HIV Protease
HIV Protease inhibitors are a class of antiretroviral drugs that specifically target the protease enzyme of the Human Immunodeficiency Virus (HIV). By inhibiting this enzyme, these compounds prevent the virus from processing its polyproteins into mature, functional proteins, thereby blocking the production of new infectious virions. HIV Protease inhibitors are a cornerstone of highly active antiretroviral therapy (HAART) used to manage HIV/AIDS. At CymitQuimica, we provide a variety of HIV Protease inhibitors to support your research in HIV treatment, drug resistance, and virology.
Found 505 products of "HIV Protease"
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Antitumor agent-191
Antitumor agent-191 (Compound 7) exhibits antiviral activity against HSV-1 and HIV, with EC50 values of 0.03 μM and 0.81 μM, respectively. It also demonstrates potential antitumor properties by inhibiting cancer cell lines HepG2, WI-38, Vero, and MCF-7, with IC50 values of 19.6, 39.3, 18.3, and 28 μM, respectively.Formula:C22H14N12S2Color and Shape:SolidMolecular weight:510.557Clathrin-IN-1
CAS:Pitstop 2 inhibits clathrin-mediated endocytosis, targeting clathrin's terminal domain, with potential in cancer research.
Formula:C20H13BrN2O3S2Purity:99.53%Color and Shape:SolidMolecular weight:473.36GP120, HIV-1 MN
GP120, HIV-1 MN, a peptide, is utilized in researching HIV infection [1] [2].Formula:C135H221N45O33Color and Shape:SolidMolecular weight:3002.5Cys-TAT(47-57) acetate(583836-55-9 Free base)
Cys-TAT(47-57) acetate is derived from the HIV-1 transactivating protein. Cys-TAT(47-57) acetate is an arginine rich peptide that can penetrate cells.Formula:C69H128N34O16SPurity:95.1100%Color and Shape:SolidMolecular weight:1722.04Schineolignin B
Schineolignin B is a useful organic compound for research related to life sciences and the catalog number is T126011.Formula:C22H30O5Color and Shape:SolidMolecular weight:374.477Elvucitabine
CAS:Elvucitabine, a reverse transcriptase inhibitor, is used potentially for the treatment of HBV infection and HIV infection.Formula:C9H10FN3O3Color and Shape:SolidMolecular weight:227.19Decanoyl-RVKR-CMK
CAS:Inhibits all seven proprotein convertases; stops proET-1 processing; hinders VGF secretion in PC12 cells.Formula:C34H66ClN11O5Purity:98%Color and Shape:SolidMolecular weight:744.42Diacetylsplenopentin HCl
CAS:Diacetylsplenopentin HCl, a synthetic immunomodulator, aids healthy bone marrow stem cell growth without triggering harmful immune reactions.Formula:C35H56ClN9O11Purity:98%Color and Shape:SolidMolecular weight:814.33Aureothin
CAS:Aureothin: a nitroaryl polyketide with antitumor, antifungal & insecticidal properties; inhibits NADH:oxidoreductase (IC50s: 0.07-22 nmol/mg).Formula:C22H23NO6Color and Shape:SolidMolecular weight:397.422-Hydroxyisoquinoline-1,3(2H,4H)-dione
CAS:Hydroxyisoquinoline-1,3(2H,4H)-dione (compound 6a) acts as an inhibitor of both HIV-1 integrase (IN) and HIV-1 reverse transcriptase ribonuclease H (RT RNase H), exhibiting IC50 values of 6.32 µM and 5.9 µM, respectively.Formula:C9H7NO3Color and Shape:SolidMolecular weight:177.16Isoquinoline
CAS:Compound PDK0035, with CAS No. 119-65-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0035 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C9H7NColor and Shape:Liquid OthersolidMolecular weight:129.15(±)-BI-D
CAS:(±)-BI-D is an effective ALLINI(An allosteric IN inhibitor) that binds integrase at the LEDGF/p75 binding site (IC50: 2.4–2.9 μM).Formula:C25H27NO4Color and Shape:SolidMolecular weight:405.49Dideoxyadenosine
CAS:2',3'-Dideoxyadenosine is an inhibitor of HIV replication with antiretroviral activity and antiviral efficacy [1].
Formula:C10H13N5O2Purity:99.28%Color and Shape:Physical Description Off-White Powder (Ntp 1992)Molecular weight:235.242'-Deoxy-2'-fluoroarabinoadenosine
CAS:2'-Deoxy-2'-fluoroarabinoadenosine is a nucleoside analogue with extensive anti-tumor activity and can be used for the study of tumor diseases.Formula:C10H12FN5O3Purity:99.95%Color and Shape:SolidMolecular weight:269.23Pseudothymidine
CAS:Pseudothymidine is a C-nucleoside analog of thymidine.Formula:C10H14N2O5Purity:98%Color and Shape:SolidMolecular weight:242.23TAT (48-57)
CAS:TAT (48-57) is a cell-permeable HIV-1 Tat protein fragment, amino acids 48-57.
Formula:C55H109N31O12Purity:98%Color and Shape:SolidMolecular weight:1396.65(Z)-9-Propenyladenine
CAS:(Z)-9-Propenyladenine is a mutagenic impurity in tenofovir disoproxil fumarate.Formula:C8H9N5Color and Shape:SolidMolecular weight:175.19Betulin diacetate
CAS:Betulin diacetate is a bioactive chemical.Formula:C34H54O4Color and Shape:SolidMolecular weight:526.8Tenofovir hydrate
CAS:Tenofovir hydrate (GS 1278 hydrate) is a nucleotide reverse transcriptase inhibitor with antiviral activity.Formula:C9H16N5O5PPurity:99.63%Color and Shape:SolidMolecular weight:305.23Etravirine D4
CAS:Etravirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used for the treatment of HIV. Etravirine D4 is the deuterium labeled Etravirine.Formula:C20H15BrN6OPurity:98%Color and Shape:SolidMolecular weight:439.3Saquinavir mesylate
CAS:Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapyFormula:C39H54N6O8SPurity:99.19%Color and Shape:White Or Pale Yellow PowderMolecular weight:766.9Abacavir hydroxyacetate
CAS:Abacavir hydroxyacetate is a nucleoside analog reverse transcriptase inhibitor used in the study of HIV infection.Formula:C16H20N6O3Purity:98.29%Color and Shape:SolidMolecular weight:344.37Cabotegravir sodium
CAS:Cabotegravir sodium inhibits HIV integrase (IC50: 2.5 nM), metabolized by UGT1A1, with minimal ARV interaction.Formula:C19H16F2N3NaO5Purity:99.63%Color and Shape:SolidMolecular weight:427.34PL 100
CAS:PL 100 could inhibit HIV-1 protease.Formula:C33H44N4O6SPurity:98%Color and Shape:SolidMolecular weight:624.79Pentosan Polysulfate Sodium (W/W 43%)
CAS:Pentosan Polysulfate Sodium: anti-HIV, anti-inflammatory, aids cartilage, treats interstitial cystitis.Purity:98%Color and Shape:SolidMolecular weight:N/ALoviride
CAS:Loviride, a reverse transcriptase inhibitor with IC50 of 0.3 μM, blocks HIV-1/2 and SIV in MT-4 cells.Formula:C17H16Cl2N2O2Color and Shape:SolidMolecular weight:351.23Cyclotriazadisulfonamide
CAS:Cyclotriazadisulfonamide (CADA) is a selective, CD4-targeted HIV and Sec61 inhibitor that downregulates CD4 T-cell receptors and restricts CD4 translocation.Formula:C31H39N3O4S2Purity:99.91% - 99.98%Color and Shape:SolidMolecular weight:581.799-Propenyladenine
CAS:9-Propenyladenine is a mutagenic impurity in tenofovir disoproxil fumarate.Formula:C8H9N5Color and Shape:SolidMolecular weight:175.19gardiquimod TFA salt
CAS:Gardiquimod diTFA is a TLR7/8 agonist that may block HIV-1 in macrophages and PBMCs, active under 10 μM.Formula:C21H25F6N5O5Color and Shape:SolidMolecular weight:541.44Ditiocarb sodium
CAS:Ditiocarb sodium (Sodium diethyldithiocarbamate) (sodium diethiocarbamate) is a copper reagent, which reacts with Cu2 + solution to form a complex and improvesFormula:C5H10NNaS2Purity:98.04%Color and Shape:White Solid CrystallineMolecular weight:171.26Doravirine
CAS:Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.Formula:C17H11ClF3N5O3Purity:99.65% - 99.79%Color and Shape:SolidMolecular weight:425.75Ref: TM-T3632
1mg50.00€2mg65.00€5mg92.00€10mg166.00€25mg318.00€50mg492.00€100mg710.00€500mg1,468.00€1mL*10mM (DMSO)124.00€Tenofovir alafenamide
CAS:Tenofovir alafenamide (GS-7340) is a nucleotide reverse transcriptase inhibitor (NRTI) and a novel ester prodrug of the antiretroviral tenofovir.Formula:C21H29N6O5PPurity:99.68% - 99.81%Color and Shape:SolidMolecular weight:476.47Lopinavir
CAS:Lopinavir (ABT-378) is a peptidomimetic HIV protease inhibitor that retains activity against HIV protease with the Val 82 mutation.Formula:C37H48N4O5Purity:98% - 99.62%Color and Shape:White Crystalline SolidMolecular weight:628.8Escin IA
CAS:Escin IA (Escin IA;Aescin IA) is a triterpene saponin isolated from horse chestnut, which inhibits HIV-1 protease with IC50 values of 35 μM.Formula:C55H86O24Purity:98.97% - 99.81%Color and Shape:SolidMolecular weight:1131.26Raltegravir sodium
CAS:Raltegravir (MK 0518) sodium is a potent, orally active HIV integrase (IN) inhibitor.Formula:C20H20FN6NaO5Color and Shape:SolidMolecular weight:466.405Didanosine
CAS:Didanosine (ddI) is a nucleoside reverse transcriptase inhibitor analog of adenosine (IC50: 0.49 μM).Formula:C10H12N4O3Purity:99.64%Color and Shape:White Crystalline PowderMolecular weight:236.23Darunavir
CAS:Darunavir (TMC114) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Formula:C27H37N3O7SPurity:99.67% - 99.76%Color and Shape:White Amorphous SolidMolecular weight:547.66Temsavir
CAS:Temsavir (BMS626529) is a novel attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T cells.Formula:C24H23N7O4Purity:99.14%Color and Shape:SolidMolecular weight:473.48Ref: TM-T4665
2mg39.00€5mg60.00€10mg92.00€25mg166.00€50mg278.00€100mg411.00€200mg578.00€1mL*10mM (DMSO)60.00€Peptide T acetate(106362-32-7 free base)
Peptide T acetate is an octapeptide from the V2 region of HIV-1 gp120.Formula:C37H59N9O18Purity:99.47%Color and Shape:SolidMolecular weight:917.91lavendustin B
CAS:Lavendustin B inhibits Tyrosine Kinase and HIV-1 integrase-LEDGF/p75 interaction.Formula:C21H19NO5Purity:95.72%Color and Shape:Off-White SolidMolecular weight:365.38Fosamprenavir sodium
CAS:Fosamprenavir sodium is an HIV protease inhibitor that is the water soluble prodrug of amprenavir.Formula:C25H34N3Na2O9PSColor and Shape:SolidMolecular weight:629.57Raltegravir
CAS:Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIVFormula:C20H21FN6O5Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:444.42BMS-707035
CAS:BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.Formula:C17H19FN4O5SPurity:99.78%Color and Shape:SolidMolecular weight:410.42Apelin-17 (human, bovine) acetate
Apelin-17 (human, bovine) acetate is an endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).Formula:C98H160N34O22SPurity:99.36%Color and Shape:SolidMolecular weight:2198.63I-XW-053 sodium
CAS:I-XW-053 sodium inhibits the replication of a diverse panel of primary HIV-1 isolates in Peripheral blood mononuclear cell with no appreciable cytotoxicity.Formula:C22H16N2NaO2Color and Shape:SolidMolecular weight:363.372Indinavir sulfate
CAS:Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.
Formula:C36H49N5O8SPurity:99.75% - >99.99%Color and Shape:White PowderMolecular weight:711.872,4-Dihydroxypyridine
CAS:2,4-Dihydroxypyridine: a pyridine derivative, chelates metals, assesses ion levels, measures enzymatic reactions, and quantifies biomolecules.Formula:C5H5NO2Purity:97.79%Color and Shape:White To Yellow-Beige Crystals OrMolecular weight:111.1Darunavir Ethanolate
CAS:Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.Formula:C29H43N3O8SPurity:99.84% - 99.86%Color and Shape:SolidMolecular weight:593.74Ref: TM-T3335
5mg37.00€10mg52.00€25mg80.00€50mg111.00€100mg165.00€200mg236.00€500mg399.00€1mL*10mM (DMSO)48.00€TAT
CAS:TAT peptide (YGRKKRRQRRR), originating from the human immunodeficiency virus-1 (HIV-1) transactivator of transcription (TAT), enhances the solubility and
Formula:C64H118N32O14Purity:>99.99%Color and Shape:SolidMolecular weight:1559.83
