GNRH Receptor
Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.
Found 84 products of "GNRH Receptor"
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Alarelin Acetate
CAS:Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.Formula:C56H78N16O12Purity:99.81% - >99.99%Color and Shape:White PowderMolecular weight:1167.34Ref: TM-T1494
5mg58.00€10mg95.00€25mg115.00€50mg156.00€100mg180.00€500mg452.00€1mL*10mM (DMSO)120.00€Degarelix acetate(214766-78-6 free base)
CAS:Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Formula:C84H107ClN18O18Purity:98.66%Color and Shape:SolidMolecular weight:1692.34(R)-Elagolix
CAS:(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Formula:C32H30F5N3O5Purity:99.08%Color and Shape:SolidMolecular weight:631.59Ref: TM-T11174
5mg50.00€10mg75.00€25mg137.00€50mg195.00€100mg306.00€200mg452.00€1mL*10mM (DMSO)70.00€Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Formula:C72H95ClN14O14Purity:>99.99%Color and Shape:SolidMolecular weight:1416.06[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide is a LHRH peptide analogue.Formula:C58H82N16O12Color and Shape:SolidMolecular weight:1195.37Onvitrelin ucalontide
CAS:Onvitrelin ucalontide is a LHRH analogue with anticancer effect; halts breast, ovarian, and prostate tumors in mice.Formula:C163H243N43O32Color and Shape:SolidMolecular weight:3316.94Kisspeptin-54(human)
CAS:Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.Formula:C258H401N79O78Purity:98%Color and Shape:SolidMolecular weight:5857.49AG 045572
CAS:AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 isFormula:C30H37NO5Purity:99.96%Color and Shape:SolidMolecular weight:491.62LHRH
CAS:Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and hasFormula:C55H74N16O14Purity:98%Color and Shape:SolidMolecular weight:1183.27LGnRH-III, lamprey
CAS:GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.Formula:C59H74N18O14Purity:98%Color and Shape:SolidMolecular weight:1259.33MI 1544
CAS:MI 1544 is a LHRH antagonist.Formula:C71H94ClN17O13Color and Shape:SolidMolecular weight:1429.09Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS:LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.Formula:C60H73N15O13Purity:98%Color and Shape:SolidMolecular weight:1212.31Phoenixin-14
CAS:Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/
Formula:C75H110N18O20Purity:98%Color and Shape:SolidMolecular weight:1583.78RS 18286
CAS:RS 18286 is a LHRH antagonist.Formula:C74H101Cl2N17O14Color and Shape:SolidMolecular weight:1523.6LHRH, Ala(6)-
CAS:LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32Avorelin
CAS:Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.Formula:C65H85N17O12Purity:98%Color and Shape:SolidMolecular weight:1296.48(D-Trp6)-LHRH free acid
CAS:(D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .Formula:C64H81N17O14Molecular weight:1312.43APTAA-LHRH
CAS:APTAA-LHRH is a gonadorelin antagonist.Formula:C69H91Cl2N17O14Purity:98%Color and Shape:SolidMolecular weight:1453.47Azaline
CAS:Azaline is a gonadorelin antagonist.Formula:C74H106ClN23O12Purity:98%Color and Shape:SolidMolecular weight:1545.26Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Formula:C27H28F3N3O8SPurity:99.64%Color and Shape:SolidMolecular weight:611.59LH-RH (4-10)
CAS:LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Formula:C33H53N11O9Color and Shape:SolidMolecular weight:747.84Lamprey LH-RH I
CAS:Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Formula:C58H79N15O15Color and Shape:SolidMolecular weight:1226.34(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS:(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Formula:C53H62N12O11Molecular weight:1043.13Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).Formula:C44H80N14O15Molecular weight:1044.59276Bim 21009
CAS:Bim 21009 is an inhibitor of gonadorelin.Formula:C74H92ClN17O13Purity:98%Color and Shape:SolidMolecular weight:1463.08[D-Phe2,6, Pro3]-LH-RH
CAS:[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).Formula:C59H80N14O13Color and Shape:SolidMolecular weight:1193.35Human follicular gonadotropin releasing peptide
CAS:Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH)Formula:C68H94N22O27Color and Shape:SolidMolecular weight:1651.61Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Formula:C162H26N56O44SColor and Shape:SolidMolecular weight:3724.17Prolactin Releasing Peptide (1-31), human
CAS:Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).Formula:C160H252N56O42SPurity:98%Color and Shape:SolidMolecular weight:3664.15Surfagon
CAS:Surfagon is an effective LHRH agonist.Formula:C56H78N16O12Purity:98%Color and Shape:SolidMolecular weight:1167.34[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.Formula:C67H84N16O13Color and Shape:SolidMolecular weight:1321.48[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Formula:C54H71N15O14Purity:98%Color and Shape:SolidMolecular weight:1154.23Fsh receptor-binding inhibitor fragment(bi-10)
CAS:FSH antagonist bi-10 suppresses ovulation, induces follicular atresia, and may help in ovarian cancer by downregulating FSHR/ERβ.Formula:C42H67N13O19Color and Shape:SolidMolecular weight:1058.06Zebrafish Kisspeptin-1
CAS:Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.Formula:C58H84N16O15Color and Shape:SolidMolecular weight:1245.39GnRH Associated Peptide (1-24), human
CAS:GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.Formula:C117H190N32O43Color and Shape:SolidMolecular weight:2732.95LH-RH (7-10)
CAS:LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.Formula:C19H36N8O4Color and Shape:SolidMolecular weight:440.54(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:Analog of LHRH, stimulates LH and FSH release, controls reproduction.
Formula:C59H84N18O14Color and Shape:SolidMolecular weight:1269.41Kisspeptin-54(human) TFA
Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.Formula:C258H401N79O78·C2HF3O2Color and Shape:SolidMolecular weight:5971.45sGnRH-A
CAS:sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Formula:C64H83N17O12Color and Shape:SolidMolecular weight:1282.45Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Formula:C75H110N18O20·xC2HF3O2Purity:99.11%Color and Shape:SolidMolecular weight:1583.78 (free base)Kisspeptin 13
CAS:Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.Formula:C78H107N21O18Color and Shape:SolidMolecular weight:1626.81Azaline B
CAS:Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.Formula:C80H102ClN23O12Color and Shape:SolidMolecular weight:1613.27A 76154
CAS:A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).Formula:C70H93FN12O12Color and Shape:SolidMolecular weight:1313.584Wy 43657
CAS:Wy 43657 is a gonadorelin antagonist.Formula:C71H86N14O13Purity:98%Color and Shape:SolidMolecular weight:1343.554LUF5771
CAS:LUF5771: potent allosteric recLH & Org 43553 inhibitor, partial LH receptor activator with low efficacy.Formula:C24H23NO2Color and Shape:SolidMolecular weight:357.44Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Formula:C59H84N16O12Color and Shape:SolidMolecular weight:1209.4Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormula:C61H88N16O14Purity:98.1%Color and Shape:SolidMolecular weight:1269.45Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurity:98.64% - 99.97%Color and Shape:SolidMolecular weight:623.63Ref: TM-T3630
2mg39.00€5mg58.00€10mg93.00€25mg167.00€50mg250.00€100mg408.00€200mg585.00€1mL*10mM (DMSO)81.00€Sufugolix
CAS:Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.Formula:C36H31F2N5O4SPurity:97.78%Color and Shape:SolidMolecular weight:667.72Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formula:C23H31FO5Purity:99.47%Color and Shape:CoaMolecular weight:406.49Ref: TM-T21335
2mg44.00€5mg67.00€10mg96.00€25mg178.00€50mg261.00€100mg374.00€200mg494.00€1mL*10mM (DMSO)80.00€Fertirelin
CAS:Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).Formula:C55H76N16O12Purity:>99.99%Color and Shape:SolidMolecular weight:1153.29Ref: TM-TP1288
1mg47.00€2mg63.00€5mg96.00€10mg135.00€50mg177.00€100mg264.00€200mg393.00€1mL*10mM (DMSO)170.00€Cetrorelix diacetate
CAS:Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.Formula:C74H100ClN17O18Purity:98.38%Color and Shape:SolidMolecular weight:1551.17Ref: TM-T5520L
1mg52.00€5mg90.00€10mg150.00€25mg291.00€50mg437.00€100mg642.00€500mg1,359.00€1mL*10mM (DMSO)251.00€Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormula:C82H117ClN18O15Purity:96.05%Color and Shape:SolidMolecular weight:1630.4LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretionFormula:C61H78N18O16Purity:99.66%Color and Shape:SolidMolecular weight:1319.38Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formula:C68H90N18O14Purity:99.92%Color and Shape:SolidMolecular weight:1383.55Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)Formula:C66H87N17O14Purity:99.84%Color and Shape:SolidMolecular weight:1342.5Buserelin Acetate (57982-77-1 free base)
CAS:Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).Formula:C62H90N16O15Purity:99.31% - 99.78%Color and Shape:SolidMolecular weight:1299.48Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formula:C66H86N18O15Purity:99.59% - 99.90%Color and Shape:White PowderMolecular weight:1371.53Ref: TM-T21410
5mg52.00€10mg78.00€25mg119.00€50mg172.00€100mg259.00€200mg388.00€1mL*10mM (DMSO)116.00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:SolidMolecular weight:653.57Ref: TM-T5031
2mg35.00€5mg52.00€10mg80.00€25mg144.00€50mg227.00€100mg359.00€200mg532.00€1mL*10mM (DMSO)74.00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurity:99.33%Color and Shape:SolidMolecular weight:508.42Goserelin acetate
CAS:Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
Formula:C61H88N18O16Purity:99.77% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:1329.46Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Formula:C70H92ClN17O14·xC2H4O2Purity:97.96%Color and Shape:SolidMolecular weight:1491.11Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Formula:C55H74N16O13Color and Shape:SolidMolecular weight:1167.29Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Formula:C80H104ClN21O14Color and Shape:SolidMolecular weight:1619.27NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Formula:C27H24F3N3O3Color and Shape:SolidMolecular weight:495.49EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Formula:C15H27N5O6Color and Shape:SolidMolecular weight:373.4BAY 1214784
CAS:BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.Formula:C29H26ClF4N3O5S2Purity:100% - 99.77%Color and Shape:SolidMolecular weight:672.11Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurity:98.60% - 98.97%Color and Shape:SolidMolecular weight:544.5BAY-784
CAS:BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).
Formula:C29H26ClF4N3O5S2Purity:98%Color and Shape:SolidMolecular weight:672.115α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFormula:C21H36O2Color and Shape:SolidMolecular weight:320.51T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFormula:C37H37F2N3O4SPurity:98%Color and Shape:SolidMolecular weight:657.77BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Formula:C27H21ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:473.93DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Formula:C11H17Cl2NOSColor and Shape:SolidMolecular weight:282.22[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32Abarelix acetate
CAS:Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formula:C72H95ClN14O14·xC2H4O2Color and Shape:SolidMolecular weight:1476.14BAY-899
CAS:BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.Formula:C25H19F2N5O2Purity:98%Color and Shape:SolidMolecular weight:459.45(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Formula:C25H19F2N5O2Color and Shape:SolidMolecular weight:459.45GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Formula:C31H28F5N7O6SPurity:98%Color and Shape:SolidMolecular weight:721.65GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Formula:C28H27F2N9O5Purity:98.08%Color and Shape:SolidMolecular weight:607.57Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Formula:C80H102ClN15O14Color and Shape:SolidMolecular weight:1533.21Merigolix
CAS:Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Formula:C36H35F7N4O6Color and Shape:SolidMolecular weight:752.68Goserelin acetate(65807-02-5 Free base)
Goserelin acetate （ICI-118630 acetate） is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.
Purity:99.77%Color and Shape:Odour SolidRef: TM-T36918L
Discontinued productDimethandrolone Undecanoate
CAS:Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.Formula:C31H50O3Purity:99.65% - >99.99%Color and Shape:SolidMolecular weight:470.73Ref: TM-T27176
Discontinued product
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