GNRH Receptor
Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.
Read more
(R)-Elagolix
CAS:834153-87-6
(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing …
Formula:
C32H30F5N3O5
Purity:
97.63%
Color and Shape:
Solid
Molecular weight:
631.59
Ref: TM-T11174
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 487.00 € | ||
| 200mg | 695.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 4 Aug 2025
Alarelin Acetate
CAS:79561-22-1
Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis …
Formula:
C56H78N16O12
Purity:
100% - 99.81%
Color and Shape:
White Powder
Molecular weight:
1167.34
Ref: TM-T1494
| 5mg | 58.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 180.00 € | ||
| 500mg | 452.00 € | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Monday 4 Aug 2025
Abarelix
CAS:183552-38-7
Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate …
Formula:
C72H95ClN14O14
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1416.06
Ref: TM-T10217L
| 2mg | 42.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 283.00 € | ||
| 100mg | 432.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Monday 4 Aug 2025
Degarelix acetate(214766-78-6 free base)
CAS:934016-19-0
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
Formula:
C84H107ClN18O18
Purity:
98.66%
Color and Shape:
Solid
Molecular weight:
1692.34
Ref: TM-T10988L
| 1mg | 77.00 € | ||
| 2mg | 99.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 266.00 € | ||
| 25mg | 477.00 € | ||
| 50mg | 695.00 € | ||
| 100mg | 938.00 € |
Estimated delivery in United States, on Monday 4 Aug 2025
Linzagolix choline
CAS:1321816-57-2
Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with …
Formula:
C27H28F3N3O8S
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
611.59
Ref: TM-T25742
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 1,872.00 € |
Estimated delivery in United States, on Tuesday 5 Aug 2025
Elagolix sodium
CAS:832720-36-2
Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of …
Formula:
C32H29F5N3NaO5
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
653.57
Ref: TM-T5031
| 2mg | 46.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 11 Aug 2025
Relugolix
CAS:737789-87-6
Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) …
Formula:
C29H27F2N7O5S
Purity:
98.64% - 99.97%
Color and Shape:
Solid
Molecular weight:
623.63
Ref: TM-T3630
| 2mg | 44.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 279.00 € | ||
| 100mg | 454.00 € | ||
| 200mg | 650.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 11 Aug 2025
Fertirelin
CAS:38234-21-8
Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist …
Formula:
C55H76N16O12
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1153.29
Ref: TM-TP1288
| 1mg | 47.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 135.00 € | ||
| 50mg | 177.00 € | ||
| 100mg | 264.00 € | ||
| 200mg | 393.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Monday 11 Aug 2025
Cetrorelix diacetate
CAS:130143-01-0
Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.
Formula:
C74H100ClN17O18
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
1551.17
Ref: TM-T5520L
| 1mg | 52.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 437.00 € | ||
| 100mg | 642.00 € | ||
| 500mg | 1,359.00 € | ||
| 1mL*10mM (DMSO) | 251.00 € |
Estimated delivery in United States, on Monday 11 Aug 2025
Ganirelix Acetate
CAS:123246-29-7
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
Formula:
C82H117ClN18O15
Purity:
96.05%
Color and Shape:
Solid
Molecular weight:
1630.4
Ref: TM-TP2337
| 1mg | 88.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 598.00 € | ||
| 100mg | 810.00 € | ||
| 200mg | 1,074.00 € |
Estimated delivery in United States, on Monday 11 Aug 2025
Linzagolix
CAS:935283-04-8
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under …
Formula:
C22H15F3N2O7S
Purity:
99.33%
Color and Shape:
Solid
Molecular weight:
508.42
Ref: TM-T27837
| 1mg | 42.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 439.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 11 Aug 2025
Goserelin acetate
CAS:145781-92-6
Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of …
Formula:
C61H88N18O16
Purity:
100% - 99.86%
Color and Shape:
White Crystalline Powder
Molecular weight:
1329.46
Ref: TM-T4102
| 2mg | 48.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 310.00 € | ||
| 100mg | 467.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Monday 11 Aug 2025
Cetrorelix Acetate
CAS:145672-81-7
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
Formula:
C70H92ClN17O14·xC2H4O2
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
1491.11
Ref: TM-T5520
| 1mg | 48.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 401.00 € | ||
| 100mg | 628.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Monday 22 Sep 2025
Opigolix
CAS:912587-25-8
Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
Formula:
C25H19F3N4O5S
Purity:
98.60% - 98.97%
Color and Shape:
Solid
Molecular weight:
544.5
Ref: TM-T17301
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,622.00 € |
Estimated delivery in United States, on Monday 29 Sep 2025
GnRH antagonist 2
CAS:1709823-61-9
GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.
Formula:
C28H27F2N9O5
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
607.57
Ref: TM-T37003
| 1mg | 157.00 € | ||
| 5mg | 383.00 € | ||
| 10mg | 604.00 € | ||
| 25mg | 1,195.00 € | ||
| 50mg | 1,892.00 € | ||
| 1mL*10mM (DMSO) | 503.00 € |
Estimated delivery in United States, on Monday 3 Nov 2025
GnRH-R antagonist 1
CAS:2826273-90-7
Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.
Formula:
C31H28F5N7O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
721.65
Ref: TM-T72492
| 25mg | 2,300.00 € | ||
| 50mg | 3,022.00 € | ||
| 100mg | 4,085.00 € |
Estimated delivery in United States, on Monday 3 Nov 2025
