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G-protein Coupled Receptors and 7-TM Receptors

G-protein Coupled Receptors and 7-TM Receptors

G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.

Found 5708 products of "G-protein Coupled Receptors and 7-TM Receptors"

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  • CYM 50769
    Targetmol
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    CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Formula:C24H17ClN2O3
    Purity:98% - 99.08%
    Color and Shape:Solid
    Molecular weight:416.86

    Ref: TM-T22702

  • Urocortin (rat) acetate
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    Urocortin (rat) acetate

    Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
    Purity:97.76%
    Color and Shape:Soild

    Ref: TM-TP1020L

  • AH 6809
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Formula:C17H14O5
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:298.29

    Ref: TM-T14148

  • Indacaterol maleate
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    Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Formula:C28H32N2O7
    Purity:99.03% - 99.67%
    Color and Shape:Solid
    Molecular weight:508.56

    Ref: TM-T1239

  • Ticlopidine hydrochloride
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    Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Formula:C14H15Cl2NS
    Purity:99.85% - >99.99%
    Color and Shape:White Powder
    Molecular weight:300.25

    Ref: TM-T0362

  • Rimonabant
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purity:98% - 99.91%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:463.79

    Ref: TM-T1519L

  • Quetiapine hemifumarate
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    Quetiapine hemifumarate

    CAS:
    Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.
    Formula:C46H54N6O8S2
    Purity:99.32% - >99.99%
    Color and Shape:White Crystalline Solid
    Molecular weight:883.09

    Ref: TM-T6241

  • Fexofenadine hydrochloride
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    Fexofenadine hydrochloride

    CAS:
    Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with
    Formula:C32H40ClNO4
    Purity:>99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:538.12

    Ref: TM-T1470L

  • Filorexant
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    Filorexant

    CAS:
    Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).
    Formula:C24H25FN4O2
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:420.48

    Ref: TM-T16096

  • Bufotenidine hydrochloride(487-91-2 Free base)
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    Bufotenidine hydrochloride(487-91-2 Free base)

    CAS:
    <p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>
    Formula:C13H19ClN2O
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:254.76

    Ref: TM-TN7062L

  • Ondansetron hydrochloride dihydrate
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    Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Formula:C18H19N3O·HCl·2H2O
    Purity:99.92%
    Color and Shape:White Crystal Powder
    Molecular weight:365.86

    Ref: TM-T1478

  • ML-180
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    ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Formula:C20H25ClN4O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:388.89

    Ref: TM-T12075

  • Blonanserin
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    Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Formula:C23H30FN3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:367.5

    Ref: TM-T1180

  • Zolmitriptan
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    Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formula:C16H21N3O2
    Purity:99.69% - 99.91%
    Color and Shape:White Or Kind Of White Powder
    Molecular weight:287.36

    Ref: TM-T1092

  • Aripiprazole
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    Aripiprazole

    CAS:
    Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
    Formula:C23H27Cl2N3O2
    Purity:99.43% - 99.62%
    Color and Shape:Colourless Flake Crystalline Solid
    Molecular weight:448.39

    Ref: TM-T1566

  • hGPR91 antagonist 1
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    hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Formula:C31H23F4N3O
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:529.53

    Ref: TM-T11560

  • Clonidine hydrochloride
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    Clonidine hydrochloride

    CAS:
    Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
    Formula:C9H10Cl3N3
    Purity:99.16% - 99.86%
    Color and Shape:Solid
    Molecular weight:266.55

    Ref: TM-T1247

  • Metaproterenol hemisulfate
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    Metaproterenol hemisulfate

    CAS:
    Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
    Formula:C11H17NO3·5H2O4S
    Purity:98.53% - 99.74%
    Color and Shape:Solid
    Molecular weight:260.3

    Ref: TM-T0277

  • Silodosin
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    Silodosin

    CAS:
    Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
    Formula:C25H32F3N3O4
    Purity:99.282% - 99.76%
    Color and Shape:Colorless To Pink Solid
    Molecular weight:495.53

    Ref: TM-T1504

  • Rimonabant hydrochloride
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    Rimonabant hydrochloride

    CAS:
    <p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂， Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>
    Formula:C22H22Cl4N4O
    Purity:98.24% - 99.5%
    Color and Shape:Off-White To White Crystalline Powder
    Molecular weight:500.25

    Ref: TM-T1519

  • Talastine
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    Talastine

    CAS:
    Talastine is an antihistamine compound that can induce an allergic rash.
    Formula:C19H21N3O
    Purity:99.44% - 99.84%
    Color and Shape:Solid
    Molecular weight:307.39

    Ref: TM-T68150

  • Olinciguat
    Targetmol
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    Olinciguat

    CAS:
    Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.
    Formula:C21H16F5N7O3
    Purity:99.33% - 99.71%
    Color and Shape:Solid
    Molecular weight:509.39

    Ref: TM-T16383

  • Terlipressin Acetate
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    Terlipressin Acetate

    CAS:
    Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).
    Formula:C56H82N16O19S2
    Purity:98.50% - 99.69%
    Color and Shape:Solid
    Molecular weight:1347.5

    Ref: TM-T13920L

  • Noradrenaline bitartrate
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    Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purity:99.53% - >99.99%
    Color and Shape:Solid
    Molecular weight:337.28

    Ref: TM-T0871

  • Fluparoxan hydrochloride
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H11ClFNO2
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:231.65

    Ref: TM-T77565

  • Ziprasidone
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    Ziprasidone

    CAS:
    <p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>
    Formula:C21H21ClN4OS
    Purity:99.55%
    Color and Shape:Tan Solid
    Molecular weight:412.94

    Ref: TM-T0031L2

  • YNT-185
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    YNT-185

    CAS:
    YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,
    Formula:C33H37N5O5S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:615.74

    Ref: TM-T39229

  • Senktide acetate
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    Senktide acetate

    <p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>
    Formula:C42H59N7O13S
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:902.02

    Ref: TM-T7633L

  • Azatadine dimaleate
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    Azatadine dimaleate

    CAS:
    <p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>
    Formula:C28H30N2O8
    Purity:99.7% - >99.99%
    Color and Shape:Powder
    Molecular weight:522.55

    Ref: TM-T0236

  • Nylidrin hydrochloride
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    Nylidrin hydrochloride

    CAS:
    Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.
    Formula:C19H26ClNO2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:335.87

    Ref: TM-T0173

  • (3aR,9aR)-Fluparoxan
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    (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H10FNO2
    Purity:97.82%
    Color and Shape:Soild
    Molecular weight:195.19

    Ref: TM-T77566

  • Phenothiazine
    Targetmol
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    Phenothiazine

    CAS:
    Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.
    Formula:C12H9NS
    Purity:99.95%
    Color and Shape:Yellow Solid Pellets
    Molecular weight:199.27

    Ref: TM-T0776

  • BIBO3304 TFA
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    BIBO3304 TFA

    CAS:
    BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).
    Formula:C31H36F3N7O5
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:643.66

    Ref: TM-T10539

  • (±) Clopidogrel hydrogen sulfate
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    (±) Clopidogrel hydrogen sulfate

    CAS:
    (±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots
    Formula:C16H16ClNO2S·H2SO4
    Purity:98.67% - 99.04%
    Color and Shape:Colorless To Light Yellow Liquid
    Molecular weight:419.9

    Ref: TM-T0182L2

  • Levodropropizine
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    Levodropropizine

    CAS:
    Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
    Formula:C13H20N2O2
    Purity:99.87% - 99.93%
    Color and Shape:White Or Off White Crystalline Powder
    Molecular weight:236.31

    Ref: TM-T0217

  • Trimipramine maleate
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    Trimipramine maleate

    CAS:
    Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.
    Formula:C24H30N2O4
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:410.51

    Ref: TM-T1045

  • Roxatidine Acetate hydrochloride
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    Roxatidine Acetate hydrochloride

    CAS:
    Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.
    Formula:C19H29ClN2O4
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:384.9

    Ref: TM-T0157

  • CP-809101 hydrochloride
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    CP-809101 hydrochloride

    CAS:
    <p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>
    Formula:C15H18Cl2N4O
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:341.24

    Ref: TM-T10871

  • Bromopride
    Targetmol
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    Bromopride

    CAS:
    Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.
    Formula:C14H22BrN3O2
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:344.25

    Ref: TM-T1175

  • Agomelatine
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    Agomelatine

    CAS:
    Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
    Formula:C15H17NO2
    Purity:99.92%
    Color and Shape:White Solid
    Molecular weight:243.3

    Ref: TM-T1445

  • Dimenhydrinate
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    Dimenhydrinate

    CAS:
    Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
    Formula:C24H28ClN5O3
    Purity:99.57% - 99.77%
    Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Molecular weight:469.96

    Ref: TM-T0298

  • Protriptyline hydrochloride
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    Protriptyline hydrochloride

    CAS:
    <p>Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.</p>
    Formula:C19H21N·HCl
    Purity:98.54% - 99.98%
    Color and Shape:Solid
    Molecular weight:299.84

    Ref: TM-T0204

  • Antazoline hydrochloride
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    Antazoline hydrochloride

    CAS:
    Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous
    Formula:C17H19N3·HCl
    Purity:98% - 99.53%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:301.82

    Ref: TM-T0092

  • CymitQuimica logo
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    Indusatumab

    CAS:
    <p>Indusatumab (5F9 Monoclonal antibody) is an anti-human GUCY2C (Guanylate cyclase 2C) monoclonal antibody that can be used to synthesize antibody-drug conjugate.</p>
    Purity:> 95% - > 95%
    Color and Shape:Liquid
    Molecular weight:145.18 kDa

    Ref: TM-T76769

  • Levosulpiride
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    Levosulpiride

    CAS:
    Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.
    Formula:C15H23N3O4S
    Purity:98.20% - 99.88%
    Color and Shape:White Crystalline Powder
    Molecular weight:341.43

    Ref: TM-T1211

  • Cefaclor monohydrate
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    Cefaclor monohydrate

    CAS:
    <p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>
    Formula:C15H16ClN3O5S
    Purity:97.36% - 99.9%
    Color and Shape:White Crystaling Powder
    Molecular weight:385.82

    Ref: TM-T1495

  • Trazodone hydrochloride
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    Trazodone hydrochloride

    CAS:
    <p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>
    Formula:C19H23Cl2N5O
    Purity:99.5% - 99.52%
    Color and Shape:Solid
    Molecular weight:408.33

    Ref: TM-T1619

  • Fezolinetant
    Targetmol
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    Fezolinetant

    CAS:
    <p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>
    Formula:C16H15FN6OS
    Purity:98.62% - 99.7%
    Color and Shape:Solid
    Molecular weight:358.39

    Ref: TM-T15278

  • Salmeterol
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    Salmeterol

    CAS:
    Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
    Formula:C25H37NO4
    Purity:99.2% - 99.9%
    Color and Shape:Solid
    Molecular weight:415.57

    Ref: TM-T12829

  • Carbetapentane citrate
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    Carbetapentane citrate

    CAS:
    Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.
    Formula:C20H31NO3·C6H8O7
    Purity:99.46%
    Color and Shape:White To Off-White Solid
    Molecular weight:525.59

    Ref: TM-T0464