G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Aripiprazole
CAS:129722-12-9
Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
Formula:
C23H27Cl2N3O2
Purity:
99.43% - 99.62%
Color and Shape:
Colourless Flake Crystalline Solid
Molecular weight:
448.39
Ref: TM-T1566
| 1g | 133.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 84.00 € | ||
| 500mg | 101.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Azatadine dimaleate
CAS:3978-86-7
Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
Formula:
C28H30N2O8
Purity:
100% - 99.70%
Color and Shape:
Powder
Molecular weight:
522.55
Ref: TM-T0236
| 25mg | 47.00 € | ||
| 50mg | 66.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 140.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Triflupromazine hydrochloride
CAS:1098-60-8
Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.
Formula:
C18H20ClF3N2S
Purity:
99.73% - 99.73%
Color and Shape:
Crystals
Molecular weight:
388.88
Ref: TM-T0302
| 25mg | 39.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 92.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Terazosin hydrochloride
CAS:63074-08-8
Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.
Formula:
C19H26ClN5O4
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
423.89
Ref: TM-T0197
| 50mg | 44.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 89.00 € | ||
| 500mg | 135.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Olopatadine hydrochloride
CAS:140462-76-6
Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in …
Formula:
C21H23NO3·HCl
Purity:
100% - 99.78%
Color and Shape:
White Solid
Molecular weight:
373.87
Ref: TM-T1170
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 163.00 € | ||
| 500mg | 264.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Loxapine succinate
CAS:27833-64-3
Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.
Formula:
C22H24ClN3O5
Purity:
99.92%
Color and Shape:
White To Of-White Solid
Molecular weight:
445.9
Ref: TM-T1412
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 84.00 € | ||
| 500mg | 164.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Trimipramine maleate
CAS:521-78-8
Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.
Formula:
C24H30N2O4
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
410.51
Ref: TM-T1045
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 74.00 € | ||
| 500mg | 110.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Pericyazine
CAS:2622-26-6
Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.
Formula:
C21H23N3OS
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
365.49
Ref: TM-T16472
| 1mg | 46.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 389.00 € | ||
| 100mg | 567.00 € | ||
| 500mg | 1,225.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Droperidol
CAS:548-73-2
Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as …
Formula:
C22H22FN3O2
Purity:
97.16% - 98%
Color and Shape:
Solid
Molecular weight:
379.43
Ref: TM-T0990
| 100mg | 47.00 € | ||
| 200mg | 60.00 € | ||
| 500mg | 89.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Mianserin hydrochloride
CAS:21535-47-7
Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce …
Formula:
C18H21ClN2
Purity:
99.63% - 99.82%
Color and Shape:
White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film Coated
Molecular weight:
300.83
Ref: TM-T0783
| 1g | 157.00 € | ||
| 50mg | 35.00 € | ||
| 100mg | 42.00 € | ||
| 500mg | 106.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Dimenhydrinate
CAS:523-87-5
Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
Formula:
C24H28ClN5O3
Purity:
99.57% - 99.77%
Color and Shape:
Crystals Physical Description Crystalline White Powder (Ntp 1992)
Molecular weight:
469.96
Ref: TM-T0298
| 1g | 97.00 € | ||
| 100mg | 37.00 € | ||
| 200mg | 52.00 € | ||
| 500mg | 77.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
MRGPRX1 agonist 1
CAS:2377379-39-8
MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).
Formula:
C23H21N3O4S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
435.5
Ref: TM-T12104
| 1mg | 88.00 € | ||
| 5mg | 210.00 € | ||
| 10mg | 338.00 € | ||
| 25mg | 612.00 € | ||
| 50mg | 838.00 € | ||
| 100mg | 1,198.00 € | ||
| 1mL*10mM (DMSO) | 233.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Tolazoline hydrochloride
CAS:59-97-2
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of …
Formula:
C10H13ClN2
Purity:
100%
Color and Shape:
Pale Yellow Crystalline Solid
Molecular weight:
196.68
Ref: TM-T1680
| 1g | 48.00 € | ||
| 5g | 90.00 € | ||
| 10g | 131.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Proglumide
CAS:6620-60-6
Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal …
Formula:
C18H26N2O4
Purity:
99.4% - 99.44%
Color and Shape:
White Crystalline Powder
Molecular weight:
334.41
Ref: TM-T1052
| 25mg | 39.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 118.00 € | ||
| 500mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Carbazochrome sodium sulfonate
CAS:51460-26-5
Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.
Formula:
C10H11N4NaO5S
Purity:
99.8%
Color and Shape:
Orange Yellow Crystalline Powder
Molecular weight:
322.03
Ref: TM-T0852
| 25mg | 35.00 € | ||
| 50mg | 65.00 € | ||
| 100mg | 96.00 € | ||
| 500mg | 221.00 € | ||
| 1mL*10mM (DMSO) | 40.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
CP-809101 hydrochloride
CAS:1215721-40-6
CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A …
Formula:
C15H18Cl2N4O
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
341.24
Ref: TM-T10871
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 107.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 432.00 € | ||
| 100mg | 652.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Dopexamine hydrochloride
CAS:86484-91-5
Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting …
Formula:
C22H34Cl2N2O2
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
429.42
Ref: TM-T11318
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 528.00 € | ||
| 100mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Nylidrin hydrochloride
CAS:849-55-8
Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast …
Formula:
C19H26ClNO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
335.87
Ref: TM-T0173
| 1g | 283.00 € | ||
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 69.00 € | ||
| 200mg | 97.00 € | ||
| 500mg | 188.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Venlafaxine hydrochloride
CAS:99300-78-4
Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.
Formula:
C17H28ClNO2
Purity:
99.69%
Color and Shape:
White Crystalline Powder
Molecular weight:
313.863
Ref: TM-T0472
| 5mg | 38.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 79.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 164.00 € | ||
| 500mg | 264.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Amantadine hydrochloride
CAS:665-66-7
Amantadine hydrochloride (CI-719) is an antiviral that is used in the prophylactic or symptomatic treatment …
Formula:
C10H18ClN
Purity:
99.86%
Color and Shape:
Solid Crystalline
Molecular weight:
187.71
Ref: TM-T1406
| 1g | 39.00 € | ||
| 5g | 57.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
