G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
GTS-21 dihydrochloride
CAS:156223-05-1
GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by …
Formula:
C19H20N2O2·2HCl
Purity:
100% - 99.62%
Color and Shape:
Solid
Molecular weight:
381.3
Ref: TM-T2663
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 213.00 € | ||
| 200mg | 320.00 € | ||
| 500mg | 532.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Clorprenaline hydrochloride
CAS:6933-90-0
Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.
Formula:
C11H17Cl2NO
Purity:
100% - 98.65%
Color and Shape:
Solid
Molecular weight:
250.16
Ref: TM-T0248
| 25mg | 39.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 75.00 € | ||
| 200mg | 94.00 € | ||
| 500mg | 157.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Roluperidone
CAS:359625-79-9
Roluperidone (CYR-101) is a novel cyclic amide derivative.
Formula:
C22H23FN2O2
Purity:
96.46% - 97.77%
Color and Shape:
Solid
Molecular weight:
366.43
Ref: TM-T15034
| 1mg | 36.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 369.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Aripiprazole Lauroxil
CAS:1259305-29-7
Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.
Formula:
C36H51Cl2N3O4
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
660.71
Ref: TM-T14319
| 10mg | 48.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 127.00 € | ||
| 200mg | 184.00 € | ||
| 500mg | 312.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Molindone hydrochloride
CAS:15622-65-8
Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking …
Formula:
C16H24N2O2·HCl
Purity:
99% - 99.93%
Color and Shape:
Solid
Molecular weight:
312.84
Ref: TM-T0716
| 10mg | 35.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 64.00 € | ||
| 100mg | 86.00 € | ||
| 500mg | 174.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Fexofenadine hydrochloride
CAS:138452-21-8
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor …
Formula:
C32H40ClNO4
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
538.12
Ref: TM-T1470L
| 10mg | 50.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 104.00 € | ||
| 100mg | 138.00 € | ||
| 200mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Azatadine dimaleate
CAS:3978-86-7
Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
Formula:
C28H30N2O8
Purity:
100% - 99.70%
Color and Shape:
Powder
Molecular weight:
522.55
Ref: TM-T0236
| 25mg | 46.00 € | ||
| 50mg | 65.00 € | ||
| 100mg | 95.00 € | ||
| 200mg | 138.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Dipivefrin hydrochloride
CAS:64019-93-8
Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of …
Formula:
C19H27NO5·HCl
Purity:
99.22% - 99.92%
Color and Shape:
Less Gas With A Sweet Odor Colorless Gas With A Sweet Odor
Molecular weight:
387.9
Ref: TM-T0103
| 25mg | 51.00 € | ||
| 50mg | 82.00 € | ||
| 100mg | 112.00 € | ||
| 200mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
JMV 2959 hydrochloride (925238-89-7 free base)
CAS:2448414-54-6
JMV 2959 hydrochloride (925238-89-7 free base) is a growth hormone secretagogue receptor type 1a (GHS-R1a) …
Formula:
C30H33ClN6O2
Purity:
98.09%
Color and Shape:
Liquid
Molecular weight:
545.08
Ref: TM-T11719
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 547.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
6-Iodopravadoline
CAS:164178-33-0
6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity …
Formula:
C23H25IN2O3
Purity:
99.86%
Color and Shape:
Off-White Solid
Molecular weight:
504.36
Ref: TM-T14204
| 1mg | 40.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 539.00 € | ||
| 1mL*10mM (DMSO) | 104.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
LIT-001
CAS:2245072-21-1
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin …
Formula:
C30H34F3N7O4S
Purity:
96.88% - 98.25%
Color and Shape:
Solid
Molecular weight:
645.7
Ref: TM-T11857
| 1mg | 71.00 € | ||
| 5mg | 154.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 437.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 917.00 € | ||
| 500mg | 1,789.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Cisatracurium besylate
CAS:96946-42-8
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.
Formula:
C53H72N2O12·2C6H5O3S
Purity:
99.57% - ≥95%
Color and Shape:
White Or White Powder Category
Molecular weight:
1243.48
Ref: TM-T1459
| 10mg | 46.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 176.00 € | ||
| 200mg | 260.00 € | ||
| 500mg | 443.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Motixafortide TFA(664334-36-5,Free)
Motixafortide TFA is a CXCR4 antagonist with ~1 nM IC50, promoting AML apoptosis by modulating …
Formula:
C99H145F4N33O21S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
2273.54
Ref: TM-T14665L
| 1mg | 72.00 € | ||
| 5mg | 182.00 € | ||
| 10mg | 272.00 € | ||
| 25mg | 435.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 817.00 € | ||
| 200mg | 1,080.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Proglumide
CAS:6620-60-6
Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal …
Formula:
C18H26N2O4
Purity:
99.44%
Color and Shape:
White Crystalline Powder
Molecular weight:
334.41
Ref: TM-T1052
| 25mg | 39.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 117.00 € | ||
| 500mg | 182.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Vincamine
CAS:1617-90-9
Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain …
Formula:
C21H26N2O3
Purity:
99.52%
Color and Shape:
White To Almost White Fine Crystalline Powder
Molecular weight:
354.44
Ref: TM-T1286
| 1g | 66.00 € | ||
| 500mg | 53.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Vapreotide acetate
CAS:849479-74-9
Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).
Formula:
C59H74N12O11S2
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
1191.42
Ref: TM-T13306L
| 1mg | 35.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 495.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Venlafaxine hydrochloride
CAS:99300-78-4
Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.
Formula:
C17H28ClNO2
Purity:
99.69%
Color and Shape:
White Crystalline Powder
Molecular weight:
313.863
Ref: TM-T0472
| 5mg | 38.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 83.00 € | ||
| 100mg | 100.00 € | ||
| 200mg | 166.00 € | ||
| 500mg | 256.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Carebastine
CAS:90729-42-3
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
Formula:
C32H37NO4
Purity:
99.06%
Color and Shape:
Off-White Solid
Molecular weight:
499.64
Ref: TM-T10680
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 407.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Dimenhydrinate
CAS:523-87-5
Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
Formula:
C24H28ClN5O3
Purity:
99.57% - 99.77%
Color and Shape:
Crystals Physical Description Crystalline White Powder (Ntp 1992)
Molecular weight:
469.96
Ref: TM-T0298
| 1g | 95.00 € | ||
| 100mg | 36.00 € | ||
| 200mg | 52.00 € | ||
| 500mg | 75.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Fluphenazine dihydrochloride
CAS:146-56-5
Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used …
Formula:
C22H28Cl2F3N3OS
Purity:
100%
Color and Shape:
Off-White Solid
Molecular weight:
510.44
Ref: TM-T0068
| 50mg | 55.00 € | ||
| 100mg | 61.00 € | ||
| 200mg | 86.00 € | ||
| 500mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
