula:C17H20F2N3O6PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.39
  • A1AR antagonist 2

    CAS:
    <p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>
    Formula:C17H12N4O
    Color and Shape:Solid
    Molecular weight:288.3
  • Adenosine receptor inhibitor 1

    CAS:
    <p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>
    Formula:C17H19ClFN5O3
    Color and Shape:Solid
    Molecular weight:395.82
  • A1/A3 AR antagonist 2

    CAS:
    <p>The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.</p>
    Formula:C22H16N2O3S
    Color and Shape:Solid
    Molecular weight:388.44
  • AB-MECA

    CAS:
    <p>AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.</p>
    Formula:C18H21N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.4
  • A2AAR/HDAC-IN-1

    CAS:
    <p>A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.</p>
    Formula:C24H21N7O2
    Color and Shape:Solid
    Molecular weight:439.47
  • LASSBio-1359

    CAS:
    <p>LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.</p>
    Formula:C17H18N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:298.34
  • PSB 11 hydrochloride

    CAS:
    <p>PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.</p>
    Formula:C16H18ClN5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.8
  • Adenosine receptor antagonist 3

    CAS:
    <p>Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].</p>
    Formula:C16H14N6S
    Color and Shape:Solid
    Molecular weight:322.39
  • Adentri

    CAS:
    <p>Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.</p>
    Formula:C18H24N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:344.41
  • A2A receptor antagonist 3

    CAS:
    <p>A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).</p>
    Formula:C26H26N6O2
    Color and Shape:Solid
    Molecular weight:454.52
  • MRS1186

    CAS:
    <p>MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).</p>
    Formula:C16H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.75
  • Adenosine receptor A1 antagonist 5

    CAS:
    <p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>
    Formula:C17H20N4O2
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:312.37
  • MRS1177

    CAS:
    <p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>
    Formula:C20H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.79
  • XU1

    CAS:
    <p>XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or</p>
    Formula:C12H8N2O
    Purity:98.58% - 99.59%
    Color and Shape:Solid
    Molecular weight:196.2
  • HEMADO

    CAS:
    <p>HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).</p>
    Formula:C17H23N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.4
  • A1AR antagonist 6

    CAS:
    <p>A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].</p>
    Formula:C17H15N3O2
    Color and Shape:Solid
    Molecular weight:293.32
  • Lu AA41063

    CAS:
    <p>Lu AA41063 is a potent and selective antagonist of the hA2A receptor.</p>
    Formula:C16H17F2N3O2S
    Color and Shape:Solid
    Molecular weight:353.39
  • Neladenoson dalanate HCl

    CAS:
    <p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>
    Formula:C35H35Cl2N7O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:752.73
  • A3AR antagonist 1

    CAS:
    <p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>
    Formula:C32H24N4O4S
    Color and Shape:Solid
    Molecular weight:560.62
  • Adenosine receptor antagonist 2

    CAS:
    <p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>
    Formula:C23H21FN8O
    Color and Shape:Solid
    Molecular weight:444.46
  • CAY10498

    CAS:
    <p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>
    Formula:C18H20N6
    Color and Shape:Solid
    Molecular weight:320.39
  • VUF8507

    CAS:
    <p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>
    Formula:C21H15N3O
    Color and Shape:Solid
    Molecular weight:325.36
  • PD 81723

    CAS:
    <p>Allosteric potentiator at the adenosine A1 receptor</p>
    Formula:C14H12F3NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.31
  • Sipagladenant

    CAS:
    <p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>
    Formula:C20H19N3O4S
    Color and Shape:Solid
    Molecular weight:397.45
  • SCH-202676 HBr

    CAS:
    <p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>
    Formula:C15H13N3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.35
  • A3AR antagonist 2

    CAS:
    <p>A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.</p>
    Formula:C22H16N6O3
    Color and Shape:Solid
    Molecular weight:412.4
  • TH-162

    CAS:
    <p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>
    Formula:C19H23N5O4
    Color and Shape:Solid
    Molecular weight:385.42
  • PQ-69

    CAS:
    <p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>
    Formula:C20H19FN4O
    Color and Shape:Solid
    Molecular weight:350.39
  • MRS 1523

    CAS:
    <p>MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels &amp; inhibits action potentials in rat DRG neurons.</p>
    Formula:C23H29NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.55
  • Inupadenant

    CAS:
    <p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>
    Formula:C25H26F2N8O4S2
    Color and Shape:Solid
    Molecular weight:604.65
  • CAY10680

    CAS:
    <p>CAY10680 inhibits MAO-B (IC50=34.9 nM) &amp; A2A receptors (Ki=39.5 nM), sparing other adenosine types &amp; MAO-A, may treat Parkinson's.</p>
    Formula:C18H16N2O2S
    Color and Shape:Solid
    Molecular weight:324.4
  • FR-194921

    CAS:
    <p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>
    Formula:C23H23N5O
    Color and Shape:Solid
    Molecular weight:385.46
  • CVT-2759

    CAS:
    <p>CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.</p>
    Formula:C17H24N6O6
    Color and Shape:Solid
    Molecular weight:408.41
  • Adenosine receptor inhibitor 2

    CAS:
    <p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>
    Formula:C17H20BrN5O2
    Color and Shape:Solid
    Molecular weight:406.28
  • Acefylline piperazine

    CAS:
    <p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>
    Formula:C9H10N4O4·xC4H10N2
    Color and Shape:Solid
    Molecular weight:562.54
  • JNJ-40255293

    CAS:
    <p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>
    Formula:C23H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.45
  • AK-IN-1

    CAS:
    <p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>
    Formula:C22H21N3O4
    Color and Shape:Solid
    Molecular weight:391.42
  • ATL-801

    CAS:
    <p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>
    Formula:C24H25N7O3
    Color and Shape:Solid
    Molecular weight:459.5
  • Kira8 Hydrochloride

    CAS:
    <p>Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.</p>
    Formula:C31H30Cl2N6O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:637.58
  • A2AAR/HDAC-IN-2

    CAS:
    <p>A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.</p>
    Formula:C23H26N6O4
    Color and Shape:Solid
    Molecular weight:450.49
  • Theophylline sodium glycinate

    CAS:
    <p>Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.</p>
    Formula:C9H12N5NaO4
    Color and Shape:Solid
    Molecular weight:277.216
  • hA2AAR antagonist 1

    CAS:
    <p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>
    Formula:C15H15N5O
    Color and Shape:Solid
    Molecular weight:281.31
  • LUF5831

    CAS:
    <p>LUF5831 is an agonist of adenosine A1 receptor.</p>
    Formula:C15H12N4O2S
    Color and Shape:Solid
    Molecular weight:312.35
  • Draflazine

    CAS:
    <p>Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.</p>
    Formula:C30H33Cl2F2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:604.52
  • LUF5981

    CAS:
    <p>LUF5981 is a selective agonist of human adenosine A1 receptor.</p>
    Formula:C24H23N3
    Color and Shape:Solid
    Molecular weight:353.46
  • Cirazoline hydrochloride

    CAS:
    <p>Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.</p>
    Formula:C13H17ClN2O
    Purity:99.863%
    Color and Shape:Solid
    Molecular weight:252.74
  • Bamifylline Hydrochloride

    CAS:
    <p>Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.</p>
    Formula:C20H28ClN5O3
    Color and Shape:Solid
    Molecular weight:421.92
  • MRS1067

    CAS:
    <p>MRS1067 is an antagonist of A3 adenosine receptor.</p>
    Formula:C19H16Cl2O3
    Color and Shape:Solid
    Molecular weight:363.23
  • MRE3008F20

    CAS:
    <p>MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.</p>
    Formula:C21H20N8O3
    Purity:97.29%
    Color and Shape:Solid
    Molecular weight:432.44
  • A2AR-antagonist-1

    CAS:
    <p>Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.</p>
    Formula:C27H25N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:451.52
  • VUF 5574

    CAS:
    <p>VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.</p>
    Formula:C21H17N5O2
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:371.39
  • ST3932

    CAS:
    <p>ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).</p>
    Formula:C12H16N8O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:288.31
  • APNEA

    CAS:
    <p>APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.</p>
    Formula:C18H22N6O4
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:386.41
  • N6-Cyclopentyladenosine

    CAS:
    <p>N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of</p>
    Formula:C15H21N5O4
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:335.36
  • Sonedenoson

    CAS:
    <p>Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.</p>
    Formula:C18H20ClN5O5
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:421.84
  • Evodenoson

    CAS:
    <p>Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.</p>
    Formula:C23H29N7O6
    Purity:99.75% - 99.83%
    Color and Shape:Solid
    Molecular weight:499.52
  • N-[(4-Aminophenyl)methyl]adenosine

    CAS:
    <p>N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).</p>
    Formula:C17H20N6O4
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:372.38
  • BAY 60-6583

    CAS:
    <p>BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3</p>
    Formula:C19H17N5O2S
    Purity:98.46% - 99.8%
    Color and Shape:Solid
    Molecular weight:379.44
  • ANR 94

    CAS:
    <p>ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.</p>
    Formula:C9H13N5O
    Purity:98.9%
    Color and Shape:Solid
    Molecular weight:207.23
  • Adenosine antagonist-1

    CAS:
    <p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>
    Formula:C18H13N7S
    Purity:99.28% - 99.95%
    Color and Shape:Solid
    Molecular weight:359.41
  • ST-1535

    CAS:
    <p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>
    Formula:C12H16N8
    Purity:99.64% - 99.69%
    Color and Shape:Solid
    Molecular weight:272.31
  • MRS1220

    CAS:
    <p>MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic</p>
    Formula:C21H14ClN5O2
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:403.82
  • N 0861

    CAS:
    <p>N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.</p>
    Formula:C13H17N5
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:243.31
  • Selodenoson

    CAS:
    <p>Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.</p>
    Formula:C17H24N6O4
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:376.41
  • ISAM-140

    CAS:
    <p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>
    Formula:C19H19N3O3
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:337.37
  • GW-493838

    CAS:
    <p>GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia</p>
    Formula:C21H21ClFN7O4
    Purity:99.11% - 99.58%
    Color and Shape:Solid
    Molecular weight:489.89
  • GS-9667

    CAS:
    <p>GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via</p>
    Formula:C21H24FN5O4S
    Purity:99.76% - 99.77%
    Color and Shape:Solid
    Molecular weight:461.51
  • A2A receptor antagonist 1

    CAS:
    <p>A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.</p>
    Formula:C16H12FN5O
    Purity:99.52% - 99.93%
    Color and Shape:Solid
    Molecular weight:309.3
  • LAS38096

    CAS:
    <p>LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .</p>
    Formula:C17H12N6O
    Purity:99.18% - 99.95%
    Color and Shape:Solid
    Molecular weight:316.32
  • N6-(2-Phenylethyl)adenosine

    CAS:
    <p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>
    Formula:C18H21N5O4
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:371.39
  • 2'-MeCCPA

    CAS:
    <p>2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.</p>
    Formula:C16H22ClN5O4
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:383.83
  • KI-7

    CAS:
    <p>KI-7 is an adenosine A2B receptor positive allosteric modulator.</p>
    Formula:C23H18N2O2
    Purity:98.33%
    Color and Shape:Solid
    Molecular weight:354.4
  • FK-453

    CAS:
    <p>FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.</p>
    Formula:C23H25N3O2
    Purity:99.44%
    Color and Shape:Solid
    Molecular weight:375.46
  • GP3269

    CAS:
    <p>GP3269 is a selective, potent, orally active human adenosine kinase (AK) inhibitor (IC50: 11 nM) with anticonvulsant effects in rats.</p>
    Formula:C23H21FN4O3
    Color and Shape:Solid
    Molecular weight:420.44
  • PSB-1115 potassium salt

    CAS:
    <p>PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1].</p>
    Formula:C14H13KN4O5S
    Color and Shape:Solid
    Molecular weight:388.44
  • MRS3558

    CAS:
    <p>MRS3558 is an agonist of A3 adenosine receptors.</p>
    Formula:C20H20Cl2N6O3
    Color and Shape:Solid
    Molecular weight:463.32
  • ABT-702 hydrochloride

    CAS:
    <p>ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].</p>
    Formula:C22H20BrClN6O
    Color and Shape:Solid
    Molecular weight:499.79
  • KFM19

    CAS:
    <p>KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.</p>
    Formula:C16H22N4O3
    Purity:98.62%
    Color and Shape:Solid
    Molecular weight:318.37
  • Neladenoson dalanate

    CAS:
    <p>Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.</p>
    Formula:C35H34ClN7O4S2
    Color and Shape:Solid
    Molecular weight:716.27
  • Sulmazole

    CAS:
    <p>Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.</p>
    Formula:C14H13N3O2S
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:287.34
  • Xanthine amine congener

    CAS:
    <p>Xanthine amine congener is an Adenosine receptor antagonist.</p>
    Formula:C21H28N6O4
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:428.48