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Other Inhibitors

Other Inhibitors

This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.

Found 37926 products of "Other Inhibitors"

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  • ASP-8731

    CAS:
    <p>ASP8731 is a selective inhibitor of BACH1 that prevents inflammation and vascular occlusion, and induces fetal hemoglobin in sickle cell disease.</p>
    Formula:C20H21N5O4
    Color and Shape:Solid
    Molecular weight:395.41
  • Naphthablin

    CAS:
    <p>Naphthablin is a naphthoquinone compound that inhibits the function of the Abl oncogene. It prevents the morphological transformation of v-ablts-NIH3T3 cells induced by Abl and also suppresses RNA synthesis.</p>
    Formula:C29H36O8
    Color and Shape:Solid
    Molecular weight:512.591
  • Sannamycin K

    CAS:
    <p>Sannamycin K is an aminoglycoside antibiotic with weak antibacterial activity against both Gram-positive and Gram-negative bacteria.</p>
    Formula:C13H26N4O4
    Color and Shape:Solid
    Molecular weight:302.37
  • Tabimorelin hemifumarate

    CAS:
    <p>orally active ghrelin receptor (GHS-R1a) agonist</p>
    Formula:C32H40N403C4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:586.72
  • Dynemicin Q

    CAS:
    <p>Dynemicin Q is an antibiotic that demonstrates potent activity against Gram-positive bacteria.</p>
    Formula:C28H19NO9
    Color and Shape:Solid
    Molecular weight:513.45
  • KHK-IN-6

    CAS:
    <p>KHK-IN-6 (compound 33) acts as a KHK inhibitor with an IC50 of 0.6nM.</p>
    Formula:C23H24F3N5O2S
    Color and Shape:Solid
    Molecular weight:491.53
  • Cephemimycin

    CAS:
    <p>Cephemimycin exhibits mild antibacterial and antifungal activity.</p>
    Formula:C16H22N4O9S
    Color and Shape:Solid
    Molecular weight:446.432
  • BAY-850 HCl


    <p>BAY-850 is a selective probe targeting Atad2A's bromine domain, displacing acetylated H4 peptides and detaching ATAD2 from chromatin at 1μm.</p>
    Formula:C38H48Cl5N5O3
    Color and Shape:Solid
    Molecular weight:800.08
  • ALK5-IN-82

    CAS:
    <p>ALK5-IN-82 is a potent and selective inhibitor of activin receptor-like kinase 5 (ALK5), demonstrating an IC50 value of 9.1 nM. This compound effectively suppresses the expression of α-smooth muscle actin (α-SMA), collagen I, and the proteinases tissue inhibitor of metalloproteinase 1 (TIMP-1) and matrix metalloproteinase 13 (MMP-13) in human umbilical vein endothelial cells induced by transforming growth factor-β. ALK5-IN-82 shows potential for use in research related to cardiac fibrosis.</p>
    Formula:C22H19N7OS
    Color and Shape:Solid
    Molecular weight:429.50
  • Eurocidin E

    CAS:
    <p>Eurocidin E is an antibiotic that inhibits degranulation and histamine release from rat mast cells.</p>
    Formula:C40H61NO14
    Color and Shape:Solid
    Molecular weight:779.911
  • Glucoallosamidin A

    CAS:
    <p>Glucoallosamidin A is a glycoside antibiotic that inhibits chitinase activity. It effectively suppresses the chitinase enzyme in Candida albicans [ATCC 10231], exhibiting an IC50 of 3.4 μg/mL.</p>
    Formula:C26H44N4O14
    Color and Shape:Solid
    Molecular weight:636.646
  • Ezomycin D2

    CAS:
    <p>Ezomycin D2 is an antifungal antibiotic effective primarily against plant pathogens such as Sclerotinia sclerotiorum and Botrytis cinerea. It helps control diseases like sclerotinia blight and gray mold in crops, as well as candidiasis.</p>
    Formula:C19H27N5O14
    Color and Shape:Solid
    Molecular weight:549.443
  • Resorcinomycin A

    CAS:
    <p>Resorcinomycin A is an antibiotic with potent antimycobacterial activity and relatively weaker activity against mycoplasma.</p>
    Formula:C14H20N4O5
    Color and Shape:Solid
    Molecular weight:324.332
  • Chrymutasin B

    CAS:
    <p>Chrymutasin B is a glycoside antitumor antibiotic known for its cytotoxic properties.</p>
    Formula:C32H31NO13
    Color and Shape:Solid
    Molecular weight:637.587
  • Glyphosate-trimesium

    CAS:
    <p>Glyphosate-trimesium is a herbicide.</p>
    Formula:C6H16NO5PS
    Color and Shape:Solid
    Molecular weight:245.23
  • 6"'-Deamino-6"'-hydroxyparomomycin I

    CAS:
    <p>6"'-Deamino-6"'-hydroxyparomomycin I is an aminoglycoside antibiotic produced by Streptomyces rimosus forma paromomycinus A67 15, exhibiting activity against both Gram-positive and Gram-negative bacteria. It serves as an intermediate in the biosynthesis of paromomycin.</p>
    Formula:C23H44N4O15
    Color and Shape:Solid
    Molecular weight:616.613
  • Milbemycin β1

    CAS:
    <p>Milbemycin β1 is a macrolide antibiotic with insecticidal properties effective against agricultural pests, aphids, larvae, and others.</p>
    Formula:C32H48O7
    Color and Shape:Solid
    Molecular weight:544.719
  • Isohematinic acid

    CAS:
    <p>Isohematinic acid exhibits mild activity against anaerobic bacteria.</p>
    Formula:C8H9NO4
    Color and Shape:Solid
    Molecular weight:183.161
  • BMS-986120

    CAS:
    BMS-986120: Oral, reversible PAR4 antagonist. IC50: 9.5 nM (human), 2.1 nM (monkey). Potent, selective antiplatelet.
    Formula:C23H23N5O5S2
    Color and Shape:Solid
    Molecular weight:513.59
  • TRPC5-IN-4

    CAS:
    <p>TRPC5-IN-4: Potent, safe inhibitor; IC50 14.07 nM (TRPC5), 65 nM (TRPC4); non-toxic to liver/kidney cells; for CKD research.</p>
    Formula:C18H11ClF4N4O3
    Color and Shape:Solid
    Molecular weight:442.75
  • Cytochalasin F

    CAS:
    <p>Cytochalasin F reversibly inhibits cytokinesis and possesses various biological activities including the inhibition of macrophage endocytosis and exocytosis.</p>
    Formula:C29H37NO5
    Color and Shape:Solid
    Molecular weight:479.608
  • Furaquinocin A

    CAS:
    <p>Furaquinocin A has the ability to kill HeLa S3 and B16 melanoma cells, yet it lacks antibacterial activity.</p>
    Formula:C22H26O7
    Color and Shape:Solid
    Molecular weight:402.438
  • TCMDC-135051 TFA (2413716-15-9 free base)


    <p>TCMDC-135051 TFA is a highly selective and potent inhibitor of protein kinase PfCLK3.</p>
    Formula:C31H34F3N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:585.61
  • PLP_Snyder530


    <p>PLP_Snyder530, a potent PL pro inhibitor, halts SARS-CoV-2 by triggering protease conformation changes.</p>
    Formula:C24H24N2O2
    Color and Shape:Solid
    Molecular weight:372.46
  • S-2,3-Dicarboxyaziridine

    CAS:
    <p>S-2,3-Dicarboxyaziridine is a metabolite that can be isolated from Streptomyces species and exhibits antibacterial activity.</p>
    Formula:C4H5NO4
    Color and Shape:Solid
    Molecular weight:131.087
  • DXR-IN-3

    CAS:
    <p>DXR-IN-3 is an anti-Toxoplasma DXR inhibitor. It exhibits in vitro activity against the TgDXR enzyme, with an IC50 value of 0.62 μM and a Ki value of 0.19 μM. Furthermore, DXR-IN-3 can inhibit the proliferation of Toxoplasma, displaying an IC50 value of 5.46 μM.</p>
    Formula:C10H12Cl2NO5PS
    Color and Shape:Solid
    Molecular weight:360.15
  • FMK-MEA

    CAS:
    <p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>
    Formula:C21H26FN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.46
  • Fostriecin (free base)

    CAS:
    <p>Fostriecin inhibits PP2A/PP4 (IC50s = 3.2/3 nM), weakly affects topoisomerase II/PP1 (IC50s = 40/131 μM), doesn't inhibit PP2B, and may modify epigenetics.</p>
    Formula:C19H27O9P
    Color and Shape:Solid
    Molecular weight:430.39
  • Thielavin B

    CAS:
    <p>Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.</p>
    Formula:C31H34O10
    Color and Shape:Solid
    Molecular weight:566.6
  • O-GlcNAcase-IN-1


    <p>O-GlcNAcase-IN-1 is a potent and novel inhibitor of O-GlcNAcase(OGA) with an IC 50 value of 46 nM.</p>
    Formula:C15H22N6
    Color and Shape:Solid
    Molecular weight:286.38
  • XD23

    CAS:
    <p>XD23 is a potent osteosarcoma inhibitor that functions by downregulating DKK1 and activating the WNT/β-catenin signaling pathway.</p>
    Formula:C22H26ClN7O3
    Color and Shape:Solid
    Molecular weight:471.94
  • Atiratecan

    CAS:
    <p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>
    Formula:C31H34N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:586.64
  • Rivasterat

    CAS:
    <p>Rivasterat is a cholesterol-derived steroid known for its anti-inflammatory properties.</p>
    Formula:C37H54O8
    Color and Shape:Solid
    Molecular weight:626.82
  • Unoprostone

    CAS:
    <p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>
    Formula:C22H38O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.53
  • Pyriftalid

    CAS:
    <p>Pyriftalid is a novel insecticide known for its potent inhibitory activity against a variety of pests. It is widely utilized in agriculture to effectively manage crop pests, thereby enhancing both the yield and quality of crops. Additionally, research is exploring the use of Pyriftalid in boosting plant resistance to pests and diseases.</p>
    Formula:C15H14N2O4S
    Color and Shape:Solid
    Molecular weight:318.35
  • Hynapene A

    CAS:
    <p>Hynapene A exhibits an inhibitory minimum inhibitory concentration (MIC) of 123 μM against Eimeria tenella.</p>
    Formula:C18H28O5
    Color and Shape:Solid
    Molecular weight:324.412
  • HYL001

    CAS:
    <p>HYL001 (compound 338) is a potent inhibitor of the TGFβ receptor 1 (ALK5), exhibiting approximately nine times the efficacy of its structurally related counterpart, galunisertib, in eliminating liver metastasis tumors generated in mice.</p>
    Formula:C21H18N4O
    Color and Shape:Solid
    Molecular weight:342.39
  • GNE-616

    CAS:
    <p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>
    Formula:C24H23F4N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.53
  • GK241

    CAS:
    <p>GK241 (compound 31a-c), a 2-oxoamide-based compound, exhibits inhibitory activity against group IIA secretory phospholipase A2 (GIIA sPLA2) in humans and mice, with IC50 values of 143 nM and 68 nM, respectively. The mechanism of inhibition has been explored through molecular dynamics simulations.</p>
    Formula:C21H39NO4
    Color and Shape:Solid
    Molecular weight:369.54
  • NRX-2663

    CAS:
    <p>NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).</p>
    Formula:C20H13F3N2O5
    Color and Shape:Solid
    Molecular weight:418.32
  • KY-02327 acetate


    <p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>
    Formula:C22H31N3O6
    Color and Shape:Solid
    Molecular weight:433.5
  • Oral antiplatelet agent 1

    CAS:
    <p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>
    Formula:C23H24N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.53
  • hTrkA-IN-2


    <p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>
    Formula:C24H22F3N5O3
    Color and Shape:Solid
    Molecular weight:485.46
  • PEN-866

    CAS:
    <p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>
    Formula:C49H49N7O9
    Color and Shape:Solid
    Molecular weight:879.95
  • Hydroxyakalone

    CAS:
    <p>Hydroxyakalone is an inhibitor of the enzyme xanthine oxidase (XOD, EC 1.2.3.2) and has an IC50 of 4.6 μM for XOD.</p>
    Formula:C5H5N5O2
    Color and Shape:Solid
    Molecular weight:167.126
  • Fipronil desulfinyl

    CAS:
    <p>Fipronil desulfinyl, a photodegradation product of the insecticide Fipronil, exhibits similar in vivo toxicity to Fipronil and possesses higher environmental toxicity.</p>
    Formula:C12H4Cl2F6N4
    Color and Shape:Solid
    Molecular weight:389.08
  • Albicidin

    CAS:
    <p>Albicidin is a DNA gyrase inhibitor produced by Xanthomonas albilineans.</p>
    Formula:C44H38N6O12
    Color and Shape:Solid
    Molecular weight:842.818
  • Antitrypanosomal agent 6


    <p>Compound 18a: potent vs. T. brucei (IC50: 0.47 μM), &gt;2x efficacy compared to Nifurtimox, good ADME, binds AT-rich DNA.</p>
    Formula:C22H29Cl2N5O
    Color and Shape:Solid
    Molecular weight:450.4
  • Protease-Activated Receptor-1 antagonist 3


    <p>PAR-1 antagonist 3: potent (IC50: 7 nM), binds hERG K+ channels (IC50: 9 μM).</p>
    Formula:C30H34N4O3
    Color and Shape:Solid
    Molecular weight:498.62
  • Falecalcitriol

    CAS:
    <p>Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.</p>
    Formula:C27H38F6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:524.58
  • MRS2279

    CAS:
    <p>Selective, high affinity competitive antagonist of the P2Y1 receptor</p>
    Formula:C13H18ClN5O8P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.71
  • Tandutinib (MLN518) HCl


    <p>Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.</p>
    Formula:C31H43ClN6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:599.16
  • ETH 157

    CAS:
    <p>ETH 157 is a synthetic neutral carrier-based Na+ selective microelectrode, with sufficient selectivity against K+, Ca2+, and Mg2+ for extracellular measurement of Na+ activity.</p>
    Formula:C36H32N2O4
    Color and Shape:Solid
    Molecular weight:556.65
  • WS-898


    <p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>
    Formula:C33H25N7OS
    Color and Shape:Solid
    Molecular weight:567.66
  • Bagremycin B

    CAS:
    <p>Bagremycin B is produced by the bacterium Streptomyces strain Tu 4128. It exhibits weak activity against Gram-positive bacteria, Saccharomyces cerevisiae, and Candida albicans.</p>
    Formula:C17H15NO4
    Color and Shape:Solid
    Molecular weight:297.305
  • UNC7467

    CAS:
    <p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>
    Formula:C20H13NO3
    Purity:98.28% - 98.64%
    Color and Shape:Soild
    Molecular weight:315.32
  • Isobetanin

    CAS:
    <p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>
    Formula:C24H26N2O13
    Color and Shape:Solid
    Molecular weight:550.47
  • SPR-00305

    CAS:
    <p>SPR-00305 is a novel potent inhibitor of the mvfr pathway</p>
    Formula:C24H19ClN2O3
    Color and Shape:Solid
    Molecular weight:418.87
  • CHNQD-01255

    CAS:
    <p>CHNQD-01255 is an orally active inhibitor of Arf-GEFs that is effective against hepatocellular carcinoma (HCC).</p>
    Formula:C23H29NO6
    Color and Shape:Solid
    Molecular weight:415.48
  • Zetomipzomib

    CAS:
    <p>KZR-616: Immunoproteasome inhibitor targeting LMP7 (IC50: 39/57 nM) &amp; LMP2 (IC50: 131/179 nM), potential in autoimmune disease research.</p>
    Formula:C30H42N4O8
    Color and Shape:Solid
    Molecular weight:586.68
  • Citreamicin β

    CAS:
    <p>Citreamicin β exhibits activity against aerobic and anaerobic Gram-positive bacteria.</p>
    Formula:C35H29NO12
    Color and Shape:Solid
    Molecular weight:655.604
  • PARP1-IN-5


    <p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>
    Formula:C25H24N2O5S
    Color and Shape:Solid
    Molecular weight:464.53
  • Depsidomycin

    CAS:
    <p>Depsidomycin is an immunomodulatory antibiotic isolated from the culture broth of Streptomyces lavendofoliae MI951-62F2, exhibiting immunosuppressive properties. It primarily shows antibacterial activity against Gram-positive bacteria.</p>
    Formula:C38H65N9O9
    Color and Shape:Solid
    Molecular weight:791.978
  • L-Tyrosyl-L-glutamic acid

    CAS:
    <p>L-Tyrosyl-L-glutamic acid acts as an inhibitor of the amino acid permease GAP1.</p>
    Formula:C14H18N2O6
    Color and Shape:Solid
    Molecular weight:310.3
  • LK-732

    CAS:
    <p>LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.</p>
    Formula:C25H29N5O3S
    Color and Shape:Solid
    Molecular weight:479.59
  • PCSK9-IN-16

    CAS:
    <p>PCSK9-IN-16, holds potential for research into hypercholesterolemia and other cardiovascular diseases [1].</p>
    Formula:C16H20N6O2S3
    Color and Shape:Solid
    Molecular weight:424.56
  • Keap1-Nrf2-IN-1 TFA


    <p>Keap1-Nrf2-IN-1 TFA (compound35) is a potent inhibitor (IC50: 43 nM) protecting against acetaminophen liver damage.</p>
    Formula:C26H25F3N2O9S
    Color and Shape:Solid
    Molecular weight:598.54
  • Jietacin A

    CAS:
    <p>Jietacin A exhibits nematocidal activity, capable of killing Burs helenchus Lignicolus at a concentration of 0.25 μg/mL.</p>
    Formula:C18H34N2O2
    Color and Shape:Solid
    Molecular weight:310.475
  • Fredericamycin A

    CAS:
    <p>Fredericamycin A exhibits activity against gram-positive bacteria and fungi, demonstrating potent antitumor effects both in vivo and in vitro.</p>
    Formula:C30H21NO9
    Color and Shape:Solid
    Molecular weight:539.489
  • Erizepine

    CAS:
    <p>Erizepine, an octopamine receptor 3 (OAR3) antagonist, exhibits a Ki value of 474 nM. This compound is utilized in insect research.</p>
    Formula:C20H22N2
    Color and Shape:Solid
    Molecular weight:290.4
  • BE-10988

    CAS:
    <p>BE-10988 is a DNA topoisomerase (DNAtopoisomerase) inhibitor. It suppresses the growth of P388 murine leukemia cell lines that are resistant to Doxorubicin and Vinblastine by promoting the formation of DNA topoisomerase complexes.</p>
    Formula:C13H10N4O3S
    Color and Shape:Solid
    Molecular weight:302.31
  • 8,9-Epoxyeicosatrienoic acid

    CAS:
    <p>8,9-Epoxyeicosatrienoic acid offers unique protective effects on the glomerulus. It inhibits the increase in glomerular albumin permeability caused by circulating permeability factors (FSPF). Additionally, 8,9-Epoxyeicosatrienoic acid is used in research related to glomerular dysfunction.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.47
  • Glycocinnasperimicin D

    CAS:
    <p>Glycocinnasperimicin D is a glycoside cinnamoyl iminohistamine antibiotic. It exhibits activity against both Gram-positive and Gram-negative bacteria. Additionally, Glycocinnasperimicin D inhibits leukemia L1210 cells, with an IC50 of 2.0 μg/mL.</p>
    Formula:C30H50N10O9
    Color and Shape:Solid
    Molecular weight:694.78
  • Curromycin B

    CAS:
    <p>Curromycin B exhibits antibacterial activity against Gram-positive bacteria such as Bacillus subtilis. It also inhibits the replication of human immunodeficiency virus (HIV) and suppresses the proliferation of mouse melanoma B16 and leukemia P388 cells.</p>
    Formula:C37H53N3O9
    Color and Shape:Solid
    Molecular weight:683.831
  • Fluopsin F

    CAS:
    <p>Fibrostatin F is a metal-containing iron antibiotic with potent activity against Gram-positive and Gram-negative bacteria, as well as antitumor properties.</p>
    Formula:C6H12FeN3O3S3
    Color and Shape:Solid
    Molecular weight:326.218
  • Heparastatin

    CAS:
    <p>Heparastatin is an inhibitor of heparanase.</p>
    Formula:C8H11F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:272.18
  • Naphthoquinomycin A

    CAS:
    <p>Naphthoquinomycin A is an antibiotic that exhibits activity against Gram-positive bacteria and fungi, and also inhibits the synthesis of fatty acids in Escherichia coli.</p>
    Formula:C40H47NO10
    Color and Shape:Solid
    Molecular weight:701.802
  • Antiproliferative agent-3


    <p>Antiproliferative agent-3 (comp 4) exhibits potent growth inhibitory effects against MCF-7 cells with IC 50 of 0.19 nM [1].</p>
    Formula:C11H12N2O5S
    Color and Shape:Solid
    Molecular weight:284.29
  • Dechloromycorrhizin A

    CAS:
    <p>Dechloromycorrhizin A is an antibiotic with weak activity against Gram-positive bacteria, yeasts, and molds, but it exhibits strong nematocidal activity.</p>
    Formula:C14H16O4
    Color and Shape:Solid
    Molecular weight:248.274
  • AT1R antagonist 2


    <p>AT1R antagonist 2 is a potent AT1R selective ligand with good AT1R affinity (Ki: 26 nM).</p>
    Formula:C29H37N5O4S2
    Color and Shape:Solid
    Molecular weight:583.77
  • SIK1 activator 1

    CAS:
    <p>SIK1 activator 1 boosts SIK1 phosphorylation, reduces type 2 diabetes hyperglycemia, and inhibits liver gluconeogenesis.</p>
    Formula:C23H32O6
    Color and Shape:Solid
    Molecular weight:404.50
  • Granaticin

    CAS:
    <p>Granaticin A inhibits the initial stages of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, as well as tumor cells.</p>
    Formula:C22H20O10
    Color and Shape:Solid
    Molecular weight:444.388
  • PrCP-7414

    CAS:
    <p>PrCP-7414 is a potent PrCP inhibitor, CAS# 1252037-41-4, named after the CAS number's last four digits.</p>
    Formula:C31H33Cl2N5O2
    Color and Shape:Solid
    Molecular weight:578.53
  • MI-1851

    CAS:
    <p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>
    Formula:C34H53N15O6
    Color and Shape:Solid
    Molecular weight:767.88
  • Resolvin E4

    CAS:
    <p>RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.</p>
    Formula:C20H30O4
    Color and Shape:Solid
    Molecular weight:334.45
  • BMS-751324

    CAS:
    <p>BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.</p>
    Formula:C32H35N6O10P
    Color and Shape:Solid
    Molecular weight:694.63
  • ABCA1 inducer 1

    CAS:
    <p>ABCA1 inducer 1, a non-lipid inducer of ABCA1, enhances ABCA1 expression in E3/4FAD mice expressing human APOE 3/4, augments the lipidation of apolipoprotein (APOE), and reverses various Alzheimer's disease (AD) phenotypes without increasing triglycerides.</p>
    Formula:C24H24Cl2N2O7S2
    Color and Shape:Solid
    Molecular weight:587.49
  • Sovesudil hydrochloride


    <p>Sovesudil (PHP-201) HCl: potent local ROCK inhibitor; targets ROCK I/II (IC50: 3.7/2.3 nM); lowers IOP, non-congesting.</p>
    Formula:C23H23ClFN3O3
    Color and Shape:Solid
    Molecular weight:443.9
  • Macquarimicin A

    CAS:
    <p>Macquarimicin A is an antibiotic.</p>
    Formula:C19H22O5
    Color and Shape:Solid
    Molecular weight:330.375
  • Glucopiericidin B

    CAS:
    <p>Glucopiericidin B exhibits antibacterial activity.</p>
    Formula:C31H47NO9
    Color and Shape:Solid
    Molecular weight:577.706
  • AM-9514

    CAS:
    <p>AM-9514: a potent Glucokinase activator with strong in vitro results, good pharmacokinetics, and efficacy in diabetes.</p>
    Formula:C18H25N5O4
    Color and Shape:Solid
    Molecular weight:375.42
  • Epihygromycin

    CAS:
    <p>Epihygromycin is a glycoside antibiotic with relatively weak activity against Gram-positive bacteria.</p>
    Formula:C23H29NO12
    Color and Shape:Solid
    Molecular weight:511.476
  • AZD-3409

    CAS:
    <p>AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.</p>
    Formula:C34H41FN4O4S2
    Color and Shape:Solid
    Molecular weight:652.84
  • NA 382

    CAS:
    <p>NA 382 is a staurosporine derivative that inhibits multidrug resistance.</p>
    Formula:C31H28N4O6
    Color and Shape:Solid
    Molecular weight:552.58
  • PAD-IN-2

    CAS:
    <p>PAD-IN-2, potent PAD4 inhibitor, IC50 &lt;1 μM; targets autoimmune/cancer disorders.</p>
    Formula:C27H28ClN5O2
    Color and Shape:Solid
    Molecular weight:490
  • Heme Oxygenase-2-IN-1


    <p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>
    Formula:C19H17N3O2
    Color and Shape:Solid
    Molecular weight:319.36
  • Gusperimus

    CAS:
    <p>Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.</p>
    Formula:C17H37N7O3
    Color and Shape:Solid
    Molecular weight:387.52
  • Methylenomycin B

    CAS:
    <p>Methylenomycin B is a cyclopentanone-derived antibiotic effective against both Gram-negative and Gram-positive bacteria.</p>
    Formula:C8H10O
    Color and Shape:Solid
    Molecular weight:122.164
  • CL656

    CAS:
    <p>CL656 is a stimulator of interferon genes (STING) activator.</p>
    Formula:C20H21F2N9O9P2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:695.51
  • Anti-TSWV agent 1


    <p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>
    Formula:C22H27ClN4OS3
    Color and Shape:Solid
    Molecular weight:495.12
  • Agosterol A

    CAS:
    <p>Agosterol A is isolated from marine sponge Spongia.</p>
    Formula:C33H52O8
    Color and Shape:Solid
    Molecular weight:576.76
  • Alkannin

    CAS:
    <p>Alkannin: potent, tumor-specific PKM2 inhibitor; non-inhibitory to PKM1/PKL; potential anticancer agent.</p>
    Formula:C16H16O5
    Color and Shape:Solid
    Molecular weight:288.3
  • AM Toxin II

    CAS:
    <p>AM Toxin II is a Cyclic tetradepsipeptide isolated from Alternaria mali.</p>
    Formula:C22H29N3O5
    Color and Shape:Solid
    Molecular weight:415.49
  • ChemR23-IN-3


    <p>ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.</p>
    Formula:C31H33N5O5S2
    Color and Shape:Solid
    Molecular weight:619.75
  • Lactonamycin Z

    CAS:
    <p>Lactonamycin Z is an antitumor antibiotic with mild activity against Gram-positive bacteria and shows inhibitory effects on human tumor cells HMO2, MCF7, and Hep G2, with GI50 (μg/mL) values of 1.9, 0.85, and 5.11, respectively.</p>
    Formula:C28H27NO13
    Color and Shape:Solid
    Molecular weight:585.513
  • Anticancer agent 79


    <p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>
    Formula:C20H12F3NO5
    Color and Shape:Solid
    Molecular weight:403.31
  • Antitumor agent-47


    <p>Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.</p>
    Formula:C30H27NO11
    Color and Shape:Solid
    Molecular weight:577.54
  • GSK268


    <p>GSK268 is a BET inhibitor.</p>
    Formula:C26H27N5O3
    Color and Shape:Solid
    Molecular weight:457.53
  • Nothramicin

    CAS:
    <p>Nothramicin is an anthracycline antibiotic that exhibits antimycobacterial activity.</p>
    Formula:C30H37NO11
    Color and Shape:Solid
    Molecular weight:587.615
  • Resolvin E2

    CAS:
    <p>RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.</p>
    Formula:C20H30O4
    Color and Shape:Solid
    Molecular weight:334.45
  • Encephalitic alphavirus-IN-1


    <p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) &amp; EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>
    Formula:C27H25FN6O2
    Color and Shape:Solid
    Molecular weight:484.52
  • FCE-27262

    CAS:
    <p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>
    Formula:C23H31N3O3
    Color and Shape:Solid
    Molecular weight:397.51
  • MMP408

    CAS:
    <p>MMP408 acts as an inhibitor of MMP-12.</p>
    Formula:C19H20N2O7S
    Color and Shape:Solid
    Molecular weight:420.44
  • (±)-HIP-B

    CAS:
    <p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>
    Formula:C6H8N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:172.14
  • CI 922

    CAS:
    <p>CI 922 is an anaphylaxis mediator release inhibitor. It inhibits the activation of human neutrophils.</p>
    Formula:C26H30N10O6
    Color and Shape:Solid
    Molecular weight:578.58
  • Thalicarpine

    CAS:
    <p>Thalicarpine, a natural anticancer alkaloid, inhibits p-glycoprotein and induces DNA damage, arresting cell cycle.</p>
    Formula:C41H48N2O8
    Color and Shape:Solid
    Molecular weight:696.83
  • Tazide


    <p>Tazide is an antitumor agent [1].</p>
    Formula:C12H16N4O
    Color and Shape:Solid
    Molecular weight:232.28
  • CS-003 HCl

    CAS:
    <p>CS-003 HCl is a TNRA - triple neurokinin receptor antagonist.</p>
    Formula:C34H39Cl3N2O6S
    Color and Shape:Solid
    Molecular weight:710.1
  • KMN-80

    CAS:
    <p>KMN-80 is a potent, selective EP4 agonist with IC50 3 nM, spurring osteoblast differentiation, and showing in vivo bone repair efficacy.</p>
    Formula:C21H33NO4
    Color and Shape:Solid
    Molecular weight:363.49
  • NS2B/NS3-IN-4

    CAS:
    <p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>
    Formula:C15H11NO4
    Color and Shape:Solid
    Molecular weight:269.25
  • 18-Deoxyherboxidiene

    CAS:
    <p>18-Deoxyherboxidiene (RQN-18690A) inhibits angiogenesis, targeting SF3b in U2 snRNP spliceosome, affects HUVEC, useful for cancer research.</p>
    Formula:C25H42O5
    Color and Shape:Solid
    Molecular weight:422.6
  • CU-2010

    CAS:
    <p>CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.</p>
    Formula:C37H42N6O6S
    Color and Shape:Solid
    Molecular weight:698.83
  • SHR0687

    CAS:
    <p>SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.</p>
    Formula:C39H60N8O5
    Color and Shape:Solid
    Molecular weight:720.94
  • mPGES1-IN-4

    CAS:
    <p>mPGES1-IN-4 (compound 32) is a multi-substituted pyrimidine compound acting as a submicromolar inhibitor of PGE2 production. It primarily exerts its anti-inflammatory effects by inhibiting mPGES-1 and significantly suppresses acute inflammation models in vivo.</p>
    Formula:C27H25F2N3O
    Color and Shape:Solid
    Molecular weight:445.50
  • Mifepristone methochloride

    CAS:
    <p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>
    Formula:C30H38ClNO2
    Color and Shape:Solid
    Molecular weight:480.08
  • N-methyl Leukotriene C4

    CAS:
    <p>N-methyl LTC4 is a stable synthetic analog of LTC4 and a selective CysLT2 agonist, useful in studying leukotriene pharmacology.</p>
    Formula:C31H49N3O9S
    Color and Shape:Solid
    Molecular weight:639.8
  • CLR01 sodium

    CAS:
    <p>CLR01 is a tweezer reducing α-synuclein in MSA, inhibits SOD1 in ALS, blocks Ebola/Zika, stabilizes proteins, and lessens mutant p53 toxicity.</p>
    Formula:C42H30Na2O8P2
    Color and Shape:Solid
    Molecular weight:770.6211
  • AS1940477

    CAS:
    <p>AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.</p>
    Formula:C24H22FN5O2
    Color and Shape:Solid
    Molecular weight:431.46
  • Antimalarial agent 9


    <p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>
    Formula:C28H32BrN3O2
    Color and Shape:Solid
    Molecular weight:522.48
  • Aspochalasin M

    CAS:
    <p>Aspochalasin M shows moderate activity on HL-60 cells (IC50=20.0 μ M). Aspochalasin M has research potential in leukemia diseases.</p>
    Formula:C24H35NO4
    Color and Shape:Solid
    Molecular weight:401.54
  • NS2B/NS3-IN-5


    <p>Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.</p>
    Formula:C14H9IN2O3S
    Color and Shape:Solid
    Molecular weight:412.2
  • ATX inhibitor 12


    <p>Oral ATX inhibitor 12 (IC50: 1.72 nM) at 60 mg/kg prevents lung damage in C57Bl/6J mice.</p>
    Formula:C30H34FN5O2
    Color and Shape:Solid
    Molecular weight:515.62
  • AGN-204396

    CAS:
    <p>AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).</p>
    Formula:C32H44FN3O4
    Color and Shape:Solid
    Molecular weight:553.71
  • SARS-CoV-2-IN-8


    <p>SARS-CoV-2-IN-8 is a major protease inhibitor of SARS-CoV-2 (IC50: 0.75 μM).</p>
    Formula:C35H38N6O3
    Color and Shape:Solid
    Molecular weight:590.71
  • ORP-101

    CAS:
    <p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>
    Formula:C60H84N2O8
    Color and Shape:Solid
    Molecular weight:961.32
  • KT2-962

    CAS:
    <p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>
    Formula:C23H27ClNNaO5S2
    Color and Shape:Solid
    Molecular weight:520.04
  • KP 10614

    CAS:
    <p>KP 10614 is a new prostacyclin analog that inhibits platelet-polymorphonuclear leukocyte interaction.</p>
    Formula:C23H32O4
    Color and Shape:Solid
    Molecular weight:372.50
  • RIPK1-IN-26

    CAS:
    <p>RIPK1-IN-26 is a potent inhibitor of Receptor-Interacting Serine/Threonine Kinase 1 (RIPK1), exhibiting anti-necrotic properties in cells. This compound demonstrates good metabolic stability and binding specificity in mice. RIPK1-IN-26 holds potential for development as a PET imaging probe and in the research of neurodegenerative diseases.</p>
    Formula:C15H20FNO2
    Color and Shape:Solid
    Molecular weight:265.32
  • D-473

    CAS:
    <p>D-473 is a novel orally active triple reuptake inhibitor targeting dopamine, serotonin and norepinephrine transporters.</p>
    Formula:C26H27F2NO3
    Color and Shape:Solid
    Molecular weight:439.49
  • Neoenactin M2

    CAS:
    <p>Neoenactin M2 exhibits strong antifungal activity against yeasts and filamentous fungi.</p>
    Formula:C19H38N2O5
    Color and Shape:Solid
    Molecular weight:374.52
  • Hoe 892

    CAS:
    <p>Hoe 892 is a stable thia-thimo-analogue of prostacyclin and acts as a platelet aggregation inhibitor.</p>
    Formula:C20H33NO4S
    Color and Shape:Solid
    Molecular weight:383.55
  • Vitamin A Propionate

    CAS:
    <p>Vitamin A Propionate, an ester derivative of vitamin A, exhibits varying effects on growth, serum biochemistry, and hematological indices in foal nutrition studies depending on the dosage administered. Both excessively high and low doses lead to adverse impacts. These effects are correlated with the concentrations of vitamin A in the plasma, liver, and kidneys.</p>
    Formula:C23H34O2
    Color and Shape:Solid
    Molecular weight:342.51
  • Mf 268

    CAS:
    <p>Mf 268 is a pseudo-reversible carbamate-type inhibitor which interacts with the catalytic and regulatory anionic site of the enzyme.</p>
    Formula:C28H46N4O3
    Color and Shape:Solid
    Molecular weight:486.69
  • Ascofuranone

    CAS:
    <p>Ascofuranone is an inhibitor of the ubiquinol oxidase activity of Trypanosoma brucei mitochondrial alternative oxidase (TAO), as well as an inhibitor of HsDHODH</p>
    Formula:C23H29ClO5
    Color and Shape:Solid
    Molecular weight:420.93
  • RORγt Inverse agonist 2

    CAS:
    <p>RORγt Inverse agonist 2 is a selective, orally active inverse agonist of RORγt(EC50 of 119 nM).</p>
    Formula:C27H25F8NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:627.54
  • Everafenib


    <p>Everafenib: potent BRAF inhibitor, crosses blood-brain barrier, hinders MAPK, effective on V600EBRAF cells, outperforms other drugs in trials.</p>
    Formula:C20H23ClFN5O2S2
    Color and Shape:Solid
    Molecular weight:484.01
  • CYP11B1-IN-2


    <p>CYP11B1-IN-2 selectively inhibits human and rat CYP11B1 (IC50: 9/25 nM) orally to research cortisol-related diseases.</p>
    Color and Shape:Solid
  • 5α-reductase-IN-1

    CAS:
    <p>5α-reductase-IN-1 is a potent inhibitor of the enzyme 5α-reductase.</p>
    Formula:C31H37NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:503.63
  • PPARγ agonist 2


    <p>PPARγ agonist 2 is a highly effective compound that acts as a partial agonist for PPARγ.</p>
    Formula:C24H20O5
    Color and Shape:Solid
    Molecular weight:388.41
  • MurB-IN-1


    <p>MurB-IN-1 (compound 44) inhibits key bacterial enzyme MurB with 3.57 μM affinity, offering treatment potential against P. aeruginosa.</p>
    Formula:C12H7Cl2F3N2O2
    Color and Shape:Solid
    Molecular weight:339.1
  • PARP-1-IN-1


    <p>PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.</p>
    Formula:C23H25FN4O
    Color and Shape:Solid
    Molecular weight:392.47
  • PF-06815345 hydrochloride

    CAS:
    <p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>
    Formula:C27H30Cl2FN9O4
    Color and Shape:Solid
    Molecular weight:634.49
  • Malioxamycin

    CAS:
    <p>Malioxamycin is an antibiotic that inhibits Gram-negative bacteria by suppressing peptidoglycan synthesis in the bacterial cell wall and promoting the formation of protoplasts.</p>
    Formula:C9H16N2O6
    Color and Shape:Solid
    Molecular weight:248.233
  • BDZ-h

    CAS:
    <p>BDZ-h inhibits both closed/open states of all 4 homomeric &amp; 2 GluA2R-complex AMPA receptors.</p>
    Formula:C21H21N5O3S
    Color and Shape:Solid
    Molecular weight:423.49
  • PPARγ agonist 1


    <p>PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.</p>
    Formula:C34H39NO3
    Color and Shape:Solid
    Molecular weight:509.68
  • DG013A

    CAS:
    <p>DG013A inhibits ERAP1 &amp; ERAP2 (IC50: 33 nM &amp; 11 nM) to research autoimmune diseases &amp; cancer.</p>
    Formula:C27H37N4O4P
    Color and Shape:Solid
    Molecular weight:512.58
  • Tembotrione

    CAS:
    <p>Tembotrione is a chemical compound that may reduce the productivity of carrots. It possesses activity that degrades the quality of carrot stems. Additionally, Tembotrione can be used in studies focusing on the overall productivity of carrot cultivation.</p>
    Formula:C17H16ClF3O6S
    Color and Shape:Solid
    Molecular weight:440.82
  • DGY-08-097

    CAS:
    <p>DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.</p>
    Formula:C60H76N10O14
    Color and Shape:Solid
    Molecular weight:1161.3
  • T-3861174

    CAS:
    <p>T-3861174 is a prolyl tRNA synthetase (PRS) inhibitor, exhibiting significant in vitro anti-tumor activity with GCN2-ATF4 pathway activation.</p>
    Formula:C26H25FN6O2
    Color and Shape:Solid
    Molecular weight:472.51
  • Dihydrokainic acid

    CAS:
    <p>EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake</p>
    Formula:C10H17NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:215.25
  • Irinotecan Carboxylate Sodium Salt

    CAS:
    <p>Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.</p>
    Formula:C33H39N4NaO7
    Color and Shape:Solid
    Molecular weight:626.68
  • ER272

    CAS:
    <p>ER272 is a natural PKC activator, inducing hippocampal neurogenesis.</p>
    Formula:C24H34O6
    Color and Shape:Solid
    Molecular weight:418.52
  • CGS 22652

    CAS:
    <p>CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.</p>
    Formula:C22H29ClN2O4S
    Color and Shape:Solid
    Molecular weight:452.99
  • IDX-320

    CAS:
    <p>IDX-320 is an HCV protease inhibitor.</p>
    Formula:C37H43F3N6O7S2
    Color and Shape:Solid
    Molecular weight:804.9
  • G12Si-1


    <p>G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.</p>
    Formula:C29H32ClN5O3
    Color and Shape:Solid
    Molecular weight:534.05
  • H 218-54

    CAS:
    <p>H 218-54 is a renin inhibitor.</p>
    Formula:C37H56N2O5S
    Color and Shape:Solid
    Molecular weight:640.92
  • P2X receptor-1


    <p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>
    Formula:C14H14ClN3O3S2
    Color and Shape:Solid
    Molecular weight:371.86
  • Lobaric acid

    CAS:
    <p>Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.</p>
    Formula:C25H28O8
    Color and Shape:Solid
    Molecular weight:456.48
  • XN methyl pyrazole


    <p>XN methyl pyrazole exhibits beneficial effects on diet-induced obesity and enhances energy expenditure in mice fed with a high-fat diet [1].</p>
    Formula:C22H24N2O4
    Color and Shape:Solid
    Molecular weight:380.44
  • ZK168281

    CAS:
    <p>ZK168281 is a 1α,25(OH)2D3 analog, VDR antagonist with 0.1 nM Kd, and blocks receptor CoA interaction.</p>
    Formula:C32H46O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.70
  • eIF4A3-IN-6

    CAS:
    <p>eIF4A3-IN-6 is a potent eIF4A inhibitor, potentially used for treating eIF4A-related diseases like cancer. (US20170145026A1)</p>
    Formula:C26H25N3O5
    Color and Shape:Solid
    Molecular weight:459.49
  • Cicaprost

    CAS:
    <p>Cicaprost (ZK 96480) is an IP agonist with artery relaxing effects; EC50 is 5.8 nM.</p>
    Formula:C22H30O5
    Color and Shape:Solid
    Molecular weight:374.47
  • AP-6

    CAS:
    AP-6, a selective TMEM175 inhibitor, enhances lysosomal macromolecular catabolism by acutely inhibiting TMEM175, thus speeding up macrophage and other digestive activities. This compound holds potential for use in Parkinson's disease research due to its role in modulating lysosomal function.
    Formula:C16H14N4
    Color and Shape:Solid
    Molecular weight:262.31
  • PNU-140457

    CAS:
    <p>PNU-140457 is a bio-active chemical.</p>
    Formula:C14H14FN5O3
    Color and Shape:Solid
    Molecular weight:319.29
  • FTI-2148

    CAS:
    <p>FTI-2148 blocks RAS-related FT-1 &amp; GGT-1; IC50: 1.4 nM &amp; 1.7 μM.</p>
    Formula:C24H28N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.57
  • Plumbemycin A

    CAS:
    <p>Plumbemycin A is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>
    Formula:C12H20N3O9P
    Color and Shape:Solid
    Molecular weight:381.28
  • GRPR antagonist-1


    <p>GRPR antagonist-1 targets GRPR, kills specific cancer cells (e.g., PC3, Pan02, HGC-27), and promotes apoptosis by modulating Bcl-2 and Bax.</p>
    Formula:C29H33F3N4O4
    Color and Shape:Solid
    Molecular weight:558.59
  • SCP1-IN-2


    <p>SCP1-IN-2: potent, selective SCP1 inhibitor; induces REST degradation, hinders its activity, may study REST-driven glioblastoma growth.</p>
    Formula:C19H17F3N2O6S2
    Color and Shape:Solid
    Molecular weight:490.47
  • UH 301

    CAS:
    <p>UH 301 is a 5-HT1A receptor antagonist.</p>
    Formula:C16H24FNO
    Color and Shape:Solid
    Molecular weight:265.37
  • DC41

    CAS:
    <p>DC41 is a CC-1065-based cancer drug, an antibody-linked DNA alkylator.</p>
    Formula:C37H34ClN5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:680.22
  • DLCI-1

    CAS:
    <p>DLCI-1 is a potent and selective oral inhibitor of cytochrome P450 2A6 (CYP2A6), significantly reducing self-administered nicotine doses in both male and female mice.</p>
    Formula:C12H14N2S
    Color and Shape:Solid
    Molecular weight:218.32
  • Theophylline EP impurity C

    CAS:
    <p>Theophylline EP impurity C, an alkaloid with anti-bronchospasm activity, is employed to assess the purity and quality of compounds. This substance also holds potential clinical value in the management of asthma and chronic obstructive pulmonary disease (COPD).</p>
    Formula:C7H10N4O3
    Color and Shape:Solid
    Molecular weight:198.18
  • VEGFR-2-IN-17


    <p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>
    Formula:C21H14ClN3O2
    Color and Shape:Solid
    Molecular weight:375.81
  • Propizepine

    CAS:
    <p>Propizepine is a tricyclic antidepressant compound.</p>
    Formula:C17H20N4O
    Color and Shape:Solid
    Molecular weight:296.37
  • 2,4-Diaminoanisole

    CAS:
    <p>2,4-Diaminoanisole is a carcinogenic aromatic primary amine compound.</p>
    Formula:C7H10N2O
    Color and Shape:Solid
    Molecular weight:138.17
  • Terfluranol

    CAS:
    <p>Terfluranol, a benzyl derivative, is utilized as an antitumor medication.</p>
    Formula:C17H17F3O2
    Color and Shape:Solid
    Molecular weight:310.31
  • 5-Fluoroorotic acid monohydrate

    CAS:
    <p>5-Fluoroorotic acid (monohydrate) (5-Fluorouracil-6-carboxylic acid Mono(hydrate); 5-FOA) is employed to detect the expression of the URA3 gene in yeast molecular genetic constructs. Yeast possessing an active URA3 gene (which encodes orotidine-5'-monophosphate decarboxylase) convert 5-FOA into 5-fluorodeoxyuridine, a substance toxic to cells. Yeast strains with mutations in the URA3 gene that confer resistance can grow in the presence of 5-FOA if uracil is added to the medium.</p>
    Formula:C5H5FN2O5
    Color and Shape:Solid
    Molecular weight:192.10
  • Porphine

    CAS:
    <p>Porphine (Porphyrin), the parent compound of the porphyrin family, plays a crucial role within biological systems.</p>
    Formula:C20H14N4
    Color and Shape:Solid
    Molecular weight:310.35
  • 2,3-Dimethoxy-4-(methylthio)benzeneethanamine

    CAS:
    <p>2,3-Dimethoxy-4-(methylthio)benzeneethanamine (compound 22) is an analog of methoxybenzothiazine, employed in researching pharmacological agents that model human psychiatric disorders.</p>
    Formula:C11H17NO2S
    Color and Shape:Solid
    Molecular weight:227.32
  • Copper(II) ionophore I

    CAS:
    Copper(II) ionophore I is an active compound.
    Formula:C26H44N2S4
    Color and Shape:Solid
    Molecular weight:512.90
  • Ledene

    CAS:
    <p>Ledene (Viridiflorene) is an essential oil produced by viridiflorene synthase.</p>
    Formula:C15H24
    Purity:98%
    Color and Shape:Solid
    Molecular weight:204.35
  • U 80215

    CAS:
    <p>U 80215 is an enzyme-competitive inhibitor.</p>
    Formula:C42H60N8O6S
    Color and Shape:Solid
    Molecular weight:805.04
  • Anti-inflammatory agent 23


    <p>Anti-inflammatory agent 23 blocks LPS-induced NO (IC50: 0.449 μM) and binds p65 well.</p>
    Formula:C34H49NO6
    Color and Shape:Solid
    Molecular weight:567.76
  • Henagliflozin

    CAS:
    <p>Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.</p>
    Formula:C22H24ClFO7
    Color and Shape:Solid
    Molecular weight:454.87
  • FCE-24379

    CAS:
    <p>FCE-24379 is a selective antagonist of vascular serotonin receptors that has been shown to lowers blood pressure in hypertensive rats.</p>
    Formula:C20H22N4O2
    Color and Shape:Solid
    Molecular weight:350.41
  • Dimesna free acid

    CAS:
    <p>Dimesna (BNP-778), when used in conjunction with active cancer chemotherapy agents, can reduce the toxicity associated with uremia.</p>
    Formula:C4H10O6S4
    Color and Shape:Solid
    Molecular weight:282.38
  • Xylarianaphthol-1

    CAS:
    <p>Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.</p>
    Formula:C16H20BrFN2O2
    Color and Shape:Solid
    Molecular weight:371.24
  • Diarylalkane derivative 1

    CAS:
    <p>Diarylalkane derivative 1 is used for the research of pancreatitis.</p>
    Formula:C34H51NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.77
  • GLS1 Inhibitor-5


    <p>GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.</p>
    Color and Shape:Solid
  • NTPDase-IN-1


    <p>NTPDase-IN-1 selectively inhibits NTPDases 1, 2, 8 with IC50 of 0.05, 0.23, 0.54 μM. Non-competitive, K m 21 μM, used in cancer, immune, infection research.</p>
    Formula:C18H25N3OS2
    Color and Shape:Solid
    Molecular weight:363.54