G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 1ml | 51.00 € | ||
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 218.00 € | ||
| 200mg | 326.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Olanzapine
CAS:132539-06-1
Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia …
Formula:
C17H20N4S
Purity:
100% - 99.92%
Color and Shape:
Yellowish Crystalline Powder
Molecular weight:
312.43
Ref: TM-T1567
| 1ml | 51.00 € | ||
| 25mg | 40.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 87.00 € | ||
| 500mg | 133.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
ML-109
CAS:1186649-91-1
ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
Formula:
C31H29N3O5
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
523.58
Ref: TM-T12073
| 1ml | 51.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 326.00 € | ||
| 200mg | 455.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ritodrine hydrochloride
CAS:23239-51-2
Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing …
Formula:
C17H21NO3·HCl
Purity:
99% - 99.89%
Color and Shape:
Solid
Molecular weight:
323.82
Ref: TM-T1433
| 1ml | 55.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 106.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Midodrine hydrochloride
CAS:3092-17-9
Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a …
Formula:
C12H19ClN2O4
Purity:
99.06% - 99.36%
Color and Shape:
Crystalline Solid
Molecular weight:
290.74
Ref: TM-T1577
| 1ml | 51.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 274.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Itopride hydrochloride
CAS:122892-31-3
Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.
Formula:
C20H27ClN2O4
Purity:
99.76%
Color and Shape:
White Or Pale Brownish Crystal
Molecular weight:
394.9
Ref: TM-T1552
| 1ml | 51.00 € | ||
| 50mg | 41.00 € | ||
| 100mg | 54.00 € | ||
| 500mg | 85.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Amitraz
CAS:33089-61-1
Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine …
Formula:
C19H23N3
Purity:
99.62%
Color and Shape:
White/Pale Yellow Crystalline Solid
Molecular weight:
293.41
Ref: TM-T1632
| 1g | 51.00 € | ||
| 1ml | 34.00 € | ||
| 500mg | 38.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
CYM50308
CAS:1345858-76-5
CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).
Formula:
C20H21F2N3O2S
Purity:
99.43% - 99.63%
Color and Shape:
Solid
Molecular weight:
405.46
Ref: TM-T15032
| 1mg | 39.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 263.00 € | ||
| 100mg | 345.00 € | ||
| 200mg | 487.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Carebastine
CAS:90729-42-3
Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.
Formula:
C32H37NO4
Purity:
99.06%
Color and Shape:
Off-White Solid
Molecular weight:
499.64
Ref: TM-T10680
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 407.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ramatroban
CAS:116649-85-5
Ramatroban (BAY u3405) (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
Formula:
C21H21FN2O4S
Purity:
98.12% - 99.96%
Color and Shape:
Crystalline Solid
Molecular weight:
416.47
Ref: TM-T2396
| 1ml | 63.00 € | ||
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 268.00 € | ||
| 200mg | 347.00 € | ||
| 500mg | 587.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Bromperidol
CAS:10457-90-6
Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.
Formula:
C21H23BrFNO2
Purity:
99.89%
Color and Shape:
Tan Solid
Molecular weight:
420.32
Ref: TM-T14830
| 1ml | 36.00 € | ||
| 10mg | 43.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Prochlorperazine Maleate
CAS:84-02-6
Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; …
Formula:
C28H32ClN3O8S
Purity:
99.99%
Color and Shape:
Off-White Powder
Molecular weight:
606.09
Ref: TM-T0385
| 1ml | 46.00 € | ||
| 25mg | 45.00 € | ||
| 50mg | 54.00 € | ||
| 100mg | 71.00 € | ||
| 200mg | 114.00 € | ||
| 500mg | 207.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Fipexide
CAS:34161-24-5
Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy …
Formula:
C20H21ClN2O4
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
388.84
Ref: TM-T0322
| 1ml | 55.00 € | ||
| 25mg | 36.00 € | ||
| 50mg | 48.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 81.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Deoxycholic acid
CAS:83-44-3
Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.
Formula:
C24H40O4
Purity:
99.35%
Color and Shape:
Crystals From Alc Solid
Molecular weight:
392.57
Ref: TM-T2965
| 1ml | 63.00 € | ||
| 100mg | 57.00 € | ||
| 500mg | 78.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Monomethyl fumarate
CAS:2756-87-8
Monomethyl fumarate is a potent agonist of GPR109A .
Formula:
C5H6O4
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
130.1
Ref: TM-T12095
| 1ml | 51.00 € | ||
| 500mg | 50.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Sodium butanoate
CAS:156-54-7
Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity.
Formula:
C4H7NaO2
Purity:
98.02% - 99.44%
Color and Shape:
White Powder
Molecular weight:
110.09
Ref: TM-T1393
| 1g | 52.00 € | ||
| 5g | 93.00 € | ||
| 10g | 139.00 € | ||
| 500mg | 38.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
(R)-Terazosin
CAS:109351-34-0
R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 …
Formula:
C19H25N5O4
Purity:
98.87% - 98.96%
Color and Shape:
Solid
Molecular weight:
387.43
Ref: TM-T12643
| 1mg | 46.00 € | ||
| 1ml | 105.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 484.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Friday 4 Oct 2024
Seltorexant
CAS:1293281-49-8
Seltorexant (JNJ-42847922) crosses the blood-brain barrier and quickly occupies OX2R binding sites in the rat …
Formula:
C21H22FN7O
Purity:
100% - 99.86%
Color and Shape:
Solid
Molecular weight:
407.44
Ref: TM-T12877L
| 1mg | 37.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 149.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 369.00 € | ||
| 500mg | 853.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Sertraline hydrochloride
CAS:79559-97-0
Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the …
Formula:
C17H18Cl3N
Purity:
99.12% - 99.86%
Color and Shape:
Solid Powder
Molecular weight:
342.691
Ref: TM-T0482
| 1ml | 57.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 101.00 € | ||
| 50mg | 176.00 € | ||
| 100mg | 230.00 € | ||
| 200mg | 298.00 € | ||
| 500mg | 507.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
CE3F4
CAS:143703-25-7
CE3F4 is a selective antagonist of exchange protein directly activated by cAMP (Epac1; IC50s of …
Formula:
C11H10Br2FNO
Purity:
97% - 97.15%
Color and Shape:
Solid
Molecular weight:
351.01
Ref: TM-T12616L
| 1ml | 57.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 273.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
