Organometallic Ligands

<p>Antagonist of serotonin receptors 5-HT3</p>

<p>An active product of vitamin A metabolism. Activates RXR and RAR receptor isoforms with high binding affinity. Induces differentiation of neural stem cells into neurons.</p>

<p>Dopamine reuptake inhibitor</p>

<p>Apatinib, also known as rivoceranib, is an inhibitor of the vascular endothelial growth factor receptor 2 (VEGFR2) tyrosine kinase. Apatinib targets VEGFR2 with its action and has proven to have strong anti-tumor effects in human cancers. In studies in mice, apatinib acted as an Inhibitor of VEGFR2 and played an antiangiogenic effect. Apatinib has been suggested for the treatment of ischemia-induced proliferative retinopathy and neovascular age-related macular degeneration.</p>

<p>Inhibitor of Abl and Src kinases; anti-proliferative; antineoplasticÂ</p>

<p>Uricosuric agent</p>

<p>Aldose reductase AKR1B10 inhibitor; hepatotoxic</p>

<p>Inhibitor of CKD1, CDK2, and CDK4 serine/threonine kinases</p>

<p>C16(Plasm) LPC is a lysophosphatidylcholine, a type of lysophospholipid derived predominantly from plasma membrane phospholipids. It originates from the enzymatic action of phospholipase A2, which cleaves the fatty acid chain, typically at the sn-2 position. This leaves behind the lysophospholipid with a single acyl chain.</p>

<p>Angiotensin-converting enzyme inhibitor; anti-hypertensive</p>

<p>MG 132 is a modified tripeptide that acts as proteasomal inhibitor. In 2006, MG 132 has been experimentally tested in in vitro cell-based and in vivo models for to assess its use in the medical treatment of Parkinson's disease.</p>

<p>Synthetic antagonist of GnRH receptor</p>

<p>Histamine (H1) antagonist; used to treat allergies, rhinitis and urticaria</p>

<p>Anti-folate inhibitor of thymidylate synthase</p>

<p>Voxelotor is an oral therapeutic agent, which is a small molecule obtained through synthetic chemistry with targeted activity on hemoglobin. Its mode of action involves the allosteric modification of hemoglobin, specifically increasing hemoglobin oxygen affinity. By stabilizing the oxygenated hemoglobin state, voxelotor reduces the sickling and polymerization of red blood cells that are characteristic of sickle cell disease (SCD).</p>

<p>Please enquire for more information about Ceralifimod including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>

<p>Iron chelator</p>

<p>Angiotensin-converting enzyme inhibitor; antioxidant</p>

<p>Inhibits acetylcholinesterase (AChE); antispasmodic agent</p>

<p>Protective agent against mercuric chloride poisoning</p>